Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.801 produits)
- Apoptose(6.278 produits)
- Cycle cellulaire/point de contrôle(4.814 produits)
- Chromatine/Épigénétique(2.476 produits)
- Signalisation du cytosquelette(1.541 produits)
- Altération de l'ADN/réparation de l'ADN(2.948 produits)
- Endocrinologie/Hormones(3.708 produits)
- Enzyme(3.671 produits)
- GPCR/G-Protéine(9.024 produits)
- Immunologie et Inflammation(3.893 produits)
- Virus de la grippe(302 produits)
- Signalisation JAK/STAT(414 produits)
- Signalisation MAPK(1.247 produits)
- Transporteur membranaire/Canal ionique(3.064 produits)
- Métabolisme(10.184 produits)
- Microbiologie/Virologie(7.614 produits)
- Neuroscience(10.377 produits)
- Autres inhibiteurs(36.011 produits)
- Oxydation-Réduction(41 produits)
- Signalisation PI3K/Akt/mTOR(1.441 produits)
- Protéases/Protéasome(1.720 produits)
- Cellules souche et Dérivés(812 produits)
- Tyrosine Kinase/Adaptateurs(2.031 produits)
- Ubiquitination(1.717 produits)
Affichez 16 plus de sous-catégories
66673 produits trouvés pour "Inhibiteurs"
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Imolamine hydrochloride
CAS :Imolamine hydrochloride is a blood platelet aggregation antagonist.Formule :C14H21ClN4OCouleur et forme :SolidMasse moléculaire :296.80BAY-850 HCl
BAY-850 is a selective probe targeting Atad2A's bromine domain, displacing acetylated H4 peptides and detaching ATAD2 from chromatin at 1μm.Formule :C38H48Cl5N5O3Couleur et forme :SolidMasse moléculaire :800.08GSK2578999A
CAS :GSK2578999A is a betulin derivative with antitumor activity.Formule :C46H62ClNO7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :776.44Dihydrophaseic acid
CAS :Dihydrophaseic acid 3'-O-b-D-glucopyranoside (D3G) can increase the proliferation and differentiation of osteoblast cells and enhance bone formation, suggestsFormule :C15H22O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :282.33Oberadilol
CAS :Oberadilol is a pyridazinone derivative with vasodilatory and beta-adrenergic blocking activities and type III phosphodiesterase inhibitory actionFormule :C25H30ClN5O3Couleur et forme :SolidMasse moléculaire :483.99GSK3527497
CAS :GSK3527497 is a novel potent and selective inhibitor of transient receptor potential vanilloid-4 (TRPV4).Formule :C17H16ClFN4O4SCouleur et forme :SolidMasse moléculaire :426.85SDM25N hydrochloride
CAS :δ receptor antagonistFormule :C26H27ClN2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :450.96SG3199
CAS :<p>SG3199, a PBD dimer, binds DNA's minor groove, forms covalent cross-links, and is cytotoxic to various human cancer cells.</p>Formule :C33H36N4O6Couleur et forme :SolidMasse moléculaire :584.66Casein Kinase II Inhibitor IV Hydrochloride
CAS :Casein Kinase II Inhibitor IV HCl promotes keratinocyte differentiation, potential for skin disorder therapy.Formule :C24H24ClN5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :465.93Silvestrol
CAS :Silvestrol is a eukaryotic translation initiation factor 4A inhibitor. Silvestrol causes autophagy and caspase-mediated apoptosis.Formule :C34H38O13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :654.66SSTR4 agonist 4
CAS :SSTR4 agonist 4, potent in pain research, shows promise in rodent pain models, with potential for Alzheimer's due to hippocampus activity.Formule :C19H26N4OCouleur et forme :SolidMasse moléculaire :326.44Freselestat
CAS :Freselestat (ONO-6818) inhibits neutrophil elastase, reduces interleukin 8, C5B-9, and inflammation in cardiopulmonary bypass.Formule :C23H28N6O4Couleur et forme :SolidMasse moléculaire :452.51PEN-866
