
Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.782 produits)
- Apoptose(6.263 produits)
- Cycle cellulaire/point de contrôle(4.792 produits)
- Chromatine/Épigénétique(2.441 produits)
- Signalisation du cytosquelette(1.528 produits)
- Altération de l'ADN/réparation de l'ADN(2.965 produits)
- Endocrinologie/Hormones(3.707 produits)
- Enzyme(3.667 produits)
- GPCR/G-Protéine(9.009 produits)
- Immunologie et Inflammation(3.875 produits)
- Virus de la grippe(301 produits)
- Signalisation JAK/STAT(414 produits)
- Signalisation MAPK(1.248 produits)
- Transporteur membranaire/Canal ionique(3.033 produits)
- Métabolisme(10.209 produits)
- Microbiologie/Virologie(7.592 produits)
- Neuroscience(10.381 produits)
- Autres inhibiteurs(36.040 produits)
- Oxydation-Réduction(42 produits)
- Signalisation PI3K/Akt/mTOR(1.442 produits)
- Protéases/Protéasome(1.724 produits)
- Cellules souche et Dérivés(826 produits)
- Tyrosine Kinase/Adaptateurs(2.035 produits)
- Ubiquitination(1.717 produits)
Affichez 16 plus de sous-catégories
66683 produits trouvés pour "Inhibiteurs"
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SB 216763
CAS :SB 216763 (SB216763) is an effective and specific GSK-3α/β inhibitor (IC50: 34.3 nM).Formule :C19H12Cl2N2O2Degré de pureté :98.9% - 99.13%Couleur et forme :SolidMasse moléculaire :371.22Ref: TM-T3077
2mg39,00€5mg52,00€10mg79,00€25mg131,00€50mg197,00€100mg334,00€500mg803,00€1mL*10mM (DMSO)52,00€3-(3,4,5-Trimethoxyphenyl)propanoic acid
CAS :3-(3,4,5-Trimethoxyphenyl)-propanoic acid is a constituent of Piper retrofractum and Piper longum and is found in herbs and spices.Formule :C12H16O5Degré de pureté :97.93%Couleur et forme :Almost White PowderMasse moléculaire :240.25Amuvatinib
CAS :Amuvatinib (MP470) is an orally bioavailable synthetic carbothioamide with potential antineoplastic activity.Formule :C23H21N5O3SDegré de pureté :99.38% - >99.99%Couleur et forme :SolidMasse moléculaire :447.51Hemokinin 1 (mouse) acetate(208041-90-1 free base)
Mouse Hemokinin-1 acetate: NK1 receptor agonist, Ki=0.175 nM; NK2 Ki=560 nM.Formule :C63H104N22O17SDegré de pureté :98.33%Couleur et forme :SolidMasse moléculaire :1473.72TC-067533
CAS :TC-067533 is a Papain-like protease inhibitor with an IC50 of 8.7 μM.Formule :C20H19NODegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :289.37Ref: TM-T9606
1mg50,00€5mg94,00€10mg144,00€25mg264,00€50mg386,00€100mg552,00€200mg745,00€1mL*10mM (DMSO)101,00€VP3.15 dihydrobromide
CAS :VP3.15 dihydrobromide: potent, oral, CNS-penetrant PDE7/GSK3 inhibitor; IC50s: PDE7- 1.59 μM, GSK- 0.88 μM.Formule :C20H24Br2N4OSDegré de pureté :99.67% - ≥95%Couleur et forme :SolidMasse moléculaire :528.3Continentalic acid
CAS :<p>Continentalic acid from Aralia continentalis has minimum inhibitory concentrations (MICs) of approximately 8-16 µg/mL against S.</p>Formule :C20H30O2Degré de pureté :98.39%Couleur et forme :SolidMasse moléculaire :302.45Kukoamine A
CAS :Kukoamine A: anticancer, cytoprotective, antioxidant, anti-inflammatory, inhibits trypanothione reductase (mixed inhibitor, Ki=1.8µM).Formule :C28H42N4O6Degré de pureté :99.28% - 99.35%Couleur et forme :SolidMasse moléculaire :530.66Epimagnolin A
