
Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.849 produits)
- Apoptose(6.366 produits)
- Cycle cellulaire/point de contrôle(4.907 produits)
- Chromatine/Épigénétique(2.623 produits)
- Signalisation du cytosquelette(1.585 produits)
- Altération de l'ADN/réparation de l'ADN(2.872 produits)
- Endocrinologie/Hormones(3.759 produits)
- Enzyme(3.673 produits)
- GPCR/G-Protéine(9.051 produits)
- Immunologie et Inflammation(3.945 produits)
- Virus de la grippe(300 produits)
- Signalisation JAK/STAT(417 produits)
- Signalisation MAPK(1.259 produits)
- Transporteur membranaire/Canal ionique(3.162 produits)
- Métabolisme(10.149 produits)
- Microbiologie/Virologie(7.672 produits)
- Neuroscience(10.549 produits)
- Autres inhibiteurs(35.857 produits)
- Oxydation-Réduction(41 produits)
- Signalisation PI3K/Akt/mTOR(1.435 produits)
- Protéases/Protéasome(1.693 produits)
- Cellules souche et Dérivés(734 produits)
- Tyrosine Kinase/Adaptateurs(1.991 produits)
- Ubiquitination(1.743 produits)
Affichez 16 plus de sous-catégories
66517 produits trouvés pour "Inhibiteurs"
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TMB-PS
CAS :TMB-PS (TMBZ-PS) is a chromogenic reagent for the detection of hydrogen peroxide e.g. in the enzymatic analysis of body fluids.Formule :C19H26N2O3SDegré de pureté :≥95%Couleur et forme :SolidMasse moléculaire :362.49WS3
CAS :WS3, a β cell proliferation inducer, regulates Erb3 binding protein-1 (EBP1) and the IκB kinase pathway.Formule :C28H30F3N7O3Degré de pureté :97.93% - 99.94%Couleur et forme :SolidMasse moléculaire :569.58PF-04802367
CAS :PF-04802367 is a highly selective GSK-3 inhibitor with an IC50 of 2.1 nM based on a recombinant human GSK-3β enzyme assay and 1.1 nM based on ADP-Glo assay.Formule :C16H16ClN5O3Degré de pureté :98.76%Couleur et forme :SolidMasse moléculaire :361.78Ref: TM-T9611
1mg49,00€5mg100,00€1mL*10mM (DMSO)111,00€10mg152,00€25mg264,00€50mg399,00€100mg532,00€200mg705,00€Argireline
CAS :Argireline (Acetyl hexapeptide-3) is a peptide that inhibits neurotransmitter release, reducing wrinkles.Formule :C34H60N14O12SDegré de pureté :96.79% - 99.65%Couleur et forme :White PowderMasse moléculaire :888.99LY3009120
CAS :LY3009120 (DP-4978) is a potent pan-Raf inhibitor with IC50 of 44 nM, 31-47 nM, and 42 nM for A-raf, B-Raf, and C-Raf in A375 cells, respectively. Phase 1.Formule :C23H29FN6ODegré de pureté :96.96% - ≥95%Couleur et forme :SolidMasse moléculaire :424.51Luteolin-3-O-β-D-glucuronide
CAS :Luteolin-3-O-beta-D-glucuronide is active in the inhibition of nitrite production in macrophages.
