Microbiologie/Virologie
Les inhibiteurs en microbiologie et virologie sont des composés qui ciblent les microorganismes, y compris les bactéries, les virus et les champignons, perturbant leur croissance, leur réplication ou leur survie. Ces inhibiteurs sont essentiels pour étudier la pathogénie microbienne, comprendre les mécanismes de résistance et développer de nouvelles thérapies antimicrobiennes et antivirales. Les inhibiteurs de cette catégorie sont utilisés pour combattre les maladies infectieuses, explorer l'écologie microbienne et étudier les interactions hôte-pathogène. Chez CymitQuimica, nous offrons une large sélection d'inhibiteurs de haute qualité en microbiologie et virologie pour soutenir vos recherches en maladies infectieuses, microbiologie et virologie.
Sous-catégories appartenant à la catégorie "Microbiologie/Virologie"
- Antibactérien(3.423 produits)
- Antibiotique(945 produits)
- Antifection(27 produits)
- DHFR(30 produits)
- Synthèse ADN/ARN(808 produits)
- VHB(186 produits)
- Protéase du VIH(507 produits)
- HSV(99 produits)
- Intégrase(2 produits)
- Ribosome(5 produits)
Affichez 2 plus de sous-catégories
6442 produits trouvés pour "Microbiologie/Virologie"
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MMV03
CAS :MMV03 is an antimalarial compound effective against Plasmodium falciparum, with an EC50 of 0.6 μM.Formule :C19H14N4OSCouleur et forme :SolidMasse moléculaire :346.406ZINC000104379474
ZINC000104379474 is a compound that targets SARS-CoV-2 endoribonuclease.Formule :C27H33N3O10Couleur et forme :SolidMasse moléculaire :559.57Antimalarial agent 9
Antimalarial 9, a quinoline-imidazole derivative, effectively targets CQ-susceptible (IC50-0.14 μM) and MDR strains (IC50-0.41 μM) with low toxicity.Formule :C28H32BrN3O2Couleur et forme :SolidMasse moléculaire :522.48Fenbenicillin potassium
CAS :Fenbenicillin (Phenbenicillin) potassium is a semi-synthetic penicillin with antibacterial spectrum activity.Formule :C22H22KN2O5SCouleur et forme :SolidMasse moléculaire :465.584GSK_WRN4
CAS :GSK_WRN4 is a WRN helicase inhibitor with anti-cancer activity, inhibiting MSI tumor cell growth by inducing DNA double-strand breaks, useful in cancer researchFormule :C16H20N2O4SDegré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :336.41Asukamycin
CAS :Asukamycin, from S. nodosus asukaensis, is a polyketide antibiotic inhibiting tumor cells by activating caspases 8 and 3.Formule :C31H34N2O7Couleur et forme :SolidMasse moléculaire :546.61Antibacterial agent 174
CAS :Compound 174 (Compound 5g), an antibacterial agent, exhibits potent anti-infective properties in vivo along with appreciable pharmacokinetic profiles. This highly active substance demonstrates favorable biofilm removal capabilities, low hemolysis, and acceptable mammalian cell toxicity [1].Formule :C25H30FN2NaO5Couleur et forme :SolidMasse moléculaire :480.5(R)-CSN5i-3
CAS :(R)-CSN5i-3 is CSN5i-3 of the R configuration.Formule :C28H29F2N5O2Degré de pureté :99.76% - 99.97%Couleur et forme :SolidMasse moléculaire :505.56CRS-3123
CAS :CRS-3123, a methionyl-tRNA synthetase inhibitor, is used potentially for the treatment of enteric infections.Formule :C19H19Br2N3O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :513.25WRN inhibitor 11
