Récepteur d'adénosine
Les récepteurs de l'adénosine sont une classe de récepteurs GPCR qui répondent à la nucléoside endogène adénosine. Ces récepteurs sont impliqués dans la régulation de divers processus physiologiques, y compris la fonction cardiovasculaire, les cycles veille-sommeil et les réponses immunitaires. Les modulateurs des récepteurs de l'adénosine ont un potentiel thérapeutique pour traiter des affections telles que les arythmies cardiaques, l'inflammation et les maladies neurodégénératives. Chez CymitQuimica, nous offrons une sélection de modulateurs des récepteurs de l'adénosine de haute qualité pour soutenir vos recherches en biologie cardiovasculaire, neurosciences et immunologie.
242 produits trouvés pour "Récepteur d'adénosine"
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CGS 15943
CAS :<p>CGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor.</p>Formule :C13H8ClN5ODegré de pureté :97.4%Couleur et forme :SolidMasse moléculaire :285.69Pentoxifylline
CAS :<p>Pentoxifylline (PTX) stimulates cytokines, inhibits phosphodiesterase, enhances blood flow, and increases cell flexibility.</p>Formule :C13H18N4O3Degré de pureté :99.26% - 99.93%Couleur et forme :SolidMasse moléculaire :278.31Acefylline
CAS :<p>Acefylline (Theophylline-7-acetic acid), a stimulant drug of the xanthine chemical class, acts as an adenosine receptor antagonist.</p>Formule :C9H10N4O4Degré de pureté :99.57%Couleur et forme :White Crystalline SolidMasse moléculaire :238.2AB928
CAS :<p>AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].</p>Formule :C23H22N8ODegré de pureté :98.09% - >99.99%Couleur et forme :SolidMasse moléculaire :426.47N6-Ethyladenosine
CAS :<p>N6-Ethyladenosine is an adenosine derivative, acts as an agonist of Adenosine receptor(hA1AR and hA3AR with Kis of 4.9 and 4.7 nM , respectively).</p>Formule :C12H17N5O4Degré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :295.29DPTN dihydrochloride
CAS :<p>DPTN dihydrochloride is a potent and selective A3AR antagonist with Ki values of 1.65, 9.61 and 8.53 nM in human, mouse and rat, respectively.</p>Formule :C22H20Cl2N4OSDegré de pureté :99.95%Couleur et forme :SoildMasse moléculaire :459.39Amp579 TFA
<p>Amp579 TFA is a novel adenosine A1/A2a receptor agonist that induces acute and delayed preconditioning against myocardial shock in vivo.</p>Formule :C24H29ClF3N5O5SDegré de pureté :96.56%Couleur et forme :SoildMasse moléculaire :592.03Theophylline
CAS :<p>Theophylline (1,3-Dimethylxanthine) is a methyl xanthine derivative from tea with diuretic, smooth muscle relaxant, bronchial dilation, cardiac and central</p>Formule :C7H8N4O2Degré de pureté :99.65% - 99.98%Couleur et forme :White Solid PowderMasse moléculaire :180.16YT 146
CAS :<p>YT 146 is a biochemical.</p>Formule :C18H25N5O4Degré de pureté :98.81% - 99.25%Couleur et forme :SolidMasse moléculaire :375.42Diphylline
CAS :<p>Diphylline is a bronchodilator with mild vasodilator and diuretic properties, used for asthma, bronchitis, and emphysema.</p>Formule :C10H14N4O4Degré de pureté :98.54%Couleur et forme :Crystals From Alcohol SolidMasse moléculaire :254.24Adenosine A1 receptor activator T62
CAS :<p>Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor, and it produces antinociception in animal models of acute pain and also</p>Formule :C15H14ClNOSDegré de pureté :97.83%Couleur et forme :SolidMasse moléculaire :291.8Adenosine 5'-monophosphate monohydrate
CAS :<p>Adenosine 5'-monophosphate monohydrate (5'-AMP) , also known as 5'-adenylic acid, is a nucleotide that is used as a monomer in RNA.</p>Formule :C10H14N5O7P·H2ODegré de pureté :97.68% - 98.49%Couleur et forme :White PowderMasse moléculaire :365.24Theophylline monohydrate
CAS :<p>Theophylline monohydrate (Quibron) appears to inhibit phosphodiesterase and prostaglandin production, regulate calcium flux and intracellular calcium</p>Formule :C7H8N4O2·H2ODegré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :198.18Ticlopidine hydrochloride
CAS :<p>Ticlopidine hydrochloride (Ticlodix) is an effective inhibitor of platelet aggregation commonly used in the placement of STENTS in CORONARY ARTERIES.</p>Formule :C14H15Cl2NSDegré de pureté :99.85% - >99.99%Couleur et forme :White PowderMasse moléculaire :300.25Aminophylline
CAS :<p>Aminophylline (Phyllocontin) is a competitive nonselective phosphodiesterase inhibitor giving a bronchodilatory effect.</p>Formule :C7H8O2·C2H8N2Degré de pureté :99.31%Couleur et forme :White Or Slightly Yellowish Granules Or Powder SolidMasse moléculaire :420.43Quercetin-3'-o-phosphate TEA
<p>Quercetin-3'-o-phosphate TEA (Quercetin 3'-phosphate TEA) is an adenosine A receptor antagonist that can be used to prevent and treat metabolic disorders.</p>Formule :C21H26NO10PDegré de pureté :95.63%Couleur et forme :SoildMasse moléculaire :483.41Pamabrom
CAS :<p>Pamabrom is a diuretic for premenstrual and menstrual bloating, swelling, and fullness.</p>Formule :C11H18BrN5O3Degré de pureté :99.84% - >99.99%Couleur et forme :CoaMasse moléculaire :348.2Doxofylline
CAS :<p>Doxofylline (Doxophylline) is a methylxanthine derivative with the presence of a dioxolane group in position 7.</p>Formule :C11H14N4O4Degré de pureté :99.958% - >99.99%Couleur et forme :SolidMasse moléculaire :266.25N6-Cyclohexyladenosine
CAS :<p>N6-Cyclohexyladenosine (CHA) is a selective agonist of A1 receptor with EC50 of 8.2 Nm.</p>Formule :C16H23N5O4Degré de pureté :99.84% - 99.98%Couleur et forme :SolidMasse moléculaire :349.38Adenosine receptor antagonist 1
CAS :<p>A2aR-selective antagonist with IC50 of 0.29 nM; 14x more selective over A2bR.</p>Formule :C22H15ClFN7OCouleur et forme :SolidMasse moléculaire :447.86Theophyllol
