
Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.524 produits)
- Apoptose(5.793 produits)
- Cycle cellulaire/point de contrôle(4.452 produits)
- Chromatine/Épigénétique(2.242 produits)
- Signalisation du cytosquelette(1.382 produits)
- Altération de l'ADN/réparation de l'ADN(2.826 produits)
- Endocrinologie/Hormones(3.507 produits)
- Enzyme(3.640 produits)
- GPCR/G-Protéine(8.333 produits)
- Immunologie et Inflammation(3.527 produits)
- Virus de la grippe(296 produits)
- Signalisation JAK/STAT(404 produits)
- Signalisation MAPK(1.203 produits)
- Transporteur membranaire/Canal ionique(2.792 produits)
- Métabolisme(9.449 produits)
- Microbiologie/Virologie(6.981 produits)
- Neuroscience(9.926 produits)
- Autres inhibiteurs(37.921 produits)
- Oxydation-Réduction(41 produits)
- Signalisation PI3K/Akt/mTOR(1.400 produits)
- Protéases/Protéasome(1.597 produits)
- Cellules souche et Dérivés(830 produits)
- Tyrosine Kinase/Adaptateurs(2.015 produits)
- Ubiquitination(1.650 produits)
Affichez 16 plus de sous-catégories
66639 produits trouvés pour "Inhibiteurs"
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VASICINE
CAS :<p>Vasicine: oxytocic, abortifacient, Alzheimer's treatment, and may aid respiratory and reproductive health.</p>Formule :C11H12N2ODegré de pureté :99.62%Couleur et forme :SolidMasse moléculaire :188.235,6,7-TRIMETHOXYFLAVONE
CAS :<p>5,6,7-Trimethoxyflavone, a natural product extracted from Japanese Callicarpa, acts as a p38-α MAPK inhibitor and exhibits anti-inflammatory properties.</p>Formule :C18H16O5Degré de pureté :99.05% - 99.49%Couleur et forme :SolidMasse moléculaire :312.32YHO-13177
CAS :<p>YHO-13177 is a potent and specific inhibitor of BCRP; potentiated the cytotoxicity of SN-38 in cancer cells.</p>Formule :C20H22N2O3SDegré de pureté :98.78%Couleur et forme :SolidMasse moléculaire :370.47Urolithin C
CAS :<p>Urolithin C is a gut metabolite of ellagic acid. Urolithin C induces apoptosis in PC12 cells through a mitochondria-mediated pathway.</p>Formule :C13H8O5Degré de pureté :98.01% - 99.53%Couleur et forme :SolidMasse moléculaire :244.2Acetagastrodin
CAS :<p>Acetagastrodin (Acegastrodine) has an antispasmodic effect on vascular smooth muscle.</p>Formule :C21H26O11Degré de pureté :95.09% - 99.36%Couleur et forme :SolidMasse moléculaire :454.42MAC-545496
CAS :MAC-545496 is a glycopeptide-resistance-associated protein R (GraR) inhibitor, is an antivirulence agent.Formule :C18H18ClN5O3SDegré de pureté :97.41%Couleur et forme :SolidMasse moléculaire :419.89Potassium 1-carboxyvinyl hydrogenphosphate
CAS :<p>Potassium 1-carboxyvinyl hydrogenphosphate (PEP-K) is involved in glycolysis and gluconeogeneis. PEP is metabolized by Pyruvate Kinase to yield pyruvate.</p>Formule :C3H4KO6PDegré de pureté :99.44% - >99.99%Couleur et forme :White To Light Yellow Fine Crystalline PowderMasse moléculaire :206.13Syn-Ake acetate
CAS :<p>Syn-Ake acetate (Dipeptide diaminobutyroyl benzylamide) is a muscarinic acetylcholine receptor antagonist.</p>Formule :C19H29N5O3·2(C2H4O2)Degré de pureté :99.60%Couleur et forme :SolidMasse moléculaire :495.58Vancomycin
