Canal calcique
Les canaux calciques sont des protéines membranaires qui régulent le flux d'ions calcium dans et hors des cellules, ce qui est essentiel pour diverses fonctions cellulaires, y compris la contraction musculaire, la libération de neurotransmetteurs et l'expression génique. La dysrégulation de l'activité des canaux calciques est associée à des conditions telles que l'hypertension, les arythmies cardiaques et les troubles neurologiques. Chez CymitQuimica, nous proposons une large sélection de modulateurs des canaux calciques pour soutenir vos recherches en santé cardiovasculaire, neurobiologie et transduction du signal.
493 produits trouvés pour "Canal calcique"
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Nifedipine
CAS :<p>Nifedipine (Procardia) is a dihydropyridine calcium channel blocking agent.</p>Formule :C17H18N2O6Degré de pureté :99.39% - 99.49%Couleur et forme :Yellow Crystals Physical Description Odorless Yellow Crystals Or Powder Tasteless (Ntp 1992)Masse moléculaire :346.33Nitrendipine
CAS :<p>Nitrendipine is a vasodilating calcium channel blocker and antihypertensive that preserves kidney function and promotes sodium excretion.</p>Formule :C18H20N2O6Degré de pureté :99% - 99.55%Couleur et forme :SolidMasse moléculaire :360.36BMS-195270
CAS :<p>BMS-195270 is a bio-active chemical.</p>Formule :C15H9ClF3N3O2Degré de pureté :98.7%Couleur et forme :SolidMasse moléculaire :355.7Norverapamil hydrochloride
CAS :<p>Norverapamil HCl, a Verapamil metabolite, blocks L-type calcium channels and inhibits P-gp function.</p>Formule :C26H37ClN2O4Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :477.04Cav 2.2 blocker 1
CAS :<p>Cav 2.2 blocker 1 is an N-type calcium channel (Cav 2.2; IC50: 1 nM) blocker for the treatment of pain.</p>Formule :C25H29ClN2O2Degré de pureté :99.44%Couleur et forme :SolidMasse moléculaire :424.96ML-9
CAS :<p>ML-9 suppresses MLCK, PKA, and PKC activity with Ki values of 4, 32, and 54 μM, respectively.</p>Formule :C15H18Cl2N2O2SDegré de pureté :99.69%Couleur et forme :Crystalline SolidMasse moléculaire :361.29Cilnidipine
CAS :<p>Cilnidipine (FRC-8653)(FRC8653) is a dual L- and N-type calcium channel blocker and displays antihypertensive, sympatholytic and neuroprotective activity.</p>Formule :C27H28N2O7Degré de pureté :98.85% - 99.83%Couleur et forme :Yellow Crystalline SolidMasse moléculaire :492.52CRAC intermediate 1
CAS :<p>CRAC intermediate 1 (5-(S)-Fluorowillardiine) is a key intermediate in the chemical synthesis of a series of CRAC channel inhibitors.</p>Formule :C10H7F2N3ODegré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :223.18Ca2+ channel agonist 1
CAS :<p>Ca2+ channel agonist 1 activates N-type Ca2+ channels and inhibits Cdk2 (EC50: 14.23 μM/3.34 μM) for motor nerve issues.</p>Formule :C19H26N6ODegré de pureté :97.71%Couleur et forme :SolidMasse moléculaire :354.45L-Ascorbic acid
CAS :<p>L-Ascorbic acid (Vitamin C) is a natural product that is a potent reducing agent and antioxidant.</p>Formule :C6H8O6Degré de pureté :99.85% - 99.89%Couleur et forme :Crystals (Usually Plates Sometimes Needles Mon°Clinic System) Taste Almost Odorless (Ntp 1992)Masse moléculaire :176.12Nisoldipine
CAS :<p>Nisoldipine (BAY-k 5552) is a dihydropyridine calcium channel antagonist that acts as a potent arterial vasodilator and antihypertensive agent.</p>Formule :C20H24N2O6Degré de pureté :98.79% - 99.57%Couleur et forme :SolidMasse moléculaire :388.41Felodipine
CAS :<p>Felodipine (CGH-869) is a longlasting 1, 4-dihydropyridine calcium channel repressor.</p>Formule :C18H19Cl2NO4Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :384.25Fendiline hydrochloride
CAS :<p>Fendiline hydrochloride (Fendiline HCl) is a non-selective blocker of calcium channel.</p>Formule :C23H26ClNDegré de pureté :98.76% - 99.75%Couleur et forme :SolidMasse moléculaire :351.91Ethosuximide
CAS :<p>Ethosuximide (Zarontin) is an anticonvulsant, blocks the low voltage-activated T-type calcium channel used in the treatment of absence seizures unaccompanied by</p>Formule :C7H11NO2Degré de pureté :98.87% - 99.72%Couleur et forme :Crystals From Acetone And Ether SolidMasse moléculaire :141.17Manidipine dihydrochloride
CAS :<p>Manidipine dihydrochloride (Manidipine 2HCl) is a potent calcium channel blocker for Ca2+ current(IC50=2.6 nM).</p>Formule :C35H40Cl2N4O6Degré de pureté :99.76% - 99.86%Couleur et forme :SolidMasse moléculaire :683.62Lercanidipine
CAS :<p>Lercanidipine (Masnidipine) is a calcium channel blocker of the dihydropyridine class.</p>Formule :C36H41N3O6Degré de pureté :99.92%Couleur et forme :White To Light Yellow SolidMasse moléculaire :611.73GV-58
CAS :<p>GV-58 agonizes N/P-Q-type Ca2+ channels (EC50: 7.21/8.81 μM) with 20x less inhibition on CDK kinases.</p>Formule :C18H26N6OSDegré de pureté :97.36%Couleur et forme :SolidMasse moléculaire :374.5Lacidipine
CAS :<p>Lacidipine (SN-305) is a slow-acting, long-duration lipophilic dihydropyridine calcium blocker that prevents reflex tachycardia and lowers blood pressure.</p>Formule :C26H33NO6Degré de pureté :99.98%Couleur et forme :White-To-Off-White Crystalline SolidMasse moléculaire :455.545,5-Dimethyloxazolidine-2,4-dione
CAS :<p>5,5-Dimethyloxazolidine-2,4-dione (Dimethadione) is an anticonvulsant that is the active metabolite of TRIMETHADIONE.</p>Formule :C5H7NO3Degré de pureté :99.12%Couleur et forme :Drypowder PelletslargecrystalsMasse moléculaire :129.11GSK-7975A
CAS :<p>GSK-7975A is a potent and orally available inhibitor of CRAC channel.</p>Formule :C18H12F5N3O2Degré de pureté :98.92%Couleur et forme :SolidMasse moléculaire :397.3Bupivacaine hydrochloride
CAS :<p>Bupivacaine hydrochloride (Vivacaine) is a long-lasting, amide local anesthetic that blocks sodium channels, inhibiting nerve impulses and sensation.</p>Formule :C18H28N2O·HClDegré de pureté :99.9% - >99.99%Couleur et forme :SolidMasse moléculaire :324.89Nilvadipine
CAS :<p>Nilvadipine (FK235), a calcium channel blocker (CCB), is utilized for treatment of hypertension.</p>Formule :C19H19N3O6Degré de pureté :99.86% - 99.93%Couleur et forme :Yellow PrismsMasse moléculaire :385.37Amlodipine Besylate
CAS :<p>Amlodipine Besylate(Amlodipine benzenesulfonate) is a long-lasting calcium channel blocker.</p>Formule :C26H31ClN2O8SDegré de pureté :96.67% - 99.92%Couleur et forme :White PowderMasse moléculaire :567.05Otilonium bromide