CAS :<p>Theophyllol (theophylline sodium acetate) can alter calcium levels in subcellular fractions of rat brain cortex.</p>Formule :C9H10N4Na2O4Couleur et forme :SolidMasse moléculaire :284.183F6-9G5
<p>3F6-9G5 is a humanized monoclonal antibody targeting AA2AR/Adenosine A2aR, used in neurodegenerative disease research.</p>Degré de pureté :>95%Couleur et forme :Odour LiquidHeterobivalent ligand-1
<p>Heterobivalent ligand-1 targets A2A-D2 receptor heteromer with affinity: Kd for A2A=2.1 nM, D2=0.13 nM.</p>Formule :C86H115FN16O21Couleur et forme :SolidMasse moléculaire :1727.93PSB 0777 ammonium salt
CAS :<p>adenosine A2A receptor full agonist</p>Formule :C18H24N6O7S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :500.55AR ligand 40
<p>AR ligand 40 (compound 19c) is an Adenosine A1 Receptor ligand with antagonistic activity. It exhibits antiproliferative effects on SW480, SW48, HCT116, K562, MDA-MB-231, and A549 cells, with EC50 values of 7, 10, 12, 13, 15, and 39 μM, respectively.</p>Formule :C21H25N5Couleur et forme :SolidMasse moléculaire :347.211MRS-1706
CAS :<p>MRS-1706: Ki of 1.39nM for A2B; selective inverse agonist; also affects A2A, A1, A3.</p>Formule :C27H29N5O5Degré de pureté :99.00%Couleur et forme :SolidMasse moléculaire :503.55A2A/A3 AR antagonist-1
<p>A2A/A3 AR antagonist-1 is a dual fluorescent AR ligand with K i of 90 nM (hA2A) & 31.8 nM (hA3).</p>Formule :C56H71N15O12S2Couleur et forme :SolidMasse moléculaire :1210.39Norisoboldine hydrochloride
CAS :<p>Norisoboldine hydrochloride: an oral AhR agonist from Radix Linderae, for Rheumatoid arthritis and Ulcerative colitis research.</p>Formule :C18H20ClNO4Couleur et forme :SolidMasse moléculaire :349.81A3AR agonist 2
<p>Compound 19, a selective A3 Adenosine Receptor (A3AR) agonist (K i : 22.1 nM), effectively stimulates β-arrestin2 recruitment with an EC 50 value of 4.36 nM.</p>Formule :C34H34N6O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :622.67LUF7690
CAS :<p>LUF7690 (Compound 9), a clickable and covalent affinity-based probe (AfBP) for the human A3 adenosine receptor (hA3AR), facilitates the detection and</p>Formule :C25H24FN5O6SCouleur et forme :SolidMasse moléculaire :541.55Apadenoson TFA
<p>Apadenoson TFA is a potent adenosine A2A receptor (A2AR) agonist that can be used to improve survival in patients infected with SARS.</p>Formule :C25H31F3N6O8Degré de pureté :98.08%Couleur et forme :SoildMasse moléculaire :600.55Xanthine amine congener dihydrochloride
CAS :<p>XAC dihydrochloride is an Adenosine A1 and A2 receptor antagonist with IC50s of 1.8 nM and 114 nM, also a mouse convulsant.</p>Formule :C21H30Cl2N6O4Couleur et forme :SolidMasse moléculaire :501.41FSCPX
CAS :<p>FSCPX is a potent and selective irreversible antagonist of the A1 adenosine receptor (A1AR), exhibiting low nanomolar binding potency.</p>Formule :C23H27FN4O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :506.55ABT-702
CAS :<p>ABT-702 is an orally active, competitive, and reversible non-nucleoside adenosine kinase (AK) inhibitor analgesic and anti-inflammatory.</p>Formule :C22H19BrN6ODegré de pureté :99.57%Couleur et forme :SoildMasse moléculaire :463.33PSB 0777 ammonium hydrate
<p>PSB 0777 ammonium hydrate is a potent and selective adenosine A2A receptor full agonist, exhibiting K i values of 44.4 nM for rat A2A receptors and 360 nM for</p>Formule :C18H20N5O7S2·NH4·75H2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :532.09Adenosine receptor agonist 1
<p>Compound 6m, an A3 adenosine receptor (AR) partial agonist, exhibits a K i value of 6.7 nM as an adenosine receptor agonist.</p>Formule :C12H14ClN5O2SeCouleur et forme :SolidMasse moléculaire :374.68A3AR modulator 1
<p>MRS8054 is an oral A3 adenosine receptor positive allosteric modulator, enhancing Cl-IB-MECA-induced activity.</p>Formule :C23H25IN4Couleur et forme :SolidMasse moléculaire :484.38hA3AR agonist 2
<p>hA3AR agonist 2 is a potent activator of A3AR, with a Ki value of 3.5 nM.</p>Formule :C11H14ClN5O2SCouleur et forme :SolidMasse moléculaire :315.78N6-Benzyl-5'-ethylcarboxamido adenosine
CAS :<p>N6-Benzyl-5'-ethylcarboxamido adenosine is a selective A3 adenosine receptor agonist.</p>Formule :C19H22N6O4Couleur et forme :SolidMasse moléculaire :398.428-Chloro caffeine
CAS :<p>8-Chloro caffeine binds to adenosine receptors with a Ki of 30 µM. It enhances UV-induced chromosomal aberrations in the Cl-I type Chinese hamster embryo lung cells. 8-Chloro caffeine is a derivative of the methylxanthine alkaloid caffeine.</p>Formule :C8H9ClN4O2Couleur et forme :SolidMasse moléculaire :228.64GW-328267
CAS :<p>GW-328267 is an agonist of the adenosine A2 receptor.</p>Formule :C21H26N10O4Couleur et forme :SolidMasse moléculaire :482.5Xanthine amine congener trihydrochloride
CAS :<p>Xanthine amine congener trihydrochloride: potent adenosine antagonist, reverses effects of N6-cyclohexyladenosine on urine, sodium excretion, heart rate.</p>Formule :C21H29ClN6O4Degré de pureté :98.81%Couleur et forme :SolidMasse moléculaire :464.95A3AR agonist 1
<p>A3AR Agonist 1 (Compound 12), with a Ki of 25.8 nM, is a potent A3 adenosine receptor (A3AR) agonist that promotes β-arrestin2 recruitment with an effective</p>Formule :C28H34N6O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :550.61Danshenol B
<p>Danshenol B is a natural product that can be used as a reference standard.</p>Formule :C22H26O4Couleur et forme :SolidMasse moléculaire :354.446A-286501
CAS :<p>A-286501: Oral adenosine kinase inhibitor, IC50=0.47 nM, reduces pain via non-opioid, non-NSAID ADO receptors.</p>Formule :C11H14BrN5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :328.17LUF6096