Formule :C21H18O12Degré de pureté :98.56% - 99.51%Couleur et forme :SolidMasse moléculaire :462.36Oxyphencyclimine Hydrochloride
CAS :Oxyphencyclimine Hydrochloride (Ulcociclinina) is a synthetic tertiary amine and antimuscarinic agent with antispasmodic and antisecretory activities.Formule :C20H29ClN2O3Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :380.91PEG6-(CH2CO2H)2
CAS :PEG6-(CH2CO2H)2 is a symmetric PEG PROTAC linker.Formule :C14H26O10Degré de pureté :≥95%Couleur et forme :SolidMasse moléculaire :354.35O-Acetyl-L-serine hydrochloride
CAS :O-Acetylserine (OASS), a cysteine precursor in bacteria/plants, enters humans via gut microbes or diet.Formule :C5H10ClNO4Degré de pureté :99.79% - ≥95%Couleur et forme :SolidMasse moléculaire :183.59Prostaglandin E2
CAS :Prostaglandin E2 (PGE2): Key in muscle function, blood flow regulation, and inflammation control.Formule :C20H32O5Degré de pureté :99.76% - 99.95%Couleur et forme :LiquidMasse moléculaire :352.47Ref: TM-T5014
1mg34,00€2mg47,00€1mL*10mM (DMSO)52,00€5mg67,00€10mg93,00€25mg167,00€50mg230,00€100mg334,00€200mg489,00€A 922500
CAS :A 922500 (DGAT-1 Inhibitor 4a) is an inhibitor for human and mouse DGAT-1, good selectivity over related acyltransferases, hERG, and a panel of anti-targets.Formule :C26H24N2O4Degré de pureté :97.34% - 97.66%Couleur et forme :SolidMasse moléculaire :428.482-Iodobenzoic acid
CAS :2-Iodobenzoic acid (o-Iodobenzoic acid) is the impact-sensitive intermediate in the synthesis of the Dess-Martin periodinane.Formule :C7H5IO2Degré de pureté :99.89%Couleur et forme :White To Off-White CrystalsMasse moléculaire :248.02Pyridostatin
CAS :Pyridostatin (RR82) is a synthetic small-molecule stabilizer of G-quadruplexes, a secondary structure of DNA that usually exists in the end of the chromosome orFormule :C31H32N8O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :596.64Fraxinellone
CAS :1.Formule :C14H16O3Degré de pureté :99.35% - 99.92%Couleur et forme :SolidMasse moléculaire :232.27Ref: TM-T6S0071
2mg34,00€5mg50,00€1mL*10mM (DMSO)81,00€10mg84,00€25mg152,00€50mg222,00€100mg334,00€200mg494,00€ML-18
CAS :ML-18 is a non-peptide bombesin receptor subtype-3 (BRS-3) antagonist with an IC50 of 4.8 μM.Formule :C32H35N5O5Degré de pureté :98.62% - >99.99%Couleur et forme :SolidMasse moléculaire :569.65Ref: TM-T4540
1mg34,00€5mg60,00€1mL*10mM (DMSO)75,00€10mg96,00€25mg170,00€50mg264,00€100mg425,00€200mg587,00€(Z)-Guggulsterone
CAS :(Z)-Guggulsterone triggers apoptosis in prostate cancer cells and blocks angiogenesis by inhibiting VEGF pathways.Formule :C21H28O2Degré de pureté :98.93% - 99.72%Couleur et forme :SolidMasse moléculaire :312.45Rucaparib acetate
CAS :Rucaparib acetate, an oral PARP-1, -2, -3 inhibitor (Ki 1.4 nM for PARP1), also moderately inhibits H6PD; promising for CRPC research.Formule :C21H22FN3O3Couleur et forme :SolidMasse moléculaire :383.423GRGDSPC acetate
GRGDSPC acetate (GRGDSPC acetate (91575-26-7 free base)) is a 7-amino acid peptide of thiolated cell adhesion.