CAS :<p>Otilonium bromide (SP63) , an antimuscarinic, is utilized as a spasmolytic agent.</p>Formule :C29H43BrN2O4Degré de pureté :98.88% - 99.78%Couleur et forme :White PowerMasse moléculaire :563.57Trimethadione
CAS :<p>Trimethadione (3,5,5,-Trimethyloxazolidine-2,4-dione) is a dione-type anticonvulsant with antiepileptic activity.</p>Formule :C6H9NO3Degré de pureté :99.67% - >99.99%Couleur et forme :SolidMasse moléculaire :143.14BX430
CAS :<p>BX430 is used for chronic pain and cardiovascular disease and it is a potent and selective noncompetitive allosteric human P2X4 receptor channels antagonist</p>Formule :C15H15Br2N3ODegré de pureté :97.34%Couleur et forme :SolidMasse moléculaire :413.11Azelnidipine
CAS :<p>Azelnidipine (UR-12592) is a dihydropyridine used as calcium channel blocker.</p>Formule :C33H34N4O6Degré de pureté :99.78%Couleur et forme :Light Yellowish PowderMasse moléculaire :582.65Amlodipine
CAS :<p>Amlodipine (UK-48340) is a synthetic dihydropyridine and a calcium channel blocker with antihypertensive and antianginal properties.</p>Formule :C20H25ClN2O5Degré de pureté :99.33% - 99.60%Couleur et forme :Solid PowderMasse moléculaire :408.88Dantrolene sodium
CAS :<p>Dantrolene sodium treats spasticity by disrupting muscle contraction; not central in action, grouped with central relaxants.</p>Formule :C14H9N4NaO5Degré de pureté :98% - 99.87%Couleur et forme :CoaMasse moléculaire :336.23Flunarizine dihydrochloride
CAS :<p>Flunarizine dihydrochloride: a calcium blocker also targeting calmodulin and histamine H1, used for migraine, vertigo, vascular disease, and epilepsy aid.</p>Formule :C26H28Cl2F2N2Degré de pureté :99.53% - 99.89%Couleur et forme :White Crystalline Powder Odorless And TastelessMasse moléculaire :477.42Nimodipine
CAS :<p>Nimodipine (BAY-e 9736), a 1, 4-dihydropyridine calcium channel blocker, acts primarily on vascular smooth muscle cells.</p>Formule :C21H26N2O7Degré de pureté :99.64% - 99.79%Couleur et forme :SolidMasse moléculaire :418.44Cromolyn sodium
CAS :<p>Cromolyn sodium (FPL-670) is a chromone complex that acts by inhibiting the release of chemical mediators from sensitized mast cells.</p>Formule :C23H14Na2O11Degré de pureté :99.4% - 99.95%Couleur et forme :Colorless Crystals From Ethanol + Ether White Crystalline PowderMasse moléculaire :512.33Clevidipine
CAS :<p>Clevidipine (Clevidipine butyrate) is a dihydropyridine L-type calcium channel blocker that is selective for vascular smooth muscle and is indicated for blood</p>Formule :C21H23Cl2NO6Degré de pureté :99.40%Couleur et forme :PowderMasse moléculaire :456.32Nicardipine hydrochloride
CAS :<p>Nicardipine hydrochloride is a potent calcium channel blocker used to dilate cerebral and coronary vessels.</p>Formule :C26H30ClN3O6Degré de pureté :99.58% - 99.89%Couleur et forme :Yellow SolidMasse moléculaire :515.99Butamben
CAS :<p>Butamben (Butyl 4-aminobenzoate) is a long-duration local anesthetic used for the treatment of chronic pain.</p>Formule :C11H15NO2Degré de pureté :99.43%Couleur et forme :Crystals From Alc Physical Description Yellow Powder Insoluble In Water (Ntp 1992)Masse moléculaire :193.24Ethaverine hydrochloride
CAS :<p>Ethaverine hydrochloride is a homologue of papaverine and is used as a vasodilator and antispasmodic.Cost-effective and quality-assured.</p>Formule :C24H30ClNO4Degré de pureté :99.66% - 99.90%Couleur et forme :SolidMasse moléculaire :431.96Catharanthine tartrate
CAS :<p>Catharanthine tartrate (Catharanthine hemitartrate) is an alkaloid from periwinkle that inhibits voltage-gated L-type calcium channels and has antitumor effect.</p>Formule :C25H30N2O8Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :486.51Praziquantel
CAS :<p>Praziquantel (Droncit) is an anthelmintic that paralyzes worms by increasing calcium in muscle cells, causing tegument damage and immune response.</p>Formule :C19H24N2O2Degré de pureté :99.67% - 99.69%Couleur et forme :SolidMasse moléculaire :312.41Gabapentin
CAS :<p>Gabapentin (Neurontin) is an Anti-epileptic Agent.</p>Formule :C9H17NO2Degré de pureté :99.55% - 99.91%Couleur et forme :White To Off-White Crystalline Solid; Crystals From Ethanol/Ether SolidMasse moléculaire :171.24Caloxin 2A1 TFA
<p>Caloxin 2A1 TFA is a PM Ca2+ pump inhibitor that inhibits human red blood cell Ca2+-Mg2+-ATPase leakage.</p>Formule :C66H92F3N19O24Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :1592.55Verapamil hydrochloride
CAS :<p>Verapamil hydrochloride (Verapamil HCl) is a calcium channel blocker that is a class IV anti-arrhythmia agent.</p>Formule :C27H39ClN2O4Degré de pureté :98.7% - 99.98%Couleur et forme :White To Off-White PowderMasse moléculaire :491.06Tetracaine hydrochloride
CAS :<p>Tetracaine HCl (Pontocaine), a potent local anesthetic and antipruritic, is used in eye care and for surface/spinal anesthesia.</p>Formule :C15H25ClN2O2Degré de pureté :99.72% - 99.94%Couleur et forme :White Or Off White Crystalline PowderMasse moléculaire :300.82Topiramate
CAS :<p>Topiramate (RWJ 17021) is a unique antiseizure medication that is used in the treatment of partial and generalized seizures.</p>Formule :C12H21NO8SDegré de pureté :99.79% - 99.92%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :339.36Flufenamic acid
CAS :<p>Flufenamic acid (Arlef) is an anthranilic acid derivative with analgesic, anti-inflammatory, and antipyretic properties.</p>Formule :C14H10F3NO2Degré de pureté :98.68%Couleur et forme :White To Light Yellow Crystalline PowderMasse moléculaire :281.23Synta66
CAS :<p>Synta66 is a store-operated calcium entry channel Orai inhibitor, and used for the research of neurological disease.</p>Formule :C20H17FN2O3Degré de pureté :99.57% - 99.84%Couleur et forme :SolidMasse moléculaire :352.361-EBIO
CAS :<p>1-EBIO (1-EBIO) is a calium channel agonist.</p>Formule :C9H10N2ODegré de pureté :98.75%Couleur et forme :SolidMasse moléculaire :162.19Ranolazine dihydrochloride
CAS :<p>Ranolazine 2HCl, an antianginal, treats arrhythmia by inhibiting sodium current without changing blood pressure or heart rate.</p>Formule :C24H35Cl2N3O4Degré de pureté :99.30% - >99.99%Couleur et forme :White Crystalline PowderMasse moléculaire :500.46Levamlodipine