CAS :PEN-866, a conjugate of HSP90i and SN-38, may control early NSCLC tumor growth.Formule :C49H49N7O9Couleur et forme :SolidMasse moléculaire :879.95MtDTBS-IN-1
MtDTBS-IN-1 is a notably potent binder (K_D = 57 nM) and inhibitor (K_i = 5 μM) of MtDTBS.Formule :C16H16N4O5Couleur et forme :SolidMasse moléculaire :344.32CB30865
CAS :CB30865 (ZM 242421) is a selective and highly effective nicotinamide phosphoribosyltransferase (Nampt) inhibitor with potential antitumor activity.Formule :C26H22BrN5O2Degré de pureté :99.04%Couleur et forme :SolidMasse moléculaire :516.39FW 34569
CAS :FW 34569, an enkephalin analog, boosts growth hormones and prolactin, reduces cortisol and LH; FSH stable.Formule :C30H43N5O7SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :617.76WF-47-JS03
<p>WF-47-JS03: RET kinase inhibitor, crosses blood-brain barrier, 500x more selective for KDR, IC50: 1.7 nM in Ba/F3 cells, 5.3 nM in LC-2/ad lung cancer cells.</p>Formule :C30H38N6O2Couleur et forme :SolidMasse moléculaire :514.66GR-71251
CAS :<p>GR-71251 is a Tachykinin receptor antagonist.</p>Formule :C74H105N19O13Couleur et forme :SolidMasse moléculaire :1468.74Guraxetan
Guraxetan can be used in the synthesis of the antitumour drug Lutetium (177Lu) zadavotide Guraxetan.Formule :C20H34N4O9Couleur et forme :SolidMasse moléculaire :474.51COX-2-IN-6
CAS :COX-2-IN-6: Potent, selective COX-2 inhibitor; oral; IC50 0.84μM, Ki 69nM; blocks PGE2 synthesis; prevents colorectal cancer.Formule :C20H27NO6SDegré de pureté :99.29% - 99.32%Couleur et forme :SoildMasse moléculaire :409.5AZD4625
AZD4625 (Compound 21) is a selective, potent, orally active, covalent and mutagenic mutant GTPaseKRASG12C inhibitor.Formule :C24H21ClF2N4O3Couleur et forme :SolidMasse moléculaire :486.9GNE684
CAS :GNE684 inhibits RIP1; Ki app: 21 nM (human), 189 nM (mouse), 691 nM (rat).Formule :C23H24N6O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :432.48TAS05567
CAS :TAS05567 is a potent, highly selective, and ATP-competitive Syk inhibitor (IC50: 0.37 nM).Formule :C21H29N9O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :439.51BI 224436
CAS :BI 224436 is an inhibitor of HIV-1 noncatalytic site integrase. With EC50 values of less than 15 nM against different HIV-1 laboratory strains.Formule :C27H26N2O4Couleur et forme :SolidMasse moléculaire :442.51CD73-IN-12
CD73-IN-12, a compound from CN114437038A, shows strong anti-tumor activity by effectively inhibiting CD73 enzyme.Formule :C17H14F2N4O2Couleur et forme :SolidMasse moléculaire :344.32ZM514
ZM514 inhibits CD73 (hCD73 IC50: 1.39 μM, mCD73 IC50: 14.65 μM) with low cytotoxicity, suitable for cancer research.Formule :C36H57NO4Couleur et forme :SolidMasse moléculaire :567.84BAY-7598
CAS :BAY-7598 is a potent, selective, and orally bioavailable MMP12 inhibitor (IC50s: 0.085, 0.67, and 1.1 nM for human/murine/rat MMP12).Formule :C28H31N3O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :505.56Spliceostatin A
CAS :Spliceostatin A is an anticancer agent and splicing inhibitor that induces apoptosis by inducing cell cycle arrest in the G1 and G2/M phases.Formule :C28H43NO8Degré de pureté :94.66%Couleur et forme :SolidMasse moléculaire :521.643FT001
CAS :FT001: Oral BET Bromodomain inhibitor, IC50=0.46μM, suppresses MYC, anti-cancer, effective in vitro/vivo.Formule :C25H29N3O4SDegré de pureté :99.9%Couleur et forme :SolidMasse moléculaire :467.58Ref: TM-T27392
1mg115,00€2mg172,00€5mg255,00€10mg374,00€25mg562,00€50mg787,00€100mg1.074,00€500mg2.147,00€1mL*10mM (DMSO)299,00€S-1033
