Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.805 produits)
- Apoptose(6.292 produits)
- Cycle cellulaire/point de contrôle(4.820 produits)
- Chromatine/Épigénétique(2.490 produits)
- Signalisation du cytosquelette(1.544 produits)
- Altération de l'ADN/réparation de l'ADN(2.940 produits)
- Endocrinologie/Hormones(3.706 produits)
- Enzyme(3.670 produits)
- GPCR/G-Protéine(9.024 produits)
- Immunologie et Inflammation(3.902 produits)
- Virus de la grippe(302 produits)
- Signalisation JAK/STAT(417 produits)
- Signalisation MAPK(1.247 produits)
- Transporteur membranaire/Canal ionique(3.078 produits)
- Métabolisme(10.178 produits)
- Microbiologie/Virologie(7.618 produits)
- Neuroscience(10.367 produits)
- Autres inhibiteurs(35.951 produits)
- Oxydation-Réduction(41 produits)
- Signalisation PI3K/Akt/mTOR(1.442 produits)
- Protéases/Protéasome(1.716 produits)
- Cellules souche et Dérivés(801 produits)
- Tyrosine Kinase/Adaptateurs(2.030 produits)
- Ubiquitination(1.722 produits)
Affichez 16 plus de sous-catégories
66630 produits trouvés pour "Inhibiteurs"
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AChE-IN-25
AChE-IN-25: selective, potent AChE inhibitor, non-competitive, IC50 = 2.95 μM, for Alzheimer's research.Formule :C20H15ClN4O4SCouleur et forme :SolidMasse moléculaire :442.88ZINC000104379474
ZINC000104379474 is a compound that targets SARS-CoV-2 endoribonuclease.Formule :C27H33N3O10Couleur et forme :SolidMasse moléculaire :559.57RORγt/DHODH-IN-1
CAS :RORγt/DHODH-IN-1 (compound (R)-14d) is a potent, orally active dual inhibitor of RORγt (IC50: 0.083 μM) and DHODH (IC50: 0.172 μM), which exhibits significantFormule :C24H26ClF6N3O3SCouleur et forme :SolidMasse moléculaire :585.99PRMT5-IN-19
PRMT5-IN-19 is a potent, selective PRMT5 inhibitor with IC50 of 23.9 nM and 47 nM, showing anti-cancer activity by inducing apoptosis.Formule :C25H24N4OCouleur et forme :SolidMasse moléculaire :396.48COX-2-IN-9
COX-2-IN-9: potent oral COX-2 blocker, selective over Celecoxib, IC50 10.17 μM, less ulcers, strong anti-inflammatory.Formule :C25H23N5O4S2Couleur et forme :SolidMasse moléculaire :521.61AChE/BACE1/GSK3β-IN-1
AChE/BACE1/GSK3β-IN-1 is an orally active, blood-brain barrier-transparent, moderately bioavailable triple inhibitor of AChE/BACE1/GSK3β.Formule :C26H27FN2O4Couleur et forme :SolidMasse moléculaire :450.5HBV-IN-12
CAS :HBV-IN-12: strong HBsAg & HBV DNA inhibitor; EC50 0.001-0.05 μM & 0.001-0.02 μM respectively. (WO2021204252A1)Formule :C23H27NO8Couleur et forme :SolidMasse moléculaire :445.46Antifungal agent 27
Antifungal agent 27 shows moderate action against MRSA, weak against C. albicans, with MICs of 8 μg/mL and 32 μg/mL, respectively.Formule :C18H23N5OSCouleur et forme :SolidMasse moléculaire :357.475(S),6(S)-DiHETE
CAS :5(S),6(S)-DiHETE: a 5,6-dihydroxy acid from LTA4 hydrolysis, lacks leukotriene activity.Formule :C20H32O4Couleur et forme :SolidMasse moléculaire :336.47A1-Phytoprostane-I
CAS :A1-Phytoprostane-I: cyclopentenone from α-linolenic acid in plants, induces gene expression & increases phytoalexin synthesis.Formule :C18H28O4Couleur et forme :SolidMasse moléculaire :308.41PDHK-IN-3
PDHK-IN-3 (compound 7) is a potent inhibitor of pyruvate dehydrogenase kinase(PDHK) with IC50s of 0.21 and 1.54 μM for PDHK2 and PDHK4, respectively [1].Formule :C17H16N2O2Couleur et forme :SolidMasse moléculaire :280.32Cap-dependent endonuclease-IN-7