CAS :<p>Levamlodipine (S-amlodipine) belongs to the dihydropyridine group of calcium channel blockers.</p>Formule :C20H25ClN2O5Degré de pureté :97.21%Couleur et forme :White Crystal PowderMasse moléculaire :408.88Cinepazide maleate
CAS :<p>Cinepazide maleate (MD-67350), a maleate salt form of cinepazide, is a vasodilator.</p>Formule :C22H31N3O5·C4H4O4Degré de pureté :99.9% - 99.97%Couleur et forme :White Or Off-White Crystalline PowderMasse moléculaire :533.57CRAC intermediate 2
CAS :<p>CRAC intermediate 2 is a intermediate compound for CRAC inhibitor synthesis.</p>Formule :C11H7F6N3Degré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :295.18Carboxyamidotriazole Orotate
CAS :<p>Carboxyamidotriazole Orotate (L-651582 Orotate) is a cytostatic inhibitor of non-voltage-operated calcium channels and calcium channel-mediated signaling</p>Formule :C22H16Cl3N7O6Degré de pureté :99.37%Couleur et forme :SolidMasse moléculaire :580.76Strontium ranelate
CAS :<p>Strontium ranelate (S12911), a strontium (II) salt of the ranelic acid, is a medication for osteoporosis and can slow the course of osteoarthritis of the knee.</p>Formule :C12H6N2O8S·2SrDegré de pureté :98.97%Couleur et forme :Crystalline SolidMasse moléculaire :513.49Caldaret HCl
CAS :<p>Caldaret HCl is an intracellular Ca2+ modulator that regulates calcium homeostasis at the sarcoplasmic reticulum and cell membrane, and can be used to study acute myocardial infarction and heart failure.</p>Formule :C11H17ClN2O3SDegré de pureté :98.99%Couleur et forme :SoildMasse moléculaire :292.78Cinnarizine
CAS :<p>Cinnarizine is a piperazine, blocks H1-receptor & Ca-channels, has vasodilating & antiemetic effects, may cause Parkinson-like symptoms.</p>Formule :C26H28N2Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :368.51Diltiazem hydrochloride
CAS :<p>Diltiazem hydrochloride (RG 83606 HCl) is a benzothiazepine calcium channel blocking agent with vasodilating action.</p>Formule :C22H27ClN2O4SDegré de pureté :98% - 99.65%Couleur et forme :Odorless White PowderMasse moléculaire :450.98Penfluridol
CAS :<p>Penfluridol (TLP-607) is a highly potent antipsychotic.</p>Formule :C28H27ClF5NODegré de pureté :98.9% - 99.87%Couleur et forme :Off-White To White Crystalline PowderMasse moléculaire :523.97Acetylcholine chloride
CAS :<p>Acetylcholine Chloride is the chloride salt form of acetylcholine, a synthetic, quaternary amino alcohol with cholinergic properties.</p>Formule :C7H16ClNO2Degré de pureté :98.02% - ≥95%Couleur et forme :White Crystalline PowderMasse moléculaire :181.66Brompheniramine maleate
CAS :<p>Brompheniramine maleate (Dimotane) is an antagonist against histamine H1 receptors.</p>Formule :C16H19BrN2·C4H4O4Degré de pureté :99.80%Couleur et forme :Crystal PowderMasse moléculaire :435.31Minocycline hydrochloride
CAS :<p>Minocycline HCl: tetracycline antibiotic, treats bacterial infections and acne, may cause acute or chronic hepatitis.</p>Formule :C23H28ClN3O7Degré de pureté :99.28% - >99.99%Couleur et forme :Bright Yellow-Orange Amorphous Solid Crystalline YellowMasse moléculaire :493.94Ebselen
CAS :<p>Ebselen is a selenium compound with anti-inflammatory and antioxidant properties, mimicking glutathione peroxidase to protect against ROS damage.</p>Formule :C13H9NOSeDegré de pureté :98.99% - 99.94%Couleur et forme :White SolidMasse moléculaire :274.18Devapamil
CAS :<p>Devapamil (Devapamilo) is a phenylalkylamine that blocks L-type calcium currents from the inner side of membrane cells in a use-dependent manner.</p>Formule :C26H36N2O3Degré de pureté :99.63%Couleur et forme :SolidMasse moléculaire :424.58Flavoxate hydrochloride
CAS :<p>Flavoxate hydrochloride (DW61) , a muscarinic AChR antagonist, is used in the therapy of various urinary syndromes and as an antispasmodic.</p>Formule :C24H26ClNO4Degré de pureté :99.78%Couleur et forme :White SolidMasse moléculaire :427.92PDDHV
CAS :<p>PDDHV: a capsaicin-like vanilloid selective for rat TRPV1; induces Ca2+ uptake in neurons, EC50 of 70 nM.</p>Formule :C49H72O11Couleur et forme :SolidMasse moléculaire :837.09JTV-519 Formate
<p>JTV-519 Formate is a Ca2+-dependent blocker of sarcoplasmic reticulum Ca2+-stimulated ATPase (SERCA).</p>Formule :C26H34N2O4SDegré de pureté :99.06%Couleur et forme :SolidMasse moléculaire :470.62NSC156529
CAS :<p>NSC156529 suppresses AKT1, reduces cancer cell growth in vitro, and inhibits prostate tumors in vivo.</p>Formule :C28H21ClS2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :457.05PACAP-38 (31-38), human, mouse, rat
CAS :<p>PACAP-38 (31-38), human, mouse, rat demonstrates potent, efficacious, and sustained stimulatory effects on sympathetic neuronal NPY and catecholamine production</p>Formule :C47H83N17O11Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1062.27Calcium Channel antagonist 2
CAS :<p>Calcium Channel antagonist 2 is a calcium channel antagonist (IC50=5-20 μM) that can be used to study diseases due to Ca2+ channels like pain and diabetes.</p>Formule :C23H25FN2O4SDegré de pureté :99.34%Couleur et forme :SolidMasse moléculaire :444.52ω-Conotoxin GVIA
CAS :<p>Peptide neurotoxin; selectively and reversibly blocks N-type calcium channels (IC50 = 0.15 nM). Reduces (RS)-3,5-DHPG -induced long term depression in vivo.</p>Formule :C120H182N38O43S6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3037Calcium Channel antagonist 4
CAS :<p>Calcium Channel antagonist 4 is a voltage-gated calcium channel inhibitor (IC50 : 5-20 μM).</p>Formule :C23H26N2O4SDegré de pureté :98.09%Couleur et forme :SolidMasse moléculaire :426.532,4,6-Tri-tert-butylphenol
CAS :<p>2,4,6-Tri-tert-butylphenol inhibits the Ca2+ ATPase activity of human red blood cell membranes and can be used in related research in the field of life sciences.</p>Formule :C18H30ODegré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :262.43Calcium Channel antagonist 5
CAS :<p>Calcium Channel antagonist5 (compound 32) is a calcium channel antagonist with a pIC50 of 5.50.</p>Formule :C17H18N2O6Couleur et forme :SolidMasse moléculaire :346.34Flunarizine
CAS :<p>Flunarizine is an orally administered peripheral vasodilator, a dual blocker of voltage-gated Na+/Ca2+ channels and a D2 dopamine receptor antagonist.</p>Formule :C26H26F2N2Degré de pureté :99.9%Couleur et forme :SolidMasse moléculaire :404.50ω-Conotoxin MVIIC TFA