Formule :C27H46N10O13SDegré de pureté :96.67%Couleur et forme :SolidMasse moléculaire :750.78AG-1557 hydrochloride (189290-58-2(free base))
AG-1557 hydrochloride is an inhibitor of the epidermal growth factor receptor (EGFR) tyrosine kinase (pIC50: 8.194).Formule :C16H15ClIN3O2Degré de pureté :98.64%Couleur et forme :SolidMasse moléculaire :443.66Trans-ACBD
CAS :Trans-ACBD (Trans-1-aminocyclobutane-1,3-dicarboxylic acid) is an effective and specific N-methyl-D-aspartate receptor agonist.Formule :C6H9NO4Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :159.14Bredinin aglycone
CAS :Bredinin aglycone (SM-108) is a purine nucleotide analog.Formule :C4H5N3O2Degré de pureté :99.06%Couleur et forme :SolidMasse moléculaire :127.1GW280264X
CAS :GW280264X (Carbamic acid) is an inhibitor of ADAM17 .Formule :C28H41N5O6SDegré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :575.72Ref: TM-T8961
1mg156,00€5mg319,00€1mL*10mM (DMSO)404,00€10mg477,00€25mg773,00€50mg1.063,00€100mg1.431,00€SB-590885
CAS :SB590885 is an effective B-Raf inhibitor (Ki: 0.16 nM, in a cell-free assay).Formule :C27H27N5O2Degré de pureté :95.42% - 99.06%Couleur et forme :SolidMasse moléculaire :453.54L-Cystine
CAS :L-Cystine (Cystine Acid) is not considered one of the 20 amino acids, L-Cystine (Cystine Acid) is a sulfur-containing derivative obtained from oxidation ofFormule :C6H12N2O4S2Degré de pureté :99.59% - 99.85%Couleur et forme :White Solid PowderMasse moléculaire :240.3Tenuifolin
CAS :Tenuifolin has no inherent toxicity to either the transfected or wild type cells at the effective concentrations, it inhibits amyloid-β secretion in vitro.Formule :C36H56O12Degré de pureté :97.37% - 99.54%Couleur et forme :SolidMasse moléculaire :680.8213,21-Dihydroeurycomanone
CAS :13,21-Dihydroeurycomanone (Pasakbumin C) is a natural product isolated from the root of Eurycoma longifolia with antiparasitic activity such as PlasmodiumFormule :C20H26O9Degré de pureté :98.01%Couleur et forme :SolidMasse moléculaire :410.42Bupranolol
CAS :Bupranolol blocks β2-adrenergic receptor; treats angina, hypertension, glaucoma, arrhythmia, and prevents clots.Formule :C14H22ClNO2Degré de pureté :97.63%Couleur et forme :SolidMasse moléculaire :271.78Ref: TM-T8580
1mg52,00€1mL*10mM (DMSO)96,00€5mg105,00€10mg159,00€25mg309,00€50mg440,00€100mg583,00€200mg785,00€UNBS5162
CAS :UNBS5162 (UNBS-5162) is a novel naphthalimide that decreases CXCL chemokine expression in experimental prostate cancers.Formule :C17H18N4O3Degré de pureté :98.37% - 99.97%Couleur et forme :SolidMasse moléculaire :326.35Ref: TM-T2477
1mg39,00€5mg81,00€1mL*10mM (DMSO)89,00€10mg116,00€25mg215,00€50mg340,00€100mg540,00€200mg787,00€Astragaloside IV
CAS :Astragaloside IV suppresses ERK1/2, JNK, MMP-2/9 in breast cancer; inhibits adenovirus and protects cardiovascular, immune, digestive, nervous systems.Formule :C41H68O14Degré de pureté :99% - 99.84%Couleur et forme :Hydroscopic Brown Or Yellow PowderMasse moléculaire :784.97Ac-DEVD-pNA
CAS :Ac-DEVD-pNA is the preferred peptidic substrate for caspase-3.Formule :C26H34N6O13Degré de pureté :>99.99%Couleur et forme :WhiteMasse moléculaire :638.58Ref: TM-T7816
2mg34,00€5mg57,00€10mg75,00€1mL*10mM (DMSO)79,00€25mg160,00€50mg231,00€100mg335,00€200mg477,00€Derenofylline
CAS :Derenofylline is a selective and potent adenosine A(1) antagonist in vitro (Ki=1 nM)Formule :C18H20N4ODegré de pureté :98.09%Couleur et forme :SolidMasse moléculaire :308.38Eprinomectin
CAS :Eprinomectin (MK-397) is an avermectin with anthelmintic and insecticidal activities.Formule :C50H75NO14Degré de pureté :97.84% - ≥95%Couleur et forme :SolidMasse moléculaire :914.13LDC-4297 HCl (1453834-21-3(free base))
LDC4297 is a potent and selective CDK7 inhibitor with an IC50 of 0.13 nM.
Formule :C23H29ClN8ODegré de pureté :100%Couleur et forme :SolidMasse moléculaire :469.02Montelukast sodium
CAS :Montelukast sodium (MK0476), an oral leukotriene antagonist for asthma, can cause rare liver injury.Formule :C35H35ClNNaO3SDegré de pureté :99.14% - 99.89%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :608.17BIM-23190 aceate
BIM-23190 aceate, a somatostatin analog, a selective agonist of SSTR2 and SSTR5. BIM-23190 can be used in cancer and acromegaly studies.