CAS :<p>LUF6096 (CF-602) is a potent allosteric enhancer of the adenosine A3 receptor, exhibiting the capability to enhance agonist binding allosterically while</p>Formule :C22H21Cl2N3ODegré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :414.33LAS101057
CAS :<p>LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma.</p>Formule :C18H14FN5ODegré de pureté :99.03% - >99.99%Couleur et forme :SolidMasse moléculaire :335.34GR79236
CAS :<p>GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.</p>Formule :C15H21N5O5Couleur et forme :SolidMasse moléculaire :351.36MRS-3777 hemioxalate
CAS :<p>MRS-3777 hemioxalate, a selective adenosine A3 receptor antagonist, reverses the anti-injury perception effects of its corresponding agonist and serves as a valuable tool for studying inflammatory pain.</p>Formule :C17H19N5OC2H2O4Degré de pureté :97.10%Couleur et forme :SolidMasse moléculaire :354.39(Rac)-Mirabegron-d5
CAS :<p>(Rac)-Mirabegron D5 is a deuterium labeled (Rac)-Mirabegron. Mirabegron is a selective agonist of β3-adrenoceptor.</p>Formule :C21H24N4O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :401.54CCPA
CAS :<p>CCPA (2-chloro-N(6)cyclopentyladenosine) is a potent and selective agonist of adenosine A1 receptor</p>Formule :C15H20ClN5O4Degré de pureté :99.1%Couleur et forme :Off-White To Light Yellow SolidMasse moléculaire :369.8A2B receptor antagonist 2
CAS :<p>A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).</p>Formule :C12H15N5Degré de pureté :100%Couleur et forme :SolidMasse moléculaire :229.28CPI-444
CAS :<p>CPI-444 (V81444) is an antagonist of the adenosine A2A receptor.It reduces tumor area in mouse model of murine Her2/neu-expressing breast cancer.</p>Formule :C20H21N7O3Degré de pureté :98.78%Couleur et forme :SolidMasse moléculaire :407.43Regadenoson hydrate
CAS :<p>Regadenoson is an A2A adenosine receptor agonist, a coronary vasodilator commonly used in pharmacologic stress testing.</p>Formule :C15H20N8O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :408.37Tecadenoson
CAS :<p>Tecadenoson (CVT-510) is a selective agonist of A1 adenosine receptor.</p>Formule :C14H19N5O5Degré de pureté :98.83%Couleur et forme :SolidMasse moléculaire :337.33Derenofylline
CAS :<p>Derenofylline is a selective and potent adenosine A(1) antagonist in vitro (Ki=1 nM)</p>Formule :C18H20N4ODegré de pureté :98.09%Couleur et forme :SolidMasse moléculaire :308.385-Iodotubercidin
CAS :<p>5-Iodotubercidin (NSC-113939) is a potent adenosine kinase inhibitor with IC50 of 26 nM.</p>Formule :C11H13IN4O4Degré de pureté :99.98%Couleur et forme :Tan SolidMasse moléculaire :392.15DPCPX
CAS :<p>DPCPX (PD 116948) is an A1 adenosine receptor antagonist</p>Formule :C16H24N4O2Degré de pureté :99.23% - 99.93%Couleur et forme :White SolidMasse moléculaire :304.39Proxyphylline
CAS :<p>Proxyphylline (7-(2-Hydroxypropyl)theophylline) is a dual of adenosine A1/A2a receptor inhibitor and phosphodiesterase (PDE) inhibitor.</p>Formule :C10H14N4O3Degré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :238.24ABT-702 dihydrochloride
CAS :<p>ABT-702 dihydrochloride is a potent adenosine kinase (AK) inhibitor.</p>Formule :C22H21BrCl2N6ODegré de pureté :98.42% - 98.98%Couleur et forme :SolidMasse moléculaire :536.25ZM241385
CAS :<p>ZM-241385 is a high-affinity antagonist ligand selective for the adenosine A2A receptor.</p>Formule :C16H15N7O2Degré de pureté :97.02% - 99.69%Couleur et forme :SolidMasse moléculaire :337.34N6,N6-Dimethyladenosine
CAS :<p>N6,N6-Dimethyladenosine is find in mycobacterium bovis Bacille Calmette-Guérin tRNA.</p>Formule :C12H17N5O4Degré de pureté :98.79%Couleur et forme :White PowderMasse moléculaire :295.29CGS 21680 Hydrochloride
CAS :<p>CGS 21680 Hydrochloride (CGS 21680 HCl)(IC50=22 nM), an adenosine receptor agonist, exhibits 140-fold potency in A2 receptor over A1 receptor.</p>Formule :C23H29N7O6·HClDegré de pureté :96.74% - 99.53%Couleur et forme :SolidMasse moléculaire :535.98Piclidenoson
CAS :<p>Piclidenoson (CF-101), a selective agonist of adenosine A3 receptor(EC50 values of 0.11 μM), induces robust anti-inflammatory effect in psoriasis patients.</p>Formule :C18H19IN6O4Degré de pureté :99.83% - ≥95%Couleur et forme :SolidMasse moléculaire :510.29Swertisin
CAS :<p>Swertisin: an herbal molecule with antihyperglycemic, antidiabetic, anti-inflammatory, and antioxidant properties; blocks adenosine A1 receptor.</p>Formule :C22H22O10Degré de pureté :99.74% - 99.89%Couleur et forme :SolidMasse moléculaire :446.42-Chloroadenosine
CAS :<p>2-Chloroadenosine (CADO) is a metabolically stable analog of adenosine that binds to adenosine A1, A2A, and A3 receptors( Ki:300, 80, and 1,900 nM, respectively</p>Formule :C10H12ClN5O4Degré de pureté :99.23%Couleur et forme :White PowderMasse moléculaire :301.69VPC171
CAS :<p>VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).</p>Formule :C18H12F3NOSDegré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :347.35BAY-545
CAS :<p>BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59 nM).</p>Formule :C18H22F3N3O4SDegré de pureté :98.05%Couleur et forme :SolidMasse moléculaire :433.451-Ethyl-6-aminouracil
CAS :<p>1-Ethyl-6-aminouracil (6-AMINO-1-ETHYL-1H-PYRIMIDINE-2,4-DIONE) is an intermediate in the synthesis of a series of new substituted Xanthines which have high</p>Formule :C6H9N3O2Degré de pureté :99.29%Couleur et forme :SolidMasse moléculaire :155.15Regadenoson
CAS :<p>Regadenoson (CVT-3146) is a selective A2A receptor agonist that increases coronary blood flow with a longer half-life than adenosine.</p>Formule :C15H18N8O5Degré de pureté :99.57% - 99.81%Couleur et forme :Off-White SolidMasse moléculaire :390.355'-N-Ethylcarboxamidoadenosine