CAS :Epimagnolin A is a lignan obtained from the flower buds of Magnolia fargesii, which is traditionally used in Asian medicine for treating headache and nasalFormule :C23H28O7Degré de pureté :99.82% - ≥98%Couleur et forme :SolidMasse moléculaire :416.46Ref: TM-TN1610
1mg111,00€2mg166,00€5mg283,00€10mg419,00€25mg682,00€50mg939,00€100mg1.264,00€1mL*10mM (DMSO)320,00€Norathiol
CAS :Norathiol (N-methyl-N-dithiocarboxyglucamine) is a metal chelator that promotes the excretion of 109Cd and may be used in the treatment of cadmium poisoning.Formule :C8H17NO5S2Couleur et forme :SolidMasse moléculaire :271.35F1063-0967
CAS :<p>F1063-0967 is a Dual-specificity phosphatase 26 (DUSP26) inhibitor with an IC50 of 11.62 μM.</p>Formule :C24H24N2O5S2Degré de pureté :97.77%Couleur et forme :SolidMasse moléculaire :484.59N-Feruloyloctopamine
CAS :N-Feruloyloctopamine is a natural product.Formule :C18H19NO5Degré de pureté :99.70%Couleur et forme :SolidMasse moléculaire :329.35Ref: TM-TN1968
1mg85,00€5mg195,00€10mg288,00€25mg485,00€50mg695,00€100mg949,00€1mL*10mM (DMSO)168,00€BD-1047 dihydrobromide
CAS :BD-1047 dihydrobromide (BD1047.2HBr) , a selective functional antagonist of sigma receptors, has antipsychotic activity in animal models predictive of efficacyFormule :C13H22Br2Cl2N2Degré de pureté :98.13% - 99.39%Couleur et forme :SolidMasse moléculaire :437.04Ref: TM-T1740
1mg37,00€2mg48,00€5mg73,00€10mg95,00€25mg168,00€50mg290,00€100mg490,00€1mL*10mM (DMSO)74,00€Hederagenin 28-O-β-D-glucopyranosyl ester
CAS :Hederagenin-28-beta-D-glucopyranoside, a triterpene saponin isolated from Ilex cornuta, protects cardiac myocytes against H2O2-induced damage.Formule :C36H58O9Degré de pureté :97.26% - 99.95%Couleur et forme :SolidMasse moléculaire :634.84NVP-TNKS656
CAS :NVP-TNKS656 (TNKS656) is a highly potent, selective, and orally active TNKS2 inhibitor.Formule :C27H34N4O5Degré de pureté :99.59%Couleur et forme :SolidMasse moléculaire :494.58Ref: TM-T3261
1mg46,00€2mg57,00€5mg88,00€10mg129,00€25mg261,00€50mg444,00€100mg652,00€1mL*10mM (DMSO)87,00€Albendazole sulfoxide
CAS :Albendazole sulfoxide (Ricobendazole) is a metabolite of Albendazole, an anthelmintic.Formule :C12H15N3O3SDegré de pureté :97.29%Couleur et forme :White To Off-White PowderMasse moléculaire :281.33Stigmasterol
CAS :Stigmasterol (Stigmasterin) is a phytosterol with a function in the maintenance of cell membranes. Stigmasterol lowers cholesterol levels. Cost-effective and quality-assured.Formule :C29H48ODegré de pureté :99.67% - 99.97%Couleur et forme :White SolidMasse moléculaire :412.69Ambazone
CAS :Ambazone (Primal) was found to be active against various transplantable tumors in mice as well as rats.Formule :C8H11N7SDegré de pureté :98.68%Couleur et forme :SolidMasse moléculaire :237.28Olivetol
CAS :Olivetol, found in lichens, is an organic antioxidant and THC synthesis precursor.Formule :C11H16O2Degré de pureté :99.98%Couleur et forme :(Melting Point 102-106°F) (Ntp 1992)Masse moléculaire :180.24Atezolizumab
CAS :Atezolizumab is an antibody inhibitor, a humanized monoclonal antibody, IgG1, which targets PD-L1. Atezolizumab has antitumor effect. Cost-effective and quality-assured.Degré de pureté :95.10% - 99.3% (SEC-HPLC)Couleur et forme :LiquidMasse moléculaire :145 kDaAviptadil Acetate