CAS :WRN inhibitor 11 (Example 17) is an orally effective inhibitor of WRN helicase, with an IC50 of 63 nM.Formule :C34H35ClF3N9O5Couleur et forme :SolidMasse moléculaire :742.15SARS-CoV-2-IN-100
CAS :SARS-CoV-2-IN-100 (Compound 172) is a broad-spectrum antiviral agent against various SARS-CoV-2 variants. It works synergistically with Nirmatrelvir to reduce the risk of antiviral resistance.Formule :C29H23NO2Couleur et forme :SolidMasse moléculaire :417.50Metallo-β-lactamase-IN-16
CAS :Metallo-β-lactamase-IN-16 (compound 18), a sulfone-containing metallo-β-lactamase inhibitor, exhibits antimicrobial activity. It effectively inhibits various metallo-β-lactamases, including NDM-1 (New Delhi metallo-β-lactamase-1), IMP-1 (imipenemase-1), VIM-1 (Verona Integron-encoded Metallo-β-lactamase), and VIM-2. The IC50 values for these enzymes are 0.16 nM, 0.23 nM, 0.31 nM, and 1.0 nM respectively.Formule :C16H16N8O4S3Couleur et forme :SolidMasse moléculaire :480.54SARS-CoV-2-IN-102
CAS :SARS-CoV-2-IN-102 (example 58) is an inhibitor of the SARS-CoV papain-like protease (SARS-CoVPLpro), demonstrating an IC50 of less than 100 nM.Formule :C29H34F2N6O2Couleur et forme :SolidMasse moléculaire :536.62Antifungal agent 113
CAS :Antifungalagent 113 (compound 9a) serves as an effective antifungal and antibacterial agent. It exhibits strong inhibitory activity against both S. aureus and methicillin-resistant S. aureus.Formule :C23H20O5Couleur et forme :SolidMasse moléculaire :376.40HRSV/HMPV-IN-1
CAS :HRSV/HMPV-IN-1 (compound 3) is an inhibitor targeting HRSV/HMPV, exhibiting EC50 values of < 0.2 μM against human RSV-A and < 0.5 μM for human MPV A2 TN/94-49. This compound is utilized in the study of bronchiolitis and pneumonia.Formule :C34H31ClF2N4O5SCouleur et forme :SolidMasse moléculaire :681.15MED6-189
CAS :MED6-189, an analog of kalihinol, disrupts the apicoplast functions and vesicular transport in the malignant malaria parasite (P. falciparum, IC50 < 50 nM). The compound specifically targets the apicoplast, which is a non-photosynthetic plastid essential for isoprenoid synthesis, found in most apicomplexan parasites.Formule :C17H26N2OCouleur et forme :SolidMasse moléculaire :274.40Ciluprevir
CAS :Ciluprevir is a selective HCV NS3 protease inhibitor, effective against non-genotype-1 HCV; less potent for genotypes 2/3.Formule :C40H50N6O8SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :774.93Palmitanilide
CAS :Palmitanilide (Palmitic acid anilide) is an antimicrobial agent effective against Gram-positive bacteria. It can electrostatically bind to components of the cell wall of Gram-positive bacteria (such as Bacillus cereus), altering the membrane structure and affecting normal cellular functions. Palmitanilide shows potential for research into infections caused by Gram-positive bacteria.Formule :C22H37NOCouleur et forme :SolidMasse moléculaire :331.535Bleomycin Free Base
CAS :Bleomycin Free Base, a glycopeptide antibiotic, halts DNA function and treats solid tumors.Formule :C55H84N17O21S3Couleur et forme :SolidMasse moléculaire :1415.555-Methylcytosine hydrochloride
