Récepteur cannabinoïde
Les récepteurs cannabinoïdes sont des GPCR qui médiatisent les effets des cannabinoïdes endogènes (endocannabinoïdes) et des phytocannabinoïdes, tels que ceux trouvés dans le cannabis. Les deux principaux types de récepteurs cannabinoïdes, CB1 et CB2, sont impliqués dans la régulation d'une large gamme de processus physiologiques, y compris la perception de la douleur, l'appétit, l'humeur et la fonction immunitaire. Les modulateurs des récepteurs cannabinoïdes ont un potentiel thérapeutique dans le traitement de conditions telles que la douleur chronique, l'épilepsie et la sclérose en plaques. Chez CymitQuimica, nous offrons une large gamme de modulateurs de récepteurs cannabinoïdes de haute qualité pour soutenir vos recherches en neuropharmacologie, gestion de la douleur et immunologie.
217 produits trouvés pour "Récepteur cannabinoïde"
Trier par
Degré de pureté (%)
0
100
|
0
|
50
|
90
|
95
|
100
CB1 antagonist 2
CAS :CB1 antagonist 2 (AM4113) is caimabinoid 1 (CB1) antagonist which inhibits CB1 in vivo with an IC50 of 25.5 nM.Formule :C17H12Cl3N3ODegré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :380.66Pregnenolone
CAS :Pregnenolone (Arthenolone) is an endogenous steroid hormone synthesized from cholesterol, used in the treatment of Alzheimer's disease.Formule :C21H32O2Degré de pureté :99.5% - 99.84%Couleur et forme :SolidMasse moléculaire :316.48JHU 75528
CAS :JHU 75528 (JHU-75528) is a novel PET tracer with inhibitory effects on CB that can be used to study the cannabinoid system in schizophrenic patients.Formule :C23H21Cl2N5O2Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :470.35EHP-101
CAS :EHP-101 is a PPARγ/CB2 dual agonist with anti-inflammatory properties, inhibits fat formation, and combats diet-related obesity.Formule :C28H35NO3Degré de pureté :98.36%Couleur et forme :SolidMasse moléculaire :433.58Ref: TM-T13289
1mg107,00€5mg227,00€10mg378,00€25mg620,00€50mg868,00€100mg1.169,00€1mL*10mM (DMSO)250,00€Rimonabant
CAS :Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.Formule :C22H21Cl3N4ODegré de pureté :98% - 99.91%Couleur et forme :White Or Almost White Crystalline PowderMasse moléculaire :463.796-Iodopravadoline
CAS :6-Iodopravadoline (AM630) is an antagonist of CB2 (Ki: 31.2 nM). And it shows 165-fold selectivity more than CB1 receptors.Formule :C23H25IN2O3Degré de pureté :99.29%Couleur et forme :Off-White SolidMasse moléculaire :504.36Ref: TM-T14204
1mg38,00€2mg52,00€5mg70,00€10mg90,00€25mg198,00€50mg326,00€100mg520,00€1mL*10mM (DMSO)99,00€Rimonabant hydrochloride
CAS :Rimonabant hydrochloride (SR 141716A) 是中心大麻素受体 1 的高效选择性反向激动剂， Ki 值为1.8 nM。它也能够抑制分枝杆菌膜蛋白3。Formule :C22H22Cl4N4ODegré de pureté :98.24% - 99.5%Couleur et forme :Off-White To White Crystalline PowderMasse moléculaire :500.25Anandamide
CAS :Anandamide ((5Z,8Z,11Z,14Z)-N-(2-Hydroxyethyl)icosa-5,8,11,14-tetraenamide), an immune modulator, acts via not only cannabinoid receptors (CB1 and CB2) but alsoFormule :C22H37NO2Degré de pureté :95.037% - 99.22%Couleur et forme :Light Yellow OilMasse moléculaire :347.53Ref: TM-T14046
1mg34,00€2mg46,00€5mg67,00€10mg117,00€25mg221,00€50mg330,00€100mg485,00€200mg675,00€1mL*10mM (DMSO)73,00€CB2 PET Radioligand 1