Formule :C59H83N13O14S2Degré de pureté :99.7%Couleur et forme :SolidMasse moléculaire :1262.5Tuftsin 3TFA
CAS :Tuftsin 3TFA is a tetrapeptide. It is a macrophage/microglial activator.Formule :C27H43F9N8O12Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :842.66Leucokinin VIII acetate
Leucokinin VIII acetate (Leucokinin 8) is an diuretic octapeptide isolated form head extracts of the cockroach.Formule :C44H56N10O13Degré de pureté :98.52%Couleur et forme :SolidMasse moléculaire :932.99antifungal-agent-6
CAS :Antifungal agent 6 shows antifungal activity.
Formule :C21H23NO5Degré de pureté :98.39%Couleur et forme :SolidMasse moléculaire :369.41SU9516
CAS :SU9516 is a potent CDK2 inhibitor, with an IC50 of 22 nM, and also has inhibitory effects on CDK1 and CDK4, with IC50s of 40 nM and 200 nM, respectively.Formule :C13H11N3O2Degré de pureté :99.34% - 99.96%Couleur et forme :SolidMasse moléculaire :241.25Ref: TM-T6167
1mg34,00€2mg48,00€5mg70,00€1mL*10mM (DMSO)71,00€10mg98,00€25mg197,00€50mg356,00€100mg530,00€500mg1.153,00€AES-350
CAS :AES-350, an HDAC6 inhibitor (IC50: 0.0244 μM), also targets HDAC-3, -8, -11, induces AML cell apoptosis, and aids AML research.Formule :C18H20N2O3Degré de pureté :98.82%Couleur et forme :SolidMasse moléculaire :312.36Propyphenazone
CAS :Propyphenazone: an anti-inflammatory, analgesic, antipyretic pyrazolone; prodrug; COX-2 inhibitor.Formule :C14H18N2ODegré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :230.31NSAH
CAS :NSAH (2-hydroxy-N'-[(E)-(2-hydroxynaphthalen-1-yl)methylidene]benzohydrazide) is a nonnucleoside inhibitor of human ribonucleotide reductase (hRR).with cell-Formule :C18H14N2O3Degré de pureté :99.27%Couleur et forme :SolidMasse moléculaire :306.32Gefarnate
CAS :Gefarnate is a synthetic compound used for the treatment of gastric ulcers,and also used in the treatment of dry eye syndrome.Formule :C27H44O2Degré de pureté :98.36%Couleur et forme :SolidMasse moléculaire :400.64JG-98
CAS :JG-98 is an allosteric Hsp70 inhibitor, displays high active against the breast cancer cell lines MDA-MB-231 and MCF-7 (EC50s: 0.4/0.7 μM).Formule :C24H21Cl2N3OS3Degré de pureté :99.13%Couleur et forme :SolidMasse moléculaire :534.53Protein kinase inhibitor 6
CAS :Protein kinase inhibitor 6 is a protein kinase inhibitor.Formule :C13H9FN2SDegré de pureté :98.01%Couleur et forme :SolidMasse moléculaire :244.29Ref: TM-T9779
2mg34,00€5mg52,00€1mL*10mM (DMSO)52,00€10mg86,00€25mg163,00€50mg222,00€100mg324,00€200mg440,00€HCGRP-(8-37) acetate
HCGRP-(8-37) acetate is a human calcitonin gene-related peptide (hCGRP) fragment acetate and also an antagonist of CGRP receptor.Formule :C141H234N44O40Degré de pureté :99.29%Couleur et forme :SolidMasse moléculaire :3185.64Alisol B
CAS :Alisol B may be a potential novel therapeutic molecule for bone disorders through targeting the differentiation of osteoclasts as well as their functions.Formule :C30H48O4Degré de pureté :99.22% - 99.77%Couleur et forme :SolidMasse moléculaire :472.70Ref: TM-T5770
1mg66,00€5mg177,00€1mL*10mM (DMSO)178,00€10mg264,00€25mg447,00€50mg623,00€100mg883,00€200mg1.189,00€CL 218872
CAS :CL 218872: selective α1 GABAA receptor agonist, anxiolytic, and anticonvulsant; Ki=130 nM for α1, less potent for α2-α6.Formule :C13H9F3N4Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :278.23P110 TFA
P110 TFA is a dynamin-related protein 1 (Drp1) inhibitor, inhibits Drp1 GTPase activity.Formule :C102H180F3N45O27Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :2525.8Ophiopogonin D'
CAS :Ophiopogonin D' can activate SIRT1 in a dose-dependent manner. Ophiopogonin D' also noncompetitively inhibits UGT1A6 and UGT1A10.
