Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.785 produits)
- Apoptose(6.253 produits)
- Cycle cellulaire/point de contrôle(4.833 produits)
- Chromatine/Épigénétique(2.588 produits)
- Signalisation du cytosquelette(1.532 produits)
- Altération de l'ADN/réparation de l'ADN(2.883 produits)
- Endocrinologie/Hormones(3.747 produits)
- Enzyme(3.670 produits)
- GPCR/G-Protéine(8.977 produits)
- Immunologie et Inflammation(3.777 produits)
- Virus de la grippe(299 produits)
- Signalisation JAK/STAT(415 produits)
- Signalisation MAPK(1.248 produits)
- Transporteur membranaire/Canal ionique(3.147 produits)
- Métabolisme(10.143 produits)
- Microbiologie/Virologie(7.585 produits)
- Neuroscience(10.341 produits)
- Autres inhibiteurs(35.820 produits)
- Oxydation-Réduction(40 produits)
- Signalisation PI3K/Akt/mTOR(1.413 produits)
- Protéases/Protéasome(1.680 produits)
- Cellules souche et Dérivés(747 produits)
- Tyrosine Kinase/Adaptateurs(1.948 produits)
- Ubiquitination(1.719 produits)
Affichez 16 plus de sous-catégories
66565 produits trouvés pour "Inhibiteurs"
Trier par
Degré de pureté (%)
0
100
|
0
|
50
|
90
|
95
|
100
Antifungal agent 13
CAS :Antifungal agent 13 demonstrates significant antifungal activity against Sclerotinia sclerotiorum, achieving an EC50 of 1.25 mg/L.Formule :C21H16ClF3N4OCouleur et forme :SolidMasse moléculaire :432.83Antitubercular agent-16
Compound 5q is a potent antitubercular with low MIC90 values (0.40-23.51 μg/mL) against M. tuberculosis strains, showing minimal cytotoxicity.Formule :C21H27N3SCouleur et forme :SolidMasse moléculaire :353.52CI-1029
CAS :CI-1029: HIV protease inhibitor, combats mutant strains, high efficacy, good bioavailability in animals.Formule :C28H37NO4SCouleur et forme :SolidMasse moléculaire :483.66FNDR-20123
FNDR-20123: First safe, effective anti-malarial HDAC inhibitor for Plasmodium (IC50: 31 nM) & human HDACs, with nanomolar potency across several subtypes.Formule :C21H24ClN5O2Couleur et forme :SolidMasse moléculaire :413.9Steroid sulfatase/17β-HSD1-IN-1
Steroid sulfatase/17β-HSD1-IN-1 is a highly effective inhibitor of both steroid sulfatase and 17β-hydroxysteroid dehydrogenase type 1 (17β-HSD1) activities,Formule :C19H18N2O5SCouleur et forme :SolidMasse moléculaire :386.42NSC 828467
NSC 828467 is one of the top five CA-IX inhibitors with significant in vitro anticancer activity (IC50: 27.2 nM).Formule :C21H19N9O2SCouleur et forme :SolidMasse moléculaire :461.5Vps34-IN-3
Vps34-IN-3 is a potent, selective, and orally bioavailable inhibitor of VPS34 kinase .Formule :C14H20N4O2Couleur et forme :SolidMasse moléculaire :276.33Fluperolone acetate
CAS :Fluperolone acetate is a Glucocorticoid/Adrenal Cortex Hormone.