CB2 PET Radioligand 1 (compound [18F]9) is a positron emission tomography (PET) radioligand with high affinity for the human cannabinoid receptor 2 (hCB2, Ki=7.Formule :C20H19F3N4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :388.39Hemopressin (human, mouse)
CAS :Endogenous peptide, inhibits ep24.15/24.16/ACE with Ki of 27.76/3.43/1.87 μM. Lowers blood pressure, CB1 inverse agonist, reduces pain in vivo.Formule :C50H79N13O12Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1054.26CB2R agonist 3
CB2R agonist 3, a potent activator of cannabinoid receptor 2 (CB2R), exhibits an EC50 value of 0.37μM, indicative of its significant role in the immune system [Degré de pureté :98%Couleur et forme :Odour SolidPSB-SB-1203
CAS :PSB-SB-1203 (Compound 25b) is a dual CB1/CB2 ligand that blocks the CB1 receptor and activates the CB2 receptor with a CB1 Ki of 0.244 μM, a CB2 Ki of 0.210 μM, and an EC50 of 0.054 μM. It shows potential for research in obesity and cancer.Formule :C25H30O4Couleur et forme :SolidMasse moléculaire :394.5GPR55 agonist 4
GPR55 agonist 4 (Compound 28), with an EC50 of 131 nM for hGPR55 and 1.41 nM for rGPR55, effectively induces β-arrestin recruitment to human GPR55 [1].Formule :C19H16FN5O2Couleur et forme :SolidMasse moléculaire :365.36Cannabigerorcin
CAS :Cannabigerorcin, a phytocannabinoid, serves as an analytical reference standard. It is designated for research and forensic applications.Formule :C17H24O2Couleur et forme :SolidMasse moléculaire :260.377Calcitonin-13C6,15N4 TFA
Calcitonin-13CIC6,15NIC4(salmon) (Salmon calcitonin-13CIC6,15NIC4) TFA is a version of calcitonin(salmon) labeled with carbon-13 and nitrogen-15. This hormone regulates calcium and acts dualistically as an agonist to both amylin and calcitonin receptors, promoting bone formation while inhibiting bone resorption.Formule :C1401C5H240N4315NO48S2·5C2HF3O2Couleur et forme :SolidMasse moléculaire :4007.93Zevaquenabant
CAS :Zevaquenabant (S-MRI-1867): oral CB1/iNOS antagonist combatting obesity-induced CKD.Formule :C25H21ClF3N5O2SCouleur et forme :SolidMasse moléculaire :547.98Hemopressin(human, mouse) TFA
CAS :Hemopressin TFA: nonapeptide from hemoglobin, oral CB1 inverse agonist, eases inflammatory pain.Formule :C52H80F3N13O14Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1168.27GFB-024
GFB-024 is a humanized antibody targeting CB1, which can be used to study obesity.Couleur et forme :LiquidMasse moléculaire :146.12 kDaNESS 0327
CAS :NESS 0327 is a high selectivity antagonist of the cannabinoid CB1 receptor. NESS 0327 is more than 60,000-fold selective for the CB1 receptor.Formule :C24H23Cl3N4ODegré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :489.82(−)-6α-hydroxy Cannabidiol
CAS :(−)-6α-Hydroxy Cannabidiol, an analytical reference standard and a phytocannabinoid metabolite, serves primarily as a metabolite of cannabidiol (CBD). This product is designed for use in research and forensic applications.Formule :C21H30O3Couleur et forme :SolidMasse moléculaire :330.46exo-Tetrahydrocannabivarin
CAS :exo-Tetrahydrocannabivarin (Compound 12) is an analog of Δ9,11-THC. It weakly binds to cannabinoid receptors (CB) with an IC50 of 1.4 μM. In mice, exo-Tetrahydrocannabivarin exhibits activity related to both motor function and analgesia.Formule :C19H26O2Couleur et forme :SolidMasse moléculaire :286.41VIP36