CAS :<p>Vancomycin is a glycopeptide antibiotic that exerts its antimicrobial activity by altering the permeability of cell membranes and selectively inhibiting</p>Formule :C66H75Cl2N9O24Degré de pureté :98.76% - 99.35%Couleur et forme :Almost White PowderMasse moléculaire :1449.255-Fluoro-2'-deoxycytidine
CAS :<p>5-Fluoro-2'-deoxycytidine (2'-DEOXY-5-FLUOROCYTIDINE) is an inhibitor of DNA methyltransferase (DNMT) .</p>Formule :C9H12FN3O4Degré de pureté :97.91%Couleur et forme :Fine White PowderMasse moléculaire :245.21Secretoneurin, rat acetate
<p>Secretoneurin, a 33-amino acid peptide from SgII, triggers dopamine release and attracts monocytes/eosinophils.</p>Degré de pureté :96.54%Couleur et forme :SolidMasse moléculaire :N/AMethyl indole-3-carboxylate
CAS :<p>Methyl indole-3-carboxylate (Methyl 3-indolecarboxylate) is a natural product isolated from Heracleum candicans.</p>Formule :C10H9NO2Degré de pureté :99.41%Couleur et forme :Light Pink PowderMasse moléculaire :175.18N-Benzyloctadecanamide
CAS :<p>N-Benzyloctadecanamide is a distinct class of secondary metabolites in Lepidium meyenii Walp. (Maca).</p>Formule :C25H43NODegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :373.612'-Hydroxy-2-methoxychalcone
CAS :<p>2'-Hydroxy-2-methoxychalcone is a synthetic chalcone with antibacterial activity.</p>Formule :C16H14O3Degré de pureté :99.36%Couleur et forme :SolidMasse moléculaire :254.28FPH1
CAS :<p>FPH1 (BRD-6125) (BRD-6125) can promote the expansion of iPS-derived hepatocytes.</p>Formule :C16H15ClF2N2O3SDegré de pureté :99.80%Couleur et forme :SolidMasse moléculaire :388.82Fosifidancitinib
CAS :<p>Fosifidancitinib is a potent inhibitor of JAK 1 and JAK 3.</p>Formule :C21H21FN5O7PDegré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :505.39GLX351322
CAS :<p>GLX351322 is NADPH Oxidase 4 Inhibitor with IC50 of 5 μM.</p>Formule :C21H25N3O5SDegré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :431.51Doxercalciferol
CAS :<p>Doxercalciferol, a synthetic vitamin D2, curbs parathyroid activity for treating secondary hyperparathyroidism and bone disorders.</p>Formule :C28H44O2Degré de pureté :99.03% - 99.69%Couleur et forme :White Crystalline PowderMasse moléculaire :412.65GSK 2830371
CAS :<p>GSK 2830371 is an orally active, allosteric Wip1 phosphatase inhibitor with IC50 of 6 nM.</p>Formule :C23H29ClN4O2SDegré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :461.02Cholesteryl oleate
CAS :<p>Cholesteryl oleate (Cholesteryl cis-9-octadecenoate) is a cholesteryl ester.</p>Formule :C45H78O2Degré de pureté :99.24%Couleur et forme :SolidMasse moléculaire :651.1VUN65671
CAS :<p>Compounds 35 are superior inhibitors of Ebola (Mayinga) and Marburg (Angola) infectious viruses.</p>Formule :C25H30F3N3O2Degré de pureté :99.79%Couleur et forme :SoildMasse moléculaire :461.52p-Hydroxybenzaldehyde
CAS :1.Formule :C7H6O2Degré de pureté :99.05% - 99.86%Couleur et forme :SolidMasse moléculaire :122.12M2I-1
CAS :<p>M2I-1 inhibits Mad2 binding to Cdc20, disrupting SAC-related PPI and Mad2 dynamics, blocks Mad2-F-Mbp1 in FP assays.</p>Formule :C19H24N4O4SDegré de pureté :99.02% - >99.99%Couleur et forme :SolidMasse moléculaire :404.48Compound 401