Formule :C24H31FO6Couleur et forme :SolidMasse moléculaire :434.50Cathepsin C-IN-4
Cathepsin C-IN-4 is a potent inhibitor (IC50: 65.6 nM) of histone C. Cathepsin C-IN-4 inhibits THP-1 cells (IC50: 203.4 nM) and U937 cells (IC50: 177.6 nM).Formule :C21H14ClF3N4SCouleur et forme :SolidMasse moléculaire :446.88Chitin synthase inhibitor 9
CHS inhibitor 9: a broad-spectrum antifungal for studying fungal infections.Formule :C24H25N3O6Couleur et forme :SolidMasse moléculaire :451.47Niravoline
CAS :Niravoline is a kappa-opioid agonist.Formule :C22H25N3O3Couleur et forme :SolidMasse moléculaire :379.45DRX-065
CAS :DRX-065, a deuterated R-enantiomer of pioglitazone, treats NASH without PPARγ weight gain issues.Formule :C19H20N2O3SCouleur et forme :SolidMasse moléculaire :357.45PD-1/PD-L1-IN-15
PD-1/PD-L1-IN-15 is a potent inhibitor of PD-1/PD-L1 (IC50: 60.1 nM) and has shown investigational potential for tumor immunotherapy.Formule :C32H30N4O3Couleur et forme :SolidMasse moléculaire :518.61Osanetant HCl
CAS :Osanetant HCl is the (R)-enantiomer; neurokinin-3 receptor antagonistFormule :C35H42Cl3N3O2Couleur et forme :SolidMasse moléculaire :643.09MRS4738
MRS4738 is a potent antagonist with high affinity for the P2Y14R receptor. It demonstrates in vivo anti-hyperallodynic and antiasthmatic activity [1].Formule :C30H24F3NO2Couleur et forme :SolidMasse moléculaire :487.51MSK-195
CAS :MSK-195 is an effective TRPV1 agonist.Formule :C28H40N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :484.63Glucosylceramide synthase-IN-3
Glucosylceramide synthase-IN-3 (BZ1) is a potent, brain-accessible, oral GCS inhibitor with a 16 nM IC50, relevant for Gaucher's disease study.Formule :C21H20FN3O3Couleur et forme :SolidMasse moléculaire :381.4Adiaft
CAS :Adiaftis a bioactive chemical.Formule :C10H11IN2O4Couleur et forme :SolidMasse moléculaire :350.11WF-47-JS03
WF-47-JS03: RET kinase inhibitor, crosses blood-brain barrier, 500x more selective for KDR, IC50: 1.7 nM in Ba/F3 cells, 5.3 nM in LC-2/ad lung cancer cells.
Formule :C30H38N6O2Couleur et forme :SolidMasse moléculaire :514.66ATUX-1215
CAS :ATUX-1215, a protein phosphatase 2A (PP2A) activator, diminishes the phosphorylation of ERK, p38, JNK, and Akt, as well as decreases the secretion of IL-12p70,Formule :C27H24F5NO4SCouleur et forme :SolidMasse moléculaire :553.54FTI-2153 TFA
FTI-2153 TFA inhibits farnesyltransferase with high selectivity (IC50: 1.4 nM), over 3000x more than Rap1A processing.Formule :C27H31F3N4O5SCouleur et forme :SolidMasse moléculaire :580.62Indoluidin E
Indoluidin E selectively inhibits DHODH and has an inhibitory effect on cancer cell growth.Formule :C28H30N4O2Couleur et forme :SolidMasse moléculaire :454.56DMP 728
CAS :DMP 728 is an antagonist of Glycoprotein IIb-IIIa.Formule :C26H40N8O10SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :656.71PD-1/PD-L1-IN-30
CAS :PD-1/PD-L1-IN-30: Cancer research inhibitor with 0.018 μM IC50.Formule :C29H28F3NO5Couleur et forme :SolidMasse moléculaire :527.53EGFR-IN-24
EGFR-IN-24 is a potent inhibitor of EGFR and inhibits EGFR (del19/T790M/C797S) and EGFR (L858R/T790M/C797S).Formule :C30H35FN6O3Couleur et forme :SolidMasse moléculaire :546.64Retezorogant
CAS :Retezorogant is a retinoic acid receptor-related orphan receptor gamma (RORγ) antagonist.Formule :C23H33ClN2O3Couleur et forme :SolidMasse moléculaire :420.97SSTR4 agonist 4
CAS :SSTR4 agonist 4, potent in pain research, shows promise in rodent pain models, with potential for Alzheimer's due to hippocampus activity.Formule :C19H26N4OCouleur et forme :SolidMasse moléculaire :326.44Annonin VI
