
Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.519 produits)
- Apoptose(5.786 produits)
- Cycle cellulaire/point de contrôle(4.444 produits)
- Chromatine/Épigénétique(2.235 produits)
- Signalisation du cytosquelette(1.382 produits)
- Altération de l'ADN/réparation de l'ADN(2.823 produits)
- Endocrinologie/Hormones(3.499 produits)
- Enzyme(3.639 produits)
- GPCR/G-Protéine(8.314 produits)
- Immunologie et Inflammation(3.516 produits)
- Virus de la grippe(296 produits)
- Signalisation JAK/STAT(404 produits)
- Signalisation MAPK(1.199 produits)
- Transporteur membranaire/Canal ionique(2.786 produits)
- Métabolisme(9.417 produits)
- Microbiologie/Virologie(6.967 produits)
- Neuroscience(9.920 produits)
- Autres inhibiteurs(37.931 produits)
- Oxydation-Réduction(41 produits)
- Signalisation PI3K/Akt/mTOR(1.399 produits)
- Protéases/Protéasome(1.596 produits)
- Cellules souche et Dérivés(832 produits)
- Tyrosine Kinase/Adaptateurs(2.015 produits)
- Ubiquitination(1.646 produits)
Affichez 16 plus de sous-catégories
66627 produits trouvés pour "Inhibiteurs"
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4μ8C
CAS :<p>4μ8C (IRE1 Inhibitor III)(IC50=76 nM) is an effective and specific IRE1 Rnase inhibitor.</p>Formule :C11H8O4Degré de pureté :97.48% - 98.45%Couleur et forme :SolidMasse moléculaire :204.183-Methyltoxoflavin
CAS :<p>3-Methyltoxoflavin (3-methyl toxoflavin) is an effective inhibitor of protein disulfide isomerase (PDI) and its IC50 value is 170 nM.</p>Formule :C8H9N5O2Degré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :207.19ODQ
CAS :<p>ODQ is an effective and selective soluble guanylyl cyclase (sGC) inhibitor.</p>Formule :C9H5N3O2Degré de pureté :98.98%Couleur et forme :Off-White To Light Yellow PowderMasse moléculaire :187.15Picloxydine
CAS :<p>Picloxydine has antiplaque and antibacterial activity.</p>Formule :C20H24Cl2N10Degré de pureté :97.11%Couleur et forme :SolidMasse moléculaire :475.38PI-103
CAS :<p>PI-103 is a potent, cell-permeable, ATP-competitive inhibitor of PI3K family members (IC50s: 2/3/3/15/30/23 nM for p110α/β/δ/γ, mTOR, and DNA-PK).</p>Formule :C19H16N4O3Degré de pureté :97.79% - 99.3%Couleur et forme :SolidMasse moléculaire :348.36Castanospermine
CAS :<p>Castanospermine (1,6,7,8-Tetrahydroxyoctahydroindolizine) is a natural compound that inhibits α- and β-glucosidases, especially glucosidase l.</p>Formule :C8H15NO4Degré de pureté :99.74% - 99.93%Couleur et forme :White Crystalline SolidMasse moléculaire :189.21RO8994
CAS :<p>RO8994: potent MDM2 spiroindolinone inhibitor, IC50: 20 nM (proliferation), 5 nM (binding).</p>Formule :C31H31Cl2FN4O4Degré de pureté :99.31% - 99.44%Couleur et forme :SolidMasse moléculaire :613.51Clodronic acid disodium salt
CAS :<p>Clodronic acid disodium salt (Lodronate), a bisphosphonate, is a potent antiosteolytic agent which inhibits bone resorption.</p>Formule :CH4Cl2O6P0·2NaDegré de pureté :>99.99% - ≥98%Couleur et forme :White SolidMasse moléculaire :288.86Dolasetron