CAS :Cap-dependent endonuclease-IN-7, a potent CEN inhibitor, blocks viral mRNA synthesis and virus spread, with research use for influenza A, B, C.Formule :C36H28FN3O7SCouleur et forme :SolidMasse moléculaire :665.69LRH-1 modulator-1
CAS :LRH-1 modulator-1: potent agonist, boosts IL-10, reduces IL-1b/TNFa, anti-inflammatory in gut.Formule :C28H36N2O2SCouleur et forme :SolidMasse moléculaire :464.66EICAR
CAS :EICAR: IMP dehydrogenase inhibitor with anticancer and antiviral properties, failed in leukemia trials, active against various viruses but not SARS.Formule :C11H13N3O5Couleur et forme :SolidMasse moléculaire :267.24LJ-4517
LJ-4517 is an effective A2AAR antagonist (Ki=18.3 nM). LJ-4517 can effectively replace the binding of [3H] ZM241385 at WT A2AAR.Formule :C19H21N5O3SCouleur et forme :SolidMasse moléculaire :399.47QTX125 TFA
QTX125 TFA: Potent, selective HDAC6 inhibitor with antitumor effects.Formule :C25H20F3N3O7Couleur et forme :SolidMasse moléculaire :531.44Longicoricin
CAS :Longicoricin is a monotetrahydrofuran Annonaceous acetogenin from Asimina longifolia.Formule :C37H68O6Couleur et forme :SolidMasse moléculaire :608.93LY 292728
CAS :LY 292728 is a highly potent antagonist of leukotriene B4 receptor.Formule :C34H29FO9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :600.59LY503430
CAS :LY503430: Oral AMPA enhancer with nootropic, neuroprotective properties, mitigates 6-OHDA/MPTP brain damage.Formule :C20H25FN2O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :392.49HER2-IN-9
HER2-IN-9, an oral HER2 inhibitor (IC50: 0.03 μM), hinders growth and spread of HER2+ breast cancer.Formule :C19H14BrF3N2OCouleur et forme :SolidMasse moléculaire :423.23MLKL-IN-1
MLKL-IN-1 is a covalent inhibitor of MLKL with a Kd value of 50 μM.Formule :C19H20N2O3Couleur et forme :SolidMasse moléculaire :324.37HPK1-IN-3
HPK1-IN-3: Selective HPK1 inhibitor, ATP-competitive, IC50=0.25nM; boosts IL-2 in PBMCs, EC50=108nM.Formule :C23H22F4N6O2Couleur et forme :SolidMasse moléculaire :490.45L-threo-Sphingosine C-18
CAS :L-threo-Sphingosine C-18 is a protein kinase C inhibitor.Formule :C18H37NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :299.49AZD-4121
CAS :<p>AZD-4121 is an oral cholesterol absorption inhibitor targeting NPC1L1 for the treatment of dyslipidaemia.</p>Formule :C36H39F2N3O7SCouleur et forme :SolidMasse moléculaire :695.77ABT 491 Hydrochloride
CAS :ABT-491 hydrochloride is an active platelet activator receptor (PAF-R) antagonist with good selectivity and oral administration.Formule :C28H23ClFN5O2Couleur et forme :SolidMasse moléculaire :515.97PDE-I2
CAS :PDE-I2 is a parasite schizogony inhibitor.Formule :C25H23N5O8Couleur et forme :SolidMasse moléculaire :521.48Metoquizine
CAS :Metoquizine is an anticholinergic compound. It is a muscarinic acetylcholine receptor antagonist that has been used to treat ulcers.Formule :C22H27N5ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :377.48Antitumor agent-78
Antitumor agent-78 blocks GPx-4, raises COX2, triggers apoptosis, halts EMT, and stifles cancer cell growth and migration.Couleur et forme :SoildPlasma kallikrein-IN-2
Plasma kallikrein-IN-2: PKal inhibitor, IC50=0.1 nM. Used in angioedema, diabetic eye disease research.Formule :C28H24ClF3N8O3Couleur et forme :SolidMasse moléculaire :612.99Tribenuron
CAS :<p>Tribenuron, a slow acting sulfonylurea herbicide, controls broadleaf weed.</p>Formule :C14H15N5O6SCouleur et forme :SolidMasse moléculaire :381.36HDAC-IN-9