CAS :<p>NECA, an adenosine receptor agonist, boosts brain extravasation of fluorescein and dextran without affecting the blood-brain barrier.</p>Formule :C12H16N6O4Degré de pureté :98.95% - ≥95%Couleur et forme :PowderMasse moléculaire :308.29Namodenoson
CAS :<p>Namodenoson (2-Cl-IB-MECA) is an adenosine A3 receptor agonist.</p>Formule :C18H18ClIN6O4Degré de pureté :98.97%Couleur et forme :SolidMasse moléculaire :544.73Taminadenant
CAS :<p>Taminadenant is an adenosine receptor antagonist.</p>Formule :C10H8BrN7Degré de pureté :99.11%Couleur et forme :SolidMasse moléculaire :306.12CHEMBL241987
CAS :<p>CHEMBL241987 targets the Adenosine receptor A3 (human)</p>Formule :C16H11N3ODegré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :261.28Xanthine amine congener hydrochloride
CAS :<p>Xanthine amine congener (XAC) hydrochloride is a non-selective adenosine receptor antagonist that induces convulsions in mice.</p>Formule :C21H29ClN6O4Couleur et forme :SolidMasse moléculaire :464.95Vipadenant
CAS :<p>Vipadenant (CEB-4520)(BIIB-014) is an adenosine A2a antagonist with Ki of 1.3 nM; less potent for A1(Ki=69 nM).</p>Formule :C16H15N7ODegré de pureté :97.25% - 97.36%Couleur et forme :SolidMasse moléculaire :321.34Fostamatinib
CAS :<p>Fostamatinib (R788)(IC50 of 41 nM), which is a prodrug of the active metabolite R406, is a Syk inhibitor. It does not work on Lyn.</p>Formule :C23H26FN6O9PDegré de pureté :93.08% - 99.38%Couleur et forme :SolidMasse moléculaire :580.46MIPS521
CAS :<p>MIPS521 ({2-Amino-4-[3,5-bis(trifluoromethyl)phenyl]thiophen-3-yl}(4-chlorophenyl)methanone) is a positive allosteric modulator of the A1R.</p>Formule :C19H10ClF6NOSDegré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :449.88-Cyclopentyl-1,3-dimethylxanthine
CAS :<p>8-Cyclopentyl-1,3-dimethylxanthine (CPT) is a potent antagonist of adenosine A1 receptor.</p>Formule :C12H16N4O2Degré de pureté :98.58% - >99.99%Couleur et forme :SolidMasse moléculaire :248.28Adenosine receptor antagonist 4
CAS :<p>Adenosine receptor antagonist 4 is an adenosine receptor antagonist.</p>Formule :C10H13N3Degré de pureté :99.63% - 99.65%Couleur et forme :Off-White PowderMasse moléculaire :175.23Inosine
CAS :<p>Inosine (NSC-20262), an endogenous purine nucleoside produced by the catabolism of adenosine, is an agonist of adenosine receptors A1R and A2AR. Low-Cost!</p>Formule :C10H12N4O5Degré de pureté :99.51% - 99.89%Couleur et forme :SolidMasse moléculaire :268.23Binodenoson
CAS :<p>Binodenoson (WRC 0470), a selective A2A adenosine receptor agonist, aids in coronary imaging.</p>Formule :C17H25N7O4Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :391.42PD 117519
CAS :<p>PD 117519 (CI947) is an agonist of adenosine receptor</p>Formule :C19H21N5O4Degré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :383.4Preladenant
CAS :<p>Preladenant (SCH-420814) is an orally bioavailable antagonist of the adenosine A2A receptor (Ki: 1.1 nM) and has >1000-fold selectivity over all other adenosine</p>Formule :C25H29N9O3Degré de pureté :98.02% - 99.68%Couleur et forme :SolidMasse moléculaire :503.56Nitrobenzylthioinosine
CAS :<p>Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.</p>Formule :C17H17N5O6SDegré de pureté :99.69% - 99.74%Couleur et forme :Off-White SolidMasse moléculaire :419.41Adenosine amine congener
CAS :<p>Adenosine amine congener (ADAC) (ADAC) is an agonist of selective A1 adenosine receptor,.</p>Formule :C28H32N8O6Degré de pureté :97.86%Couleur et forme :SolidMasse moléculaire :576.6Alloxazine
CAS :<p>Alloxazine (Isoalloxazine) is an A2 receptor antagonist, which is approximately 10-fold more selective for the A2B receptor than for the A2A receptor.</p>Formule :C10H6N4O2Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :214.18SDZ WAG 994
CAS :<p>SDZ WAG 994 is an A1 adenosine receptor agonist.</p>Formule :C17H25N5O4Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :363.41Istradefylline
CAS :<p>Istradefylline (KW-6002)(Ki of 2.2 nM) is a selective adenosine A2A receptor (A2AR) antagonist, which is under development in Phase 3 trails.</p>Formule :C20H24N4O4Degré de pureté :98.18% - 99.95%Couleur et forme :SolidMasse moléculaire :384.43Norisoboldine
CAS :<p>Norisoboldine, potential rheumatoid arthritis therapy, protects joints and modulates immunity by inhibiting MAPKs, not NF-κB.</p>Formule :C18H19NO4Degré de pureté :98.12% - 99.7%Couleur et forme :SolidMasse moléculaire :313.35SCH442416
CAS :<p>SCH442416: selective A2A adenosine receptor antagonist; Ki: 0.048 nM (human), 0.5 nM (rat).</p>Formule :C20H19N7O2Degré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :389.41Tozadenant
CAS :<p>Tozadenant (SYN115) is an adenosine A2A receptor antagonist(Ki of 11.5 nM and 6 nM on human and rhesus,respectively)</p>Formule :C19H26N4O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :406.5SCH 58261
CAS :<p>SCH 58261 is a potent and selective A2a adenosine receptor antagonist.The Ki =2.3 nM for rat A2a and 2 nM is for bovine A2a.</p>Formule :C18H15N7ODegré de pureté :99.07% - 99.75%Couleur et forme :SolidMasse moléculaire :345.36Enprofylline
CAS :<p>Enprofylline (Enprofilina), a bronchodilator, acts primarily as a competitive nonselective phosphodiesterase inhibitor.</p>Formule :C8H10N4O2Degré de pureté :98.37%Couleur et forme :SolidMasse moléculaire :194.19Capadenoson
CAS :<p>Capadenoson (BAY 68-4986) is a selective adenosine-A1 receptor agonist.</p>Formule :C25H18ClN5O2S2Degré de pureté :98.85% - 99.57%Couleur et forme :SolidMasse moléculaire :520.03Reversine