CAS :<p>Compound 401 (2-morpholino-4H-pyrimido[2,1-a]isoquinolin-4-one) is a synthetic DNA-PK inhibitor (IC50 = 0.28 μM) that also targets mTOR but not PI3K.</p>Formule :C16H15N3O2Degré de pureté :99.73% - 99.78%Couleur et forme :SolidMasse moléculaire :281.31NG-Nitroarginine methyl ester
CAS :<p>NG-Nitroarginine methyl ester (ω-Nitroarginine methyl) is a non-selective nitric oxide synthase inhibitor.</p>Formule :C7H15N5O4Degré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :233.23Brilanestrant
CAS :Brilanestrant (GDC-0810) is a selective estrogen receptor degrader (IC50: 0.7 nM).Formule :C26H20ClFN2O2Degré de pureté :99.07% - 99.17%Couleur et forme :Solid PowderMasse moléculaire :446.9Ufenamate
CAS :<p>Ufenamate (Flufenamic acid butyl ester) is an anthranilic acid-based anti-inflammatory drug developed for skin diseases</p>Formule :C18H18F3NO2Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :337.34T0070907
CAS :<p>T0070907(IC50=1 nM) , an effective and specific PPARγ inhibitor, with the >800-fold selectivity over PPARα and PPARδ.</p>Formule :C12H8ClN3O3Degré de pureté :98.25% - 99.98%Couleur et forme :SolidMasse moléculaire :277.66Dianemycin
CAS :<p>Dianemycin (Nanchangmycin (free acid)) is a broad spectrum polyether antibiotic, inhibits gram-positive bacteria.</p>Formule :C47H78O14Degré de pureté :98% - 99.86%Couleur et forme :SolidMasse moléculaire :867.1116,17-Epoxypregnenol
CAS :<p>16,17-Epoxypregnenol is a useful organic compound for research related to life sciences. The catalog number is T3222 and the CAS number is 974-23-2.</p>Formule :C21H30O3Degré de pureté :99.19% - 99.93%Couleur et forme :SolidMasse moléculaire :330.4620-(tert-Butoxy)-20-oxoicosanoic acid
CAS :<p>20-(tert-Butoxy)-20-oxoicosanoic acid: a non-cleavable alkyl-chain-based PROTAC and ADC linker.</p>Formule :C24H46O4Degré de pureté :≥98%Couleur et forme :SolidMasse moléculaire :398.624-(6,7-dimethoxyquinolin-4-yl)oxyaniline
CAS :<p>4-(6,7-dimethoxyquinolin-4-yl)oxyaniline is a quinoline used in creating drugs and pesticides.</p>Formule :C17H16N2O3Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :296.32Selisistat R-enantiomer
CAS :<p>Selisistat R-enantiomer (EX-527 (R-enantiomer)) is a SIRT1 inhibitor with much less activity than the R-enantiomer of Selisistat (IC50 of SIRT1 > 100 μM).</p>Formule :C13H13ClN2ODegré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :248.71Galgravin
CAS :<p>Galgravin combats inflammation, safeguards neurons, promotes neurite growth, and resists Abeta25-35 and MPP+ toxicity.</p>Formule :C22H28O5Degré de pureté :99.75% - 99.88%Couleur et forme :SolidMasse moléculaire :372.45D-tetrahydropalmatine
CAS :<p>D-Tetrahydropalmatine inhibits OCT1, reducing MCT uptake and hepatocyte damage in MDCK-hOCT1 cells and rat livers.</p>Formule :C21H25NO4Degré de pureté :99.34%Couleur et forme :SolidMasse moléculaire :355.43Perilipin-1/5 Inhibitor 1