HDAC-IN-9, a dual tubulin/HDAC inhibitor, impedes A549 cell invasion/migration and shows strong anti-tumor/angiogenic effects.Formule :C33H38N2O4Couleur et forme :SolidMasse moléculaire :526.67(2R,3S)-Azelaprag
CAS :(2R,3S)-N-(4-(2,6-dimethoxyphenyl)-5-(5-methylpyridin-3-yl)-4H-1,2,4-triazol-3-yl)-3-(5-methylpyrimidin-2-yl)butane-2-sulfonamide is an Apelin receptor agonistFormule :C25H29N7O4SDegré de pureté :97.47% - >99.99%Couleur et forme :SoildMasse moléculaire :523.61MRGPRX1 agonist 3
Compound 1f, a potent MRGPRX1 agonist, has an EC50 of 0.22 μM, useful for neuropathic pain studies.Formule :C14H11FN2OSCouleur et forme :SolidMasse moléculaire :274.31cis-RdRP-IN-5
Cis-RdRP-IN-5 is an effective inhibitor of the influenza virus RNA-dependent RNA polymerase (RdRP), employed in influenza virus research.Formule :C23H21N3O5Couleur et forme :SolidMasse moléculaire :419.43AS1940477
CAS :AS1940477 selectively inhibits p38 MAPK α/β, blocks proinflammatory cytokines in cells, and has anti-inflammatory effects in rats.Formule :C24H22FN5O2Couleur et forme :SolidMasse moléculaire :431.46DJT06001
CAS :DJT06001 is a selective Factor Xa inhibitor, reducing thrombus formation with low risk of bleeding.Formule :C21H20ClN3O5SCouleur et forme :SolidMasse moléculaire :461.92PAIR2
CAS :PAIR2 is a selective IRE1α RNase partial antagonist, blocking its ATP site and preventing KIRA from hindering XBP1 splicing.Formule :C27H26F4N6O3SCouleur et forme :SolidMasse moléculaire :590.59NPEC-caged-(S)-3,4-DCPG
CAS :mGlu8a agonistFormule :C19H16N2O10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :432.34K027
K027 is a potent organophosphate (OP) inhibitor of acetylcholinesterase (AChE) reactivation. k027 can be used to study Alzheimer's disease.Formule :C15H18Br2N4O2Couleur et forme :SolidMasse moléculaire :446.14Tuberculosis inhibitor 5
Compound 11i: potent, non-toxic anti-tuberculosis biphenyl analogue.Formule :C25H18N2O2SCouleur et forme :SolidMasse moléculaire :410.4912(S)-HETE
CAS :<p>Enpatoran hydrochloride (M5049 hydrochloride) is a TLR7/8 inhibitor with antiviral activity that is used in the study of autoimmune diseases.</p>Formule :C20H32O3Couleur et forme :SolidMasse moléculaire :320.47AB 5046A
CAS :AB 5046A is a chlorosis inducing substance isolated from Nodulisporium SP.Formule :C10H14O4Couleur et forme :SolidMasse moléculaire :198.22SMP-797 HCl
CAS :SMP-797 HCl, an ACAT (acyl-CoA-cholesterol acyltransferase) inhibitor, is used potentially for the treatment of Hyperlipidemia.Formule :C34H44ClN5O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :622.20EGFR-IN-58
EGFR-IN-58 is a potent, selective, ATP-competitive inhibitor of EGFR. EGFR-IN-58 exhibits significant cytotoxicity against melanoma, colon and blood cancers.Formule :C31H30FN7OCouleur et forme :SolidMasse moléculaire :535.61T01-1
CAS :T01-1, a derivative of camptothecin, is an anticancer agent demonstrating significant anti-proliferative activity.Formule :C26H29N3O6SCouleur et forme :SolidMasse moléculaire :511.59FR 900452
CAS :FR 900452 is a platelet activating factor antagonist from fermentatiion products of Streptomyces phaeofaciens.Formule :C22H25N3O3SCouleur et forme :SolidMasse moléculaire :411.52Netupitant metabolite Monohydroxy Netupitant
CAS :Monohydroxy Netupitant is a highly selective antagonist of NK1 receptor, and is Netupitant metabolite.Formule :C30H32F6N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :594.59Tipelukast