CAS :Annonin VI is a natural inhibitor of NADH:ubiquinone oxidoreductase.Formule :C37H66O7Couleur et forme :SolidMasse moléculaire :622.92HCV-IN-38
Potent oral HCV inhibitor HCV-IN-38 has 15 nM EC50, 431 SI, high efficacy, and low toxicity.Formule :C22H24ClF3N4O4Couleur et forme :SolidMasse moléculaire :500.9CCT369260
CAS :CCT369260 (compound 1), an orally active inhibitor targeting B-cell lymphoma 6 (BCL6), demonstrates anti-tumor efficacy with an IC50 value of 520 nM [1].Formule :C24H31ClF2N6O2Couleur et forme :SolidMasse moléculaire :508.99BRD0418
CAS :BRD0418 acts as an upregulator of TRIB1 expression by leading to reprogramming of hepatic lipoprotein metabolism from adipogenesis to clearance it.Formule :C29H32N2O5Degré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :488.57MK-7445
CAS :MK-7445 is a conformationally constrained inhibitor of non-nucleoside reverse transcriptase.Formule :C21H13Cl2N7OCouleur et forme :SolidMasse moléculaire :450.28Carumonam Sodium
CAS :Carumonam Sodium is a monobactam, penicillin-binding protein inhibitor. It is used as antibacterials.Formule :C12H12N6Na2O10S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :510.37Triphen diol
CAS :Triphen diol, a phenol diol, fights pancreatic cancer & cholangiocarcinoma, inducing apoptosis via caspase-dependent & -independent paths.Formule :C22H20O4Couleur et forme :SolidMasse moléculaire :348.39LpxC-IN-10
CAS :LpxC-IN-10 is a selective LpxC inhibitor with an MIC of 0.5 μg/mL against E. coli and K. pneumoniae and is capable of being used to study bacterial infections.Formule :C30H31N5O3Couleur et forme :SolidMasse moléculaire :509.6ABT-072
CAS :ABT-072 is a nonnucleoside NS5B polymerase inhibitor and a candidate drug evaluated for treatment of hepatitis C virus.Formule :C24H27N3O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :469.55BAY-693
CAS :BAY-693 is a ERK5 negative control agent with IC50 (ERK5) = 6400 nM. Its analog, BAY-885, is a potent and selective ERK5 (MAPK7) inhibitor with IC50 of 40 nMFormule :C26H30F3N7O2Couleur et forme :SolidMasse moléculaire :529.564'-Ethynyl-2'-deoxyadenosine
CAS :4'-E-dA is a potent nucleoside RT inhibitor for drug-resistant HIV (EC50: 98 nM in MT-4 cells).Formule :C12H13N5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :275.26Plm IV inhibitor-2
CAS :"Plm IV inhibitor-2: Potent for Plm IV (IC50=24nM), affects Plm II/Plm I; malaria research compound."Formule :C39H54N4O4Couleur et forme :SolidMasse moléculaire :642.87EB-0150
EB-0150 inhibits ER α-Glu I/II (IC50: 0.73/0.0337 μM), is an N-substituted valerian with antiviral effects, and has drug discovery potential.Formule :C19H30N6O7Couleur et forme :SolidMasse moléculaire :454.48MtTMPK-IN-7
MtTMPK-IN-7 inhibits MtbTMPK (IC50: 47 μM), active against M. brevis (MIC: 2.3-4.7 μM), useful for tuberculosis research.Formule :C27H29ClN6O3Couleur et forme :SolidMasse moléculaire :521.01Ornoprostil
CAS :Ornoprostil, a prostaglandin E1 analogue, acts as a mucosal protectant.Formule :C23H38O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :410.54GABAA receptor agonist 2
Compound 4c, a potent GABAA agonist with anti-depressive effects in mouse FST/TST, shows promise in depression research.Formule :C22H36O5Couleur et forme :SolidMasse moléculaire :380.52Glycyl H-1152 hydrochloride
CAS :Glycyl-H-1152 is a potent ROCK-II inhibitor (IC50=11.8 nM) with high selectivity over CaMKII, PKG, Aurora A, PKA, and PKC. Better than Y-27632 and HA-1077.Formule :C18H26Cl2N4O3SCouleur et forme :SolidMasse moléculaire :449.39SCH-1473759