CAS :<p>Reversine, a small synthetic purine analogue (2, 6-disubstituted purine), is a potent inhibitior of Aurora A/B/C(IC50s=150-500 nM).</p>Formule :C21H27N7ODegré de pureté :98% - 98.42%Couleur et forme :SolidMasse moléculaire :393.49AZD4635
CAS :<p>AZD4635 (HTL1071) is a new-type adenosine 2A receptor (A2AR) inhibitor(Ki=1.7 nM).</p>Formule :C15H11ClFN5Degré de pureté :99.15% - 99.90%Couleur et forme :SolidMasse moléculaire :315.735'-Amino-5'-deoxyadenosine
CAS :<p>5'-Amino-5'-deoxyadenosine (NH2dAdo) is an adenosine kinase inhibitor targeting malignant tumors of the inert lymphatic system with antitumor and anticancer</p>Formule :C10H14N6O3Degré de pureté :95.55%Couleur et forme :SolidMasse moléculaire :266.26Rolofylline
CAS :<p>Rolofylline (KW-3902) is an adenosine A1 receptor antagonist used to study acute congestive heart failure and renal dysfunction.</p>Formule :C20H28N4O2Degré de pureté :99.53%Couleur et forme :SolidMasse moléculaire :356.46Theobromine
CAS :<p>Theobromine (3,7-Dimethylxanthine), a xanthine alkaloid, is used as a bronchodilator and as a vasodilator.</p>Formule :C7H8N4O2Degré de pureté :99.69% - 99.91%Couleur et forme :White To Yellow Crystalline PowderMasse moléculaire :180.16Trabodenoson
CAS :<p>Trabodenoson (INO-8875) is a selective and potent adenosine A1 receptor agonist, an adenosine analog, for the study of primary open-angle glaucoma.</p>Formule :C15H20N6O6Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :380.36Blontuvetmab
CAS :<p>Blontuvetmab (AT 004), a caninized CD20 monoclonal antibody, is utilized in the study of Canine B-cell lymphoma [1].</p>Couleur et forme :LiquidTC-G 1004
CAS :<p>adenosine A2A receptors antagonist</p>Formule :C22H27N7O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :421.5A2AR-agonist-1
CAS :<p>A2AR-agonist-1 targets A2A Receptor/ENT1 for neuroprotection; potent with Ki of 4.39 (A2AR), 3.47 (ENT1).</p>Formule :C20H22N6O4Degré de pureté :99.9%Couleur et forme :SolidMasse moléculaire :410.43hA2A/hCA XII modulator 1
CAS :<p>Potent hA2AAR antagonist & hCA XII inhibitor; Ki: hA2AAR 6.4 nM, hCA XII 6.2 nM. Possible cancer research use.</p>Formule :C24H19N7O4SCouleur et forme :SolidMasse moléculaire :501.52IHCH-3064
CAS :<p>IHCH-3064: dual-action cancer immunotherapy, A2AR affinity (Ki 2.2 nM), selective HDAC1 inhibitor (IC50 80.2 nM).</p>Formule :C25H21N9O2Couleur et forme :SolidMasse moléculaire :479.49MRS 1334
CAS :<p>antagonist for the human adenosine A3 receptor</p>Formule :C31H26N2O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :522.55LUF6000
CAS :<p>LUF6000 is an allosteric modulator of the human A3 adenosine receptor (AR).</p>Formule :C22H20Cl2N4Couleur et forme :SolidMasse moléculaire :411.33A2A/A1 AR antagonist-1
CAS :<p>A2A/A1 AR antagonist-1 is a potent dual antagonist for ischemic stroke research with Ki values of 5.58 nM (A2A) and 24.2 nM (A1).</p>Formule :C15H12N6O2Couleur et forme :SolidMasse moléculaire :308.29LUF 5834
CAS :<p>A2A and A2B adenosine receptor partial agonist</p>Formule :C17H12N6OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :348.385'-(N-Cyclopropyl)carboxamidoadenosine
CAS :<p>adenosine A2 receptor agonist</p>Formule :C13H16N6O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :320.3A1AR antagonist 5
CAS :<p>A1AR antagonist 5 (compound 20) is a potent and selective antagonist of A1 adenosine receptor (A1AR) with a pKi of 6.11 and a pIC 50 of 5.83 [1].</p>Formule :C17H15ClN4OCouleur et forme :SolidMasse moléculaire :326.78A1AR antagonist 3
CAS :<p>Compound 13: selective A1AR antagonist, Ki human A1: 9.69 nM, rat A1: 0.529 nM, useful for neurological research.</p>Formule :C25H20N2O3SCouleur et forme :SolidMasse moléculaire :428.5XCC
CAS :<p>XCC is an Adenosine receptor antagonist.</p>Formule :C19H22N4O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :386.4A1AR antagonist 4
CAS :<p>Compound 22: A1AR antagonist, pIC50 5.51, pKi 6.29, potent and selective.</p>Formule :C23H25N3O2Couleur et forme :SolidMasse moléculaire :375.46MRS1097
CAS :<p>MRS1097 is a selective antagonist A3 adenosine receptor.</p>Formule :C26H27NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :417.5MRS-1191
CAS :<p>MRS-1191 is an effective and selective A3 adenosine receptor antagonist (KB: 92 nM, a Ki: 31.4 nM for human A3 receptor and an IC50: 120 nM for CHO cells).</p>Formule :C31H27NO4Couleur et forme :SolidMasse moléculaire :477.55Apadenoson
CAS :<p>Apadenoson: potent A2 agonist, A3 inhibitor (IC 45 nM), anti-inflammatory, for neurological research.</p>Formule :C23H30N6O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :486.52Lu AA 47070
CAS :<p>adenosine A2A receptor antagonist</p>Formule :C17H20F2N3O6PSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :463.39A1AR antagonist 2
CAS :<p>Compound 18h is a potent A1 adenosine receptor blocker with Ki of 1.49 nM for hA1, 10.2 nM for hA2A, 50.1 nM for hA2B.</p>Formule :C17H12N4OCouleur et forme :SolidMasse moléculaire :288.3Adenosine receptor inhibitor 1
CAS :<p>Potent, selective adenosine receptor blocker with strong affinity, especially A2A (Ki 68.5 nM). Promising for cancer, neurodegeneration study.</p>Formule :C17H19ClFN5O3Couleur et forme :SolidMasse moléculaire :395.82A1/A3 AR antagonist 2
CAS :<p>The compound is an a1/a3 adenosine receptor antagonist, which helps to treat (neurological) inflammatory diseases.</p>Formule :C22H16N2O3SCouleur et forme :SolidMasse moléculaire :388.44AB-MECA
CAS :<p>AB-MECA is a high affinity A3 adenosine receptor agonist. It has high affinity for recombinant A1 and A3 receptors.</p>Formule :C18H21N7O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :399.4A2AAR/HDAC-IN-1