CAS :Aviptadil Acetate (Vasoactive Intestinal Peptide acetate salt) induces pulmonary vasodilation and inhibits the proliferation of vascular SMCs.Formule :C147H238N44O42S·C2H4O2Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :3385.9Alisol F
CAS :Alisol F is a natural product from Alisma plantago-aquatica Linn and has many activities.Formule :C30H48O5Degré de pureté :98.74% - 99.89%Couleur et forme :SolidMasse moléculaire :488.7trans-3-Indoleacrylic acid
CAS :trans-3-Indoleacrylic acid (trans-IAA) is a Tryptophan metabolite.Formule :C11H9NO2Degré de pureté :97.25% - 99.51%Couleur et forme :White To Light Yellow PowderMasse moléculaire :187.19TRC051384
CAS :<p>TRC051384 is a HSP70 inducer that reduces stroke-associated neuronal damage and increases survival in a rat model of transient ischemic stroke.</p>Formule :C25H31N5O4Degré de pureté :98.79%Couleur et forme :SolidMasse moléculaire :465.54PF-04859989
CAS :PF-04859989: irreversible hKAT II inhibitor; brain-penetrable; 1000x selectivity over other KATs; IC50=23 nM (human), 263 nM (rat).Formule :C9H10N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :178.19TG6-10-1
CAS :TG6-10-1 is an EP2 antagonist.Formule :C23H23F3N2O4Degré de pureté :99.66% - ≥95%Couleur et forme :SolidMasse moléculaire :448.43SPOP-IN-6b dihydrochloride
SPOP-IN-6b dihydrochloride is a potent inhibitor of spotted POZ protein (SPOP) (IC50: 3.58 μM).Formule :C28H34Cl2N6O3Couleur et forme :SolidMasse moléculaire :573.51OUL35
CAS :OUL35 (NSC-39047) is a selective PARP-10 inhibitor, and small-molecule ARTD10 inhibitor. OUL35 has been shown to rescue cells from ARTD10-induced cell death.Formule :C14H12N2O3Degré de pureté :99.2%Couleur et forme :SolidMasse moléculaire :256.26ADOS
CAS :ADOS (82692-96-4) is a biochemical reagent/chromogenic reagent.Formule :C12H18NNaO5SDegré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :311.33Pristimerin
CAS :Pristimerin has anticancer properties, counters hypoxia-induced cancer spread, and reduces inflammation by inhibiting ROS/IKK/NF-κB pathways.Formule :C30H40O4Degré de pureté :98.59% - 99.79%Couleur et forme :SolidMasse moléculaire :464.64Ref: TM-T4S1050
1mg39,00€5mg81,00€10mg127,00€25mg279,00€50mg499,00€100mg710,00€500mg1.444,00€1mL*10mM (DMSO)85,00€Ciprofibrate
CAS :Ciprofibrate (Win35833) is a fibrate derivative with antilipidemic activity.Formule :C13H14Cl2O3Degré de pureté :99.63% - >99.99%Couleur et forme :White Or Almost White Crystalline PowderMasse moléculaire :289.15OTS964
CAS :OTS964 is an oral TOPK inhibitor (IC50: 28nM), also targets CDK11, especially CDK11B (Kd: 40nM).Formule :C23H24N2O2SCouleur et forme :SolidMasse moléculaire :392.51Toddaculin
CAS :Toddaculine may be beneficial for the prevention and treatment of osteoporosis, it can not only inhibit the differentiation of osteoclasts via activation of theFormule :C16H18O4Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :274.31Thalidomide-O-amido-C6-NH2 TFA
CAS :Thalidomide-O-amido-C6-NH2 TFA (Cereblon Ligand-Linker Conjugates 11 TFA), a synthesized E3 ligase ligand-linker conjugate containing a Thalidomide-basedFormule :C46H53F6N8O16Degré de pureté :95.16%Couleur et forme :SolidMasse moléculaire :1087.95Tebipenem Pivoxil
CAS :Tebipenem Pivoxil (Orapenem) , an orally activity carbapenem antibiotic, is utilized in treating otolaryngologic and respiratory infections.Formule :C22H31N3O6S2Degré de pureté :97.96%Couleur et forme :SolidMasse moléculaire :497.63N2-methylguanine