Formule :C44H70O16Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :855.02L-778123 free base
CAS :L-778123, an FPTase and GGPTase-I inhibitor, has tolerable toxicity with radiotherapy in advanced pancreatic cancer.Formule :C22H20ClN5OCouleur et forme :SolidMasse moléculaire :405.88NPS-1034
CAS :NPS-1034 is a dual Met/Axl inhibitor with IC50 of 48 nM and 10.3 nM, respectively.Formule :C31H23F2N5O3Degré de pureté :98.48%Couleur et forme :SolidMasse moléculaire :551.54Ref: TM-T6907
1mg34,00€2mg46,00€5mg66,00€1mL*10mM (DMSO)82,00€10mg92,00€25mg167,00€50mg245,00€100mg356,00€200mg530,00€Potassium 1H-indol-3-yl sulfate
CAS :Potassium 1H-indol-3-yl sulfate (Potassium 3-indoxyl sulfate) is an agonist for the human Aryl Hydrocarbon Receptor (AhR).Formule :C8H6KNO4SDegré de pureté :99.52% - >99.99%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :251.3Punicalagin
CAS :Punicalagin, an ellagitannin in pomegranates, has antioxidant, anti-inflammatory, anticancer properties, and combats heart issues from high-fat diets.Formule :C48H28O30Degré de pureté :98% - 99.7%Couleur et forme :White Crystalline PowderMasse moléculaire :1084.72Fenclozic acid
CAS :[2-(4-Chlorophenyl)-1,3-thiazol-4-yl]acetic acid (2-[2-(4-CHLOROPHENYL)-1,3-THIAZOL-4-YL]ACETIC ACID) is an anti-inflammatory thiazoleFormule :C11H8ClNO2SDegré de pureté :98.05%Couleur et forme :SolidMasse moléculaire :253.7UDP-a-D-Galactose disodium salt
CAS :UDP-a-D-Galactose disodium salt is a donor substrate for galactosyltransferases employed in the biosynthesis of galactose-containing oligosaccharides[1].Formule :C15H22N2Na2O17P2Degré de pureté :95.00%Couleur et forme :SolidMasse moléculaire :610.265Palmitoyl Tetrapeptide-3
CAS :Palmitoyl Tetrapeptide-3, a synthetic peptide, boosts GCP-2 to recruit cells for repair and cleanup.Formule :C34H62N8O7Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :694.91Genipin
CAS :Genipin ((+)-Genipin), an active aglycone derived from an iridoid glycoside called geniposide, is found in the fruit of Gardenia jasminoides Ellis.Formule :C11H14O5Degré de pureté :99.09% - 99.21%Couleur et forme :SolidMasse moléculaire :226.23Amifostine Hydrate
CAS :Amifostine Hydrate is a radiation protective agent that induces splenic vasodilation and blocks autonomic ganglion.Formule :C5H17N2O4PSCouleur et forme :SolidMasse moléculaire :232.24SW106065
CAS :SW106065 is a novel pharmacologic inducer of apoptosis in MPNST (malignant peripheral nerve sheath tumors). SW106065 inhibits ATP consumption of sMPNST.Formule :C10H8N2OSDegré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :204.25Ibiglustat
CAS :Ibiglustat (GZ402671) inhibits Glucosylceramide synthase, may treat Fabry disease by preventing GL-3 synthesis.Formule :C20H24FN3O2SDegré de pureté :97.97% - 98.81%Couleur et forme :SolidMasse moléculaire :389.49Theliatinib tartrate
CAS :Theliatinib: oral EGFR blocker, Ki 0.05 nM, IC50 3 nM (wild-type), 22 nM (T790M/L858R), >50x kinase selectivity.Formule :C29H32N6O8Couleur et forme :SolidMasse moléculaire :592.6Creatine-d3 hydrate