CAS :<p>A2AAR/HDAC-IN-1 (compound 14c) is an orally active, balanced A2AAR/HDAC dual inhibitor of A2AAR (Ki: 163.5 nM), HDAC1 (IC50: 145.3 nM). effect.</p>Formule :C24H21N7O2Couleur et forme :SolidMasse moléculaire :439.47LASSBio-1359
CAS :<p>LASSBio-1359 is an adenosine receptor agonist. It acts by inducing relaxation of the corpus cavernosum. It also acts as a novel selective phosphodiesterase.</p>Formule :C17H18N2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :298.34PSB 11 hydrochloride
CAS :<p>PSB 11 hydrochloride is a human adenosine A3 receptor antagonist.</p>Formule :C16H18ClN5ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :331.8Adenosine receptor antagonist 3
CAS :<p>Adenosine receptor antagonist 3 has the potential for cancer disease research which is a potent adenosine receptor antagonist [1].</p>Formule :C16H14N6SCouleur et forme :SolidMasse moléculaire :322.39Adentri
CAS :<p>Adentri is a novel antagonist of adenosine A1 receptor with unique diuretic activity.</p>Formule :C18H24N4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :344.41A2A receptor antagonist 3
CAS :<p>A2A receptor antagonist 3 (Example 92) is an adenosine A2a receptor antagonist (Ki: 0.4 nM). receptor (Ki: 1467 nM).</p>Formule :C26H26N6O2Couleur et forme :SolidMasse moléculaire :454.52MRS1186
CAS :<p>MRS1186 is an effective and selective antagonist of the human Adenosine A3 receptor (Ki: 7.66 nM).</p>Formule :C16H12ClN5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :341.75Adenosine receptor A1 antagonist 5
CAS :<p>1,3-Dipropyl-8-phenylxanthine is an adenosine antagonist, oxypurine, insecticide, and reduces high blood pressure.</p>Formule :C17H20N4O2Degré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :312.37MRS1177
CAS :<p>MRS1177 is an effective and selective antagonist of the human Adenosine A3 receptor (hA3AR) (Ki: 0.3 nM).</p>Formule :C20H12ClN5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :389.79XU1
CAS :<p>XU1（Benzo[c][1,8]naphthyridin-6(5h)-One） is an Aurora protein kinase inhibitor used for the treatment of diseases suitable for inhibition, regulation or</p>Formule :C12H8N2ODegré de pureté :98.58% - 99.59%Couleur et forme :SolidMasse moléculaire :196.2HEMADO
CAS :<p>HEMADO is a potent and selective agonist of adenosine A3 receptor (Ki: 1.1 nM at the human A3 subtype).</p>Formule :C17H23N5O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :361.4A1AR antagonist 6
CAS :<p>A1AR antagonist 6 (compound 15) is a potent and selective antagonist of A1 adenosine receptor(A1AR) with a pKi of 7.13 and a pIC 50 of 6.38[1].</p>Formule :C17H15N3O2Couleur et forme :SolidMasse moléculaire :293.32Lu AA41063
CAS :<p>Lu AA41063 is a potent and selective antagonist of the hA2A receptor.</p>Formule :C16H17F2N3O2SCouleur et forme :SolidMasse moléculaire :353.39Neladenoson dalanate HCl
CAS :<p>Neladenoson dalanate HCl is a potent, selective, orally active partial agonist of adenosine A1 receptor (EC50: 0.1 nM).</p>Formule :C35H35Cl2N7O4S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :752.73A3AR antagonist 1
CAS :<p>A3AR antagonist 1 is a potent and selective human A3adenosine receptor (AR) antagonist (Ki: 4.63) and has no affinity for the rat A3AR.</p>Formule :C32H24N4O4SCouleur et forme :SolidMasse moléculaire :560.62Adenosine receptor antagonist 2
CAS :<p>Adenosine receptor antagonist 2 is an orally active A2a (IC50: 1 nM), A2b (IC50: 3 nM) adenosine receptor antagonist that exhibits antitumour effects.</p>Formule :C23H21FN8OCouleur et forme :SolidMasse moléculaire :444.46CAY10498
CAS :<p>A3 AR antagonist CAY10498, with Ki of 37 nM, is 60-200x selective over A1/A2A receptors; no dedifferentiation effects shown.</p>Formule :C18H20N6Couleur et forme :SolidMasse moléculaire :320.39VUF8507
CAS :<p>Vuf8507 is an allosteric regulator of adenosine receptor.</p>Formule :C21H15N3OCouleur et forme :SolidMasse moléculaire :325.36PD 81723
CAS :<p>Allosteric potentiator at the adenosine A1 receptor</p>Formule :C14H12F3NOSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :299.31Sipagladenant
CAS :<p>Sipagladenant: oral inverse agonist for A2A adenosine receptor, may aid frontal lobe dysfunction research.</p>Formule :C20H19N3O4SCouleur et forme :SolidMasse moléculaire :397.45SCH-202676 HBr
CAS :<p>SCH-202676 HBr is an allosteric agonist. It also an GPCR antagonist.</p>Formule :C15H13N3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :267.35A3AR antagonist 2
CAS :<p>A3AR antagonist 2 is a potent antagonist of the human A3 adenosine receptor, exhibiting a Ki value of 4.54 nM.</p>Formule :C22H16N6O3Couleur et forme :SolidMasse moléculaire :412.4TH-162
CAS :<p>TH-162 (R)-PIA is an A1 adenosine receptor agonist with ~100× higher affinity than its (+)-isomer.</p>Formule :C19H23N5O4Couleur et forme :SolidMasse moléculaire :385.42PQ-69
CAS :<p>PQ-69 is a selective adenosine A1 receptor antagonist with inverse agonist activity.</p>Formule :C20H19FN4OCouleur et forme :SolidMasse moléculaire :350.39MRS 1523
CAS :<p>MRS 1523: selective adenosine A3 antagonist, Ki 18.9/113 nM (human/rat), blocks N-type Ca channels & inhibits action potentials in rat DRG neurons.</p>Formule :C23H29NO3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :399.55Inupadenant
CAS :<p>Inupadenant is an orally active, highly selective A2A receptor antagonist. Inupadenant is not brain-penetrant. Inupadenant has potent anti-tumor activity[1].</p>Formule :C25H26F2N8O4S2Couleur et forme :SolidMasse moléculaire :604.65CAY10680
CAS :<p>CAY10680 inhibits MAO-B (IC50=34.9 nM) & A2A receptors (Ki=39.5 nM), sparing other adenosine types & MAO-A, may treat Parkinson's.</p>Formule :C18H16N2O2SCouleur et forme :SolidMasse moléculaire :324.4FR-194921