CAS :Tipelukast (KCA 757), an oral drug for asthma research, blocks leukotrienes and fights inflammation and fibrosis.Formule :C29H38O7SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :530.67BET-IN-6
CAS :BET-IN-6: Potent BRD2/4 inhibitor and ligand for PROTAC BRD2/BRD4 degrader-1 synthesis.Formule :C22H20N2O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :440.47Lp-PLA2-IN-6
CAS :Lp-PLA2-IN-6: Potent tetracyclic inhibitor of rhLp-PLA2, with pIC50 of 10.0, and potential in neurodegenerative research.Formule :C25H21F5N4O3Couleur et forme :SolidMasse moléculaire :520.45KDOAM-25 citrate
CAS :KDOAM-25 citrate inhibits KDM5A/B/C/D (IC50: 71, 19, 69, 69 nM); boosts H3K4 methylation, hinders MM1S cell growth. [1]Formule :C21H33N5O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :499.51(Rac)-PT2399
CAS :(Rac)-PT2399 is a potent and specific inhibitor of hypoxia-inducible factor 2a (HIF-2α)(IC50 of 0.01 μM).Formule :C17H10F5NO4SCouleur et forme :SolidMasse moléculaire :419.32BSc5367
CAS :<p>BSc5367 inhibits Nek1 kinase (IC50: 11.5 nM), key in cell cycle, DNA repair, impacting ALS, PKD, cancer.</p>Formule :C20H15N3O2Couleur et forme :SoildMasse moléculaire :329.35Luffolide
CAS :Luffolide, a Luffariella sponge metabolite, shares manoalide's anti-inflammatory traits and fully inhibits PLA2's cleavage of phosphatidylcholine.Formule :C27H40O6Couleur et forme :SolidMasse moléculaire :460.60Mesulergine hydrochloride
CAS :5-HT2A and 2C receptor antagonistFormule :C18H27ClN4O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :398.95CPPG
CAS :CPPG: potent group II/III mGlu receptor antagonist, 20x more selective for group III (IC50: 2.2 nM) than II (46.2 nM) in rat cortex.Formule :C11H14NO5PCouleur et forme :SolidMasse moléculaire :271.21BM635 hydrochloride
BM635 hydrochloride, an MmpL3 inhibitor, strongly blocks Divergent bacteriophage H37Rv (MIC50: 0.08 μM), with doubled in vivo potency.Formule :C25H30ClFN2OCouleur et forme :SolidMasse moléculaire :428.97RET-IN-7
CAS :RET-IN-7 exhibits strong inhibitory effects against RET kinase in vitro and shows significant efficacy in treating RET-driven tumor xenografts in mice throughFormule :C22H24ClFN6O2Couleur et forme :SolidMasse moléculaire :458.92D18
CAS :D18: Dual agonist for TLR7/8, boosts PD-L1, aids tumor sensitivity to PD-1/PD-L1 inhibitors, and is a cytotoxin for ADC HE-S2.Formule :C21H28N6Couleur et forme :SolidMasse moléculaire :364.49Antitumor agent-43
Antitumor agent-43 (Compound 4B) is a potent antitumor agent that induces cell cycle arrest at G2/M phase.Formule :C16H8N2O3Couleur et forme :SolidMasse moléculaire :276.25Tonantzitlolone
CAS :Tonantzitlolone activates TRPC1/4/5 channels, PKCα/θ, inhibits IRS1/PI3K/AKT, and triggers HSF1 to induce glucose dependence.Formule :C26H40O7Couleur et forme :SolidMasse moléculaire :464.59BTK-IN-7
BTK-IN-7 is a potent inhibitor for BTK with 4.0 nM IC50, highly selective over ITK and EGFR, showing strong antitumor activity.Formule :C30H32N6O4Couleur et forme :SolidMasse moléculaire :540.61Carbonic anhydrase inhibitor 4
CA inhibitor 4, photoprobe; targets hCA I-XIV; Ki: 640-1166 nM.Formule :C21H18N2O4SCouleur et forme :SolidMasse moléculaire :394.44Xylarianaphthol-1
CAS :Xylarianaphthol-1 is an activator of p21 promoter in a p53-independent manner.Formule :C16H20BrFN2O2Couleur et forme :SolidMasse moléculaire :371.24PF-07054894
CAS :PF-07054894: potent CCR6 antagonist, targets GPCR, for inflammatory bowel disease research.Formule :C24H30N6O4Couleur et forme :SolidMasse moléculaire :466.53SI-109