CAS :5-Methylcytosine hydrochloride plays a critical role in regulating gene expression, promoting genomic imprinting, and inhibiting transposon factors. It is also closely associated with translation fidelity and tRNA recognition.Formule :C5H8ClN3OCouleur et forme :SolidMasse moléculaire :161.59RhlR antagonist 1
RhlR antagonist 1: IC50 of 26 μM, selective for RhlR, inhibits P. aeruginosa biofilm and virulence factors.Formule :C12H10F2OCouleur et forme :SolidMasse moléculaire :208.2DXR-IN-3
CAS :DXR-IN-3 is an anti-Toxoplasma DXR inhibitor. It exhibits in vitro activity against the TgDXR enzyme, with an IC50 value of 0.62 μM and a Ki value of 0.19 μM. Furthermore, DXR-IN-3 can inhibit the proliferation of Toxoplasma, displaying an IC50 value of 5.46 μM.Formule :C10H12Cl2NO5PSCouleur et forme :SolidMasse moléculaire :360.15Antibacterial agent 88
Antibacterial agent 88 is an effective antibacterial agent against B. subtilis (MIC: 4 μg/ml) with MIC values of ≤0.0156 μg/mL for MRSA, MRSE and S. aureus.Formule :C31H44N2O6SCouleur et forme :SolidMasse moléculaire :572.76PptT-IN-3
PptT-IN-3 (5p), an inhibitor of PptT in Mycobacterium tuberculosis, IC50=3.5μM, is key for TB research.Formule :C16H27N5O3SCouleur et forme :SolidMasse moléculaire :369.48(R)-ZG197
(R)-ZG197: Activates Sa ClpP (EC50=1.5μM) & Hs ClpP (EC50=31.4μM); selective for Sa ClpP.Formule :C28H35F3N4O3Couleur et forme :SolidMasse moléculaire :532.6Arterolane maleate
CAS :Arterolane, an adenosine triphosphatase inhibitor, is used potentially for the treatment of malaria.Formule :C26H40N2O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :508.612Urease-IN-16
CAS :Urease-IN-16, with an IC50 of 132 µmol/L, is a urease inhibitor that coordinates with nickel atoms through the oxygen atoms of either carbonyl or boronic acid groups. This compound holds significant potential as an additive in the development of efficient fertilizers and medical applications.Formule :C14H17BN2O4SCouleur et forme :SolidMasse moléculaire :320.17Anticaries agent-1
CAS :Anticaries agent-1 (Compound 21b) is utilized as an anticaries agent. It effectively inhibits biofilm formation with an IC50 of 77 μM and restricts the growth of S. mutans.Formule :C15H12O4Couleur et forme :SolidMasse moléculaire :256.253DC-159a
CAS :DC-159a, an 8-methoxy fluoroquinolone, possesses broad-spectrum antibacterial activity, with a particular efficacy against Gram-positive pathogens. The MIC90 values for DC-159a are 0.5 μg/mL against Streptococcus anginosus group, 4 μg/mL against Clostridium difficile, and 2 μg/mL against Bacteroides fragilis.Formule :C21H23F2N3O40·5H2OCouleur et forme :SolidMasse moléculaire :428.4295Pyriftalid
CAS :Pyriftalid is a novel insecticide known for its potent inhibitory activity against a variety of pests. It is widely utilized in agriculture to effectively manage crop pests, thereby enhancing both the yield and quality of crops. Additionally, research is exploring the use of Pyriftalid in boosting plant resistance to pests and diseases.Formule :C15H14N2O4SCouleur et forme :SolidMasse moléculaire :318.35SARS-CoV-2 nsp3-IN-1
Compound 15c selectively inhibits SARS-CoV-2 nsp3 Mac1 with IC50 of 6.1 μM.Formule :C17H15N5O2Couleur et forme :SolidMasse moléculaire :321.33CM-728
CAS :CM-728 is an oxazanonaphthoquinone that exhibits cytotoxic and antibacterial properties. It acts as a human peroxidase-1 inhibitor and serves as a source of oxidative stress affecting mitochondrial function.Formule :C22H14N2O5Couleur et forme :SolidMasse moléculaire :386.357Chitinase-IN-5