CAS :SCH-1473759 is an inhibitor of the aurora (IC50s: 4 and 13 nM for Aurora A and B, respectively).Formule :C20H26N8OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :426.54PPO-IN-1
PPO-IN-1 is a potent inhibitor of protoporphyrinogen IX oxidase (PPO) (Ki: 2.5 nM).Formule :C18H10F3N3O4SCouleur et forme :SolidMasse moléculaire :421.35ATX inhibitor 22
ATX inhibitor 22 is a novel inhibitor of ATX (autotaxin) (IC50: 218.9 μM) that lacks inhibitory activity against LPAR1.Formule :C19H17Cl3F2N2O4SCouleur et forme :SolidMasse moléculaire :513.77NPEC-caged-(S)-3,4-DCPG
CAS :mGlu8a agonistFormule :C19H16N2O10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :432.34NNTA
CAS :NNTA is a highly selective and potent activator of μ/κ-opioid heteromers.Formule :C31H32N2O4Couleur et forme :SolidMasse moléculaire :496.60MDL-27788
CAS :MDL-27788 is a tricyclic inhibitor.Formule :C24H26N2O5SCouleur et forme :SolidMasse moléculaire :454.54BCL6-IN-9
CAS :BCL6-IN-9 (compound 1) is a potent inhibitor of B-cell lymphoma 6 protein (BCL6) (IC50: 3.9 nM) and can be used to study cancer.Formule :C22H18ClF2N5O2Couleur et forme :SolidMasse moléculaire :457.86MM-589
CAS :MM-589 is a potent WD repeat domain 5 (WDR5) inhibitor and mixed lineage leukemia (MLL) protein-protein interaction.Formule :C28H44N8O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :572.70Human carbonic anhydrase II-IN-1
Compound S-13: Potent hCA II inhibitor, Kis 4.4, 9.2, 480.2, 14.7 nM for hCA II, I, IV, IX. Used in glaucoma research.Formule :C20H25N3O4SCouleur et forme :SolidMasse moléculaire :403.5Galectin-8-IN-1
Galectin-8-IN-1 selectively binds galectin-8N with 48 μM affinity, 15x more than galectin-3.Formule :C16H18N2O6Couleur et forme :SolidMasse moléculaire :334.32Antibacterial agent 99
CAS :Compound 7b (Antibacterial agent 99) is an effective agent with antibacterial, antifungal properties and no haemolytic activity.Formule :C27H27BrN2Couleur et forme :SolidMasse moléculaire :459.42Albicidin
CAS :Albicidin is a DNA gyrase inhibitor produced by Xanthomonas albilineans.Formule :C44H38N6O12Couleur et forme :SolidMasse moléculaire :842.818SphK1-IN-1
SphK1-IN-1: SphK1 ATPase inhibitor, IC50=2.48 μM, potential for cancer research.Formule :C22H22N6O2Couleur et forme :SolidMasse moléculaire :402.45MRS2279
CAS :Selective, high affinity competitive antagonist of the P2Y1 receptorFormule :C13H18ClN5O8P2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :469.71BW A868C
CAS :BW A868C is a potent, selective PGD2 antagonist and a BW245C analogue, inert to other prostaglandin receptors.Formule :C25H37N3O5Couleur et forme :SolidMasse moléculaire :459.58MEIS-IN-3
MEIS-IN-3 is a potent inhibitor of MEIS.Formule :C25H26N2O4Couleur et forme :SolidMasse moléculaire :418.48FP0429
CAS :FP0429 is an agonist of mGlu4.Formule :C10H12N2O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :272.21ABD957
CAS :ABD957: covalent ABHD17 depalmitoylases inhibitor, IC50 0.21µM for ABHD17B, blocks N-Ras, halts NRAS-mutant AML cell growth.Formule :C27H36F3N7O5SCouleur et forme :SolidMasse moléculaire :627.684,5'-Dimethylangelicin-NHS
NHS-modified coumarin, 4,5'-Dimethylangelicin-NHS, shows photochemical activity & photosensitivity.Formule :C21H19NO7SCouleur et forme :SolidMasse moléculaire :429.44BAY-364
CAS :BAY-364 (BAY-299N) functions as an inhibitor targeting the second bromine domain in TAF1, demonstrating inhibitory effects on TAF1 in Kasumi-1 cells, CD34+Formule :C23H19N3O4Couleur et forme :SolidMasse moléculaire :401.41DH376
CAS :DH376 inhibits DAGLα in a time and dose dependent manner in mouse brain. DH376 shows picomolar activity.Formule :C31H28F2N4O3Couleur et forme :SolidMasse moléculaire :542.58CB1/2 agonist 1