<p>ω-Conotoxin MVIIC TFA is a peptide and neurotoxin blocks P-type and q-type voltage-sensitive neuronal Ca ++ channels (VGCCs) radiolabel immunoprecipitation.</p>Formule :C106H178N40O32S7·C2HF3O2Couleur et forme :SolidMasse moléculaire :2863.272-Nitrobenzoic acid
CAS :<p>2-Nitrobenzoic acid is an anti-growth agent with an IC50 of 8.3 μM against Jurkat cells with T-type Ca²⁺ channel alpha 1H/delta 25.</p>Formule :C7H5NO4Degré de pureté :99.97%Couleur et forme :SoildMasse moléculaire :167.12CALP3
CAS :<p>Cell-permeable CaM agonist, binds EF-hand, activates phosphodiesterase without Ca2+, inhibits Ca2+ toxicity, IC50=33μM.</p>Formule :C44H68N10O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :881.08(R)-IDHP
CAS :<p>(R)-IDHP, a salvia derivative, relaxes blood vessels by blocking calcium channels, aiding cardiovascular research.</p>Formule :C12H16O5Couleur et forme :SolidMasse moléculaire :240.25Isotachysterol 3
CAS :<p>Isotachysterol 3 boosts calcium transport in gut and bone mobilization in kidneyless rats.</p>Formule :C27H44OCouleur et forme :SolidMasse moléculaire :384.64UK-59811 hydrochloride
CAS :<p>UK-59811 hydrochloride, Br-dihydropyridine derivative, blocks Ca V Ab channels in bacteria, IC50: 194 nM.</p>Formule :C22H30BrClN2O5Couleur et forme :SolidMasse moléculaire :517.85Budiodarone tartrate
CAS :<p>Budiodarone tartrate (ATI-2042 tartrate) is an antiarrhythmic agent that inhibits calcium channels, and can be used in atrial fibrillation research.</p>Formule :C31H37I2NO11Degré de pureté :97.44%Couleur et forme :SolidMasse moléculaire :853.44ILS-920
CAS :<p>ILS-920, a Rapamycin analog, has reduced immunosuppression, enhanced neuroprotection, and preferentially binds FKBP52 and L-type VGCC β1.</p>Formule :C57H86N2O14Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1023.3NAADP tetrasodium salt
CAS :<p>Ca2+ mobilizing agent</p>Formule :C21H27N6O18P3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :744.39Ion Channel Targeted Library
<p>A unique collection of 931 compounds targeting ion channels for research in ion channels-related diseases and ion channel drug discovery;</p>Couleur et forme :Odour SolidIns(1,4,5)-P3 hexapotassium salt
CAS :<p>D-myo-Inositol 1,4,5-trisphosphate hexapotassium salt is promotes endoplasmic The second messenger of net calcium ions.</p>Formule :C6H9K6O15P3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :648.64SNX-482
CAS :<p>Potent CaV2.3 calcium channel blocker, selective, voltage-dependent, with 30 nM IC50. Offers antinociceptive effects on C and Aδ fibres.</p>Formule :C192H274N52O60S7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4495.01ω-Agatoxin IVA
CAS :<p>Selective blocker of P-type calcium channels (IC50 < 1 - 3 nM). Also inhibits N-type channels at micromolar concentrations.</p>Formule :C217H360N68O60S10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :5202.25D-myo-Inositol-1,3,4,5-tetraphosphate (sodium salt)
CAS :<p>Ins(1,3,4,5)-P4, made via Ins(1,4,5)P3 phosphorylation, boosts calcium by opening ER and plasma membrane channels.</p>Formule :C6H8Na8O18P4Couleur et forme :SolidMasse moléculaire :675.93SG-094
CAS :<p>SG-094 inhibits TPC2, halts RIL175 cell growth, IC50: 3.7 μM for cancer research.</p>Formule :C30H29NO3Degré de pureté :97.06%Couleur et forme :SoildMasse moléculaire :451.56Sulcardine 2HCl
CAS :<p>Sulcardine 2HCl is a multi-ion channel blocker that blocks the properties of hERG and hNav1.5 channels and can be used to study atrial fibrillation.</p>Formule :C24H35Cl2N3O4SDegré de pureté :99.33% - 99.76%Couleur et forme :SoildMasse moléculaire :532.523Mipsagargin
CAS :<p>Mipsagargin (G-202) is a new antibiotic that inhibits DNA biosynthesis.</p>Formule :C66H100N6O27Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1409.52GTx1-15
<p>GTx1-15, an inhibitor cystine knot (ICK) peptide, antagonizes the voltage-dependent calcium channel Cav3.1, as well as voltage-dependent sodium channels Nav1.3</p>Formule :C176H271N53O45S7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4073.82Nesiritide
CAS :<p>Nesiritide, recombinant human B-type natriuretic peptide, binds NPR-A/C with Kd 7.3/13 pM.</p>Formule :C143H244N50O42S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3464.04Ryanodine
CAS :<p>Ryanodine: a diterpenoid modulating Ca2+ release via ryanodine receptors; concentration-dependent effects; found in Ryania speciosa; toxic.</p>Formule :C25H35NO9Degré de pureté :98%Couleur et forme :White SolidMasse moléculaire :493.553Kurtoxin
<p>Kurtoxin is a selective Cav3 (T-type) voltage-gated Ca2+ channel gating inhibitor, exhibiting a dissociation constant (Kd) of 15 nM for the Cav3.1 (α1G T-type)</p>Formule :C324H478N94O90S8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :7386.36G-Glu-Ser
CAS :<p>G-Glu-Ser is a calcium receptor activator and Flavor-enriching agent.</p>Formule :C8H14N2O6Couleur et forme :SolidMasse moléculaire :234.21Mast cell degranulating peptide (28-49)
CAS :<p>Mast cell degranulating peptide (28-49) is a bee venom depolarizer that can improve the cGMP content of cerebellum tablets in mice.</p>Formule :C110H196N40O24S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2591.25γ-Glutamylserine TFA
<p>γ-Glutamylserine TFA (γ-Glu-Ser TFA) serves as a calcium receptor activator and is utilized in research focused on Parkinson's disease, diabetes, and obesity [1</p>Formule :C10H15F3N2O8Degré de pureté :98%Couleur et forme :SoildMasse moléculaire :348.23Lyso-Globotriaosylceramide (d18:1)
CAS :<p>Lyso-Gb3, lacking fatty acyl, binds Stx1 with cholesterol and phosphatidylcholine, not Stx2; lowers neutrophil viability; accumulates in Fabry disease.</p>Formule :C36H67NO17Couleur et forme :SolidMasse moléculaire :785.922Calcium Ionophore I
CAS :<p>Calcium Ionophore I has a wide range of applications in life science related research.</p>Formule :C38H72N2O8Couleur et forme :SolidMasse moléculaire :685.0LY393615
<p>LY393615 (NCC1048) is a novel blocker of both neuronal Ca²⁺ (calcium) and Na⁺ (sodium) channels, exhibiting half-maximal inhibitory concentrations (IC₅₀) of 1.9</p>Degré de pureté :98%Couleur et forme :Odour SolidOxodipine
CAS :<p>Oxodipine blocks rabbit aortic contraction and weakens rat cardiac force; reduces Ca currents in myocytes; side effects: mouse constipation, dog gum swelling.</p>Formule :C19H21NO6Degré de pureté :99.24%Couleur et forme :SolidMasse moléculaire :359.37O-Desmethylcarvedilol