CAS :S-1033 is an FP receptor agonist.Formule :C20H33NaO4Couleur et forme :SolidMasse moléculaire :360.4698Vps34-IN-3
Vps34-IN-3 is a potent, selective, and orally bioavailable inhibitor of VPS34 kinase .Formule :C14H20N4O2Couleur et forme :SolidMasse moléculaire :276.33Mcl-1 inhibitor 9
CAS :Mcl-1 Inhibitor 9 (Example 2) is a potent inhibitor of myeloid cell leukemia 1 (Mcl-1), demonstrating anti-tumor activity with an IC50 value of 0.21889 nM.Formule :C32H39ClN2O5SCouleur et forme :SolidMasse moléculaire :599.18SENP2-IN-1
CAS :SENP2-IN-1 selectively inhibits SENP2, SENP1, and SENP5 with low IC50 values; useful in cancer studies.Formule :C32H29N3O5S2Couleur et forme :SolidMasse moléculaire :599.72MEIS-IN-2
MEIS-IN-2 is an inhibitor of MEIS1. MEIS-IN-2 can be used in studies of cardiac regeneration and haematopoietic stem cell (HSC) regulation.Formule :C23H21ClN2O4Couleur et forme :SolidMasse moléculaire :424.88K203
K203 is a potent tabun-inhibited AChE reactivator and is an important antidote to organophosphorus poisoning.Formule :C16H18Br2N4O2Couleur et forme :SolidMasse moléculaire :458.15I-BET282E
I-BET282E inhibits eight BET bromodomains (pIC50 6.4-7.7) with selectivity for other bromodomain proteins.Formule :C26H34N4O7SCouleur et forme :SolidMasse moléculaire :546.64PARP1/BRD4-IN-2
PARP1/BRD4-IN-2, a potent inhibitor of PARP1 and BRD4, halts cell cycle, triggers apoptosis, and has antitumor effects on TNBC.Formule :C25H20N4O4Couleur et forme :SolidMasse moléculaire :440.45BRL-42715
CAS :BRL-42715 is an effective inhibitor of bacterial beta-lactamases.Formule :C10H7N4NaO3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :286.24Luffariellolide
CAS :Luffariellolide is a terpene compound obtained from the marine sponge Hyrtios communis that is an HSF-PLA2 inhibitor and a RAR agonist.Formule :C25H38O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :386.57PDE4-IN-14
CAS :PDE4-IN-14 (Compound 1) serves as an inhibitor of phosphodiesterase 4 (PDE4), applicable in research concerning diseases associated with PDE4, includingFormule :C19H20F2N4O3SCouleur et forme :SolidMasse moléculaire :422.45Cathepsin C-IN-4
Cathepsin C-IN-4 is a potent inhibitor (IC50: 65.6 nM) of histone C. Cathepsin C-IN-4 inhibits THP-1 cells (IC50: 203.4 nM) and U937 cells (IC50: 177.6 nM).Formule :C21H14ClF3N4SCouleur et forme :SolidMasse moléculaire :446.88Streptothricin F
CAS :Streptothricin F is a biochemical.Formule :C19H34N8O8Couleur et forme :SolidMasse moléculaire :502.52TTT 3002
CAS :TTT 3002: oral FLT3 inhibitor for AML research, blocks D835 mutations, potent at 0.2 nM IC50.Formule :C27H23N5O3Couleur et forme :SolidMasse moléculaire :465.50Napsagatran hydrate
CAS :Napsagatran hydrate is a novel and specific inhibitor of thrombin.Formule :C26H36N6O7SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :576.66BAY-364
CAS :BAY-364 (BAY-299N) functions as an inhibitor targeting the second bromine domain in TAF1, demonstrating inhibitory effects on TAF1 in Kasumi-1 cells, CD34+Formule :C23H19N3O4Couleur et forme :SolidMasse moléculaire :401.41MRTX-EX185
MRTX-EX185 inhibits GDP-KRAS/G12D; IC50=90 nM on G12D. It also binds GDP-HRAS.Formule :C33H33FN6O2Couleur et forme :SolidMasse moléculaire :564.65Monoamine Oxidase B inhibitor 2
MAO-B inhibitor 2: potent, reversible, oral, selective (IC50=1.33 nM), BBB-penetrant, with anti-oxidant and anti-inflammatory effects for Parkinson's study.Formule :C19H19FO3Couleur et forme :SolidMasse moléculaire :314.35GS-9160