CAS :<p>Dolasetron (MDL-73147)(MDL-73147) is a serotonin 5-HT3 receptor antagonist. Dolasetron is used to treat nausea and vomiting following chemotherapy.</p>Formule :C19H20N2O3Degré de pureté :99.84% - 99.86%Couleur et forme :White PowderMasse moléculaire :324.37SAR405
CAS :<p>SAR-405 inhibits PIK3C3/Vps34 (IC50: 1.2 nM, Kd: 1.5 nM), blocks autophagy, and enhances MTOR inhibitor effects on cancer cells.</p>Formule :C19H21ClF3N5O2Degré de pureté :99.42% - 99.79%Couleur et forme :SolidMasse moléculaire :443.85A66
CAS :<p>A66 is a specific and effective p110α inhibitor(IC50=32 nM).</p>Formule :C17H23N5O2S2Degré de pureté :99.51% - ≥95%Couleur et forme :SolidMasse moléculaire :393.53Methyl 5-hydroxypyridine-2-carboxylate
CAS :<p>Methyl 5-hydroxypyridine-2-carboxylate from Mahonia stems inhibits NO in vitro.</p>Formule :C7H7NO3Degré de pureté :97.04%Couleur et forme :SolidMasse moléculaire :153.14LDN-57444
CAS :<p>LDN-57444 is a reversible, competitive proteasome Uch-L1 inhibitor(IC50=0.88 μM) .</p>Formule :C17H11Cl3N2O3Degré de pureté :97.8% - 99.87%Couleur et forme :SolidMasse moléculaire :397.64Itasetron HCl
CAS :<p>Itasetron HCl is a potent 5HT-3 receptor antagonist.</p>Formule :C16H21ClN4O2Couleur et forme :SolidMasse moléculaire :336.82Mavodelpar
CAS :<p>Mavodelpar (REN001), a PPARδ agonist, may treat PMM and LC-FAOD by reducing renal damage.</p>Formule :C31H29FNNaO5Couleur et forme :SolidMasse moléculaire :537.55AL 082D06
CAS :<p>AL 082D06 (D-06), a selective nonsteroidal glucocorticoid receptor (GR) antagonist (Ki: 210 nM), exhibits outstanding selectivity against AR, ER, MR and PR.</p>Formule :C23H24ClN3O2Degré de pureté :99.05% - 99.06%Couleur et forme :SolidMasse moléculaire :409.91Sodium ionophore III
CAS :<p>Sodium ionophore III (ETH2120) is a Na+ ionophore suitable for the test of sodium activity in plasma, serum, and blood.</p>Formule :C34H52N2O4Degré de pureté :99.51% - 99.78%Couleur et forme :SolidMasse moléculaire :552.79NRX-252262
CAS :<p>NRX-252262 is a potent enhancer of the interaction between β-Catenin, and its cognate E3 ligase, SCFβ-TrCP, induces mutant β-catenin degradation(EC50:3.8 nM)</p>Formule :C23H17Cl2F3N2O4SDegré de pureté :98.94% - 99.87%Couleur et forme :SolidMasse moléculaire :545.36Senexin A
CAS :<p>Senexin A is an effective and selective CDK8 inhibitor that also inhibits CDK19 with Kd values of 0.83 microns and 0.31 microns, respectively.</p>Formule :C17H14N4Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :274.32RU 24969 free base
CAS :<p>RU 24969 (5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole) is a selective agonist of 5-HT1A and 5-HT1B receptors.</p>Formule :C14H16N2ODegré de pureté :97.38%Couleur et forme :SolidMasse moléculaire :228.29Neoeriocitrin
CAS :<p>Neoeriocitrin, from Drynaria Rhizome, boosts MC3T3-E1 growth & bone differentiation; strong AChE inhibitor.</p>Formule :C27H32O15Degré de pureté :99.92% - 99.93%Couleur et forme :SolidMasse moléculaire :596.53GW4869