CAS :<p>O-Desmethylcarvedilol (Desmethylcarvedilol) is an active metabolite of Carvedilol, a non-selective β-adrenergic receptor (β-AR) antagonist. This compound inhibits store overload-induced calcium release in HEK293 cells expressing the RyR2 R4496C mutation (IC50= 7.62 µM). Additionally, O-Desmethylcarvedilol slows the increase in heart rate and prevents diastolic pressure reduction induced by Isoproterenol in conscious rabbits (ED50s = 32 and 5 µg/kg).</p>Formule :C23H24N2O4Couleur et forme :SolidMasse moléculaire :392.45SB-237376
CAS :<p>SB-237376 is a calcium and potassium channel antagonist used to treat cardiac arrhythmias.</p>Formule :C20H25N3O5Degré de pureté :98.88% - 99.81%Couleur et forme :SoildMasse moléculaire :387.43D-myo-Inositol-1,3-diphosphate (sodium salt)
CAS :<p>D-myo-Inositol-1,3-phosphate (Ins(1,3)P) is an inositol phosphate involved in cellular signal transduction.</p>Formule :C6H12Na2O12P2Couleur et forme :SolidMasse moléculaire :384.08TPC2-A1-P
CAS :<p>TPC2-A1-P is a TPC2 agonist that can differentially activate two-pore channel 2 (TPC2) and mimic the activation of TPC2 with NAADP and PIP (2).</p>Formule :C20H21BrF3NO3Degré de pureté :98.49%Couleur et forme :SolidMasse moléculaire :460.29OPC 8490 free base
CAS :<p>OPC 8490 free base is a positive inotropic vasodilator and a cardiotonic agent that can be used to study cardiovascular diseases.</p>Formule :C24H27N3O3Degré de pureté :99.53%Couleur et forme :SoildMasse moléculaire :405.49D-myo-Inositol-1,4,5-triphosphate trisodium
CAS :<p>D-myo-Inositol-1,4,5-triphosphate trisodium (Inositol 1,4,5-trisphosphate trisodium) is a second messenger produced in cells by phospholipase C-mediated</p>Formule :C6H15Na3O15P3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :489.06Elgodipine
CAS :<p>Elgodipine decreases angina severity, inhibits muscle growth, and is voltage-sensitive, showing promise for angina treatment.</p>Formule :C29H33FN2O6Degré de pureté :98.95% - 99.50%Couleur et forme :SolidMasse moléculaire :524.58Cavα2δ-IN-1
CAS :<p>Cavα2δ-IN-1 demonstrates exceptional specificity for voltage-gated calcium channels Cavα2δ-1 (with a Ki value of 6 nM), in comparison to Cavα2δ-2 (with a Ki</p>Formule :C18H27N5OCouleur et forme :SolidMasse moléculaire :329.448Ser-Ala-alloresact acetate
<p>Ser-Ala-alloresact acetate is a sperm-activating peptide (SAP) that is released by marine invertebrate eggs and plays an important role in fertilization.</p>Formule :C44H75N13O16S2Degré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :1106.281-(aminomethyl)cyclopropanecarboxylic acid hydrochloride
CAS :<p>1-(aminomethyl)cyclopropanecarboxylic acid hydrochloride inhibits L amino acid transporter proteins and the α2δ subunit of voltage-gated calcium channels.1-(</p>Formule :C5H10ClNO2Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :151.59Triphenylethylene
CAS :<p>Compound PDK0283, with CAS No. 58-72-0, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0283 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.</p>Formule :C20H16Couleur et forme :White PowderMasse moléculaire :256.34ω-Conotoxin MVIIC
CAS :<p>Peptide neurotoxin; wide spectrum blocker of N, P and Q type calcium channels.</p>Formule :C106H178N40O32S7Degré de pureté :98%Couleur et forme :White Lyophilised SolidMasse moléculaire :2749Myomodulin
CAS :<p>Myomodulin is a neuropeptide present in molluscs, insects, and gastropods.Myomodulin is present in two identified aplysia neurons that contain myomodulin A the</p>Formule :C36H67N11O8S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :846.12PACAP-38 (31-38), human, mouse, rat TFA
<p>PACAP-38 (31-38), human, mouse, rat (TFA) demonstrates potent, efficacious, and sustained stimulatory effects on sympathetic neuronal.</p>Formule :C49H84F3N17O13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1176.29BTT-266
CAS :<p>BTT-266 is a blocker of voltage-gated calcium channel for pain management.</p>Formule :C34H28N4O4Degré de pureté :98.34%Couleur et forme :SolidMasse moléculaire :556.61Calcium Channel Compound Library
<p>A unique collection of 140 calcium channel blockers and agonists for high throughput and high content screening;</p>Couleur et forme :Odour SolidPD 0299685
CAS :<p>PD 0299685 is a potent α2δ ligand of the Ca2+ channel for the treatment of interstitial cystitis.</p>Formule :C10H21NO2Degré de pureté :97.20%Couleur et forme :SoildMasse moléculaire :187.28Calcium Channel antagonist 3
CAS :<p>Calcium Channel antagonist 3 is a voltage-gated calcium channel inhibitor (IC50 : 5-20 μM).</p>Formule :C23H26N2O4SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :426.53Fasudil
CAS :<p>Fasudil (HA-1077) is a potent inhibitor of ROCK1, PKA, PKC, and MLCK.</p>Formule :C14H17N3O2SDegré de pureté :99.79% - 99.84%Couleur et forme :SolidMasse moléculaire :291.37Linoleic Acid Amide
CAS :<p>Linoleic Acid Amide (Linoleamide) is derived from linoleic acid and regulates Ca2+ flux by inhibiting the sarco/endoplasmic reticulum Ca2+-ATPase.</p>Formule :C18H33NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :279.46Flosatidil
CAS :<p>Flosatidil is a small molecule voltage-gated calcium channel complex (VDCCs) blocker for the treatment of neurological disorders and cardiovascular diseases,</p>Formule :C26H34F3N3O3SDegré de pureté :98.29% - 99.60%Couleur et forme :SolidMasse moléculaire :525.63Ziconotide
CAS :<p>Ziconotide: analgesic from cone snail for severe, chronic pain; synthetic ω-conotoxin.</p>Formule :C102H172N36O32S7Degré de pureté :98%Couleur et forme :White PowderMasse moléculaire :2639.13Atagabalin HCl
CAS :<p>Atagabalin HCl is a novel voltage-dependent calcium channel (VDCC) α2δ subunit (1 and 2) ligand that affects slow-wave sleep and can be used to treat insomnia.</p>Formule :C10H20ClNO2Degré de pureté :99.96% - ≥98%Couleur et forme :SoildMasse moléculaire :221.72Huwentoxin I
CAS :<p>Huwentoxin I (HWTX-I) is a peptide toxin that targets and inhibits both voltage-gated sodium channels and N-type calcium channels.</p>Formule :C161H246N48O44S6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3750.36KT-362 free base
CAS :<p>KT-362 is a calcium channel blocker with antihypertensive properties that can be used in the study of cardiovascular disease.</p>Formule :C22H28N2O3SDegré de pureté :99.76%Couleur et forme :SoildMasse moléculaire :400.5317R(18S)-EpETE