CAS :GS-9160 is a novel and potent inhibitor of human immunodeficiency virus type 1 (HIV-1) integrase (IN) that specifically targets the process of strand transfer.Formule :C20H18FN3O4SCouleur et forme :SolidMasse moléculaire :415.44FK-906 HCl
CAS :FK-906 HCl is a human renin inhibitor used for the long-term treatment of patients with essential hypertension.Formule :C40H64ClN7O7Couleur et forme :SolidMasse moléculaire :790.44LPM4870108
LPM4870108: Potent, oral pan-Trk inhibitor, selective over ALK, with anti-tumor effects. TrkC IC50=0.2nM, TrkA IC50=2.4nM.Formule :C20H19FN6O3Couleur et forme :SolidMasse moléculaire :410.4DNA crosslinker 3 dihydrochloride
CAS :Compound 1: a DNA minor groove binder with 1.4°C ΔTm; useful in cancer research.Formule :C15H22Cl2N8OCouleur et forme :SolidMasse moléculaire :401.29Methyl Streptonigrin
CAS :Methyl Streptonigrin is an ABCG2 transporter function inhibitor.Formule :C26H24N4O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :520.49VEGFR-2-IN-12
VEGFR-2-IN-12 (compound 6g), a 2-oxoquinoxalinyl-1,2,4-triazole, is a potent inhibitor of VEGFR-2 (IC50: 0.037 μM). VEGFR-2-IN-12 has anti-tumour effects.Formule :C22H24N6O3SCouleur et forme :SolidMasse moléculaire :452.53PDE4B-IN-3
PDE4B-IN-3 is a potent inhibitor of PDE4B (IC50: 0.94 μM) and exhibits anti-inflammatory effects.Formule :C30H35N3O4S2Couleur et forme :SolidMasse moléculaire :565.75AZD0424
CAS :AZD0424: oral Src/Abl kinase inhibitor; potential anticancer; induces apoptosis, cell cycle arrest in lymphoma.Formule :C25H29ClN6O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :528.99J-104132
CAS :J-104132: potent human ETA/B antagonist; Ki: ETA=0.034nM, ETB=0.104nM; prevents ET-1 effects, ED50 i.v.=0.045mg/kg, p.o.=0.35mg/kg.Formule :C31H33NO7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :531.60Nedocromil sodium
CAS :Nedocromil sodium is a pharmacologic stabilizer of mast cells, has been shown to normalize cytokine levels and attenuate cardiac remodeling.Formule :C19H17NNaO7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :394.335RS 2135
CAS :RS 2135 is a novel class I antiarrhythmic agent to inhibit ischemia-induced ventricular arrhythmias.Formule :C18H21ClN2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :332.83ONO-AE1-329
CAS :ONO-AE1-329 is a novel agonist of the prostaglandin PGE2 receptor EP4.Formule :C22H30O6S2Couleur et forme :SolidMasse moléculaire :454.6LSD1-IN-21
LSD1-IN-21: potent LSD1 inhibitor, crosses blood-brain barrier, IC50 of 0.956 μM; lowers TNF-α, anti-cancer, anti-inflammatory.Formule :C24H25N5O2SCouleur et forme :SolidMasse moléculaire :447.55XP-524
CAS :XP-524: BET & EP300 inhibitor, suppresses KRAS tumors in vivo, targets PDAC, boosts immune response.Formule :C30H28N6O3SCouleur et forme :SolidMasse moléculaire :552.65JAK1/TYK2-IN-3
JAK1/TYK2-IN-3, orally active, selectively inhibits TYK2 (IC50: 6 nM), JAK1 (37 nM), JAK2 (140 nM), JAK3 (362 nM), and has anti-inflammatory effects.Couleur et forme :Solid2R,4S-Sacubitril
CAS :<p>2R,4S-Sacubitril (Sacubitril Enantiomer) is the impurity of Sacubitril which is a neprilysin inhibitor.</p>Formule :C24H28NO51CaDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :430.49Pyridoxatin
CAS :Pyridoxatin: fungal metabolite; blocks TBARS production, prevents AAPH-induced hemolysis, and acts against C. albicans.Formule :C15H21NO3Couleur et forme :SolidMasse moléculaire :263.33β-Glucuronidase/hCAII-IN-1
CAS :β-Glucuronidase/hCAII-IN-2 (Compound 12e) is a compound that effectively inhibits both β-glucuronidase and human Carbonic Anhydrase II (hCA II), exhibiting IC50Formule :C30H21NO9Couleur et forme :SolidMasse moléculaire :539.49AChE-IN-22