Chitinase-IN-5 (8i) blocks OfChi-h (IC50: 0.051 μM), has insecticidal qualities, useful for eco-friendly pest control.Formule :C20H21ClFN7Couleur et forme :SolidMasse moléculaire :413.88MurA-IN-6
CAS :MurA-IN-6 (Compound L16) is a selective MurA inhibitor with an IC50 of 26.63 μM. It exhibits antibacterial activity by inhibiting the function of MurA, a key protein essential for bacterial cell wall synthesis.Formule :C22H17N3O3SCouleur et forme :SolidMasse moléculaire :403.454LpxA-IN-1
CAS :LpxA-IN-1, a novel UDP-N-acetylglucosamine acyltransferase (LpxA) inhibitor exhibiting potent activity (IC 50 2 nM), effectively targets Pseudomonas aeruginosaFormule :C21H11D7F3N5O3Couleur et forme :SolidMasse moléculaire :452.44Cap-dependent endonuclease-IN-17
CAS :CEN inhibitor IN-17 targets influenza A/H3N2; IC50: 1.29 μM. From patent CN112898346A, DSC701.Formule :C24H20F2N3O7PSCouleur et forme :SolidMasse moléculaire :563.47SAG-524
CAS :SAG-524 is a powerful oral small molecule that inhibits HBV viral replication. In HepG2.2.15 cells, SAG-524 reduced HBV-DNA and HbsAg levels in the supernatant with IC₅₀ values of 0.92 nM and 1.4 nM, respectively [1].Formule :C30H32ClN5O4SCouleur et forme :SolidMasse moléculaire :594.12Antibacterial agent 262
CAS :Antibacterialagent 262 (compound A23) is a potent antibacterial agent that inhibits the activity of Xanthomonas oryzae pv oryzae. It also disrupts the integrity of bacterial cell membranes by preventing the formation of biofilms of Xanthomonas oryzae pv oryzae.Formule :C17H18F2N6O4S3Couleur et forme :SolidMasse moléculaire :504.554LpxH-IN-2
CAS :LpxH-IN-2 (compound 014), a potent inhibitor of LpxH, exhibits antibacterial activity against E. coli.Formule :C27H33ClF2N6O4SCouleur et forme :SolidMasse moléculaire :611.10Antibacterial agent 87
Antibacterial agent 87 is an effective antibacterial agent that acts on MRSA (MIC: 0.125 μg/ml), MRSE (MIC: 0.0625 μg/ml) and S. aureus (MIC: 0.0625 μg/ml).Formule :C31H46N2O6SCouleur et forme :SolidMasse moléculaire :574.77FPI-1465
CAS :FPI-1465: Dual serine-β-lactamase & PBP inhibitor; IC50 PBP2=1.0 μg/mL; Kd CTX-M-15=0.011μM, OXA-48=5.3μM.Formule :C11H18N4O7SCouleur et forme :SolidMasse moléculaire :350.35Lentiginosine
CAS :Lentiginosine is a selective amyloglucosidase inhibitor.Formule :C8H15NO2Couleur et forme :SolidMasse moléculaire :157.21TREX1-IN-3
CAS :TREX1-IN-3 (Compound 95) is an inhibitor of TREX1 and TREX2, with an IC50 of less than 0.1 μM for TREX1 and less than 1 μM for TREX2, as well as an EC50 of less than 1 μM for HCT116 cells. It is applicable for research in the field of cancer.Formule :C24H19ClN6O4Couleur et forme :SolidMasse moléculaire :490.898HPH-15
CAS :HPH-15 is an anti-cell migration compound that inhibits cell movement by binding to hnRNP U or suppressing TGF-β. Additionally, it prevents epithelial-to-mesenchymal transition (EMT). HPH-15 holds potential for research in areas such as anti-tumor metastasis and anti-fibrosis.Formule :C19H31N3S4Couleur et forme :SolidMasse moléculaire :429.73(4-Aminobenzoyl)-D-glutamic acid