CAS :<p>17R(18S)-EpETE: Oxylipin, eicosapentaenoic acid metabolite, activates BKCa channels, has negative chronotropic effects.</p>Formule :C20H30O3Couleur et forme :SolidMasse moléculaire :318.4571,4-Dihydropyridine
<p>1,4-Dihydropyridine acts as an antagonist for calcium channels (calcium channel), specifically blocking the L-type calcium channels. This action reduces the influx of calcium ions into cardiac and vascular smooth muscle cells, consequently decreasing cardiac contractility and heart rate, dilating blood vessels, and lowering blood pressure.</p>Formule :C12H17NO4Couleur et forme :SolidMasse moléculaire :239.27Chlorocresol
CAS :<p>Chlorocresol (4-Chloro-3-methylphenol) is an antiseptic medication.</p>Formule :C7H7ClOCouleur et forme :SolidMasse moléculaire :142.58Levamlodipine besylate Hemipentahydrate
CAS :<p>Levamlodipine besylate hemipentahydrate is the besylate hemipentahydrate salt form of Levamlodipine. It is an orally effective calcium channel blocker with antioxidative and vasodilatory properties. This compound can reduce serum malondialdehyde (MDA) levels, enhance the activity of superoxide dismutase (SOD), and alleviate oxidative stress. Levamlodipine besylate hemipentahydrate is relevant for research in vascular dementia, hypertension, and cerebrovascular diseases.</p>Formule :C20H25ClN2O5·C6H6O3SH2OCouleur et forme :SolidMasse moléculaire :1224.18NAADP sodium
<p>NAADP sodium is a Ca2+ motor second messenger that targets Ca(2+) channels and can be used to study cancer and immune dysfunction.</p>Formule :C21H27N6O18P3Couleur et forme :SolidMasse moléculaire :744.39D-myo-Inositol-1,4,5-triphosphate tripotassium
CAS :<p>D-myo-Inositol-1,4,5-triphosphate tripotassium is a second messenger in the intracellular signaling system that induces Ca2+ mobilization.</p>Formule :C6H12K3O15P3Couleur et forme :SolidMasse moléculaire :534.37Ethacrynic acid D5
CAS :<p>Ethacrynic acid: a diuretic, anti-inflammatory, inhibits calcium channels, GSTs, NF-kB pathway, and modulates leukotriene; has deuterium-labeled form.</p>Formule :C13H12Cl2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :308.17Cyclic ADP-ribose ammonium
<p>cADPR ammonium is a second messenger that boosts cytosolic calcium via Ryanodine receptors and TRPM2 channels.</p>Couleur et forme :LiquidsFTX-3.3
CAS :<p>sFTX-3.3 is a calcium ion channel antagonist, exhibiting IC50 values of approximately 0.24 mM and 0.70 mM against P-type and N-type channels respectively.</p>Formule :C12H29N7OCouleur et forme :SolidMasse moléculaire :287.412Candidalysin
CAS :<p>Candidalysin is a cytolytic peptide toxin initially isolated from *Candida albicans*, exhibiting both toxic and non-toxic properties. It activates epithelial cell signaling pathways by interacting with the epithelial growth factor receptor (EGFR) on host cells, leading to the activation of matrix metalloproteinases (MMP) and calcium ion influx, which results in inflammatory responses and immune cell recruitment. Additionally, Candidalysin exhibits cytotoxicity by causing membrane damage to host cells.</p>Formule :C153H266N38O38S2Couleur et forme :SolidMasse moléculaire :3310.11Ethyl 4-chloro-2-oxo-1,2-dihydroquinoline-3-carboxylate
CAS :<p>ethyl 4-chloro-2-oxo-1,2-dihydroquinoline-3-carboxylate inhibits NAD(P)H: quinone oxidoreductase 1.</p>Formule :C12H10ClNO3Degré de pureté :99.19%Couleur et forme :SolidMasse moléculaire :251.67ProTx-I
CAS :<p>Selective blocker for CaV3.1 (IC50 = 0.2 μM), CaV3.2 (31.8 μM), also inhibits NaV1.8 and blocks KV2.1 channels.</p>Formule :C171H245N53O47S6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3987.51(±)5(6)-DiHETE
CAS :<p>Eicosapentaenoic acid is an ω-3 polyunsaturated fatty acid that is abundant in marine organisms and fish oils.</p>Formule :C20H32O4Couleur et forme :SolidMasse moléculaire :336.472MMK 1
CAS :<p>Potent hFPR2 agonist; EC50: 1 nM (mFPR2), 2 nM (hFPR2), >10,000 nM (hFPR1). Induces monocyte/neutrophil migration, boosts IL-1β/IL-6, activates NADPH-oxidase.</p>Formule :C75H123N19O18SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1610.97ω-Agatoxin TK
CAS :<p>Selective blocker of CaV2.1 P/Q-type calcium channels.</p>Formule :C215H337N65O70S10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :5273.02Catharanthine
CAS :<p>Catharanthine ((+)-3,4-Didehydrocoronaridine) suppresses nicotinic receptor-mediated diaphragm contractions (IC50=59.6 μM).</p>Formule :C21H24N2O2Degré de pureté :99.11%Couleur et forme :White PowderMasse moléculaire :336.43CCT129957
CAS :<p>CCT129957 is a novel and potent phospholipase C-γ (PLC-γ) inhibitor with an IC50 of about 3 μM and a GC50 of 15 μM.CCT129957 exhibits anticancer activity and</p>Formule :C17H15N3O3Degré de pureté :99.44%Couleur et forme :SolidMasse moléculaire :309.32(R)-(+)-Bay-K-8644
CAS :<p>(R)-(+)-Bay-K-8644, a Ca2+ channel agonist, is a dihydropyridine agonist that induces central respiratory depression and inhibits platelet activation in cats.</p>Formule :C16H15F3N2O4Degré de pureté :96.51% - 96.51%Couleur et forme :SolidMasse moléculaire :356.3N-Palmitoyl Glycine
CAS :<p>Acyl amides like AEA modulate pain/inflammation. PalGly, similar to N-acyl ethanolamines, inhibits nociception and induces calcium influx in cells.</p>Formule :C18H35NO3Couleur et forme :SolidMasse moléculaire :313.48TPC2-A1-N
CAS :<p>TPC2-A1-N is a TPC2 small molecule agonist that can be used to detect different functions of TPC2 channels in intact cells.</p>Formule :C17H9Cl2F3N2O2Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :401.17(S)-Lercanidipine D3 hydrochloride
CAS :<p>(S)-Lercanidipine D3 hydrochloride is a deuterium labeled Lercanidipine D3 hydrochloride. (S)-Lercanidipine hydrochloride is an agent of antihypertensive.</p>Formule :C36H42ClN3O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :651.21(R)-Nicardipine
CAS :<p>(R)-Nicardipine is the less active R enantiomer of Nicardipine. Nicardipine is a blocker of calcium channel(IC50 of 1 μM for blocking cardiac calcium channels).</p>Formule :C26H29N3O6Couleur et forme :SolidMasse moléculaire :479.53β-Cyfluthrin
CAS :<p>β-Cyfluthrin is a type II synthetic pyrethroid compound commonly utilized as an active ingredient in agricultural insecticide products.</p>Formule :C22H18Cl2FNO3Couleur et forme :SolidMasse moléculaire :434.29(R)-Lercanidipine-d3 hydrochloride