AChE-IN-22 (10q) selectively inhibits AChE (IC50: 0.88 μM), less on BuChE (IC50: 10 μM), targets CAS and PAS, useful in Alzheimer's research.Formule :C21H20N4O5SCouleur et forme :SolidMasse moléculaire :440.47QTX125 TFA
QTX125 TFA: Potent, selective HDAC6 inhibitor with antitumor effects.Formule :C25H20F3N3O7Couleur et forme :SolidMasse moléculaire :531.44PD-L1-IN-1
PD-L1-IN-1, potent PD-L1 inhibitor with 115 nM IC50, suppresses tumors, boosts immune response, and spares healthy cells.Formule :C21H23N5O2Couleur et forme :SolidMasse moléculaire :377.44AEP-IN-1
APE-IN-1, a potent AEP inhibitor (IC50: 89 nM), aids Alzheimer's diagnosis and drug research.Formule :C18H27N3O3Couleur et forme :SolidMasse moléculaire :333.43iNOs-IN-1
iNOs-IN-1 (YPW) is a strong iNOS inhibitor with dose-dependent anti-inflammatory properties, reducing IL-6, iNOS, and NO levels.Formule :C25H30N4O5Couleur et forme :SolidMasse moléculaire :466.53LXR agonist 2
LXR agonist 2 is a potent agonist of the LXR (liver X receptor). LXR agonist 2 stabilises NCOA1 (coactivator), which in turn agonises the LXR.Formule :C35H40ClN3O3Couleur et forme :SolidMasse moléculaire :586.16SR 140333
CAS :SR 140333 is a NK1 receptor antagonist.Formule :C37H45Cl3N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :656.12HSP90-IN-9
HSP90-IN-9: potent HSP90 inhibitor, dose-dependent fungicide, impedes biofilm/morphology with FLC, reverses FLC resistance.Couleur et forme :SolidAnti-ToCV agent 1
Anti-ToCV agent 1 can be used as a potential anti-ToCV drug.Formule :C22H19FN2O5SCouleur et forme :SolidMasse moléculaire :442.46SMCypI C31
SMCypIC31, a non-peptide cyclophilin inhibitor, blocks PPIase at 0.1 μM IC50 and fights various HCV genotypes (EC50: 1.20-7.76 μM).Formule :C27H30N4O2SCouleur et forme :SolidMasse moléculaire :474.62Tasidotin hydrochloride
CAS :Tasidotin hydrochloride, a dolastatin 15 analog, inhibits microtubule assembly and dynamics.Formule :C32H59ClN6O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :643.30GSK1820795A
CAS :GSK1820795A: Telmisartan analog, selective hGPR132a antagonist, blocks yeast activation by N-acylamides, angiotensin II antagonist, partial PPARγ agonist.Formule :C35H34N8Couleur et forme :SolidMasse moléculaire :566.7LJ-4517
LJ-4517 is an effective A2AAR antagonist (Ki=18.3 nM). LJ-4517 can effectively replace the binding of [3H] ZM241385 at WT A2AAR.Formule :C19H21N5O3SCouleur et forme :SolidMasse moléculaire :399.47VEGFR-2/DHFR-IN-2
VEGFR-2/DHFR-IN-2 inhibits VEGFR-2 & DHFR (IC50: 0.623 & 9.085 μM), toxic to C26, HepG2, MCF7 cells (IC50: 3.59-8.38 μM), promising for cancer study.Formule :C21H21NO4Couleur et forme :SolidMasse moléculaire :351.4VEGFR-2-IN-10
VEGFR-2-IN-10 has enhanced antiangiogenic potency against VEGFR2 phosphorylation induced by VEGF with an IC50 value of 0.7 μM and no cytotoxic effects.Formule :C20H21N3O2Couleur et forme :SolidMasse moléculaire :335.4Abarelix acetate
CAS :Abarelix acetate: synthetic GnRHR antagonist, spikes histamine, lowers LH and testosterone temporarily, used in advanced prostate cancer.Formule :C72H95ClN14O14·xC2H4O2Couleur et forme :SolidMasse moléculaire :1476.14Nikkomycin Z
CAS :Nikkomycin Z (Nikkomycin Z from Streptomyces tendae) is a competitive chitin synthase inhibitor.It inhibitor of the growth of filamentous fungi, insects,Formule :C20H25N5O10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :495.44TEI-9063
CAS :TEI-9063 is a stable and highly specific prostacyclin analogue of prostacyclin receptor in mast cell tumor p-815 cells.Formule :C23H38O4Couleur et forme :SolidMasse moléculaire :378.55(S)-JDQ-443