CAS :<p>GW4869 (GW69A) is a selective and non-competitive inhibitor of neutral sphingomyelinase N-SMase (IC50=1 μM).</p>Formule :C30H30Cl2N6O2Degré de pureté :98.12% - 98.47%Couleur et forme :SolidMasse moléculaire :577.5HZ-1157
CAS :<p>HZ-1157 (DHFR-inhibitor) is a hepatitis C virus (HCV) inhibitor with inhibitory activities toward HCV NS3/4A protease.</p>Formule :C12H16N4ODegré de pureté :98.23%Couleur et forme :SolidMasse moléculaire :232.28AMP-945
CAS :<p>AMP-945 is a proprietary focal adhesion kinase (FAK) inhibitor.</p>Formule :C28H32F3N5O2Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :527.58Paeoniflorin
CAS :<p>Paeoniflorin (Peoniflorin) is a herbal constituent extracted from the root of Paeonia albiflora Pall.</p>Formule :C23H28O11Degré de pureté :96.9% - 97.43%Couleur et forme :White Fine PowderMasse moléculaire :480.46Eniporide hydrochloride
CAS :<p>Eniporide hydrochloride (EMD-96785 hydrochloride) serves as a robust inhibitor of the sodium/hydrogen (Na+/H+) exchange process.</p>Formule :C14H17ClN4O3SCouleur et forme :SolidMasse moléculaire :356.83Isavuconazole
CAS :<p>Isavuconazole (RO-0094815) is an azole antifungal with MICs 0.002-0.5 mg/liter against C. albicans to C. glabrata.</p>Formule :C22H17F2N5OSDegré de pureté :99.74% - >99.99%Couleur et forme :SolidMasse moléculaire :437.47KPT185
CAS :<p>KPT185 (KPT 185) is a selective CRM1 inhibitor, inducing apoptosis, cell-cycle arrest.</p>Formule :C16H16F3N3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :355.31Keracyanin chloride
CAS :<p>Keracyanin chloride (Cyanidin 3-rutinoside chloride), an anthocyanin compound, exhibits antioxidant properties.</p>Formule :C27H31ClO15Degré de pureté :95% - 99.79%Couleur et forme :SolidMasse moléculaire :630.98SGX-523
CAS :<p>SGX-523 is a selective Met inhibitor (IC50: 4 nM), no inhibitory to Abl, BRAFV599E, p38α, and c-Raf.</p>Formule :C18H13N7SDegré de pureté :99% - >99.99%Couleur et forme :SolidMasse moléculaire :359.41CZC-25146 hydrochloride
CAS :<p>CZC-25146 is a selective LRRK2 inhibitor with IC50 of 4.76 nM/6.87 nM for wild type LRRK2 and G2019S LRRK2, respectively.</p>Formule :C22H26ClFN6O4SDegré de pureté :98.76%Couleur et forme :SolidMasse moléculaire :525Gastrin-Releasing Peptide, human(TFA)
<p>Gastrin-releasing peptide (GRP) prompts gastrin release, controls stomach acid, and affects gut motility; vagus nerve fibers stimulate G cells for secretion.</p>Formule :C132H205F3N38O33S2Degré de pureté :98.55%Couleur et forme :SolidMasse moléculaire :2973.4Oleanonic acid
CAS :<p>Oleanonic acid (3-Ketooleanolic Acid) is relatively non-toxic, hepatoprotective, and exhibits antitumor and andantiviral properties.</p>Formule :C30H46O3Degré de pureté :98.35% - 99.22%Couleur et forme :SolidMasse moléculaire :454.68Fluparoxan HCl
CAS :<p>Fluparoxan is a potent α2-adrenergic receptor antagonist (pKB = 7.9) with excellent α2/α1 selectivity (2630 fold).</p>Formule :C10H11ClFNO2Couleur et forme :SolidMasse moléculaire :231.65Avibactam sodium