CAS :<p>1-[4-(2,3-dihydro-1,4-benzodioxine-6-sulfonyl)piperazin-1-yl]-2-(6-methyl-1-benzofuran-3-yl)ethan-1-one, a building block for organic synthesis.</p>Formule :C23H24N2O6SDegré de pureté :95.69%Couleur et forme :SolidMasse moléculaire :456.51PD 169316
CAS :<p>PD 169316 is a potent, cell-permeable and selective p38 MAP kinase inhibitor.</p>Formule :C20H13FN4O2Degré de pureté :98.65%Couleur et forme :SolidMasse moléculaire :360.34Pracinostat
CAS :<p>Pracinostat (SB939) is a novel HDAC inhibitor with improved in vivo properties compared to other HDAC inhibitors currently in Clinicalal trials, allowing oral</p>Formule :C20H30N4O2Degré de pureté :99.15% - 99.67%Couleur et forme :SolidMasse moléculaire :358.48Senexin B
CAS :<p>Senexin B is a potent and selective inhibitor of CDK8/19(CDK8 and CDK19 with Kds of 140 nM and 80 nM).</p>Formule :C27H26N6ODegré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :450.53Milacemide
CAS :<p>Milacemide is a glycine prodrug and MAO-B inhibitor.</p>Formule :C7H16N2ODegré de pureté :98.04%Couleur et forme :SolidMasse moléculaire :144.21UNC1999
CAS :<p>UNC1999 is a orally bioavailable, effective and specific inhibitor of EZH2 (IC50=2 nM) and EZH1 (IC50=45).</p>Formule :C33H43N7O2Degré de pureté :99.19% - >99.99%Couleur et forme :SolidMasse moléculaire :569.74VO-Ohpic trihydrate
CAS :<p>VO-Ohpic trihydrate (VO-Ohpic) is a potent inhibitor of PTEN (phosphatase and tensin homolog) with IC50 of 35 nM.</p>Formule :C12H9N2O8V·3H2O·HDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :415.21-Stearoyl-2-arachidonoyl-sn-glycero-3-phosphocholine
CAS :<p>1-Stearoyl-2-arachidonoyl-sn-glycero-3-phosphocholine is an endogenous metabolite that has been found in the aging mouse brain.</p>Formule :C46H84NO8PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :810.13Acetyl tetrapeptide-9 Acetate
<p>Acetyl tetrapeptide-9 Acetate plays a role in the stimulation of basement membrane polysaccharide (lumican) and the synthesis of collagen I.</p>Formule :C24H37N7O11Degré de pureté :96.91%Couleur et forme :SolidMasse moléculaire :599.59EBE-A22
CAS :<p>EBE-A22 (PD153035 Analog 63) is a derivative of PD 153035 which can inhibit ErbB-1-phosphorylation, whereas EBE-A22 is inactive.</p>Formule :C17H16BrN3O2Degré de pureté :99.087% - 99.88%Couleur et forme :SolidMasse moléculaire :374.23Hydroxyprogesterone caproate
CAS :<p>Hydroxyprogesterone caproate (Delalutin) is a synthetic progestin that activates progesterone receptors and inhibits ovulation.</p>Formule :C27H40O4Degré de pureté :99.70%Couleur et forme :White Or Almost White Crystalline PowerMasse moléculaire :428.60α,α-Dimethylglycine
CAS :<p>NSC-16590 (2-Aminoisobutyric acid) is a nonprotein amino acid (is an end product of pyrimidine Metabolism) excreted in the urine of about 5% of healthy</p>Formule :C4H9NO2Degré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :103.12BPR1J-097 hydrochloride (1327167-19-0(free base))
<p>BPR1J-097, a new-type small molecule FLT-3 inhibitor(IC50=11±7 nM), is with great anti-tumor activities in vivo.</p>Formule :C27H29ClN6O3SDegré de pureté :98% - 98.54%Couleur et forme :SolidMasse moléculaire :553.07AR42