CAS :(4-Aminobenzoyl)-D-glutamic acid (Compound 17) exhibits competitive inhibitory activity against the H2-pterin synthesis system, affecting folic acid synthesis and subsequently inhibiting bacterial growth.Formule :C12H14N2O5Couleur et forme :SolidMasse moléculaire :266.25SPB07935
CAS :SPB07935 inhibits plasmepsin II in the malaria-causing parasite Plasmodium falciparum and serves as an antimalarial agent. It affects the life cycle of P. falciparum, hindering the growth of the parasite's FcB1 and 3D7 strains, with IC50 values of 8 μM and 4.7 μM, respectively.Formule :C22H15N5O4S2Couleur et forme :SolidMasse moléculaire :477.516Cap-dependent endonuclease-IN-7
CAS :Cap-dependent endonuclease-IN-7, a potent CEN inhibitor, blocks viral mRNA synthesis and virus spread, with research use for influenza A, B, C.Formule :C36H28FN3O7SCouleur et forme :SolidMasse moléculaire :665.69MT0703
CAS :MT0703 is a cephalosporin antibiotic featuring an aminothiazolylglycyl moiety with a 1,5-dihydroxy-4-pyridinone-2-carbonyl group, displaying potent activity against Pseudomonas species.Formule :C26H25N7O9S3Couleur et forme :SolidMasse moléculaire :675.71AB25583
CAS :AB25583 is a small molecule inhibitor of Polθ helicase (Polθ-hel) with an IC50 of 6 nM. It selectively kills cells deficient in BRCA1/2 and synergizes with Olaparib in cancer cells harboring pathogenic BRCA1/2 mutations. AB25583 can be utilized in tumor research.Formule :C22H17ClN4O3SCouleur et forme :SolidMasse moléculaire :452.91EBOV-IN-10
CAS :EBOV-IN-10 is an orally active inhibitor of the Ebola virus (EBOV) with an EC50 value of 0.19 μM.Formule :C22H22N2O2SCouleur et forme :SolidMasse moléculaire :378.49WQ3810 TFA
WQ3810 TFA is an orally available fluoroquinolone with antimicrobial activity against Mycobacterium tuberculosis and inhibits the DNA rotamase activity ofFormule :C24H23F6N5O5Degré de pureté :99.52%Couleur et forme :SoildMasse moléculaire :575.46KL-50
CAS :KL-50, a selective toxin, effectively targets tumors deficient in the DNA repair protein O6-methylguanine-DNA-methyltransferase (MGMT), which corrects O6-alkylguanine lesions. This compound induces both DNA damage response pathways and cell cycle arrest in MGMT-deficient cells, regardless of mismatch repair (MMR) status. KL-50 shows promise in the study of brain tumors lacking MGMT.Formule :C7H7FN6O2Couleur et forme :SolidMasse moléculaire :226.17NS2B/NS3-IN-3
CAS :NS2B/NS3-IN-3 (Compd 66) is an inhibitor of Flavivirus NS2B-NS3 protease [1] .Formule :C19H21N3O2Couleur et forme :SolidMasse moléculaire :323.39A 76889
CAS :A 76889 is an inhibitor of HIV-1 protease.Formule :C44H58N8O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :794.98Metallo-β-lactamase-IN-14
CAS :Metallo-β-lactamase-IN-14 (Compound 17e) serves as an inhibitor of Metallo-β-Lactamase, displaying inhibitory activity against VIM-1 and VIM-2. This compound also exhibits antibacterial effects on Gram-negative (GN) bacteria and P. aeruginosa [1].Formule :C20H22N8O2S2Couleur et forme :SolidMasse moléculaire :470.57MRL-494
MRL-494, a small-molecule BamA inhibitor, resists efflux and outer membrane permeability, with antibacterial properties.Formule :C26H35FN16O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :622.66Antifungal agent 12