Potent CB1/2 agonist 1; crosses blood-brain barrier; anti-inflammatory, analgesic; for multiple sclerosis research.Formule :C21H24BrFN2O2Couleur et forme :SolidMasse moléculaire :435.33Methyl 5-thia-6,8,11,14-eicosatetraenoate
CAS :Methyl 5-thia-6,8,11,14-eicosatetraenoate is a bioactive chemical.Formule :C20H32O2SCouleur et forme :SolidMasse moléculaire :336.53c(phg-isoDGR-(NMe)k)
CAS :c (phg-isoDGR- (NMe) k) is a selective and effective α5β1-integrin ligand with IC50 of 2.9 nM.Formule :C27H41N9O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :603.67Antitumor agent-74
Antitumor agent-74, a quinazoline derivative, inhibits DNA, arrests cell cycle, and induces apoptosis with agent-75.Formule :C26H23FN6Couleur et forme :SolidMasse moléculaire :438.5LEO 134310
CAS :LEO 134310: Selective, non-steroidal GR agonist with 14 nM EC50, for topical skin disease treatment.Formule :C34H40N2O8Couleur et forme :SolidMasse moléculaire :604.69CAII-IN-1
CAII-IN-1 (3n) is a selective bovine CA-II inhibitor with 10.3 μM IC50, used in carbonic anhydrase disorder studies.Formule :C19H21FN4SCouleur et forme :SolidMasse moléculaire :356.46Fonadelpar
CAS :Fonadelpar is an agonist of PPARδ. It also is used in the research of neuroparalytic keratopathy.Formule :C25H23F3N2O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :504.52MCTR2
CAS :MCTR2, synthesized from DHA in macrophages, aids in tissue repair and reduces inflammation by promoting eicosanoid PGD2 and PGF2α decrease.Formule :C27H40N2O6SCouleur et forme :SolidMasse moléculaire :520.68Isoleucyl tRNA synthetase-IN-1
CAS :Isoleucyl tRNA synthetase-IN-1 is a selective and potent inhibitor (Ki: 88 nM) that targets isoleucyl tRNA synthetase (IleRS).Formule :C23H35N5O7SCouleur et forme :SolidMasse moléculaire :525.62JBJ-09-063
CAS :JBJ-09-063: EGFR inhibitor, IC50s 0.147-0.396 nM for various mutants; hinders EGFR/Akt/ERK1/2 phosphorylation; targets TKI-sensitive/resistant lung cancer.Formule :C31H29FN4O3SCouleur et forme :SolidMasse moléculaire :556.65PNU-248686A
CAS :PNU-248686A is an inhibitor of matrix metalloproteinase (MMP).Formule :C22H18ClNaO5S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :484.95Taprostene
CAS :Taprostene (CG-4203), a stable Prostacyclin analogue, protects endothelium and myocardium post-ischemia in cats, with minimal hemodynamic impact.Formule :C24H30O5Couleur et forme :SolidMasse moléculaire :398.49GSK-3β inhibitor 7
GSK-3β inhibitor 7 is a GSK-3β inhibitor (IC50: 5.25 μM).Formule :C27H23BrN4O2SCouleur et forme :SolidMasse moléculaire :547.47COX-2-IN-13
COX-2-IN-13 is a potent, selective COX-2 inhibitor with 0.98 μM IC50; shows strong anti-inflammatory properties and low acute toxicity.Formule :C19H18N2O5SCouleur et forme :SolidMasse moléculaire :386.42Tubulin inhibitor 17
Compound 3b inhibits tubulin polymerization, IC50 12.38 µM, with anticancer properties and promotes cell apoptosis.Formule :C17H16N2OCouleur et forme :SolidMasse moléculaire :264.32DBCO-Sulfo-Link-biotin
CAS :DBCO-Sulfo-Link-biotin is a cleavable linker employed in the synthesis of antibody-drug conjugates (ADCs) [1].Formule :C31H35N5O7S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :653.77Aeroplysinin 1
CAS :Aeroplysinin I is an antibacterial compound from the sponge. It has cytotoxic activity against colon cancer cells by promoting β-catenin degradation.Formule :C9H9Br2NO3Couleur et forme :SolidMasse moléculaire :338.98MK-8318
CAS :MK-8318 is an effective and selective antagonist of the CRTh2 receptor (Ki: 5.0 nM).Formule :C27H26F4N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :534.5AN-12-H5