CAS :N2-methylguanine (N2-methylguanine) is an endogenous methylated nucleoside found in human fluids and a modified nucleoside.Formule :C6H7N5ODegré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :165.15MK2-IN-1 hydrochloride
CAS :MK2-IN-1 hydrochloride (MK 25) selectively inhibits MK2 with IC50 of 0.11 μM, non-ATP competitive.Formule :C27H26Cl2N4O2Degré de pureté :97.32%Couleur et forme :SolidMasse moléculaire :509.435-AIQ
CAS :5-aminoisoquinolin-1(2H)-one is the inhibitor of calf thymus PARP1.Formule :C9H8N2ODegré de pureté :95.95%Couleur et forme :SolidMasse moléculaire :160.17NAcM-OPT HCl(2089293-61-6 free base)
CAS :NAcM-OPT HCL: Oral DCN1 inhibitor targeting N-Acetyl-UBE2M & DCN1, IC50=79 nM.Formule :C23H30Cl3N3ODegré de pureté :99.43%Couleur et forme :SolidMasse moléculaire :470.86Ref: TM-T9140
2mg38,00€5mg51,00€10mg92,00€25mg148,00€50mg240,00€100mg391,00€500mg929,00€1mL*10mM (DMSO)87,00€Afuresertib
CAS :Afuresertib (GSK2110183) is an orally bioavailable inhibitor of the serine/threonine protein kinase Akt (protein kinase B) with potential antineoplasticFormule :C18H17Cl2FN4OSDegré de pureté :97.51% - 99.51%Couleur et forme :SolidMasse moléculaire :427.32Ref: TM-T1911
1mg39,00€2mg50,00€5mg79,00€10mg97,00€25mg170,00€50mg274,00€100mg477,00€500mg1.035,00€1mL*10mM (DMSO)79,00€Toddalolactone
CAS :Toddalolactone ((+)-Toddalolactone) is an anti-inflammatory and analgesic.Formule :C16H20O6Degré de pureté :99.8% - 99.85%Couleur et forme :SolidMasse moléculaire :308.33Ref: TM-T4S0592
2mg39,00€5mg55,00€10mg77,00€25mg111,00€50mg160,00€100mg227,00€200mg339,00€1mL*10mM (DMSO)66,00€GSK2578215A
CAS :GSK2578215A is a potent and selective LRRK2 kinase inhibitor.Formule :C24H18FN3O2Degré de pureté :99.57% - 99.94%Couleur et forme :SolidMasse moléculaire :399.42LC3-mHTT-IN-AN2
CAS :LC3-mHTT-IN-AN2 (5,7-Dihydroxy-4-phenylcoumarin) is found in the plant Passiflora serratodigitata with the antibacterial activity.Formule :C15H10O4Degré de pureté :98.82% - ≥98%Couleur et forme :SolidMasse moléculaire :254.24Resmetirom
CAS :Resmetirom (MGL-3196) is a THR-β agonist (EC50=0.21 μM), with high selectivity and oral activity. High-Quality, Low-Cost!Formule :C17H12Cl2N6O4Degré de pureté :99.05% - >99.99%Couleur et forme :SolidMasse moléculaire :435.22Ref: TM-T3595
1mg39,00€2mg51,00€5mg87,00€10mg126,00€25mg213,00€50mg343,00€100mg509,00€500mg1.130,00€1mL*10mM (DMSO)92,00€Elemicin
CAS :Elemicin (Elemicine) is a constituent of several plant species' essential oils with anticholinergic effects in human.Formule :C12H16O3Degré de pureté :95.68%Couleur et forme :Less Oil-Like Liquid Colorless Oil-Like LiquidMasse moléculaire :208.25Trifloxystrobin
CAS :Trifloxystrobin is a fungicide against R. solani in sugar beets with EC50s: 23.0 μg/L for Daphnia neonates, 1.7 μg/L for embryos.Formule :C20H19F3N2O4Degré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :408.37Progoitrin
CAS :Progoitrin, a glucosinolate in certain foods, turns into goitrin after consumption, reducing thyroid hormones and yielding CHB and CHEB.Formule :C11H19NO10S2Degré de pureté :98.26%Couleur et forme :SolidMasse moléculaire :389.4AZD8931 diFuMaric acid