CAS :Creatine-d3 hydrate (CREATINE-(METHYL-D3) MONOHYDRATE) is a deuterium labeled Creatine hydrate. Creatine hydrate is pivotal in energy metabolism of muscle cell.Formule :C4H11N3O3Degré de pureté :92.96%Couleur et forme :SolidMasse moléculaire :152.17Pyrrole-2-carboxylic acid
CAS :Minaline is a degradation product of sialic acids and D-hydroxyproline, found in urine post D-isomers ingestion, linked to hyperprolinemia symptoms.Formule :C5H5NO2Degré de pureté :99.61% - 99.62%Couleur et forme :SolidMasse moléculaire :111.1Batimastat
CAS :Batimastat (BB94) (BB-94) is an effective, broad-spectrum matrix metalloprotease (MMP) inhibitor.Formule :C23H31N3O4S2Degré de pureté :98.15% - 99.5%Couleur et forme :SolidMasse moléculaire :477.64Furanodienone
CAS :1.Formule :C15H18O2Degré de pureté :98% - 99.91%Couleur et forme :SolidMasse moléculaire :230.3Lys-Bradykinin acetate(342-10-9 free base)
CAS :Lys-Bradykinin acetate is an endogenous bradykinin receptor agonist.Formule :C58H89N17O14Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :1248.43Zanamivir
CAS :Zanamivir (GG167) is a guanido-neuraminic acid that is used to inhibit NEURAMINIDASE.Formule :C12H20N4O7Degré de pureté :98.84% - 99.98%Couleur et forme :Colorless Crystalline SolidMasse moléculaire :332.31N-Isovaleroylglycine
CAS :N-Isovaleroylglycine, a leucine catabolism byproduct, is an acyl glycine elevated in some metabolic disorders and indicates IVA when accumulated.Formule :C7H13NO3Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :159.18Puromycin dihydrochloride
CAS :Puromycin dihydrochloride, from Streptomyces alboniger, blocks protein synthesis, acting as an antineoplastic and antitrypanosomal agent.Formule :C22H31Cl2N7O5Degré de pureté :98.65% - 99.89%Couleur et forme :Physical Description White Powder (Ntp 1992)Masse moléculaire :544.44Coralyne chloride
CAS :Coralyne chloride is a protoberberine with strong anticancer activity.Formule :C22H22ClNO4Degré de pureté :98.88%Couleur et forme :SolidMasse moléculaire :399.87Fedratinib
CAS :Fedratinib (TG-101348) (TG101348) is an ATP-competitive inhibitor of JAK2 (IC50: 3 nM) with significantly less potent activity against JAK3.Formule :C27H36N6O3SDegré de pureté :97.31% - 99.96%Couleur et forme :SolidMasse moléculaire :524.68Ref: TM-T1995
5mg50,00€1mL*10mM (DMSO)54,00€10mg65,00€50mg107,00€100mg127,00€200mg205,00€500mg447,00€1g592,00€CU-CPT-9a
CAS :CU-CPT-9a is a potent TLR8 inhibitor (IC50 : 0.5 nM), that suppresses TLR8-mediated proinflammatory signaling in various cell lines and human primary cells-Formule :C17H15NO2Degré de pureté :99.01%Couleur et forme :SolidMasse moléculaire :265.31Ref: TM-T7317
1mg38,00€2mg50,00€5mg84,00€1mL*10mM (DMSO)93,00€10mg119,00€25mg225,00€50mg409,00€100mg605,00€CLP-3094
CAS :CLP-3094 (2-([2-(4-CHLOROPHENOXY)ETHYL]THIO)-1H-BE) is a potent androgen receptor BF3 (binding function 3) inhibitor.Formule :C15H13ClN2OSDegré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :304.79Pomalidomide-C3-NH2 hydrochloride
CAS :Pomalidomide-C3-NH2 HCl: a synthetic E3 ligase for PROTAC, with CRBN ligand-linker.Formule :C16H19ClN4O4Degré de pureté :99.60%Couleur et forme :SolidMasse moléculaire :366.8Pseudoginsenoside RT5