CAS :<p>AR42 (OSU-HDAC42) is an HDAC inhibitor (IC50: 30 nM).</p>Formule :C18H20N2O3Degré de pureté :98.46% - 98.96%Couleur et forme :SolidMasse moléculaire :312.36Minodronic acid monohydrate
CAS :<p>Minodronic acid monohydrate 是一种法尼基二磷酸合成酶抑制剂,可作为骨吸收抑制剂。</p>Formule :C9H14N2O8P2Degré de pureté :≥95%Couleur et forme :SolidMasse moléculaire :340.16Phenazine-1-carboxylic acid
CAS :<p>Phenazine-1-carboxylic acid, with 90-100% efficacy, is a potent antifungal against phytopathogens and could protect grapevines.</p>Formule :C13H8N2O2Degré de pureté :98.52% - 99.61%Couleur et forme :SolidMasse moléculaire :224.21Lithocholic acid
CAS :<p>Lithocholic acid (3α-Hydroxy-5β-cholanic acid) is a toxic secondary bile acid, They were FXR antagonists (IC50=0.7, 1.4 μM). High-Quality, Low-Cost!</p>Formule :C24H40O3Degré de pureté :99.69% - 99.93%Couleur et forme :Hexagonal Leaflets From Alc Prisms From Acetic Acid Powder (Ntp 1992)Masse moléculaire :376.57Chrysophanol 8-O-glucoside
CAS :<p>Chrysophanol glycosides show mild cytotoxicity, boast anti-diabetic benefits, and aid insulin-driven glucose transport.</p>Formule :C21H20O9Degré de pureté :98.86% - 99.67%Couleur et forme :SolidMasse moléculaire :416.38PfDHODH-IN-2
CAS :<p>PfDHODH-IN-2: powerful antimalarial, blocks PfDHODH (IC50: 1.11 μM), for malaria research.</p>Formule :C13H12ClNO3SDegré de pureté :98.9%Couleur et forme :SolidMasse moléculaire :297.76Mozavaptan
CAS :<p>Mozavaptan (OPC-31260) is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively.</p>Formule :C27H29N3O2Degré de pureté :98.98% - 99.12%Couleur et forme :SolidMasse moléculaire :427.54PZM21
CAS :<p>PZM21 is an effective and selective μ opioid receptor agonist (EC50: 1.8 nM).</p>Formule :C19H27N3O2SDegré de pureté :99.93% - >99.99%Couleur et forme :SolidMasse moléculaire :361.5SI-113
CAS :<p>SI-113 is a potent and selective inhibitor of SGK1, a serine/threonine protein kinase, that modulates several oncogenic signaling cascades.</p>Formule :C23H24N6ODegré de pureté :98.93%Couleur et forme :SolidMasse moléculaire :400.48Hexa-His
CAS :<p>Hexa His, or 6xHis-tag, is a 6-residue His sequence used for GM2 gangliosides degradation and other molecules in tissues.</p>Formule :C36H44N18O7Degré de pureté :99.223% - 99.79%Couleur et forme :SolidMasse moléculaire :840.85AKOS025692697
CAS :<p>AKOS025692697 is a biochemical.</p>Formule :C19H23ClF3N3O3SDegré de pureté :97.70%Couleur et forme :SolidMasse moléculaire :465.917Pardoprunox hydrochloride
CAS :<p>Pardoprunox hydrochloride (SLV-308 hydrochloride) is a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist, D2 (pKi = 8.1)</p>Formule :C12H16ClN3O2Degré de pureté :98.95% - 99.13%Couleur et forme :SolidMasse moléculaire :269.73Polygodial
CAS :<p>Polygodial (Tadeonal) is an antifungal potentiator and an antibiotic, particularly against Saccharomyces cerevisiae, Candida utilis, and Sclerotinia libertiana.</p>Formule :C15H22O2Degré de pureté :98.74%Couleur et forme :SolidMasse moléculaire :234.33Cytosporone B