CAS :AZD8931 is a reversible and ATP competitive inhibitor of EGFR, ErbB2 and ErbB3 (IC50 of 4 nM, 3 nM and 4 nM, respectively).Formule :C31H33ClFN5O11Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :706.1Ref: TM-T8751
1mg62,00€5mg125,00€10mg180,00€25mg298,00€50mg419,00€100mg567,00€200mg752,00€1mL*10mM (DMSO)178,00€SB-366791
CAS :SB-366791 is a new and selective cinnamide TRPV1 antagonist.Formule :C16H14ClNO2Degré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :287.74AM-2394
CAS :AM-2394 is an effective and specific Glucokinase agonist (GKA, EC50: 60 nM), which catalyzes the phosphorylation of glucose to glucose-6-phosphate.Formule :C22H25N5O4Degré de pureté :99.01% - 99.62%Couleur et forme :SolidMasse moléculaire :423.46Ref: TM-T3312
2mg35,00€5mg52,00€10mg70,00€25mg111,00€50mg175,00€100mg279,00€200mg415,00€1mL*10mM (DMSO)52,00€Helichrysetin
CAS :Helichrysetin shows mild anti-HIV-1 activity and potential as an anticancer agent with cytotoxic effects on A549, MCF-7, Ca Ski, HT-29 cells.Formule :C16H14O5Degré de pureté :96.32% - ≥95%Couleur et forme :SolidMasse moléculaire :286.28TN-16
CAS :TN-16 is a microtubule polymerization inhibitor (IC50 :0.4-1.7 μM)Formule :C19H18N2O2Degré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :306.36(E)-Daporinad
CAS :(E)-Daporinad (FK866) is a highly specific, non-competitive inhibitor of nicotinamide phosphoribosyltransferase (NAMPT) .Cost-effective and quality-assured.Formule :C24H29N3O2Degré de pureté :98.44% - >99.99%Couleur et forme :SolidMasse moléculaire :391.51Ref: TM-T2644
2mg43,00€5mg65,00€10mg96,00€25mg188,00€50mg368,00€100mg557,00€500mg1.169,00€1mL*10mM (DMSO)70,00€VLX600
CAS :VLX600 is an iron-chelating oxidative phosphorylation (OXPHOS) inhibitor, is a cell-permeable anticancer agent.Formule :C17H15N7Degré de pureté :98.62%Couleur et forme :SolidMasse moléculaire :317.35(S)-Indoximod
CAS :(S)-Indoximod (L-Abrine) is an indoleamine-2,3-dioxygenase (IDO) inhibitor for cancer research.Formule :C12H14N2O2Degré de pureté :95.39% - 99.69%Couleur et forme :SolidMasse moléculaire :218.25Ononetin
CAS :<p>Ononetin (2',4'-Dihydroxy-2-(4-methoxyphenyl)acetophenone) is a TRPM3 channel blocker(IC50: 0.3 μM).</p>Formule :C15H14O4Degré de pureté :98.06%Couleur et forme :SolidMasse moléculaire :258.27DL-α-Tocopherol
CAS :<p>DL-alpha-Tocopherol (Ephanyl) is a synthetic vitamin E that protects skin fibroblasts from the cytotoxic effects of UV light and has antioxidant properties.</p>Formule :C29H50O2Degré de pureté :99.61% - 99.90%Couleur et forme :Light Yellow Liquid ViscousMasse moléculaire :430.71Procaterol hydrochloride hydrate
CAS :Short-acting β2-adrenergic receptor agonist used to treat asthma.Formule :C32H48Cl2N4O7Degré de pureté :99.71% - 99.97%Couleur et forme :SolidMasse moléculaire :671.65Ref: TM-T4548
1mg57,00€5mg120,00€10mg170,00€25mg305,00€50mg512,00€100mg727,00€200mg938,00€1mL*10mM (DMSO)164,00€Debrisoquin hydriodide
CAS :Debrisoquin hydriodide is an organic antioxidant with potential for treating neurological issues like Parkinson's and depression.Formule :C10H14IN3Degré de pureté :99%Couleur et forme :SolidMasse moléculaire :303.14Ginkgolic Acid
CAS :<p>Ginkgolic Acid (Romanicardic acid) C15:1 represses curli genes and prophage genes in EHEC.</p>Formule :C22H34O3Degré de pureté :98.69% - 99.9%Couleur et forme :White PowderMasse moléculaire :346.5Nudifloramide