CAS :SI-109 is a potent inhibitor of STAT3 SH2 domain (Ki=9 nM),and with antitumor activity.Formule :C40H44F2N7O9PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :835.79ACSS2-IN-1
CAS :ACSS2-IN-1, a potent ACSS2 inhibitor, has IC50 0.01-<1 nM; useful in cancer research.Formule :C27H25ClN6O2Couleur et forme :SolidMasse moléculaire :500.98L 365209
CAS :L 365209 is an oxytocin antagonist.Formule :C40H50N8O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :738.88Galectin-8-IN-1
Galectin-8-IN-1 selectively binds galectin-8N with 48 μM affinity, 15x more than galectin-3.Formule :C16H18N2O6Couleur et forme :SolidMasse moléculaire :334.32(±)-ANAP hydrochloride (1185251-08-4 free base)
(±)-ANAP hydrochloride is the amino acid analog of prodan. It can be used as a fluorescent probes and enhance environmental sensitivity.Formule :C15H17ClN2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :308.76Abarelix acetate
CAS :Abarelix acetate: synthetic GnRHR antagonist, spikes histamine, lowers LH and testosterone temporarily, used in advanced prostate cancer.Formule :C72H95ClN14O14·xC2H4O2Couleur et forme :SolidMasse moléculaire :1476.14Antibacterial agent 81
CAS :Antibacterial agent 81 blocks DNA transcription, targets S. aureus (MIC 12.5μM) & M. smegmatis (MIC 7.8μM). Used in infection research.Formule :C33H28N2O8Couleur et forme :SolidMasse moléculaire :580.58SGLT1/2-IN-1
CAS :SGLT1/2-IN-1 is a dual SGLT1/SGLT2 inhibitor.Formule :C25H28O8Couleur et forme :SolidMasse moléculaire :456.48CDK8-IN-11 hydrochloride
CDK8-IN-11 HCl: potent, selective CDK8 inhibitor (IC50: 46 nM), blocks WNT/β-catenin pathway, used in colon cancer research.Formule :C19H16ClF3N4O2Couleur et forme :SolidMasse moléculaire :424.8E7090 succinate
CAS :E7090 succinate inhibits FGFR1, FGFR2, and FGFR3 with IC50: 0.71, 0.50, 1.2 nM; less so FGFR4 at 120 nM.Formule :C76H92N10O24Couleur et forme :SolidMasse moléculaire :1529.60Cap-dependent endonuclease-IN-5
CAS :Cap-dependent endonuclease-IN-5 inhibits CEN and fights influenza with low toxicity and good in vivo properties.Formule :C27H21F2N3O4S2Couleur et forme :SolidMasse moléculaire :553.60NS2B/NS3-IN-5
Compound 25b inhibits DENV2/ZIKV NS2B/NS3 proteases; IC50: ZIKV 0.67μM, DENV2 4.38μM.Formule :C14H9IN2O3SCouleur et forme :SolidMasse moléculaire :412.2DC4SMe
CAS :DC4SMe, a prodrug for targeted tumor therapy and ADC synthesis, has IC50s: 1.9 nM (Ramos), 2.9 nM (Namalwa), 1.8 nM (HL60/s).Formule :C35H31ClN5O7PS2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :764.21UCN-01
CAS :inhibitor of Akt, protein kinase C, PDK1 and cyclin-dependent kinasesFormule :C28H26N4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :482.53Flurandrenolone Acetate
CAS :Flurandrenolone Acetate, a synthetic glucocorticoid derived from Flurandrenolide, is used to study skin issues like eczema and psoriasis.Formule :C26H35FO7Couleur et forme :SolidMasse moléculaire :478.55C5aR-IN-3
CAS :C5aR-IN-3, a potent C5aR inhibitor, may treat autoimmune and inflammatory diseases.Formule :C36H40FN5O3Couleur et forme :SolidMasse moléculaire :609.73Omesdafexor
CAS :Omesdafexor is an FXR agonist that can be used to study diseases caused by liver disease or metabolic inflammation.Formule :C34H43N3O3Couleur et forme :SolidMasse moléculaire :541.72Dinordrin
CAS :Dinordrin is an implantation inhibitor and hormone.Formule :C27H36O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :424.57FT3967385