CAS :<p>Cytosporone B is a Nur77 agonist (IC50 = 0.278 nM), induces apoptosis in cancer cells, affects gluconeogenesis, and has antibacterial properties.</p>Formule :C18H26O5Degré de pureté :95.78% - ≥95%Couleur et forme :SolidMasse moléculaire :322.4BCMA72-80 acetate(2293841-58-2 free base)
<p>BCMA72-80 acetate: HLA-A2 specific BCMA peptide for studying multiple myeloma and certain tumors.</p>Formule :C61H101N13O13SDegré de pureté :98.78%Couleur et forme :SolidMasse moléculaire :1256.6IDO-IN-7
CAS :<p>IDO-IN-7 (NLG-919 analogue) is a potent IDO (indoleamine-(2, 3)-dioxygenase) pathway inhibitor.</p>Formule :C18H22N2ODegré de pureté :99.32% - 99.9%Couleur et forme :SolidMasse moléculaire :282.38Azido-PEG11-azide
CAS :<p>Azido-PEG11-azide is a PEG-based PROTAC linker that can be used in PROTAC synthesis.</p>Formule :C24H48N6O11Degré de pureté :≥98%Couleur et forme :SolidMasse moléculaire :596.67Afatinib Dimaleate
CAS :<p>Afatinib Dimaleate (BIBW 2992MA2) is an orally bioavailable anilino-quinazoline derivative and inhibitor of the EGFR family, with antineoplastic activity.</p>Formule :C32H33ClFN5O11Degré de pureté :98.11% - 99.87%Couleur et forme :SolidMasse moléculaire :718.08SKLB1002
CAS :<p>SKLB1002 is a potent and ATP-competitive VEGFR2 inhibitor with IC50 of 32 nM.</p>Formule :C13H12N4O2S2Degré de pureté :98.51% - >99.99%Couleur et forme :SolidMasse moléculaire :320.39Methylophiopogonanone A
CAS :<p>Methylophiopogonanone A may treat cerebral I/R injury by reducing inflammation, oxidative stress, and protecting the blood-brain barrier.</p>Formule :C19H18O6Degré de pureté :99.78% - 99.99%Couleur et forme :SolidMasse moléculaire :342.34Navtemadlin
CAS :<p>Navtemadlin (AMG232) is a potent, selective and orally available inhibitor of p53-MDM2 interaction (IC50: 0.6 nM).Cost-effective and quality-assured.</p>Formule :C28H35Cl2NO5SDegré de pureté :95.55% - 99.08%Couleur et forme :SolidMasse moléculaire :568.55EHT 1864 2HCl
CAS :<p>EHT 1864 (EHT 1864 2HCl) is a Rac family GTPase inhibitor that blocks activation by direct binding to Rac1, Rac1b, Rac2, and Rac3. Cost effective and quality assured.</p>Formule :C25H29Cl2F3N2O4SDegré de pureté :98.39% - 99.42%Couleur et forme :SolidMasse moléculaire :581.47Pomalidomide-PEG4-C2-NH2
CAS :<p>Pomalidomide-PEG4-C2-NH2 (E3 Ligase Ligand-Linker Conjugates 22) is a synthesized E3 ligase ligand-linker conjugate incorporating the Pomalidomide-based</p>Formule :C23H32N4O8Degré de pureté :95.73%Couleur et forme :SolidMasse moléculaire :492.52PHPS1
CAS :<p>PHPS1 blocks Shp2, halts Shp2-E76K-induced Erk1/2 activation, and stops tumor cell growth.</p>Formule :C21H15N5O6SDegré de pureté :99.08%Couleur et forme :SolidMasse moléculaire :465.44Epirosmanol
CAS :<p>Epirosmanol is a neutral diterpene lactone, a diterpenoid with a lactone group.</p>Formule :C20H26O5Degré de pureté :98.21% - 99.12%Couleur et forme :SolidMasse moléculaire :346.42Omberacetam
CAS :<p>Omberacetam (Noopept), a synthetic dipeptide, enhances cognition similarly to racetams.</p>Formule :C17H22N2O4Degré de pureté :≥95%Couleur et forme :White PowderMasse moléculaire :318.37ASP-9521