CAS :Pseudoginsenoside RT5: anti-epileptic, anti-depressant, boosts nerve growth/cognition, fights bacteria, tumors, malaria.Formule :C36H62O10Degré de pureté :99.46% - >99.99%Couleur et forme :SolidMasse moléculaire :654.87Ibuprofen Lysine
CAS :Ibuprofen Lysine (Neoprofen) is a non-steroidal anti-inflammatory drug.Formule :C19H32N2O4Degré de pureté :99.26%Couleur et forme :CoaMasse moléculaire :352.47Endomorphin 1
CAS :Endomorphin 1 is a high affinity and selective agonist of the μ-opioid receptor and displays reasonable affinities for kappa3 binding sites (Ki: 20~30 nM).Formule :C34H38N6O5Degré de pureté :95.92%Couleur et forme :Solid (Solid Powder )Masse moléculaire :610.7SANT-1
CAS :SANT-1 directly binds to Smoothened (Smo) receptor (Kd: 1.2 nM) and inhibits Smo agonist effects (IC50: 20 nM).Formule :C23H27N5Degré de pureté :99.93% - >99.99%Couleur et forme :SolidMasse moléculaire :373.49Ceftobiprole medocaril
CAS :Ceftobiprole medocaril: injectable prodrug; its active form fights broad-range infections including MRSA.Formule :C26H26N8O11S2Degré de pureté :98.15%Couleur et forme :SolidMasse moléculaire :690.663,4-(Methylenedioxy)cinnamic acid
CAS :3,4-(Methylenedioxy)cinnamic acid (3-(Benzo[d][1,3]dioxol-5-yl)acrylic acid) is a plant-derived compound first extracted from roots of Asparagus officinalis andFormule :C10H8O4Degré de pureté :98.95%Couleur et forme :SolidMasse moléculaire :192.17CGP 71683 (free base)
CAS :CGP 71683 (free base) is a potent and highly selective non-peptide antagonist of the NPY Y(5) receptor in the study of obesity.Formule :C26H29N5O2SCouleur et forme :SolidMasse moléculaire :475.61BX471
CAS :BX471 (BX 471) is a potent, selective non-peptide CCR1 antagonist.Formule :C21H24ClFN4O3Degré de pureté :98% - 99.98%Couleur et forme :SolidMasse moléculaire :434.89Ref: TM-T2375
1mg35,00€5mg86,00€1mL*10mM (DMSO)95,00€10mg117,00€25mg200,00€50mg313,00€100mg489,00€200mg740,00€Disufenton sodium
CAS :Disufenton sodium (NXY-059), a new-type nitrone, exhibits potently neuroprotective effects.Formule :C11H13NNa2O7S2Degré de pureté :98.66% - 99.88%Couleur et forme :SolidMasse moléculaire :381.33Ref: TM-T6201
5mg42,00€1mL*10mM (DMSO)46,00€10mg63,00€25mg110,00€50mg175,00€100mg268,00€200mg413,00€500mg668,00€N-terminally acetylated Leu-enkephalin
Leu-enkephalin, an endogenous 5-amino acid peptide, activates opioid receptors; its acetylated form exists.Formule :C30H39N5O8Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :597.66L-DABA
CAS :L-DABA (L-2,4-Diaminobutyric acid) is an inhibitor of GABA transaminase (IC50 > 500 μM).Formule :C4H10N2O2Degré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :118.13CP 424174
CAS :CP 424174 blocks IL-1β processing (IC50: 210 nM), halts mature IL-1β formation, limits NLRP3, and is effective orally in vivo.Formule :C22H29ClN2O4SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :452.99Ombuin
CAS :Ombuin has anti-inflammatory activity, it inhibits some macrophage functions involved in the inflammatory process.Formule :C17H14O7Degré de pureté :98.85% - 99.71%Couleur et forme :SolidMasse moléculaire :330.29Leonurine