Antifungal agent 12 is a new fluconazole-like compound that exhibits good antifungal effects.Formule :C20H16F3N7O2S2Couleur et forme :SolidMasse moléculaire :507.51MIV-150
CAS :MIV-150 is a nonnucleoside inhibitor of reverse transcriptase (NNRT). MIV-150 also blocking HIV-1 and HIV-2 infections (EC50<1 nM against HIV-1/HIV-2MN).Formule :C19H17FN4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :368.36GSK3739936
CAS :GSK3739936 inhibits HIV-1 integrase (IC50: 11.1 nM, EC50: 1.7 nM), weak on CYP (IC50 >24.3 μM), rapid absorption, moderate clearance, high oral availability.Formule :C34H43FN2O4Couleur et forme :SolidMasse moléculaire :562.71ONO-5334
CAS :ONO-5334: selective cathepsin K inhibitor, potential for osteoporosis study; Ki: 0.10 nM (human), 0.049 nM (rabbit), 0.85 nM (rat).Formule :C21H34N4O4SDegré de pureté :98.22% - 99.60%Couleur et forme :SolidMasse moléculaire :438.58Thiolactomycin
CAS :Thiolactomycin is a novel reversible dual inhibitor of D-amino acid oxidase (DAO) and D-Aspartate oxidase (DDO).Formule :C11H14O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :210.29Antibacterial agent 113
Antibacterial agent 113 targets multiple bacteria including P. aeruginosa and E. coli, showing efficacy at MIC 15625 μM.Formule :C29H18ClN5OCouleur et forme :SolidMasse moléculaire :487.94SARS-CoV-2-IN-99
CAS :SARS-CoV-2-IN-99 (compound 58) is an inhibitor of the main protease of SARS-CoV-2.Formule :C20H16Br2NO4PCouleur et forme :SolidMasse moléculaire :525.13PolQi1
CAS :PolQi1 is a highly efficient and selective Polϴ (DNA polymerase theta) inhibitor with an IC50 of 2 nM, showing potential for cancer therapy.Formule :C18H14ClF5N4O2Degré de pureté :98.97%Couleur et forme :SolidMasse moléculaire :448.77Antitubercular agent-29
Compound 6xa inhibits drug-resistant tuberculosis with MICs 0.03 μg/mL for DS-Mtb and 0.03-0.06 for DR-Mtb, SI>40 for Vero cells.Formule :C20H12ClN3O5Couleur et forme :SolidMasse moléculaire :409.78Urease-IN-1
Urease -IN-1 is a urease inhibitor (IC50: 2.21±0.45 μM).Formule :C17H12BrFN4O2SCouleur et forme :SolidMasse moléculaire :435.27HIV-1 inhibitor-14
HIV-1 inhibitor-14: potent, broad HIV-1 RT inhibitor. IC50=0.14μM. Effective against wild-type and resistant strains, EC50=5.79-28.3nM.Formule :C29H32N6O4SCouleur et forme :SolidMasse moléculaire :560.67HBV-IN-18
HBV-IN-18 (Compound 3) is an HBV capsid assembly modulator (CpAM) (EC50: 2790 nM).Formule :C17H15F6N5O2Couleur et forme :SolidMasse moléculaire :435.32RdRP-IN-5
CAS :RdRP-IN-5 (compound 20), a potent inhibitor of the influenza virus RNA-dependent RNA polymerase (RdRP), has potential application in influenza research [1].Formule :C23H21N3O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :419.43SARS-CoV-2-IN-97
CAS :SARS-CoV-2-IN-97 (Compound CO-01) is an inhibitor of the SARS-CoV-2Nsp15 endoribonuclease, exhibiting an IC50 of 53.5 μM. It demonstrates low cytotoxicity in A549-AT cells with an IC50 value of 134 μM.Formule :C11H3Br2N3OCouleur et forme :SolidMasse moléculaire :352.97N'-(2-Fluorophenyl)pyrazine-2-carbohydrazide
N'-(2-Fluorophenyl)pyrazine-2-carbohydrazide is a Ole1p desaturase inhibitor as well as antifungal agent [1].Formule :C11H9FN4OCouleur et forme :SolidMasse moléculaire :232.21K13787