CAS :<p>FR-194921: potent oral adenosine A1 antagonist, improves cognition, reduces anxiety, similar efficacy in humans, rats, mice.</p>Formule :C23H23N5OCouleur et forme :SolidMasse moléculaire :385.46CVT-2759
CAS :<p>CVT-2759, potential A(1)-ADOR partial agonist, could slow ventricular rate without severe cardiac side effects.</p>Formule :C17H24N6O6Couleur et forme :SolidMasse moléculaire :408.41Adenosine receptor inhibitor 2
CAS :<p>Compound 14b is a potent AR inhibitor with dual affinity, stronger for A1 (Ki = 52.2 nM) than A2A (Ki = 167 nM) ARs.</p>Formule :C17H20BrN5O2Couleur et forme :SolidMasse moléculaire :406.28Acefylline piperazine
CAS :<p>Acefylline piperazine, a less toxic theophylline derivative, treats asthma and bronchitis by bronchodilation, stimulating respiration and CNS.</p>Formule :C9H10N4O4·xC4H10N2Couleur et forme :SolidMasse moléculaire :562.54JNJ-40255293
CAS :<p>JNJ-40255293 is an antagonist of adenosine A2A/A1.</p>Formule :C23H22N4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :402.45AK-IN-1
CAS :<p>AK-IN-1: competitive adenosine inhibitor, not ATP; inhibits AK 86-89% at 2-10 µM; promising for ischaemia, inflammation, seizure research.</p>Formule :C22H21N3O4Couleur et forme :SolidMasse moléculaire :391.42ATL-801
CAS :<p>ATL-801 is anselective antagonist of A2B receptor with herapeutic activity for colitis.</p>Formule :C24H25N7O3Couleur et forme :SolidMasse moléculaire :459.5Kira8 Hydrochloride
CAS :<p>Kira8 Hydrochloride is a mono-selective IRE1α inhibitor that allosterically attenuates IRE1α RNase activity with an IC50 of 5.9 nM.</p>Formule :C31H30Cl2N6O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :637.58A2AAR/HDAC-IN-2
CAS :<p>A2AAR/HDAC-IN-2: potent dual A2AAR/HDAC inhib., Ki 10.3 nM, IC50 18.5 nM, anti-tumor potential.</p>Formule :C23H26N6O4Couleur et forme :SolidMasse moléculaire :450.49Theophylline sodium glycinate
CAS :<p>Theophylline sodium glycinate inhibits PDE3, treats asthma/COPD, blocks adenosine receptors, activates HDAC, reduces inflammation and induces apoptosis.</p>Formule :C9H12N5NaO4Couleur et forme :SolidMasse moléculaire :277.216hA2AAR antagonist 1
CAS :<p>Compound 4a, also known as hA2AAR antagonist 1, is a highly selective hA2AAR antagonist with a Ki value of 5 nM. It is useful in the field of immuno-oncology research.</p>Formule :C15H15N5OCouleur et forme :SolidMasse moléculaire :281.31LUF5831
CAS :<p>LUF5831 is an agonist of adenosine A1 receptor.</p>Formule :C15H12N4O2SCouleur et forme :SolidMasse moléculaire :312.35Draflazine
CAS :<p>Draflazine: ENT1 inhibitor, reverses hypersensitivity in CFA and carrageenan-induced hyperalgesia.</p>Formule :C30H33Cl2F2N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :604.52LUF5981
CAS :<p>LUF5981 is a selective agonist of human adenosine A1 receptor.</p>Formule :C24H23N3Couleur et forme :SolidMasse moléculaire :353.46Cirazoline hydrochloride
CAS :<p>Cirazoline hydrochloride is a synthetic competitive full agonist of α1A-AR (Ki 120 nM) and partial agonist at α1B-AR and α1D-AR.</p>Formule :C13H17ClN2ODegré de pureté :99.863%Couleur et forme :SolidMasse moléculaire :252.74Bamifylline Hydrochloride
CAS :<p>Bamifylline Hydrochloride, an adenosine A1 receptor antagonist, is uesd to treat bronchiectasis and chronic obstructive pulmonary disease.</p>Formule :C20H28ClN5O3Couleur et forme :SolidMasse moléculaire :421.92MRS1067
CAS :<p>MRS1067 is an antagonist of A3 adenosine receptor.</p>Formule :C19H16Cl2O3Couleur et forme :SolidMasse moléculaire :363.23MRE3008F20
CAS :<p>MRE3008F20 is an AA3R antagonist that inhibits Cl-IB-MECA-induced cAMP production and can be used to study glaucoma and asthma.</p>Formule :C21H20N8O3Degré de pureté :97.29%Couleur et forme :SolidMasse moléculaire :432.44A2AR-antagonist-1
CAS :<p>Oral A2AR-antagonist-1, IC50 29 nM; anti-tumor, stable in mice (t1/2 86.1 min), boosts T cells, impedes LAG-3/TIM-3.</p>Formule :C27H25N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :451.52VUF 5574
CAS :<p>VUF 5574 is a selective antagonist of adenosine A3 receptor with a Ki of 4.03 nM for the recombinant human receptor.</p>Formule :C21H17N5O2Degré de pureté :99.53%Couleur et forme :SolidMasse moléculaire :371.39ST3932
CAS :<p>ST3932 is a ST1535 metabolite, is a adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively).</p>Formule :C12H16N8ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :288.31APNEA
CAS :<p>APNEA ((2R,3R,4S,5R)-2-[6-[2-(4-aminophenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol) is a non-selective agonist of adenosine A3 receptor.</p>Formule :C18H22N6O4Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :386.41N6-Cyclopentyladenosine
CAS :<p>N6-Cyclopentyladenosine (CPA) is a selective agonist of the adenosine A1 receptor and can be used to mimic the action of the adenosine A1 receptor, with Ki's of</p>Formule :C15H21N5O4Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :335.36Sonedenoson
CAS :<p>Sonedenoson (MRE0094) is an adenosine A(2A) receptor agonist and potential inhibitor potentially targeting SARS-CoV-2 coronavirus 2;-O-ribose methyltransferase.</p>Formule :C18H20ClN5O5Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :421.84Evodenoson
CAS :<p>Evodenoson (ATL313), a potent A2aR agonist, treats eye diseases, tumors, and immune disorders; potential for glaucoma and blood cancer studies.</p>Formule :C23H29N7O6Degré de pureté :99.75% - 99.83%Couleur et forme :SolidMasse moléculaire :499.52N-[(4-Aminophenyl)methyl]adenosine
CAS :<p>N-[(4-Aminophenyl)methyl]adenosine is an adenosine receptor inhibitor (Ki: 29 nM for Rat ecto-5′-Nucleotidase).</p>Formule :C17H20N6O4Degré de pureté :98.75%Couleur et forme :SolidMasse moléculaire :372.38BAY 60-6583