CAS :<p>Avibactam sodium (NXL-104) is a β-lactamase inhibitor that inhibits TEM-1, P99, and KPC-2. Avibactam sodium has antimicrobial activity. Cost-effective and quality-assured.</p>Formule :C7H10N3NaO6SDegré de pureté :99.16% - >99.99%Couleur et forme :SolidMasse moléculaire :287.22[4-(4-phenylpiperazin-1-yl)oxan-4-yl]methanamine
CAS :<p>[4-(4-Phenylpiperazin-1-yl)oxan-4-yl]methanamine: A piperazine partial agonist for serotonin and dopamine, potential for treating depression/schizophrenia.</p>Formule :C16H25N3ODegré de pureté :98.15%Couleur et forme :SolidMasse moléculaire :275.39Paroxetine maleate
CAS :<p>Paroxetine maleate is a selective inhibitor of serotonin reuptake and an antidepressant.</p>Formule :C23H24FNO7Couleur et forme :SolidMasse moléculaire :445.443Imperialine 3-β-D-glucoside
CAS :<p>Imperialine 3-β-D-glucoside (Sipeimine-3-beta-D-glucoside) is a natural product.</p>Formule :C33H53NO8Degré de pureté :99.9%Couleur et forme :SolidMasse moléculaire :591.78ML327
CAS :<p>ML327 is a MYC blocker. ML327 can also de-repress E-cadherin transcription and reverse Epithelial-to-Mesenchymal Transition (EMT).</p>Formule :C19H18N4O4Degré de pureté :98.47%Couleur et forme :SolidMasse moléculaire :366.37THPP-1
CAS :<p>THPP-1 is a potent and orally bioavailable inhibitor of PDE10A(Ki of 1 nM and 1.3 nM for human and rat PDE10A, respectively).</p>Formule :C23H21ClN6O3Degré de pureté :99.46%Couleur et forme :SolidMasse moléculaire :464.9Phytic acid sodium salt
CAS :<p>Phytic acid sodium salt (Sodium phytate hydrate) functions as a [PO4]3- storage depot and a precursor for other inositol phosphates and pyrophosphates.</p>Formule :C6H18O24P6·xNaDegré de pureté :99.67%Couleur et forme :White Hygroscopic PowderMasse moléculaire :923.82Mogrol
CAS :<p>Mogrol, a biometabolite of mogrosides, functions by inhibiting the ERK1/2 and STAT3 pathways, diminishing CREB activation, and activating AMPK signaling.</p>Formule :C30H52O4Degré de pureté :99.85% - 99.90%Couleur et forme :SolidMasse moléculaire :476.73ERK5-IN-1
CAS :<p>ERK5-IN-1 is a potent ERK5 inhibitor (IC50: 87 nM). It also inhibits LRRK2[G2019S] (IC50: 26 nM).</p>Formule :C25H29N7O2Degré de pureté :97.70%Couleur et forme :SolidMasse moléculaire :459.545,7,3'-Trihydroxy-6,4',5'-trimethoxyflavone
CAS :<p>5,7,3'-Trihydroxy-6,4',5'-trimethoxyflavone is a natural product from Artemisia argyi.</p>Formule :C18H16O8Degré de pureté :99.35% - 99.90%Couleur et forme :SolidMasse moléculaire :360.31Orientin
CAS :<p>1.</p>Formule :C21H20O11Degré de pureté :98.77% - 99.88%Couleur et forme :Yellow PowderMasse moléculaire :448.38NADP disodium salt
CAS :<p>NADP disodium salt: a redox cofactor in metabolism, alternates between oxidized NADP+ and reduced NADPH forms.</p>Formule :C21H26N7Na2O17P3Degré de pureté :97.2% - 99.56%Couleur et forme :White Solid CrystallineMasse moléculaire :787.37SPOP-IN-6b hydrochloride
CAS :<p>SPOP-IN-6b hydrochloride is a highly effective inhibitor of speckle-type POZ protein (SPOP), exhibiting an IC50 value of 3.58 μM.</p>Formule :C28H33ClN6O3Couleur et forme :SolidMasse moléculaire :537.06Caudatin