CAS :Leonurine (SCM-198) is an alkaloid that has been found in H. leonuri and with anti-oxidative and anti-inflammatory.Formule :C14H21N3O5Degré de pureté :98.55%Couleur et forme :White Crystalline PowderMasse moléculaire :311.33Theaflavin 3,3′-digallate
CAS :Theaflavin 3,3'-digallate, a major polyphenol found in black tea, is an inducer of oxidative stress which has anti-inflammatory and cancerFormule :C43H32O20Degré de pureté :98.71% - 99.86%Couleur et forme :SolidMasse moléculaire :868.70Ref: TM-T5429
1mg87,00€5mg169,00€10mg268,00€1mL*10mM (DMSO)268,00€25mg462,00€50mg647,00€100mg873,00€200mg1.153,00€Radezolid
CAS :Radezolid (RX-1741) is a novel oxazolidinone antibiotic agent.Formule :C22H23FN6O3Degré de pureté :97.52%Couleur et forme :SolidMasse moléculaire :438.45Ref: TM-T16718
1mg52,00€5mg111,00€1mL*10mM (DMSO)124,00€10mg187,00€25mg339,00€50mg525,00€100mg748,00€6-(4-methylpiperazin-1-yl)-4-o-tolylnicotinamide
CAS :6-(4-methylpiperazin-1-yl)-4-o-tolylnicotinamide can be used in the synthesis of befetupitant and netupitant.Formule :C18H22N4ODegré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :310.39BRL 52537 hydrochloride
CAS :BRL 52537 hydrochloride: selective KOR agonist, may protect against ischemic brain injury, used in stroke and heart attack research.Formule :C18H25Cl3N2ODegré de pureté :99.04%Couleur et forme :SolidMasse moléculaire :391.76Panaxadiol
CAS :Panaxadiol (20(R)-Panaxadiol) is a novel antitumor agent extracted from the Chinese medical herb Panax ginseng.Formule :C30H52O3Degré de pureté :98% - 99.9%Couleur et forme :SolidMasse moléculaire :460.73Sulbactam sodium
CAS :Sulbactam sodium (CP-45899-2) (Unasyn) is an irreversible β-lactamase inhibitor.Formule :C8H10NO5S·NaDegré de pureté :99.76% - 99.83%Couleur et forme :White Or Off-White Crystalline PowderMasse moléculaire :255.22Ergothioneine
CAS :Ergothioneine (L-(+)-Ergothioneine) is synthesized by certain bacteria and fungi. It is generally considered an antioxidant.Formule :C9H15N3O2SDegré de pureté :98.56% - ≥95%Couleur et forme :SolidMasse moléculaire :229.30N-(4-bromo-2-chlorophenyl)-5-chloro-2-hydroxybenzamide
CAS :N-(4-bromo-2-chlorophenyl)-5-chloro-2-hydroxybenzamide is a benzamide analog with anti-tumor, anti-inflammatory, anti-bacterial and anti-fungal activities.
Formule :C13H8BrCl2NO2Degré de pureté :97.47%Couleur et forme :SolidMasse moléculaire :361.02Pyridone 6
CAS :Pyridone 6, a selective JAK1/2/3 and Tyk2 inhibitor with IC50s: JAK1=15 nM, JAK2=1 nM, JAK3 (Ki=5 nM), Tyk2=1 nM; weakly binds other kinases (130 nM-10 μM).Formule :C18H16FN3ODegré de pureté :97.1% - 98.74%Couleur et forme :SolidMasse moléculaire :309.34Ref: TM-T3080
1mg50,00€2mg71,00€5mg105,00€1mL*10mM (DMSO)110,00€10mg173,00€25mg358,00€50mg587,00€100mg888,00€200mg1.198,00€Bromothymol Blue
CAS :Bromothymol Blue is a pH indicator. It is yellow when it is acidic and blue when it is alkaline.Formule :C27H28Br2O5SDegré de pureté :98.36% - 99.51%Couleur et forme :Purple To Pink PowderMasse moléculaire :624.38Tetradecyl Phosphonate
CAS :Tetradecyl Phosphonate 是溶血磷脂酸 1 (LPA1)、LPA2 和 LPA3 受体的泛拮抗剂。Formule :C14H31O3PDegré de pureté :99.95%Couleur et forme :White To Off-White PowderMasse moléculaire :278.37