VIP36 is an agonist of the cannabinoid type 1 receptor (CB1) with analgesic properties. It reduces the recruitment of inhibitory proteins, thereby exerting its pain-relieving effects, and is applicable in research related to chronic pain.Formule :C27H35FN6O4Couleur et forme :SolidMasse moléculaire :526.603Δ8-THC-C8
CAS :Δ8-THC-C8 is a semi-synthetic cannabinoid. It acts as an agonist for the cannabinoid receptor 1 (CB1) with an EC50 value of 13.8 nM.Formule :C24H36O2Couleur et forme :SolidMasse moléculaire :356.54RVD-Hpα
CAS :N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist.Formule :C65H105N19O17Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1424.66CB2 receptor antagonist 2
Compound 39, also known as CB2 receptor antagonist 2, is a potent CB2 antagonist exhibiting an IC50 of 0.33 μM.Couleur et forme :Odour SolidN-(1-(3,4-Dihydroxyphenyl)propan-2-yl)oleamide
CAS :N-(1-(3,4-Dihydroxyphenyl)propan-2-yl)oleamide: binds CB1 (Ki=365 nM), activates PPARα (EC50=698 nM), reduces rat food intake, no FAAH inhibition.Formule :C27H45NO3Couleur et forme :SolidMasse moléculaire :431.661Cannabigerorcinic Acid
CAS :Cannabigerorcinic acid, structurally akin to recognized phytocannabinoids, serves as an analytical reference standard designed for research and forensic purposes.Formule :C18H24O4Couleur et forme :SolidMasse moléculaire :304.386(R)-Zevaquenabant
(R)-Zevaquenabant ((R)-MRI-1867) is the enantiomer of Zevaquenabant. Zevaquenabant ((S)-MRI-1867) is a peripherally restricted, orally bioavailable dual antagonist of the cannabinoid CB1 receptor and inducible nitric oxide synthase (iNOS). It is beneficial in improving chronic kidney disease (CKD) caused by obesity.Couleur et forme :Odour SolidCB2R agonist 2
CB2R agonist 2 (cis-17-para) is a CB2R agonist [1].Degré de pureté :98%Couleur et forme :Odour SolidCB2R/FAAH modulator-3
CAS :CB2R/FAAH modulator-3 (compound 27) is a modulator targeting at CB2R and FAAH.Formule :C22H31NO2Degré de pureté :99.81%Couleur et forme :SoildMasse moléculaire :341.49Vicasinabin
CAS :Vicasinabin: potent CB2 agonist; researches chronic pain, atherosclerosis, bone mass, neuroinflammation.Formule :C15H22N10OCouleur et forme :SolidMasse moléculaire :358.41CB2 receptor agonist 2
CAS :CB2 receptor agonist 2 (ZINC72105556): potent, Ki=8.5 nM, high selectivity for CB2.
Formule :C30H36N2O4Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :488.62Drinabant
CAS :Drinabant (AVE-1625) is an orally active CB1 receptor antagonist.Formule :C23H20Cl2F2N2O2SDegré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :497.38Cannabinol methyl ether
CAS :Cannabinol methyl ether, a phytocannabinoid, serves as an analytical reference standard. This compound can be obtained through isolation from Cannabis plants, derived from cannabinol, or synthesized. The physiological and toxicological properties of cannabinol methyl ether remain unknown. It is designed exclusively for research and forensic applications.Formule :C22H28O2Couleur et forme :SolidMasse moléculaire :324.5Hemopressin(rat)
CAS :Peptide inhibitor for ep24.15, neurolysin & ACE with Ki 27.76, 3.43, 1.87 μM. Lowers blood pressure, modulates CB1 receptor, reduces pain & food intake.Formule :C53H77N13O12Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1088.27Tocrifluor T1117
CAS :Fluorescent form of AM 251, CB1 receptor antagonistFormule :C56H53Cl2N7O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :974.97(±)-9-Nor-9α-hydroxy Hexahydrocannabinol