CAS :<p>Caudatin is one of the species of C-21 steroidal glycosides mainly isolated from the root of Cynanchum bungei Decne and exhibits potent anticancer activities.</p>Formule :C28H42O7Degré de pureté :98.83% - 99.9%Couleur et forme :SolidMasse moléculaire :490.63RRX-001
CAS :<p>RRx-001 is a potent inhibitor ofglucose 6-phosphate dehydrogenase(G6PD) and with potent antimalarial activity</p>Formule :C5H6BrN3O5Degré de pureté :99.91% - ≥95%Couleur et forme :SolidMasse moléculaire :268.02CX-5461 dihydrochloride
<p>CX-5461 dihydrochloride: Oral Pol I inhibitor, HCT-116 (IC50: 142 nM), A375 (IC50: 113 nM), MIA PaCa-2 (IC50: 54 nM), weak on Pol II (IC50 ≥ 25 μM).</p>Formule :C27H29Cl2N7O2SCouleur et forme :SolidMasse moléculaire :586.54S 14506 HCl
CAS :<p>S 14506 HCl: Strong 5-HT1A agonist; pKi - 9.0 (5-HT1A), 6.6 (5-HT1B/C), <6.0 (5-HT3).</p>Formule :C24H26FN3O2Couleur et forme :SolidMasse moléculaire :407.48Oxyresveratrol
CAS :<p>1.</p>Formule :C14H12O4Degré de pureté :98.09% - 99.69%Couleur et forme :Yellow SolidMasse moléculaire :244.24(Z)-LFM-A13
CAS :<p>(Z)-LFM-A13(IC50=2.5 μM), a specific Bruton's tyrosine kinase (BTK), is more than 100-fold specificity than other protein kinases, such as JAK1, JAK2, HCK, EGFR, and IRK.</p>Formule :C11H8Br2N2O2Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :360Difloxacin HCl
CAS :<p>Difloxacin is a second-generation, synthetic fluoroquinolone antimicrobial antibiotic.</p>Formule :C21H19F2N3O3Couleur et forme :Whtie-Cream To Yellowish Crystalline PowderMasse moléculaire :399.39KX2-361
CAS :<p>KX2-361 is a orally bioavailable small molecule dual Src/tubulin inhibitor that provides long term survival in a murine model of glioblastoma</p>Formule :C24H24FN3O2Degré de pureté :99.64% - 99.68%Couleur et forme :SolidMasse moléculaire :405.46GNE-7915 tosylate
CAS :<p>GNE-7915 tosylate is a potent, selective, and brain-penetrant LRRK2 inhibitor, boasting an IC50 value of 9 nM.</p>Formule :C26H29F4N5O6SCouleur et forme :SolidMasse moléculaire :615.6JNJ-7777120
CAS :<p>JNJ-7777120 is the first potent and selective non-imidazole histamine H4 receptor antagonist, exhibits >1000-fold selectivity over the other histamin receptors.</p>Formule :C14H16ClN3ODegré de pureté :99.83% - 99.96%Couleur et forme :SolidMasse moléculaire :277.75Filgotinib maleate
CAS :<p>Filgotinib maleate, a selective oral JAK1 inhibitor, treats RA and Crohn's. IC50s: JAK1-10nM, JAK2-28nM, JAK3-810nM, TYK2-116nM.</p>Formule :C25H27N5O7SCouleur et forme :SolidMasse moléculaire :541.58Triadimefon
CAS :<p>Triadimefon is an azole fungicide used to control powdery mildew.</p>Formule :C14H16ClN3O2Degré de pureté :99.66%Couleur et forme :Less To Pale Yellow Crystalline Solid With A Slight Odor (Ntp 1992) Physical Description Colorless To Pale Yellow Crystalline Solid With A Slight Odor (Ntp 1992)Masse moléculaire :293.75TG100-115
CAS :<p>TG100-115 is a PI3Kγ/δ inhibitor (IC50: 83/235 nM), with fewer effects on PI3Kα/β.</p>Formule :C18H14N6O2Degré de pureté :99.22% - 99.26%Couleur et forme :SolidMasse moléculaire :346.34Solanesol