CAS :<p>ASP-9521 is a selective, potent and orally active indole-based AKR1C3 inhibitor with an IC50 of 11 nM for human AKR1C3.Cost-effective and quality-assured.</p>Formule :C19H26N2O3Degré de pureté :95.11% - 96.96%Couleur et forme :SolidMasse moléculaire :330.42VU 0357121
CAS :<p>VU0357121, a positive allosteric modulator of mGlu5 (EC50: 33 nM), is inactive or very weakly antagonizing at other mGlu receptor subtypes.</p>Formule :C17H17F2NO2Degré de pureté :99% - >99.99%Couleur et forme :SolidMasse moléculaire :305.32Pinoresinol 4-O-β-D-glucopyranoside
CAS :<p>(+)-Pinoresinol-β-D-glucoside, also known as (+)-pinor, is a major active lignan furanoid found in Forsythia.</p>Formule :C26H32O11Degré de pureté :99.32% - >99.99%Couleur et forme :SolidMasse moléculaire :520.53Histrelin acetate
CAS :<p>Histrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency.</p>Formule :C68H90N18O14Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :1383.55Anthracene-9-carboxylic acid
CAS :<p>Anthracene-9-carboxylic acid is an inhibitor of chloride transport with a moderate to strong inhibitory action on PKA activated cardiac IcI.</p>Formule :C15H10O2Degré de pureté :99.05%Couleur et forme :Yellow Cystalline PowderMasse moléculaire :222.24Tenovin-6 Hydrochloride
CAS :<p>Tenovin-6 HCl: Inhibits SIRT1 (21µM), SIRT2 (10µM), HDAC8; potent p53 activator.</p>Formule :C25H35ClN4O2SDegré de pureté :99.36%Couleur et forme :SolidMasse moléculaire :491.09Naluzotan
CAS :<p>Naluzotan(PRX 00023) is a novel and potent 5-HT1A agonist with IC50 and Ki values of approximately 20 nM and 5.1 nM, respectively.Naluzotan is a potent hERG K+</p>Formule :C23H38N4O3SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :450.64HC-030031
CAS :<p>HC-030031 (TOSLAB 829227) is a potent TRPA1 inhibitor, which antagonizes AITC- and formalin-evoked calcium influx with IC50s of 6.2 and 5.3 μM, respectively.</p>Formule :C18H21N5O3Degré de pureté :99.69% - ≥95%Couleur et forme :SolidMasse moléculaire :355.39(±)-Abscisic acid
CAS :<p>(±)-Abscisic acid (Dormin) is a compound isolated from fruits and plants.</p>Formule :C15H20O4Degré de pureté :98.98% - 99.87%Couleur et forme :White To Pale-Yellow PowderMasse moléculaire :264.32Simeprevir
CAS :<p>Simeprevir (TMC435) is a potent HCV NS3/4A protease inhibitor, and inhibits HCV replication with EC50 of 8 nM.</p>Formule :C38H47N5O7S2Degré de pureté :99.45% - 99.92%Couleur et forme :SolidMasse moléculaire :749.94Fluorometholone
CAS :<p>Fluorometholone (Fluoromethalone) is a corticosteroid, most often used after laser-based refractive surgery.</p>Formule :C22H29FO4Degré de pureté :99% - 99.15%Couleur et forme :SolidMasse moléculaire :376.46KL001
CAS :<p>KL001 stabilizes CRY, extends circadian rhythm, inhibits gluconeogenesis, and could help develop diabetes treatments.</p>Formule :C21H22N2O4SDegré de pureté :99.22%Couleur et forme :SolidMasse moléculaire :398.483-Methoxyflavone
CAS :<p>3-Methoxyflavone is a Flavonoids, with antiviral activity</p>Formule :C16H12O3Degré de pureté :99.29% - 99.97%Couleur et forme :SolidMasse moléculaire :252.26Prasugrel Hydrochloride