CAS :(S)-JDQ-443, an isomer of JDQ-443, is a selective, potent oral KRAS G12C inhibitor with antitumor properties.Formule :C29H28ClN7OCouleur et forme :SolidMasse moléculaire :526.03Tamitinol
CAS :Tamitinol is a neurotropic drug. It has been found to help symptoms of obsessive rumination in conjunction with maprotiline.Formule :C12H20N2OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :240.37Cenicriviroc Sulfone
CAS :Cenicriviroc Sulfone, a Cenicriviroc derivative, inhibits CCR2/CCR5 to block HIV entry into cells.Formule :C41H52N4O5SCouleur et forme :SolidMasse moléculaire :712.94Antitumor agent-47
Antitumor agent-47, a silibinin derivative, shows cytotoxicity in NCI-H1299 (IC50: 8.07µM) and HT29 (IC50: 6.27µM) cells.Formule :C30H27NO11Couleur et forme :SolidMasse moléculaire :577.54Sesamodil
CAS :Sesamodil (SD 3211) is a novel calcium antagonist that can be used to study hypertension.Formule :C29H32N2O6SDegré de pureté :98.87% - 99.87%Couleur et forme :SolidMasse moléculaire :536.64(R)-ONO-2952
(R)-ONO-2952 is the R-enantiomer of ONO-2952. ONO-2952 is selective and oral effective TSPO antagonist, with Kis of 0.330-9.30 nM inhibiting rat and human TSPO.Formule :C22H20ClFN2O2Couleur et forme :SolidMasse moléculaire :398.86(S)-Purvalanol B
CAS :(S)-Purvalanol B is the S enantiomer of Purvalanol B. Purvalanol B is an inhibitor of cyclin-dependent kinase(CDK) .Formule :C20H25ClN6O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :432.9BRD5631
CAS :BRD5631 is an autophagy enhancer, enhances autophagy through an mTOR-independent pathway.Formule :C30H35N3O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :501.62SX 3202
CAS :SX 3202 is an aldose reductase inhibitor being developed for the treatment of diabetic neuropathy.Formule :C17H11BrFN3O4Couleur et forme :SolidMasse moléculaire :420.19Aniline-MPB-amino-C3-PBD
CAS :Aniline-MPB-amino-C3-PBD is a cytotoxic agent comprised of the non-alkylating group. It is a sequence-selective DNA minor-groove binding agent.Formule :C42H46N8O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :758.86MRS2279
CAS :Selective, high affinity competitive antagonist of the P2Y1 receptorFormule :C13H18ClN5O8P2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :469.71ALK5-IN-7
CAS :ALK5-IN-7 inhibits ALK5, useful in TGF-β disease research like cancer, fibrosis, and autoimmune disorders. See WO2021129621A1.Formule :C26H28N4O3SCouleur et forme :SolidMasse moléculaire :476.59KPC-2-IN-2
KPC-2-IN-2 (6c) inhibits KPC-2 enzyme in Klebsiella pneumoniae (Ki 0.038 μM) and boosts cefotaxime in E. coli KPC-2.Formule :C12H10BN3O2SCouleur et forme :SolidMasse moléculaire :271.1Antiviral agent 15
Compound 15f, a Clofazimine derivative, inhibits rabies (EC50: 1.45 μM) and SARS-CoV-2 (EC50: 14.6 μM).Formule :C27H24FN5OCouleur et forme :SolidMasse moléculaire :453.51UAWJ9-36-1
CAS :UAWJ9-36-1: potent broad-spectrum coronavirus Protease inhibitor; IC50 = 51 nM.Formule :C23H29N3O5Couleur et forme :SolidMasse moléculaire :427.49IDO2-IN-1
CAS :IDO2-IN-1: potent oral IDO2 inhibitor, IC50 = 112 nM, for inflammatory autoimmunity research.Formule :C21H21BrN10O3Couleur et forme :SolidMasse moléculaire :541.36NNC 55-0396
CAS :NNC 55-0396: Selective T-type calcium channel blocker, IC50 6.8 μM, inhibits human ovarian cancer cell growth.Formule :C30H40Cl2FN3O2Degré de pureté :99.00%Couleur et forme :SolidMasse moléculaire :564.56Ref: TM-T12238
1mg66,00€5mg126,00€10mg202,00€25mg354,00€50mg550,00€100mg787,00€1mL*10mM (DMSO)160,00€