CAS :(±)-9-Nor-9α-hydroxy Hexahydrocannabinol is a cannabinoid-structured compound that exhibits potent cannabinoid-like activity in both dogs and mice.Formule :C20H30O3Couleur et forme :SolidMasse moléculaire :318.45CB2R/FAAH modulator-1
CAS :CB2R/FAAH modulator-1: agonizes CB2R, inhibits FAAH (IC50=4 μM), alters cytokine production; used in inflammation research. Ki: CB2R=14.8 nM, CB1R=241.3 nM.Formule :C24H27NO2Degré de pureté :99.77%Couleur et forme :SoildMasse moléculaire :361.48Ref: TM-T67896
1mg50,00€5mg105,00€10mg154,00€25mg224,00€50mg314,00€100mg427,00€200mg575,00€1mL*10mM (DMSO)108,00€Noladin ether
CAS :Noladin ether (2-AG ether) is a cannabinoid CB1 receptor agonist.Formule :C23H40O3Couleur et forme :SolidMasse moléculaire :364.56CB1R agonist 1
CB1R agonist 1 (Compound '1350) is a potent full agonist of the cannabinoid-1 receptor (CB1R) with a Ki value of 0.95 nM. It demonstrates significant pain-relieving effects in various pain models, including acute thermal pain, inflammatory pain, and neuropathic pain.Formule :C20H18F3N3O3SCouleur et forme :SolidMasse moléculaire :437.4358β-Hydroxy-exo-THC
CAS :8β-Hydroxy-exo-THC, a cannabinoid ether analog, exhibits weak affinity for receptor sites with an IC50 of 1.2 μM.Formule :C21H30O3Couleur et forme :SolidMasse moléculaire :330.46CB2R probe 1
CAS :CB2R Probe 1, a cannabinoid 2 receptor (CB2R) fluorescent probe, exhibits both safety and environmental friendliness, boasting a dissociation constant (K i) of
Formule :C36H42N4O4Couleur et forme :SolidMasse moléculaire :594.74TRPV1/CB2 agonist 1
TRPV1/CB2 agonist 1 (compound 41) is a dual agonist targeting hTRPV1 and CB2 receptors, with an EC50 value of 26.8 μM for hTRPV1. It is applicable in research related to the nervous system.Couleur et forme :Odour SolidCB2R/FAAH modulator-2
CAS :CB2R/FAAH modulator-2 (compound 26) is a dual modulator targeting at CB2R and FAAH.Formule :C24H33NO2Degré de pureté :99.15%Couleur et forme :SoildMasse moléculaire :367.52Afubiata
CAS :ADB-FUBIATA is a synthetic cannabinoid studied for its metabolic profile, along with AFUBIATA, CH-FUBIATA, and CH-PIATA. This in vitro analysis by Watanabe S, et al., examines these compounds, as published in "Arch Toxicol," 2023 Dec;97(12):3085-3094.Formule :C27H29FN2OCouleur et forme :SolidMasse moléculaire :416.53APP-FUBINACA
CAS :APP-FUBINACA is a cannabinoid receptor agonist, classified as a phenylalanine amide-based indazole-3-carboxamide derivative. It exhibits neurostimulatory effects.Formule :C24H21FN4O2Couleur et forme :SolidMasse moléculaire :416.45δ8-THC acetate
CAS :Delta8-THC acetate (Delta8-tetrahydrocannabinol) is a psychoactive cannabinoid that binds to the cannabinoid receptor 1 (CB1 receptor) and exhibits anti-nausea, appetite-stimulating, and anti-inflammatory effects. It may also offer neuroprotective benefits and has potential applications in research on anxiety and depression.Formule :C23H32O3Couleur et forme :SolidMasse moléculaire :356.5CB1R antagonist 2
CB1R antagonist 2 (Compound 11g) functions as an antagonist of the cannabinoid receptor 1 (CB1R), inhibiting the MAPK/NF-κB signaling pathway and exhibiting anti-inflammatory properties. In RAW264.7 cells, it suppresses LPS-induced expression of IL-6, IL-1β, and TNF-α. In murine models, it improves OVA-induced allergic rhinitis.Formule :C24H26N4OCouleur et forme :SolidMasse moléculaire :386.49Δ8-THC methyl ether