CAS :Nudifloramide (1-Methyl-6-oxo-1,6-dihydropyridine-3-carboxamide) is one of the end degradation products of nicotinamide-adenine dinucleotide (NAD).Formule :C7H8N2O2Degré de pureté :99.7% - ≥95%Couleur et forme :SolidMasse moléculaire :152.15N-Formyl-Met-Leu-Phe-Lys
CAS :<p>fMLFK: potent FPR1 agonist; EC50=3.5 nM (FPR1), 6.7 μM (FPR2), 0.88 μM (FPR2-D2817.32G); binds leukocytes; aids neutrophil assessment.</p>Formule :C27H43N5O6SDegré de pureté :99.7%Couleur et forme :SolidMasse moléculaire :565.73Chlorotriphenylmethane
CAS :Chlorotriphenylmethane (TriphenylMethyl chloride) is a biochemical substance.Formule :C19H15ClDegré de pureté :99.56%Couleur et forme :Needles Or Prisms From Benzene Or Petroleum Ether DrypowderMasse moléculaire :278.78Hexetidine
CAS :Hexetidine (NSC-17764) is a bactericidal and fungicidal antiseptic. It is used as a 0.1% mouthwash for local infections and oral hygiene.Formule :C21H45N3Degré de pureté :97.48%Couleur et forme :Liquid SolidMasse moléculaire :339.61Methyl pentadecanoate
CAS :<p>Methyl pentadecanoate is a natural product.Methyl pentadecanoate is a saturated fatty acid methyl ester obtained from the esterification of myristic acid.</p>Formule :C16H32O2Degré de pureté :98.61%Couleur et forme :SolidMasse moléculaire :256.42DSRM-3716
CAS :Isoquinoline, 5-iodo- (9CI) is a potent and selective inhibitor of SARM1(IC50 = 75 nM) by preventing axonal degeneration and by allowing functional recovery ofFormule :C9H6INDegré de pureté :97.28% - 99.785%Couleur et forme :SolidMasse moléculaire :255.06Dinotefuran
CAS :Dinotefuran (MTI-446), a neonicotinoid insecticide, targets pests by blocking their nervous system.Formule :C7H14N4O3Degré de pureté :99.89%Couleur et forme :White Crystalline PowderMasse moléculaire :202.21Thiophanate-Methyl
CAS :Thiophanate-Methyl (TM), a methyl benzimidazole carbamate (MBC) fungicide,Formule :C12H14N4O4S2Degré de pureté :99.22% - 99.58%Couleur et forme :Colourless Crystals Or White Or Light Brown PowderMasse moléculaire :342.39Ginsenoside Rb3
CAS :Ginsenoside Rb3 (Gypenoside IV) is a natural triterpenoid saponin, exhibiting inhibition effect on TNFα-induced NF-κB transcriptional activity.Formule :C53H90O22Degré de pureté :98% - 99.98%Couleur et forme :SolidMasse moléculaire :1079.27ABT-751
CAS :ABT-751 (E7010) has been investigated for the treatment of Lung Cancer, Non-Small Cell Lung Cancer, and Non-Small-Cell Lung Cancer.Formule :C18H17N3O4SDegré de pureté :98.84% - 99.50%Couleur et forme :SolidMasse moléculaire :371.41Ruthenium Red
CAS :Ruthenium Red (Ammoniated ruthenium oxychloride) is a polycationic dye widely used for electron microscopy (EM) of cells, tissues and vegetative bacteria.Formule :Cl6H42N14O2Ru3Degré de pureté :95%Couleur et forme :Purple PowderMasse moléculaire :786.34TNCA
CAS :<p>TNCA (Lycoperodine-1) is a high-affinity CaSR ligand (CaSRL) with co-agonist activity.</p>Formule :C12H12N2O2Degré de pureté :97.33% - 97.73%Couleur et forme :SolidMasse moléculaire :216.24[Sar9,Met(O2)11]-Substance P acetate
[Sar9,Met(O2)11]-Substance P acetate is an NK1 agonist, raising MAP and HR equally to septide but with unique timing and behaviors.Formule :C66H106N18O18SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :1471.75Pamapimod