CAS :<p>BAY 60-6583 is a potent, high-affinity adenosine A2B receptor agonist (EC50 = 3 nM) with affinity for A2B receptors that exceeds that for A1, A2A, and A3</p>Formule :C19H17N5O2SDegré de pureté :98.46% - 99.8%Couleur et forme :SolidMasse moléculaire :379.44ANR 94
CAS :<p>ANR94 is a potent hAA2AR antagonist (Ki 46 nM) with potential for Parkinson's research.</p>Formule :C9H13N5ODegré de pureté :98.9%Couleur et forme :SolidMasse moléculaire :207.23Adenosine antagonist-1
CAS :<p>Adenosine antagonist-1 acts as an adenosine A3 receptor (AA3R) antagonist.</p>Formule :C18H13N7SDegré de pureté :99.28% - 99.95%Couleur et forme :SolidMasse moléculaire :359.41ST-1535
CAS :<p>ST 1535: potent, oral A2A adenosine receptor antagonist with antiparkinsonian and antitremor effects, promising for Parkinson's research.</p>Formule :C12H16N8Degré de pureté :99.64% - 99.69%Couleur et forme :SolidMasse moléculaire :272.31MRS1220
CAS :<p>MRS1220, a selective and potent antagonist for the human A3 adenosine receptor (hA3AR) with a dissociation constant (Ki) of 0.59 nM, exhibits therapeutic</p>Formule :C21H14ClN5O2Degré de pureté :98.43%Couleur et forme :SolidMasse moléculaire :403.82N 0861
CAS :<p>N 0861 is a selective adenosine A1 receptor antagonist that attenuates renal insufficiency during adenosine-controlled hypotension in rats.</p>Formule :C13H17N5Degré de pureté :98.78%Couleur et forme :SolidMasse moléculaire :243.31Selodenoson
CAS :<p>Selodenoson (RG-14202) is a selective adenosine A1 receptor agonist used to slow the heart rate in patients with atrial fibrillation and to treat arrhythmias.</p>Formule :C17H24N6O4Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :376.41ISAM-140
CAS :<p>ISAM-140 is a potent and highly selective antagonist of A2B adenosine receptor.</p>Formule :C19H19N3O3Degré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :337.37GW-493838
CAS :<p>GW-493838 is a potent adenosine A1A receptor agonist for the treatment of dyslipidemia and neuropathic pain, with analgesic effects on post-herpetic neuralgia</p>Formule :C21H21ClFN7O4Degré de pureté :99.11% - 99.58%Couleur et forme :SolidMasse moléculaire :489.89GS-9667
CAS :<p>GS-9667, a selective and partial agonist of the A(1) adenosine receptor (AR), represents an effective therapy for Type 2 diabetes (T2DM) and dyslipidemia via</p>Formule :C21H24FN5O4SDegré de pureté :99.76% - 99.77%Couleur et forme :SolidMasse moléculaire :461.51A2A receptor antagonist 1
CAS :<p>A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.</p>Formule :C16H12FN5ODegré de pureté :99.52% - 99.93%Couleur et forme :SolidMasse moléculaire :309.3LAS38096
CAS :<p>LAS38096 is an A2B adenosine receptor antagonist (Ki : 17 nM) that is potent, selective and efficient .</p>Formule :C17H12N6ODegré de pureté :99.18% - 99.95%Couleur et forme :SolidMasse moléculaire :316.32N6-(2-Phenylethyl)adenosine
CAS :<p>N6-(2-Phenylethyl)adenosine (N6-Phenethyladenosine) is an adenosine derivative and an agonist of adenosine receptors with Ki values of 11.8 nM and 30.1 nM for</p>Formule :C18H21N5O4Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :371.392'-MeCCPA
CAS :<p>2'-MeCCPA is an A1AR agonist that inhibits trichothecene-stimulated adenylate cyclase activity and has analgesic activity for the study of HCV.</p>Formule :C16H22ClN5O4Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :383.83KI-7
CAS :<p>KI-7 is an adenosine A2B receptor positive allosteric modulator.</p>Formule :C23H18N2O2Degré de pureté :98.33%Couleur et forme :SolidMasse moléculaire :354.4FK-453
CAS :<p>FK-453 is a potent antagonist of non-xanthine adenosine A1 receptor with diuretic and renal vasodilatory activity.</p>Formule :C23H25N3O2Degré de pureté :99.44%Couleur et forme :SolidMasse moléculaire :375.46GP3269
CAS :<p>GP3269 is a selective, potent, orally active human adenosine kinase (AK) inhibitor (IC50: 11 nM) with anticonvulsant effects in rats.</p>Formule :C23H21FN4O3Couleur et forme :SolidMasse moléculaire :420.44PSB-1115 potassium salt
CAS :<p>PSB-1115 potassium salt, a selective A2B Adenosine Receptor antagonist, inhibits the 2,4,6-trinitrobenzenesulfonic acid (TNBS)-induced contraction inhibition of acetylcholine (ACh) [1].</p>Formule :C14H13KN4O5SCouleur et forme :SolidMasse moléculaire :388.44MRS3558
CAS :<p>MRS3558 is an agonist of A3 adenosine receptors.</p>Formule :C20H20Cl2N6O3Couleur et forme :SolidMasse moléculaire :463.32ABT-702 hydrochloride
CAS :<p>ABT-702 hydrochloride effectively inhibits adenosine kinase, exhibiting an IC50 value of 1.7 nM [1] [2].</p>Formule :C22H20BrClN6OCouleur et forme :SolidMasse moléculaire :499.79KFM19
CAS :<p>KFM19 is a potent and selective adenosine receptor (A1-receptor) antagonist (IC50 : 50 nM) for the study of neurological disorders.</p>Formule :C16H22N4O3Degré de pureté :98.62%Couleur et forme :SolidMasse moléculaire :318.37Neladenoson dalanate
CAS :<p>Neladenoson dalanate (BAY-1067197), an oral Adenosine A1 receptor partial agonist, is safe with good pharmacokinetics for chronic heart disease.</p>Formule :C35H34ClN7O4S2Couleur et forme :SolidMasse moléculaire :716.27Sulmazole
CAS :<p>Sulmazole (AR-L 115-BS) is a small molecule Sulmazole is a small molecule cGMP-PDE inhibitor.Sulmazole is a competitive inhibitor of A1 adenosine receptors.</p>Formule :C14H13N3O2SDegré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :287.34Xanthine amine congener
CAS :<p>Xanthine amine congener is an Adenosine receptor antagonist.</p>Formule :C21H28N6O4Degré de pureté :99.7%Couleur et forme :SolidMasse moléculaire :428.48
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