CAS :Δ8-THC methyl ether (compound 3) demonstrates a strong docking score of -10.167 kcal/mol for the CB2 receptor. Additionally, Δ8-THC methyl ether exhibits antinociceptive activity in mice.Formule :C22H32O2Couleur et forme :SolidMasse moléculaire :328.49CB2 receptor agonist 9
CAS :CB2 receptor agonist 9 (Compound 33) is an orally active agonist of cannabinoid receptor 2 (CB2 receptor) with an EC50 of 16.2 nM. It inhibits the expression of TNF-α, IL-1β, and IL-6, demonstrating anti-inflammatory activity in a DSS-induced acute colitis model in mice.Formule :C16H23N3O2SCouleur et forme :SolidMasse moléculaire :321.44Δ9-THCH
CAS :Δ9-THCH, a phytocannabinoid analytical reference standard, is present in a Cannabis variety cultivated for medicinal use. In the United States, it is classified as a Schedule I compound. This product is designated for research and forensic applications.Formule :C22H32O2Couleur et forme :SolidMasse moléculaire :328.49CB1-IN-3
CB1-IN-3 (Compound 6i) is a potent inhibitor of the cannabinoid receptor type 1 (CB1). It holds potential for research in obesity, inflammation, and neurological disorders.Couleur et forme :Odour SolidCannabidivarinic acid
CAS :Cannabidivarinic acid (CBDVA), the carboxylic acid precursor to cannabidivarin (CBDV), is a non-psychoactive cannabinoid found in Cannabis and known for its anti-inflammatory properties.Formule :C20H26O4Couleur et forme :SolidMasse moléculaire :330.42Taranabant racemate
CAS :Taranabant racemate is an antagonist and/or inverse agonist of the Cannabinoid-1 (CB1) receptor.Formule :C27H25ClF3N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :515.95Virodhamine
CAS :Virodhamine (O-arachidonoyl ethanolamine), an endocannabinoid, is an antagonist of CB1 receptor and an agonist of CB2 receptor.Formule :C22H37NO2Degré de pureté :98%Couleur et forme :SoildMasse moléculaire :347.53WIN 55,212-2 Mesylate
CAS :WIN 55,212-2 Mesylate ((R)-(+)-WIN 55212) is a potent aminoalkylindole cannabinoid (CB) receptor agonist with Kis of 62.3 and 3.3 nM for human recombinant CB1 and CB2 receptors, respectively. Cannabinoid analogue WIN 55,212-2 Mesylate exhibited a novel anticancer effect against human tumors.Formule :C28H30N2O6SDegré de pureté :98% - 99.71%Couleur et forme :White To Off-White SolidMasse moléculaire :522.61AM251
CAS :AM251: potent CB1 blocker (IC50: 8 nM), 306x CB2 selective; GPR55 activator (EC50: 39 nM).Formule :C22H21Cl2IN4ODegré de pureté :97.43% - 98.79%Couleur et forme :A Crystalline SolidMasse moléculaire :555.24Hemopressin (human, mouse) acetate
Hemopressin: Nonapeptide, α1-hemoglobin derivative, CB1 inverse agonist, isolated from rats, oral, reduces inflammatory pain.Formule :C52H83N13O14Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :1114.29Cannabigerol
CAS :Cannabigerol is a high affinity α±2-adrenergic receptor agonist, moderate affinity 5-HT1A receptor antagonist, and low affinity CB1 receptor antagonist ; alsoFormule :C21H32O2Degré de pureté :99.59% - 99.92%Couleur et forme :SolidMasse moléculaire :316.48Ref: TM-TN1465
1mg138,00€2mg203,00€5mg298,00€10mg449,00€25mg765,00€50mg1.054,00€100mg1.423,00€1mL*10mM (DMSO)306,00€PSB-SB-487