CAS :Pamapimod (R1503) (R-1503, Ro4402257) is a novel, selective inhibitor of p38 mitogen-activated protein kinase.Formule :C19H20F2N4O4Degré de pureté :99.52% - 99.99%Couleur et forme :SolidMasse moléculaire :406.38AG 1406
CAS :<p>AG 1406 is a selective inhibitor of the receptor tyrosine kinase VEGF receptor 2.</p>Formule :C16H18N2ODegré de pureté :98.12%Couleur et forme :SolidMasse moléculaire :254.33MK6-83
CAS :MK6-83 is the transient receptor potential channel ML3 agonist.Formule :C16H20N2O2S2Degré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :336.47Disufenton sodium
CAS :Disufenton sodium (NXY-059), a new-type nitrone, exhibits potently neuroprotective effects.Formule :C11H13NNa2O7S2Degré de pureté :98.66% - 99.88%Couleur et forme :SolidMasse moléculaire :381.33Ref: TM-T6201
5mg44,00€10mg66,00€25mg116,00€50mg185,00€100mg283,00€200mg435,00€500mg705,00€1mL*10mM (DMSO)48,00€Tiplaxtinin
CAS :<p>Tiplaxtinin (Tiplasinin)(PAI-039) is a selective and orally efficacious inhibitor of plasminogen activator inhibitor-1 (PAI-1) with IC50 of 2.7 uM.</p>Formule :C24H16F3NO4Degré de pureté :99.16% - 99.93%Couleur et forme :SolidMasse moléculaire :439.384-Oxoisotretinoin
CAS :4-Oxoisotretinoin (Ro 22-6595) is the major blood metabolite.Formule :C20H26O3Degré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :314.42Ref: TM-T3559
1mg35,00€5mg70,00€10mg97,00€25mg188,00€50mg311,00€100mg502,00€200mg715,00€1mL*10mM (DMSO)80,00€11-Maleimidoundecanoic acid
CAS :11-Maleimidoundecanoic acid is an alkyl chain-based PROTAC linker that can be used in PROTAC synthesis.Formule :C15H23NO4Degré de pureté :≥98%Couleur et forme :SolidMasse moléculaire :281.35TCPOBOP
CAS :TCPOBOP is a constitutive androstane receptor agonist that induces robust hepatocyte proliferation and hepatomegaly.Formule :C16H8Cl4N2O2Degré de pureté :99.7%Couleur et forme :SolidMasse moléculaire :402.06Lys-[Des-Arg9]Bradykinin,TFA
Lys-[Des-Arg9]Bradykinin,TFA is Endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and B2Formule :C54H75F6N13O15Degré de pureté :97.35%Couleur et forme :SolidMasse moléculaire :1260.24Acotiamide
CAS :Acotiamide, an oral AChE inhibitor (IC50: 1.79μM), improves gastric motility, targeting functional dyspepsia.Formule :C21H30N4O5SCouleur et forme :SolidMasse moléculaire :450.55Pinosylvin
CAS :Pinosylvin (5-Styrylresorcinol) induces autophagy via AMPK activation. Pinosylvin is likely to act as a pro-angiogenic factor.Formule :C14H12O2Degré de pureté :99.89% - 99.91%Couleur et forme :SolidMasse moléculaire :212.24Sulfachloropyridazine
CAS :<p>Sulfachloropyridazine (Sulfachlorpyridazine) is a sulfonamide antimicrobial used for urinary tract infections and in veterinary medicine.</p>Formule :C10H9ClN4O2SDegré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :284.72D-Isoleucine
CAS :D-Isoleucine ((2R,3R)-2-Amino-3-methylpentanoic acid) is a selective activator of Asc-1 antiporter, which enhances long-term potentiation at the hippocampal CA1Formule :C6H13NO2Degré de pureté :99.16%Couleur et forme :White To Light Yellow PowderMasse moléculaire :131.17For-Met-OH
CAS :For-Met-OH (N-Formyl-L-methionine) is a type of endogenous metabolite, effective in the initiation of protein synthesis.Formule :C6H11NO3SDegré de pureté :99.298% - 99.72%Couleur et forme :SolidMasse moléculaire :177.22PALATINOSE