CAS :<p>Solanesol (Betulanonaprenol) is a phytochemical present in tobacco leaf. Starting material for synthesis of co-enzyme Q10. Exhibits antiulcer activity.</p>Formule :C45H74ODegré de pureté :97.60%Couleur et forme :Brown Waxy SolidMasse moléculaire :631.07Sodium gualenate
CAS :<p>Sodium gualenate is an unstable, hydrophilic guaiazulene derivative with anti-inflammatory and wound-healing properties.</p>Formule :C15H17NaO3SDegré de pureté :99.70%Couleur et forme :SolidMasse moléculaire :300.35S-(5'-Adenosyl)-L-methionine tosylate
CAS :<p>S-(5'-Adenosyl)-L-methionine tosylate (SAMe) is a ubiquitous methyl donor involved in a wide variety of biological reactions, including those mediated by DNA</p>Formule :C22H30N6O8S2Degré de pureté :80% - 98.18%Couleur et forme :SolidMasse moléculaire :570.64GNE-3511
CAS :<p>GNE-3511 is a potent and selective dual leucine zipper kinase inhibitors.</p>Formule :C23H26F2N6ODegré de pureté :98.3% - 99.51%Couleur et forme :SolidMasse moléculaire :440.49Selective PI3Kδ Inhibitor 1
CAS :<p>Selective PI3Kδ Inhibitor 1 is a PI3Kδ Inhibitor( IC50 = 0.9 nM).</p>Formule :C23H20FN7ODegré de pureté :97.96%Couleur et forme :SolidMasse moléculaire :429.45Quercetagitrin
CAS :<p>Quercetagitrin (Quercetagetin-7-O-glucoside), isolated from the African Marigold (Tagetes erecta), has anti-inflammatory activity.</p>Formule :C21H20O13Degré de pureté :99.05% - 99.79%Couleur et forme :SolidMasse moléculaire :480.38Sitagliptin phosphate
CAS :<p>Sitagliptin phosphate (MK-0431 phosphate) is a dipeptidyl peptidase-4 (DPP4) inhibitor.</p>Formule :C16H18F6N5O5PDegré de pureté :99.72% - 99.91%Couleur et forme :White SolidMasse moléculaire :505.31Taselisib
CAS :<p>Taselisib (GDC-0032) is an oral PI3K alpha inhibitor with potential cancer-treating properties.</p>Formule :C24H28N8O2Degré de pureté :99.62% - 99.79%Couleur et forme :SolidMasse moléculaire :460.53KHS101 hydrochloride
CAS :<p>KHS101 is a TACC3 inhibitor and can selectively induce a neuronal differentiation phenotype.</p>Formule :C18H22ClN5SDegré de pureté :99.6%Couleur et forme :SolidMasse moléculaire :375.92MPEP hydrochloride
CAS :<p>MPEP hydrochloride is an effective and highly specific non-competitive antagonist at the mGlu5 receptor subtype (IC50: 36 nM).</p>Formule :C14H12ClNDegré de pureté :99.87% - >99.99%Couleur et forme :SolidMasse moléculaire :229.7(S,R,S)-AHPC-Me
CAS :<p>(S,R,S)-AHPC-Me is a VHL ligand for synthesizing the BET degrader ARV-771, which targets CRPC cells.</p>Formule :C23H32N4O3SDegré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :444.59ACTH (1-39) human
CAS :<p>Adrenocorticotropic Hormone (ACTH) (1-39), human (ACTH (1-39), human) is an agonist of melanocortin receptor.</p>Formule :C207H308N56O58SDegré de pureté :99.6%Couleur et forme :White Lyophilised SolidMasse moléculaire :4541.14Allatostatin IV TFA(123338-13-6 free base)
<p>Allatostatin IV TFA, an octapeptide in insects, regulates juvenile hormone, inhibiting or stimulating its synthesis.</p>Formule :C47H69F3N12O14Degré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :1083.13Dibenzoyl Thiamine