CAS :PSB-SB-487 is antagonist of GPR55.Formule :C26H32O4Degré de pureté :98.53%Couleur et forme :SolidMasse moléculaire :408.53Ref: TM-T8975
1mg35,00€5mg80,00€10mg119,00€25mg231,00€50mg344,00€100mg480,00€200mg660,00€1mL*10mM (DMSO)87,00€ML-191
CAS :ML-191 is an inhibitor of LPI-induced phosphorylation of ERK1/2.Formule :C24H25N3O3Degré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :403.47ML-184
CAS :ML-184 (CID2440433) is a potent synthetic agonist of GPR55 with EC50 of 0.26 μM.Formule :C25H34N4O3SDegré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :470.63JD-5037
CAS :JD-5037 is a novel, peripherally restricted CB1R antagonist with an IC50 of 1.5 nM.Formule :C27H27Cl2N5O3SDegré de pureté :99.54% - 99.84%Couleur et forme :SolidMasse moléculaire :572.51Ref: TM-T4453
1mg42,00€2mg55,00€5mg90,00€10mg133,00€25mg234,00€50mg350,00€100mg522,00€1mL*10mM (DMSO)101,00€ML-193
CAS :ML-193: GPR55 antagonist, IC50 221nM, 27x selective over GPR35/CB1/CB2, may aid Parkinson's symptoms.Formule :C28H25N5O4SDegré de pureté :97.74%Couleur et forme :SolidMasse moléculaire :527.59Otenabant hydrochloride
CAS :Otenabant hydrochloride (Otenabant) (CP-945598) is a competitive, high affinity, selective antagonist of the CB1 receptor (Ki: 0.7 nM).Formule :C25H26Cl3N7ODegré de pureté :99.79% - ≥95%Couleur et forme :SolidMasse moléculaire :546.88Olivetol
CAS :Olivetol, found in lichens, is an organic antioxidant and THC synthesis precursor.Formule :C11H16O2Degré de pureté :99.98%Couleur et forme :(Melting Point 102-106°F) (Ntp 1992)Masse moléculaire :180.24CB1 antagonist 4
CAS :TM38837 is an antagonist of cannabinoid receptor type 1 (CB1), with potential for the treatment of obesity and type 2 diabetes.Formule :C30H25Cl2F3N4OSDegré de pureté :98.97%Couleur et forme :SolidMasse moléculaire :617.51Ref: TM-T8511
2mg46,00€5mg92,00€10mg152,00€25mg259,00€50mg405,00€100mg597,00€200mg848,00€1mL*10mM (DMSO)155,00€Bay 59-3074
CAS :Bay 59-3074 is a CB1/CB2 receptor partial agonist (Ki: 48.3/45.5 nM).
Formule :C18H13F6NO4SDegré de pureté :97.68% - 99.69%Couleur et forme :SolidMasse moléculaire :453.36AM1241
CAS :AM-1241 is a selective cannabinoid CB2 receptor agonist with Ki of 3.4 nM, exhibits 82-fold selectivity over CB1 receptor.Formule :C22H22IN3O3Degré de pureté :98.937% - 99.1%Couleur et forme :SolidMasse moléculaire :503.33Ref: TM-T6755
2mg35,00€5mg49,00€10mg84,00€25mg168,00€50mg275,00€100mg495,00€500mg1.071,00€1mL*10mM (DMSO)87,00€Org 27569
CAS :Org 27569, an allosteric modulator of cannabinoid CB1 receptor, can induce a CB1 receptor state that is characterized by decreased inverse agonist affinity andFormule :C24H28ClN3ODegré de pureté :>99.99% - ≥95%Couleur et forme :SolidMasse moléculaire :409.95A-836339
CAS :A-836339: Potent cannabinoid, CB2-focused (Ki=0.64nM), lesser CB1 affinity (Ki=270nM); analgesic, anti-inflammatory in mice.Formule :C16H26N2O2SDegré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :310.45Ref: TM-T7375
2mg34,00€5mg67,00€10mg109,00€25mg177,00€50mg260,00€100mg369,00€200mg500,00€1mL*10mM (DMSO)63,00€RTICBM-189
CAS :RTICBM-189 is a potent, brain-penetrant allosteric modulator of the cannabinoid type-1 (CB1) receptor with a pIC50 of 7.54 in Ca2+ mobilization assay.Formule :C15H14Cl2N2ODegré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :309.19Ref: TM-T9466