CAS :Palatinose (TNP-470), a natural disaccharide, links glucose to fructose, aids liver metabolism, and can replace sucrose.Formule :C12H22O11Degré de pureté :98.71%Couleur et forme :White CrystalsMasse moléculaire :342.3GNE-3511
CAS :GNE-3511 is a potent and selective dual leucine zipper kinase inhibitors.Formule :C23H26F2N6ODegré de pureté :98.3% - 99.51%Couleur et forme :SolidMasse moléculaire :440.49Acein acetate
<p>ACE ligand with Kd 2.79 nM, inactive on ACE up to 500 nM. Boosts NMDA/D-serine-induced dopamine release in striatum.</p>Formule :C45H72N10O15Degré de pureté :99.43%Couleur et forme :SolidMasse moléculaire :993.11Arginine-glycine-aspartic acid
CAS :RGD (RGD (Arg-Gly-Asp) Peptides) (Arg-Gly-Asp) Peptides is a cell adhesion motif which can mimic cell adhesion proteins and bind to integrins.Formule :C12H22N6O6Degré de pureté :99.11%Couleur et forme :SolidMasse moléculaire :346.34CK1-IN-1
CAS :CK1-IN-1, a CK1 inhibitor with IC50: 15nM CK1δ, 16nM CK1ε, 73nM p38σ; patent WO2015119579A1.Formule :C24H15F2N3Degré de pureté :98.79%Couleur et forme :SolidMasse moléculaire :383.39Ref: TM-T5393
1mg49,00€2mg65,00€5mg97,00€10mg160,00€25mg305,00€50mg472,00€100mg707,00€1mL*10mM (DMSO)106,00€(−)-Myrtenal
CAS :(−)-Myrtenal ameliorates hyperglycemia by enhancing GLUT2 through Akt in the skeletal muscle and liver of diabetic rats.Formule :C10H14ODegré de pureté :97.65%Couleur et forme :SolidMasse moléculaire :150.226-ethyl-7-hydroxy-4-methylchromen-2-one
CAS :<p>6-Ethyl-7-hydroxy-4-methylchromen-2-one is a fluorescent dye.</p>Formule :C12H12O3Degré de pureté :99.38% - 99.61%Couleur et forme :SolidMasse moléculaire :204.22Pyridone 6
CAS :Pyridone 6, a selective JAK1/2/3 and Tyk2 inhibitor with IC50s: JAK1=15 nM, JAK2=1 nM, JAK3 (Ki=5 nM), Tyk2=1 nM; weakly binds other kinases (130 nM-10 μM).Formule :C18H16FN3ODegré de pureté :97.1% - 98.74%Couleur et forme :SolidMasse moléculaire :309.34Ref: TM-T3080
1mg52,00€2mg74,00€5mg111,00€10mg183,00€25mg378,00€50mg620,00€100mg938,00€200mg1.264,00€1mL*10mM (DMSO)116,00€AZD-8835
CAS :AZD-8835 is a mixed inhibitor of PI3Kα/δ (IC50: 6.2/5.7 nM), also with selectivity against PI3Kβ/γ (IC50: 431/90 nM).Formule :C22H31N9O3Degré de pureté :98.22% - 99.88%Couleur et forme :SolidMasse moléculaire :469.54Thiazole Orange
CAS :Thiazole Orange is a dye that can be used for reticulocyte analysis.Formule :C26H24N2O3S2Degré de pureté :99.29% - 99.93%Couleur et forme :SolidMasse moléculaire :476.61PF-9366
CAS :PF-9366 is a human methionine adenosyltransferase 2A (Mat2A) inhibitor (IC50: 420 nM; Kd: 170 nM).Formule :C20H19ClN4Degré de pureté :97.28% - 99.88%Couleur et forme :SolidMasse moléculaire :350.84Ref: TM-T5191
1mg48,00€5mg92,00€10mg137,00€25mg240,00€50mg339,00€100mg465,00€200mg677,00€1mL*10mM (DMSO)97,00€10058-F4
CAS :10058-F4 inhibits c-Myc-Max, blocking c-Myc target gene activation, causing cell-cycle arrest & apoptosis.Formule :C12H11NOS2Degré de pureté :98% - 99.87%Couleur et forme :SolidMasse moléculaire :249.35Cycloguanil hydrochloride
CAS :Cycloguanil hydrochloride, proguanil's metabolite, inhibits Plasmodium/human dihydrofolate reductase (Ki: 0.3/1.5 nM).Formule :C11H14ClN5·ClHDegré de pureté :98.72%Couleur et forme :SolidMasse moléculaire :288.18