CAS :<p>Dibenzoyl Thiamine (Bentiamine), a lipophilic derivative of vitamin B (thiamine), is a kind of food additive</p>Formule :C26H26N4O4SDegré de pureté :99.18%Couleur et forme :SolidMasse moléculaire :490.57NVP-BSK805 trihydrochloride
CAS :<p>NVP-BSK805 trihydrochloride inhibits JAK2 (0.48 nM IC50); also affects JAK1, JAK3, TYK2.</p>Formule :C27H31Cl3F2N6OCouleur et forme :SolidMasse moléculaire :599.93Meloside A
CAS :<p>Meloside A, a barley-derived phenylpropanoid, provides antioxidant benefits and UV-B protection.</p>Formule :C27H30O15Degré de pureté :99.261% - 99.71%Couleur et forme :SolidMasse moléculaire :594.523-Methyl-L-histidine
CAS :<p>3-Methylhistidine is a basic histidine derivative and eukaryotic biomarker for soy and meat consumption, linked to muscular metabolism and various diseases.</p>Formule :C7H11N3O2Degré de pureté :99.90% - ≥98%Couleur et forme :SolidMasse moléculaire :169.18Desoximetasone
CAS :<p>Desoximetasone (Topicort) is a topical corticosteroid for treating skin conditions like rashes.</p>Formule :C22H29FO4Degré de pureté :99.06% - 99.89%Couleur et forme :SolidMasse moléculaire :376.462-Chloro-4-nitrophenol
CAS :<p>2-Chloro-4-nitrophenol: phenolic COX inhibitor, reduces prostaglandins, lessens inflammation and pain.</p>Formule :C6H4ClNO3Degré de pureté :97.88%Couleur et forme :White Or Kind Of Whith Powder Or Needle Form CrystallizationMasse moléculaire :173.55Opromazine hydrochloride
CAS :<p>Opromazine hydrochloride, a phenothiazine antipsychotic, blocks brain dopamine receptors to treat schizophrenia and psychosis.</p>Formule :C17H20Cl2N2OSDegré de pureté :98.03%Couleur et forme :SolidMasse moléculaire :371.32BO-264
CAS :<p>BO-264 is a highly potent and orally active inhibitor of transforming acidic coiled-coil 3 (TACC3, IC50 of 188 nM and a Kd of 1.5 nM).</p>Formule :C18H19N5O3Degré de pureté :98.03% - 99.81%Couleur et forme :SolidMasse moléculaire :353.381-Naphthyl acetate
CAS :<p>1-Naphthyl acetate is usually used in a rapid staining method for identification of macrophages.</p>Formule :C12H10O2Degré de pureté :99.84%Couleur et forme :WhiteMasse moléculaire :186.21Dalcetrapib
CAS :<p>Dalcetrapib (RO4607381), a rhCETP inhibitor (IC50=0.2 μM), increases the plasma HDL cholesterol.</p>Formule :C23H35NO2SDegré de pureté :97.98% - >99.99%Couleur et forme :SolidMasse moléculaire :389.59BV6
CAS :<p>BV6 is an antagonist of c-IAP1 and XIAP, members of the inhibitors of apoptosis (IAP) family.</p>Formule :C70H96N10O8Degré de pureté :97.46% - 99.82%Couleur et forme :SolidMasse moléculaire :1205.57Molibresib
CAS :<p>Molibresib (GSK525762) is an inhibitor of BET proteins (IC50: about 35 nM).</p>Formule :C22H22ClN5O2Degré de pureté :97.70% - 99.08%Couleur et forme :SolidMasse moléculaire :423.9PF-573228
CAS :<p>PF-573228 is an ATP-competitive FAK inhibitor. In a cell-free assay, the IC50 of FAK is 4 nM.</p>Formule :C22H20F3N5O3SDegré de pureté :96.58% - 99.51%Couleur et forme :SolidMasse moléculaire :491.49Isomazole hydrochloride