CAS :K13787 is an acetohydroxy acid synthase (AHAS) inhibitor with antibacterial properties. It exhibits antimicrobial activity against various non-tuberculous mycobacteria (NTM) as well as clarithromycin (CLR) resistant strains.Formule :C14H11F2N5O4SCouleur et forme :SolidMasse moléculaire :383.33HIV-1 inhibitor-44
HIV-1 inhibitor-44 (compound 11l) is an HIV-1 reverse transcriptase inhibitor that exhibits activity against wild-type HIV-1 strains (EC50: 0.209 μM).Formule :C23H26N2O4SCouleur et forme :SolidMasse moléculaire :426.53Lamivudine, (+/-)-trans-
CAS :Lamivudine, a drug for HIV-1 and HBV, inhibits reverse transcriptase and resembles zalcitabine.Formule :C8H11N3O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :229.26AK-968-11563024
CAS :AK-968-11563024 is an inhibitor targeting marine V. vulnificus NAT [(VIBVN)NAT] with an IC50 value of 18.86 µM. In V. vulnificus, NAT (aromatic amine N-acetyltransferase) plays a role in drug metabolism, contributing to drug resistance. Thus, AK-968-11563024 can be used for research related to drug tolerance.Formule :C18H13I2N9O5Couleur et forme :SolidMasse moléculaire :689.162Antifungal agent 13
CAS :Antifungal agent 13 demonstrates significant antifungal activity against Sclerotinia sclerotiorum, achieving an EC50 of 1.25 mg/L.Formule :C21H16ClF3N4OCouleur et forme :SolidMasse moléculaire :432.83GR 122222X
CAS :GR 122222X is an inhibitor of topoisomerase II.Formule :C26H35N5O11SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :625.65MraY-IN-2
MraY-IN-2 (compound 6) is an effective inhibitor of bacterial transposase MraY (IC50=4.5 μ M), and can be used for antibacterial research.Formule :C16H23N3O9Couleur et forme :SolidMasse moléculaire :401.37G092
G092 is a potent inhibitor of MsbA. MsbA is an ABC transporter protein. G092 has potential for antibacterial drug research.Formule :C23H20Cl2N2O3Couleur et forme :SolidMasse moléculaire :443.32AN-12-H5
CAS :AN-12-H5 is an anti-enteroviral compound that targets the replication process of PV and EV71 viruses.Formule :C24H23N3O4S3Couleur et forme :SolidMasse moléculaire :513.65Cefempidone
CAS :Cefempidone (GR 50692) is a third-generation cephalosporin antibiotic. It exhibits antibacterial activity by inhibiting penicillin-binding proteins involved in the synthesis of bacterial cell walls.Formule :C22H21N7O6S2Masse moléculaire :543.587-APRA
CAS :7-APRA is a semisynthetic intermediate of the cephalosporin class of antibiotics. It exhibits antibacterial activity and is primarily used in the synthesis of other cephalosporin antibiotics, such as Cefaclor and Cefprozil.Formule :C10H12N2O3SMasse moléculaire :240.28Elongation factor P-IN-2
Elongation factor P-IN-2, a β-lysine derivative, is a potent EFP inhibitor reducing E. coli growth.Formule :C16H35N3O2Couleur et forme :SolidMasse moléculaire :301.47Griseofulvic Acid
CAS :Griseofulvic Acid ((±)-Griseofulvic acid) is a metabolite of the antifungal agent Griseofulvin. It induces protein aggregation and tubulin polymerization in cell-free assays.Formule :C16H15ClO6Masse moléculaire :338.74(Z)-Lanoconazole
(Z)-Lanoconazole, an imidazole antifungal for dermatophytosis and onychomycosis, inhibits fungal ergosterol production.Formule :C14H10ClN3S2Couleur et forme :SolidMasse moléculaire :319.835-Fluorouridine 5'-phosphate