2mg34,00€5mg52,00€10mg84,00€25mg161,00€50mg250,00€100mg369,00€200mg522,00€1mL*10mM (DMSO)67,00€GW842166X
CAS :GW842166X: Potent CB2 agonist, EC50=63 nM, inactive at CB1, in Phase 2 trials.Formule :C18H17Cl2F3N4O2Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :449.25β-Caryophyllene
CAS :β-Caryophyllene ((-)-(E)-Caryophyllene) acts as an CB2 receptor agonist.Formule :C15H24Degré de pureté :95.43% - 99.11%Couleur et forme :Turpentine (Ntp 1992)Masse moléculaire :204.35RVD-Hpα acetate(1193362-76-3 free base)
RVD-Hpα acetate is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist.Formule :C67H109N19O19Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :1484.71Hemopressin (rat) acetate(568588-77-2 free base)
Hemopressin is a nonapeptide, CB2 agonist, derived from rat hemoglobin, with antinociceptive properties.Formule :C5H81N13O14Degré de pureté :99.37%Couleur et forme :SolidMasse moléculaire :1148.31N-Oleoyl glycine
CAS :N-Oleoyl glycine, a lipoamino acid, was able to promote 3T3-L1 adipogenesis through the activation of CB1 receptor and the enhancement of insulin-mediated AktFormule :C20H37NO3Degré de pureté :97.43%Couleur et forme :SolidMasse moléculaire :339.51ARN272
CAS :ARN272 is a FAAH-like anandamide transporter (FLAT) inhibitor (IC50: 1.8 μM).Formule :C27H20N4O2Degré de pureté :98.23%Couleur et forme :SolidMasse moléculaire :432.47Voacamine
CAS :Voacamine: an indole alkaloid, CB1 antagonist, inhibits P-gp, may affect rhythm.
Formule :C43H52N4O5Degré de pureté :98.54% - 99.82%Couleur et forme :SolidMasse moléculaire :704.9yangonin
CAS :Yangonin (Y100550) is a novel CB1 receptor ligand with affinity for human recombinant CB1 receptors.Formule :C15H14O4Degré de pureté :98.82% - 99.55%Couleur et forme :Pale Yellow PowderMasse moléculaire :258.27Ref: TM-T3S0738
1mg70,00€5mg135,00€10mg207,00€25mg349,00€50mg515,00€100mg735,00€1mL*10mM (DMSO)177,00€(±)-Ibipinabant
CAS :(±)-Ibipinabant ((±)-SLV319) has been used in trials studying the treatment of Obesity and Obesity and Type 2 Diabetes.Formule :C23H20Cl2N4O2SDegré de pureté :99.28% - 99.83%Couleur et forme :SolidMasse moléculaire :487.4GW 405833
CAS :GW 405833 (L-768242) is an agonist of cannabinoid-2 (CB(2)) receptor-selectiveFormule :C23H24Cl2N2O3Degré de pureté :99.82% - 99.93%Couleur et forme :SolidMasse moléculaire :447.35Linoleoyl Ethanolamide
CAS :Linoleoyl Ethanolamide is an endocannabinoid agent.Formule :C20H37NO2Degré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :323.51Ref: TM-T8425
1mg35,00€5mg67,00€10mg90,00€25mg164,00€50mg239,00€100mg348,00€200mg522,00€1mL*10mM (DMSO)85,00€AM281
CAS :AM 281, a cannabinoid antagonist, reduces neurologic dysfunction and mortality rate after cecal ligation and puncture in rats.Formule :C21H19Cl2IN4O2Degré de pureté :98.6% - >99.99%Couleur et forme :White To Off-White SolidMasse moléculaire :557.21Ref: TM-T2264
1mg80,00€5mg169,00€10mg259,00€25mg523,00€50mg750,00€100mg1.035,00€500mg2.062,00€1mL*10mM (DMSO)233,00€AM-2232
CAS :AM-2232 (UNII-40KCH8YIKP) is a potent and unselective agonist of the cannabinoid receptors.Formule :C24H20N2ODegré de pureté :99.37%Couleur et forme :SolidMasse moléculaire :352.43LY2828360
CAS :LY2828360: CB2 agonist, Ki=40.3 nM; biases CB2 over CB1 with EC50s of 20.1 nM and >100 μM.Formule :C22H27ClN6ODegré de pureté :98.45% - 99.51%Couleur et forme :SolidMasse moléculaire :426.94CID 16020046