CAS :<p>Isomazole hydrochloride is a cardiotonic.</p>Formule :C14H14ClN3O2SCouleur et forme :SolidMasse moléculaire :323.8Romidepsin
CAS :<p>Romidepsin (NSC-630176), an IV histone deacetylase inhibitor, treats refractory cutaneous/peripheral T-cell lymphomas.</p>Formule :C24H36N4O6S2Degré de pureté :99.4% - 99.94%Couleur et forme :SolidMasse moléculaire :540.7Felbinac Trometamol
CAS :<p>Felbinac Trometamol is an intravenous preparation used to treat severe postoperative pain.</p>Formule :C18H23NO5Couleur et forme :SolidMasse moléculaire :333.38Senkyunolide I
CAS :<p>1. Senkyunolide I has neuroprotective effect, associated with its anti-oxidation and anti-apoptosis properties.</p>Formule :C12H16O4Degré de pureté :99.73% - 99.88%Couleur et forme :SolidMasse moléculaire :224.25Netarsudil mesylate
CAS :<p>Netarsudil mesylate (AR-13324 mesylate) is a Rho-related protein kinase inhibitor used to study glaucoma and hypertension.</p>Formule :C30H35N3O9S2Degré de pureté :99.7%Couleur et forme :SolidMasse moléculaire :645.743-Hydroxymandelic Acid
CAS :<p>3-Hydroxymandelic Acid is a metabolite of Phenylephrine.</p>Formule :C8H8O4Degré de pureté :98.47%Couleur et forme :SolidMasse moléculaire :168.15MK-8033
CAS :<p>MK-8033 is a new and selective dual ATP competitive c-Met/Ron inhibitor (IC50: 1 nM Wt c-Met).</p>Formule :C25H21N5O3SDegré de pureté :97.16%Couleur et forme :SolidMasse moléculaire :471.53Corosolic acid
CAS :<p>Corosolic acid inhibits angiogenesis, suppresses FAK, fights various cancers, induces apoptosis, and degrades β-catenin.</p>Formule :C30H48O4Degré de pureté :99.46% - 99.88%Couleur et forme :Fine-Brown Yellow PowderMasse moléculaire :472.7ASP3026
CAS :<p>ASP3026 has been used in trials studying the treatment of Solid Tumor, B-Cell Lymphoma, Advanced Malignancies,and Positive for Anaplastic Lymphoma Kinase.</p>Formule :C29H40N8O3SDegré de pureté :98.78% - 99.81%Couleur et forme :SolidMasse moléculaire :580.74BWX 46 Acetate
<p>BWX 46 Acetate is a potent, highly selective neuropeptide Y (NPY) receptor agonist with IC50 of 0.5 nM.</p>Formule :C118H190N36O30S2Degré de pureté :96.86%Couleur et forme :SolidMasse moléculaire :2657.12MCOPPB triHydrochloride
CAS :<p>MCOPPB triHydrochloride (MCOPPB 3HCl) is a nociceptin receptor agonist.</p>Formule :C26H43Cl3N4Degré de pureté :99.89% - 99.91%Couleur et forme :SolidMasse moléculaire :518.01Ethyl 2-carbamoyloxybenzoate
CAS :<p>ECXB, a synthetic derivative of benzoyloxybenzoic acid, is used in drug synthesis and biochemical studies.</p>Formule :C10H11NO4Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :209.2VU 0364439
CAS :<p>VU 0364439 is a mGlu4 positive allosteric modulator (C50: 19.8 nM).</p>Formule :C18H13Cl2N3O3SDegré de pureté :97.9%Couleur et forme :SolidMasse moléculaire :422.29Isosakuranetin
CAS :<p>Isosakuranetin is cytotoxic, fungicidal, lowers blood pressure, and reduces pain sensitivity.</p>Formule :C16H14O5Degré de pureté :98.62% - 99.82%Couleur et forme :SolidMasse moléculaire :286.28