FT3967385: New USP30 inhibitor boosts mitochondrial ubiquitylation via PINK1-PARKIN.Formule :C21H19N5O2Couleur et forme :SolidMasse moléculaire :373.41Antibacterial agent 112
Compound 112: Powerful antibacterial, MIC 1250 μM against B. subtilis, E. coli, E. faecalis, S. typhimurium, S. aureus; also an HIV-1 antibody.Formule :C35H23N5O5Couleur et forme :SolidMasse moléculaire :593.59URAT1 inhibitor 3
URAT1 inhibitor 3: potent oral URAT1 blocker, IC50=0.8 nM, for gout/hyperuricemia study.Formule :C14H8Cl2N2O2Couleur et forme :SolidMasse moléculaire :307.13Lipoxin A5
CAS :LXA5 is made from EPA by leukocytes, contracts guinea pig lungs like LXA4/LXB4, but doesn't dilate aorta.Formule :C20H30O5Couleur et forme :SolidMasse moléculaire :350.45UNC7467
CAS :UNC7467, potent IP6K2/1/6 inhibitor (4.9/8.9/1320 nM); lowers inositol pyrophosphates, minimal impact on other inositol phosphates; for obesity research.Formule :C20H13NO3Degré de pureté :98.28% - 98.64%Couleur et forme :SoildMasse moléculaire :315.32Anti-ToCV agent 1
Anti-ToCV agent 1 can be used as a potential anti-ToCV drug.Formule :C22H19FN2O5SCouleur et forme :SolidMasse moléculaire :442.46HDAC/HSP90-IN-4
HDAC/HSP90-IN-4 inhibits HDAC (20 IC50=194nM, 26 IC50=360nM) & HSP90α (20 IC50=153nM, 26 IC50=77nM), affects cancer cell survival and invasion.Formule :C20H23N3O6Couleur et forme :SolidMasse moléculaire :401.15869Lasonolide A
CAS :Lasonolide A, an anticancer compound from Forcepia sponge, shows nanomolar growth inhibition and unique cytotoxicity in the NCI 60-cell-line screen.Formule :C41H60O9Couleur et forme :SolidMasse moléculaire :696.91DNDI-8219
CAS :DNDI-8219 is an antitubercular agent. It has potent antileishmanial effects.Formule :C13H10F3N3O5Couleur et forme :SolidMasse moléculaire :345.23MDL-27088
CAS :MDL-27088 is an angiotensin-covering enzyme inhibitor.Formule :C25H28N2O5Couleur et forme :SolidMasse moléculaire :436.50CRM1 degrader 1
CRM1 degrader 1 (1l) is a low-toxic CRM1 degrader that induces apoptosis in gastric carcinoma and selectively inhibits the proliferation of gastric cancer[1].Formule :C16H20O3Couleur et forme :SolidMasse moléculaire :260.33β-Glucuronidase/hCAII-IN-1
CAS :β-Glucuronidase/hCAII-IN-2 (Compound 12e) is a compound that effectively inhibits both β-glucuronidase and human Carbonic Anhydrase II (hCA II), exhibiting IC50Formule :C30H21NO9Couleur et forme :SolidMasse moléculaire :539.49HIV-IN-3
HIV-IN-3 (Compound 22a) is a potent inhibitor of HIV (IC50: 1.5 μM). HIV-IN-3 has potential for the study of HIV-related diseases.Formule :C21H32ClN7O3Couleur et forme :SolidMasse moléculaire :465.98(+)-Sparteine sulfate pentahydrate
(+)-sparteine (sulfate pentahydrate) is a ganglion blocker that competitively blocks nicotinic acetylcholine receptors in neurons.Formule :C15H38N2O9SCouleur et forme :SolidMasse moléculaire :422.54DMGF
CAS :DMGF, a biflavonoid from Taxus, induces apoptosis, autophagy, and inhibits B16F10 cell motility and MMP-2 expression, hindering melanoma metastasis.Formule :C32H22O10Couleur et forme :SolidMasse moléculaire :566.51MtTMPK-IN-9
MtTMPK-IN-9 moderately inhibits MtbTMPK (IC50: 48 μM), has submicromolar Mycobacterium activity, and is non-toxic, aiding tuberculosis research.Formule :C25H26N6O7Couleur et forme :SolidMasse moléculaire :522.51Spliceostatin A
CAS :Spliceostatin A is an anticancer agent and splicing inhibitor that induces apoptosis by inducing cell cycle arrest in the G1 and G2/M phases.Formule :C28H43NO8Degré de pureté :94.66%Couleur et forme :SolidMasse moléculaire :521.643