CAS :5-Fluorouridine 5'-phosphate acts as an ODCase (uridine 5'-monophosphate decarboxylase) inhibitor, exhibiting a Ki value of 98 µM for human ODCase and 645 µM for Methanococcus jannaschii ODCase. This compound also shows inhibitory activity on leukemia and lymphoma cell lines, making it useful for cancer research studies.Formule :C9H12FN2O9PCouleur et forme :SolidMasse moléculaire :342.172DENV-IN-6
CAS :DENV-IN-6, a potent anti-DENV (I-IV) and HIV-1 IIIB inhibitor with EC50 ranging 6.8-17.5 μM for DENV and EC50 0.0181 μM for HIV-1.Formule :C23H26ClFN4OSCouleur et forme :SolidMasse moléculaire :461Plm IV inhibitor-2
CAS :"Plm IV inhibitor-2: Potent for Plm IV (IC50=24nM), affects Plm II/Plm I; malaria research compound."Formule :C39H54N4O4Couleur et forme :SolidMasse moléculaire :642.87VNI
CAS :VNI is an effective inhibitor of CYP51. It suppresses sterol synthesis in Trypanosoma cruzi, exhibiting anti-Trypanosoma cruzi activity.Formule :C26H19Cl2N5O2Couleur et forme :SolidMasse moléculaire :504.37TAN-1057C
CAS :TAN-1057C is a potent antibiotic with antimicrobial activity against both Gram-negative and Gram-positive bacteria, including Methicillin-resistant Staphylococcus aureus (MRSA).Formule :C13H25N9O3Couleur et forme :SolidMasse moléculaire :355.4Secutrelvir
CAS :Secutrelvir inhibits the 3CL protease (3CL protease), thereby exhibiting antiviral activity by preventing the replication of SARS-CoV-2.Formule :C23H16Cl2F3N5O2Couleur et forme :SolidMasse moléculaire :522.307Antifungal agent 43
Antifungal agent 43 inhibits biofilms with low toxicity to human cancer cells.Formule :C24H26N4Se2Couleur et forme :SolidMasse moléculaire :528.41Carumonam Sodium
CAS :Carumonam Sodium is a monobactam, penicillin-binding protein inhibitor. It is used as antibacterials.Formule :C12H12N6Na2O10S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :510.37Lavendomycin
CAS :Lavendomycin can be extracted from Streptomyces lavendulae and has active against Gram-positive bacteria.Formule :C29H50N10O8Couleur et forme :SolidMasse moléculaire :666.77RAD51-IN-6
CAS :RAD51-IN-6, a potent RAD51 gene inhibitor, may help research mitochondrial disorders. (WO2021164746A1, cmpd 23)Formule :C27H40N3O5PSCouleur et forme :SolidMasse moléculaire :549.66Dioxidine
CAS :Dioxidine is an antimicrobial agent that can inhibit bacterial growth. It is utilized in research on pyogenic infections.Formule :C10H10N2O4Couleur et forme :SolidMasse moléculaire :222.197HIV-1 inhibitor-52
CAS :HIV-1 inhibitor-52: potent, broad-spectrum with EC50s 1.6-6.4 nM against various HIV-1 strains.Formule :C46H72FNO5SCouleur et forme :SolidMasse moléculaire :770.13SMCypI C31
SMCypIC31, a non-peptide cyclophilin inhibitor, blocks PPIase at 0.1 μM IC50 and fights various HCV genotypes (EC50: 1.20-7.76 μM).Formule :C27H30N4O2SCouleur et forme :SolidMasse moléculaire :474.62NDM-1 inhibitor-3
NDM-1 inhibitor-3 is a New Delhi Metallo-β-lactamase-1 (NDM-1) inhibitor (Ki : 4 μM) widely found in nature and is associated with antibiotic resistance.Formule :C16H12O4Degré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :268.26HBV-IN-31
CAS :HBV-IN-31: strong cccDNA inhibitor, anti-HBV, IC50=0.13 µM HBsAg, hampers cell growth.Formule :C23H18ClNO6Couleur et forme :SolidMasse moléculaire :439.85