CAS :<p>(R)-lercanidipine D3 hydrochloride is a deuterium labeled (R)-Lercanidipine hydrochloride. (R)-Lercanidipine D3 (hydrochloride) is a calcium channel blocker.</p>Formule :C36H42ClN3O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :651.21YM-244769
CAS :<p>YM-244769 (3-Pyridinecarboxamide, N-[(3-aminophenyl)methyl]-6-[4-[(3-fluorophenyl)methoxy]phenoxy]-) is an effective inhibitor of Na+/Ca2+ exchange 3 (NCX3)</p>Formule :C26H22FN3O3Degré de pureté :95.62%Couleur et forme :SolidMasse moléculaire :443.47Nicardipine-d3 hydrochloride
CAS :<p>Nicardipine D3 hydrochloride is the deuterium labeled Nicardipine hydrochloride.</p>Formule :C26H30ClN3O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :519YM-244769 dihydrochloride
CAS :<p>YM-244769 dihydrochloride is an effective inhibitor of Na+/Ca2+ exchange 3 (NCX3) with an IC50 of 18 nM.</p>Formule :C26H24Cl2FN3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :516.39HSK16149
CAS :<p>HSK16149 is a novel ligand of voltage-gated calcium channel (VGCC) α 2 δ subunit with analgesic activity.</p>Formule :C12H19NO2Couleur et forme :SolidMasse moléculaire :209.28MRS1845
CAS :<p>MRS1845 is a selective inhibitor of store-operated calcium (SOC) channel (IC50 of 1.7 μM).</p>Formule :C21H22N2O6Degré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :398.41(S)-Nicardipine
CAS :<p>(S)-Nicardipine is the less active S enantiomer of Nicardipine. Nicardipine is a blocker of calcium channel(IC50 of 1 μM for blocking cardiac calcium channels).</p>Formule :C26H29N3O6Couleur et forme :SolidMasse moléculaire :479.53Almorexant hydrochloride
CAS :<p>Almorexant hydrochloride (ACT 078573 hydrochloride) is a dual orexin receptor antagonist that induces apoptosis and can be used to study sleep disorders.</p>Formule :C29H32ClF3N2O3Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :549.02Norverapamil-d7
CAS :<p>Norverapamil D7 is a deuterium labeled Norverapamil . Norverapamil is a blocker of L-type calcium channel and an inhibitor of P-glycoprotein (P-gp) function .</p>Formule :C26H36N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :447.62Hexadecylphosphoserine TFA
<p>Hexadecylphosphoserine is a type of phospholipid molecule that incorporates a long-chain alkyl group (hexadecyl) and a phosphatidylserine group, granting it high affinity for cell membranes. This compound exhibits antitumor activity by modulating [Ca++]i and related signaling pathways, making it useful for breast cancer research.</p>Formule :C21H41F3NO8PCouleur et forme :SolidMasse moléculaire :523.52Dronedarone
CAS :<p>Dronedarone (SR 33589) is an amiodarone analogue which has an effective and promising treatment for Atrial fibrillation.</p>Formule :C31H44N2O5SDegré de pureté :98.85% - 99.58%Couleur et forme :SolidMasse moléculaire :556.76Azumolene
CAS :<p>Azumolene (EU4093 free base)</p>Formule :C13H9BrN4O3Degré de pureté :98.1% - 98.35%Couleur et forme :SolidMasse moléculaire :349.14Ginsenoside Rd
CAS :<p>Ginsenoside Rd (Gypenoside VIII) may have properties that inhibit or prevent the growth of tumors.</p>Formule :C48H82O18Degré de pureté :99.13% - 99.92%Couleur et forme :SolidMasse moléculaire :947.15JNJ-26990990
CAS :<p>"JNJ-26990990: broad-spectrum anticonvulsant, less side effects than topiramate, potential for pain and depression treatment; Phase II in 2007."</p>Formule :C9H10N2O2S2Degré de pureté :97.37%Couleur et forme :SolidMasse moléculaire :242.32Efonidipine
CAS :<p>Efonidipine (NZ-105)(NZ-105) is a dihydropyridine calcium channel blocker, blocking both T-type and L-type calcium channels.</p>Formule :C34H38N3O7PDegré de pureté :98.35% - 99.47%Couleur et forme :SolidMasse moléculaire :631.66Bepridil hydrochloride
CAS :<p>Bepridil hydrochloride (CERM 1978) is a calcium channel blocker and also inhibits Na+/Ca2+ exchange (NCX), sodium channels and cardiac sarcolemmal KATP channels</p>Formule :C24H35ClN2ODegré de pureté :99.45% - 99.68%Couleur et forme :SolidMasse moléculaire :4032,5-Di-tert-butylhydroquinone
CAS :<p>2,5-Di-tert-butylhydroquinone (BHQ) is an effective and selective endoplasmic reticulum Ca2+-ATPase inhibitor.</p>Formule :C14H22O2Degré de pureté :97.11%Couleur et forme :PelletslargecrystalsMasse moléculaire :222.32DHBP dibromide
CAS :<p>DHBP dibromide (1,1'-DI-N-HEPTYL-4,4'-BIPYRIDINIUM DIBRO) is calcium release and a muscle relaxant inhibitor.</p>Formule :C24H38Br2N2Degré de pureté :99.73%Couleur et forme :Yellow To Yellow-Green Powder Or FlakesMasse moléculaire :514.38L-Phenylalanine
CAS :<p>L-Phenylalanine (3-Phenyl-L-alanine) is an essential amino acid and the precursor of the amino acid tyrosine, acts as an antagonist at α2δ calcium channels.</p>Formule :C9H11NO2Degré de pureté :99.37% - 99.87%Couleur et forme :Solid CrystallineMasse moléculaire :165.19GSK1016790A
CAS :<p>GSK1016790A (GSK101) (GSK101) is a novel, potent activator of TRPV4 (transient receptor potential vanilloid 4) with EC50 of 34 nM in choroid plexus epithelial</p>Formule :C28H32Cl2N4O6S2Degré de pureté :97.37% - 99.38%Couleur et forme :SolidMasse moléculaire :655.61Propiverine hydrochloride
CAS :<p>Propiverine is a widely used antimuscarinic drug with a mixed mode of action in the treatment of symptoms associated with overactive bladder (OAB).</p>Formule :C23H30ClNO3Degré de pureté :99.93%Couleur et forme :White Crystalling PowerMasse moléculaire :403.94Dantrolene sodium hemiheptahydrate
CAS :<p>Dantrolene depresses excitation-contraction coupling in skeletal muscle by binding to the ryanodine receptor 1 and decreasing intracellular calcium</p>Formule :C14H9N4NaO5·5H2ODegré de pureté :99.72%Couleur et forme :Orange PowderMasse moléculaire :399.29Pranidipine
CAS :<p>Pranidipine (OPC-13340) is a novel, long-acting 1,4-dihydropyridine calcium channel blocker.</p>Formule :C25H24N2O6Degré de pureté :99.95%Couleur et forme :Yellow SolidMasse moléculaire :448.47Aranidipine
CAS :<p>Aranidipine (MPC1304) (MPC1304) is a calcium channel antagonist with potent and long-lasting antihypertensive effects.</p>Formule :C19H20N2O7Degré de pureté :99.15%Couleur et forme :SolidMasse moléculaire :388.37(±)-Praeruptorin A
CAS :<p>(±)-Praeruptorin A could exhibit its anti-osteoclastogenic activity by inhibiting p38/Akt-c-Fos-NFATc1 signaling and PLCγ-independent Ca(2+) oscillation.</p>Formule :C21H22O7Degré de pureté :98.9% - 99.73%Couleur et forme :SolidMasse moléculaire :386.4(+)-Kavain