CAS :<p>Prasugrel Hydrochloride (LY 640315 Hydrochloride) is pletelet aggregation inhibitor that is used to prevent thrombosis in patients with acute coronary syndrome.</p>Formule :C20H20FNO3S·HClDegré de pureté :99.39% - 99.79%Couleur et forme :SolidMasse moléculaire :409.9Aminopterin
CAS :<p>Aminopterin (4-Aminofolic acid) is a synthetic folic acid derivative whose metabolite is a competitive inhibitor of dihydrofolate reductase</p>Formule :C19H20N8O5Degré de pureté :≥98%Couleur et forme :Orange-Yellow Powder Rodenticide In The U S (Epa 1998)Masse moléculaire :440.41Z-VAD-FMK
CAS :<p>Z-VAD-FMK (Caspase Inhibitor VI) is a broad-spectrum inhibitor of caspases.Z-VAD-FMK binds to activated caspases and inhibits apoptosis.Z-VAD-FMK does not</p>Formule :C21H28FN3O7Degré de pureté :98.24% - 99.79%Couleur et forme :SolidMasse moléculaire :453.46Ginsenoside F1
CAS :<p>Ginsenoside F1, a derivative of Rg1, inhibits CYP3A4 strongly and CYP2D6 weakly.</p>Formule :C36H62O9Degré de pureté :98% - 99.86%Couleur et forme :SolidMasse moléculaire :638.87Amine-PEG-CH2COOH (MW 2000)
<p>Amine-PEG-CH2COOH (MW 5000) is a PEG-based PROTAC linker that can be used in PROTAC synthesis.</p>Degré de pureté :≥98%Couleur et forme :SolidMasse moléculaire :20004-Hydroxybenzylamine
CAS :<p>4-Hydroxybenzylamine (4-HOBA) is a less reactive isomer of 2-HOBA as well as related compounds in a mouse model of hypertension.</p>Formule :C7H9NODegré de pureté :98.58% - 99.66%Couleur et forme :White CrystalMasse moléculaire :123.1512-Epinapelline
CAS :<p>12-Epinapelline, a diterpene alkaloid, acts as an anesthetic and neurotoxin, modulating voltage-gated Na+ channels like aconitine.</p>Formule :C22H33NO3Degré de pureté :99.53% - >99.99%Couleur et forme :SolidMasse moléculaire :359.5Laquinimod
CAS :<p>Laquinimod (LAQ) is an effective immunomodulator, which is currently under development in phase III trials for the treatment of multiple sclerosis as an oral</p>Formule :C19H17ClN2O3Degré de pureté :98.42% - 98.84%Couleur et forme :SolidMasse moléculaire :356.8LY900009
CAS :<p>LY900009 is a small molecule inhibitor of Notch signalling via selective inhibition of the γ-secretase protein.</p>Formule :C23H27N3O4Degré de pureté :97.07%Couleur et forme :SolidMasse moléculaire :409.48Carbidopa monohydrate
CAS :<p>Carbidopa monohydrate (S(-)-Carbidopa) is an inhibitor of DOPA decarboxylase, preventing the conversion of levodopa to dopamine.</p>Formule :C10H16N2O5Degré de pureté :98.11% - 98.30%Couleur et forme :SolidMasse moléculaire :244.241,3-dimethyl-2-oxobenzimidazole-5-carbaldehyde
CAS :<p>1,3-Dimethyl-2-oxobenzimidazole-5-carbaldehyde serves as an intermediate.</p>Formule :C10H10N2O2Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :190.2SM-324405
CAS :<p>SM-324405 is an agonist of TLR7.</p>Formule :C19H23N5O4Degré de pureté :97.83%Couleur et forme :SolidMasse moléculaire :385.42Kasugamycin hydrochloride hydrate
CAS :<p>Kasugamycin (Ksg) HCl hydrate blocks translation initiation in canonical mRNAs, not leaderless ones, by competing with initiator tRNA.</p>Formule :C14H28ClN3O10Degré de pureté :99.82% - >99.99%Couleur et forme :SolidMasse moléculaire :433.84