CAS :CID 16020046 (C390-0219) is a selective GPR55 antagonist, inhibiting GPR55 constitutive activity with IC50 of 0.15 μM in yeast.Formule :C25H19N3O4Degré de pureté :99.03%Couleur et forme :SolidMasse moléculaire :425.44Otenabant
CAS :Otenabant (CP-945598) has been investigated for the treatment of Obesity.Formule :C25H25Cl2N7ODegré de pureté :99.43%Couleur et forme :SolidMasse moléculaire :510.42CB1-IN-1
CAS :CB1-IN-1 (DBPR211) is a peripherally restricted CB1R antagonist, for CB1R and CB2R with Ki of 0.3 nM and 21 nM,respectively.Formule :C33H31Cl2F3N6O3S2Degré de pureté :99.08% - 99.76%Couleur et forme :SolidMasse moléculaire :751.67Ref: TM-T5996
1mg82,00€2mg110,00€5mg180,00€10mg258,00€25mg423,00€50mg588,00€100mg793,00€500mg1.594,00€1mL*10mM (DMSO)215,00€Tetrahydromagnolol
CAS :Tetrahydromagnolol can activate cannabinoid (CB) receptors.Formule :C18H22O2Degré de pureté :99.86% - >99.99%Couleur et forme :SolidMasse moléculaire :270.37Ref: TM-TN2268
2mgÀ demander5mg52,00€10mg81,00€25mgÀ demander50mg170,00€100mg243,00€1mL*10mM (DMSO)63,00€BML-190
CAS :BML-190 (Indomethacin morpholinylamide) 是一种 CB2 受体的配体，其对 CB2 受体 (Ki:435 nM) 和 CB1受体 (Ki> 2 μM)。Formule :C23H23ClN2O4Degré de pureté :97.70%Couleur et forme :SolidMasse moléculaire :426.89CB1/2 agonist 3
CAS :CB1/2 agonist 3 is a competitive and potent CB1/CB2 agonist with high affinity for hCB1 and hCB2 and can be used to study neurological disorders.Formule :C25H41NO2Degré de pureté :98.78%Couleur et forme :SolidMasse moléculaire :387.6S-Methoprene
CAS :S-Methoprene (ZR2458), a juvenile hormone analog, acts as an insecticide influencing redox activity and male sex differentiation.
Formule :C19H34O3Degré de pureté :97.05% - 98.55%Couleur et forme :SolidMasse moléculaire :310.47Dehydroabiethylamine
CAS :Dehydroabiethylamine (NSC-2955) boosts liver CYP2B, blocks PDKs & cholesterol transport, and has anti-tumor effects.Formule :C20H31NDegré de pureté :98.79%Couleur et forme :Pale Yellow Viscous Liquid /Technical Grade/ Viscous Colorless To Amber LiquidMasse moléculaire :285.47PSB-KK1445
CAS :PSB-KK1445 is a potent and selective agonist of GPR18, exhibiting EC50 values of 45.4 nM for humans and 124 nM for mice. The selectivity of PSB-KK1445 for GPR18 over the CB receptor subtypes GPR55 and GPR183 exceeds 200-fold.Formule :C24H23FN6O2Masse moléculaire :446.48GPR55 agonist 3
CAS :Compound 26, a GPR55 agonist, exhibits potent activity with EC50 values of 0.239 nM for hGPR55 and 1.76 nM for rGPR55.Formule :C19H16F4N4Couleur et forme :SolidMasse moléculaire :376.35PM226
CAS :CB2 agonist with Ki of 12.8 nM; EC50 of 38.67 nM. Negligible CB1 affinity, no GPR55 activity. Anti-inflammatory, neuroprotective, crosses BBB.Formule :C22H31NO3Couleur et forme :SolidMasse moléculaire :357.49CID1792197
CAS :CID1792197 is a selective agonist of GPR55.Formule :C24H23N3O4S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :481.59VSN-16
CAS :VSN-16, a cannabinoid receptor agonist, is used potentially for the treatment of spasticity in multiple sclerosis.Formule :C18H26N2O3Couleur et forme :SolidMasse moléculaire :318.41GAT229
CAS :GAT229 is a CB1 positive modulator, enhancing CB agonist activity without direct activation; influences binding, signaling, and lowers ocular pressure in mice.Formule :C22H18N2O2Couleur et forme :SolidMasse moléculaire :342.39