CAS :<p>(+)-Kavain ((R)-KAWAIN) is one of the six major kavalactones found in the Piper methysticum (kava) plant; reversible inhibitor of MAO-B.</p>Formule :C14H14O3Degré de pureté :97% - ≥95%Couleur et forme :White Fine PowderMasse moléculaire :230.26Suvecaltamide
CAS :<p>Suvecaltamide (MK-8998) as potent inhibitors of T-type calcium channels.</p>Formule :C20H23F3N2O2Degré de pureté :99.29% - 99.70%Couleur et forme :SolidMasse moléculaire :380.4NS-638
CAS :<p>NS-638 is a Ca2+-channel blocker. It can block K+-stimulated intracellular Ca2+-elevation (IC50: 3.4 μM).</p>Formule :C15H11ClF3N3Degré de pureté :98.44%Couleur et forme :SolidMasse moléculaire :325.72NFAT Inhibitor-2
CAS :<p>NFAT Inhibitor-2 is a compound used as a molecular building block.</p>Formule :C22H20F2N2O4SDegré de pureté :97.37%Couleur et forme :SolidMasse moléculaire :446.47Efonidipine hydrochloride monoethanolate
CAS :<p>Efonidipine HCl monoethanolate is a calcium blocker, boosts dehydroepiandrosterone sulfate in NCI-H295R cells.</p>Formule :C36H45ClN3O8PDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :714.18Praeruptorin E
CAS :<p>Praeruptorin C/E relaxes arteries, reduces heart contractility, acting like calcium blockers. D/E protect mice from acid lung injury by halting PMNs and IL-6.</p>Formule :C24H28O7Degré de pureté :98.04% - 99.95%Couleur et forme :SolidMasse moléculaire :428.47SR33805
CAS :<p>SR33805 is a potent antagonist of Ca2+ channel(EC50s of 4.1 nM and 33 nM in depolarized and polarized conditions, respectively)</p>Formule :C32H40N2O5SDegré de pureté :99.15%Couleur et forme :SolidMasse moléculaire :564.74Ibutilide Fumarate
CAS :<p>Ibutilide Fumarate is a class III antiarrhythmic, prolonging action potentials by enhancing sodium influx, and can extend QT interval.</p>Formule :(C20H36N2O3S)2·C4H4O4Degré de pureté :99.68% - 99.74%Couleur et forme :SolidMasse moléculaire :885.23Azumolene sodium anhydrous
CAS :<p>Azumolene sodium, a muscle relaxant, blocks calcium release from muscles and halts SOCE linked to RyR1 except when induced by thapsigargin.</p>Formule :C13H8BrN4NaO3Couleur et forme :SolidMasse moléculaire :371.13Argireline
CAS :<p>Argireline (Acetyl hexapeptide-3) is a peptide that inhibits neurotransmitter release, reducing wrinkles.</p>Formule :C34H60N14O12SDegré de pureté :96.79% - 99.65%Couleur et forme :White PowderMasse moléculaire :888.99TGR5 Receptor Agonist
CAS :<p>TGR5 is a potent TGR5(GPCR19) agonist.</p>Formule :C18H14Cl2N2O2Degré de pureté :99.77% - ≥95%Couleur et forme :SolidMasse moléculaire :361.22Ethacrynic acid
CAS :<p>Ethacrynic acid (Edecrin) 是谷胱甘肽 S-转移酶抑制剂，也是NF-κB 信号传导途径的有效抑制剂，并且还调节白三烯的形成。它还可抑制 L 型电压依赖性和储存操作的钙通道，从而导致气道平滑肌细胞松弛。它是利尿剂，具有抗炎特性，可减轻类维生素 A 诱导的小鼠耳部水肿。</p>Formule :C13H12Cl2O4Degré de pureté :98.61% - 99.85%Couleur et forme :Crystals Physical Description White Solid (Ntp 1992)Masse moléculaire :303.14Glaucine
CAS :<p>Glaucine: antitussive, antioxidative, antiviral, may fight arthritis, boosts IL-10, hinders breast cancer cell spread by inhibiting MMP-9 and NF-κB.</p>Formule :C21H25NO4Degré de pureté :99.42% - 99.56%Couleur et forme :SolidMasse moléculaire :355.43HC-056456
CAS :<p>HC-056456 (3,4-Bis(2-thienoyl)-1,2,5-oxadiazole-N-oxide) is a CatSper channel modulator.</p>Formule :C12H6N2O4S2Degré de pureté :99.62% - 99.65%Couleur et forme :SolidMasse moléculaire :306.32Psoralenoside
CAS :<p>Psoralenoside: a compound from Psoralea fruit; has estrogenic, osteoblastic, antitumor, and antibacterial properties.</p>Formule :C17H18O9Degré de pureté :99.03% - 99.49%Couleur et forme :SolidMasse moléculaire :366.32Quadrol
CAS :<p>Quadrol (EDTP) is an immunostimulant, accelerated wound healing.</p>Formule :C14H32N2O4Degré de pureté :99.91% - 99.92%Couleur et forme :Viscous Liquid Liquid ViscousMasse moléculaire :292.41Mirogabalin
CAS :<p>Mirogabalin (DS5565) is a calcium channel blocker with analgesic effects.</p>Formule :C12H19NO2Degré de pureté :98.57%Couleur et forme :SolidMasse moléculaire :209.28Efonidipine hydrochloride
CAS :<p>Efonidipine HCl (NZ-105) blocks T-type/L-type calcium channels; used in hypertension treatment.</p>Formule :C34H39ClN3O7PCouleur et forme :SolidMasse moléculaire :668.12NP118809
CAS :<p>NP118809 (39-1B4) is a potent N-type calcium channel blocker(IC50 : 0.11 μM).</p>Formule :C32H32N2ODegré de pureté :97.74% - 98.68%Couleur et forme :SolidMasse moléculaire :460.61Praeruptorin C
CAS :<p>Praeruptorin C: an antioxidant, calcium antagonist, protects neurons, reduces vascular hypertrophy, affects cellular signals.</p>Formule :C24H28O7Degré de pureté :99.6% - 99.92%Couleur et forme :SolidMasse moléculaire :428.47CDN1163
CAS :<p>CDN1163 is a small molecule activator of sarco/endoplasmic reticulum Ca2+-ATPase (SERCA).</p>Formule :C20H20N2O2Degré de pureté :99.83% - ≥95%Couleur et forme :SolidMasse moléculaire :320.39ABT-639 hydrochloride
CAS :<p>ABT-639 hydrochloride is a selective, novel T-type Ca2+ channel blocker.</p>Formule :C20H21Cl2F2N3O3SCouleur et forme :SolidMasse moléculaire :492.36Pyr6
CAS :<p>Pyr6 (N-[4-[3,5-Bis(trifluoromethyl)-1H-pyrazol-1-yl]phenyl]-3-fluoro-4-pyridinecarboxamide) is a selective TRPC3 inhibitor with IC50 of 0.49 uM(Ca2+ influx</p>Formule :C17H9F7N4ODegré de pureté :98.89%Couleur et forme :SolidMasse moléculaire :418.27Gabapentin hydrochloride
CAS :<p>Gabapentin hydrochloride (Neurontin HCl) is a GABA analogue, used to treat seizures and neuropathic pain.</p>Formule :C9H17NO2·HClDegré de pureté :99.71%Couleur et forme :Off-White SolidMasse moléculaire :207.7Pinaverium bromide
CAS :<p>Pinaverium bromide is an calcium channel blocker with Antispasmodic and effectively relieves pain, diarrhea and intestinal discomfort.</p>Formule :C26H41Br2NO4Degré de pureté :99.52%Couleur et forme :White Crystalline PowderMasse moléculaire :591.42Taurolithocholic acid sodium salt
CAS :<p>Taurolithocholic acid sodium salt (Sodium taurolithocholate) is the major human metabolite, a bile acid which inhibits radioligand binding to muscarinic M1, but</p>Formule :C26H44NNaO5SDegré de pureté :99.79% - 99.93%Couleur et forme :SolidMasse moléculaire :505.69FPL64176
CAS :<p>FPL64176 is a L-type calcium channels activator.</p>Formule :C22H21NO3Degré de pureté :98.68%Couleur et forme :SolidMasse moléculaire :347.41