CAS :AN-12-H5 is an anti-enteroviral compound that targets the replication process of PV and EV71 viruses.Formule :C24H23N3O4S3Couleur et forme :SolidMasse moléculaire :513.65Dihydro-β-erythroidine hydrobromide
CAS :Dihydro-β-erythroidine hydrobromide(DHβE) is a potent, oral active and competitive antagonist of neuronal nicotinic acetylcholine receptors (nAChRs).Formule :C16H22BrNO3Degré de pureté :98%Couleur et forme :White SolidMasse moléculaire :356.26Cbl-b-IN-1
CAS :Cbl-b-IN-1 is a potent Cbl-b inhibitor (IC50 <100 nM) with potential anticancer activity for the study of intestinal inflammation.Formule :C29H34N6O2Degré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :498.631ent-8-iso-15(S)-Prostaglandin F2α
CAS :Isoprostanes are produced by the non-enzymatic, free radical peroxidation of phospholipid-esterified arachidonic acid.Formule :C20H34O5Couleur et forme :SolidMasse moléculaire :354.48DNA crosslinker 1 dihydrochloride
CAS :DNA Crosslinker 1 binds DNA minor groove with 1.1°C affinity increase; used in cancer research.Formule :C15H22Cl2N8OCouleur et forme :SolidMasse moléculaire :401.29Utrophin modulator 1
UM1 upregulates utrophin, has EC50 of 0.11 μM, useful in DMD research.Formule :C22H18N6OCouleur et forme :SolidMasse moléculaire :382.42LRRK2-IN-4
CAS :LRRK2-IN-4: Potent, selective LRRK2 inhibitor, oral, BBB-penetrating, IC50=2.6 nM, potential for Parkinson's.Formule :C25H29ClF2N6O2Couleur et forme :SolidMasse moléculaire :518.99Protease-Activated Receptor-1 antagonist 3
PAR-1 antagonist 3: potent (IC50: 7 nM), binds hERG K+ channels (IC50: 9 μM).Formule :C30H34N4O3Couleur et forme :SolidMasse moléculaire :498.62Cilobamine mesylate
CAS :Cilobamine mesylate is a drug which acts as a norepinephrine-dopamine reuptake inhibitor (NDRI) and has stimulant and antidepressant effects.Formule :C18H27Cl2NO4SCouleur et forme :SolidMasse moléculaire :424.38TLR7/8 antagonist 1
Compound 16c, an imidazoquinoline, is a TLR7/8 agonist; IC50: 3.91 μM (TLR7), 2.19 μM (TLR8); targets TLR-2050 for disease treatment.Formule :C24H27N5O2Couleur et forme :SolidMasse moléculaire :417.5Homopteroic Acid
CAS :Homopteroic Acid, a precursor to Homofolic Acid, inhibits L1210 mouse leukemia growth by targeting folate uptake.Formule :C15H14N6O3Couleur et forme :SolidMasse moléculaire :326.31U92016A hydrochloride
CAS :U92016A hydrochloride: potent, orally active 5-HT1A agonist, metabolically stable, high intrinsic activity, Ki=0.2 nM.Formule :C19H26ClN3Couleur et forme :SolidMasse moléculaire :331.89Lycopodine
CAS :Lycopodine, a bioactive compound derived from Lycopodium clavatum spores, effectively inhibits the proliferation of HeLa cells through the induction of
Formule :C16H25NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :247.38O4
CAS :O4 is a novel stabilizer of amyloid- fibrils. O4 used for accelerating the formation of end-stage mature fibrils.Formule :C24H15NO7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :429.38Novokinin
CAS :Angiotensin AT2 receptor agonistFormule :C39H61N11O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :795.97Glutaminyl cyclases-IN-1
Glutaminyl cyclase inhibitor IsoQC-IN-1: IC50=12 nM for QC, 73 nM for isoQC; blocks CD47/SIRPα; boosts THP-1, U937 macrophage phagocytosis.Formule :C25H30N6O2SCouleur et forme :SolidMasse moléculaire :478.61Antitumor agent-43
Antitumor agent-43 (Compound 4B) is a potent antitumor agent that induces cell cycle arrest at G2/M phase.Formule :C16H8N2O3Couleur et forme :SolidMasse moléculaire :276.25
