Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.542 produits)
- Apoptose(5.816 produits)
- Cycle cellulaire/point de contrôle(4.466 produits)
- Chromatine/Épigénétique(2.252 produits)
- Signalisation du cytosquelette(1.381 produits)
- Altération de l'ADN/réparation de l'ADN(2.830 produits)
- Endocrinologie/Hormones(3.518 produits)
- Enzyme(3.640 produits)
- GPCR/G-Protéine(8.362 produits)
- Immunologie et Inflammation(3.540 produits)
- Virus de la grippe(296 produits)
- Signalisation JAK/STAT(405 produits)
- Signalisation MAPK(1.201 produits)
- Transporteur membranaire/Canal ionique(2.809 produits)
- Métabolisme(9.462 produits)
- Microbiologie/Virologie(7.003 produits)
- Neuroscience(9.942 produits)
- Autres inhibiteurs(37.827 produits)
- Oxydation-Réduction(40 produits)
- Signalisation PI3K/Akt/mTOR(1.399 produits)
- Protéases/Protéasome(1.598 produits)
- Cellules souche et Dérivés(830 produits)
- Tyrosine Kinase/Adaptateurs(2.012 produits)
- Ubiquitination(1.651 produits)
Affichez 16 plus de sous-catégories
66618 produits trouvés pour "Inhibiteurs"
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VEGFR-2-IN-10
<p>VEGFR-2-IN-10 has enhanced antiangiogenic potency against VEGFR2 phosphorylation induced by VEGF with an IC50 value of 0.7 μM and no cytotoxic effects.</p>Formule :C20H21N3O2Couleur et forme :SolidMasse moléculaire :335.4PI3K-IN-26
CAS :<p>PI3K-IN-26 is an effective PI3K inhibitor. PI3K-IN-26 inhibits the proliferation of SU-DHL-6 cells, IC50= 36 nM.</p>Formule :C21H18N6OSCouleur et forme :SolidMasse moléculaire :402.47GSK 366
CAS :GSK 366 is a potent kynurenine-3-monooxygenase (KMO) inhibitor (IC50s: 0.7 nM and 2.3 nM for P. fluorescens-KMO and human KMO).Formule :C17H16ClN3O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :361.78MLKL-IN-1
<p>MLKL-IN-1 is a covalent inhibitor of MLKL with a Kd value of 50 μM.</p>Formule :C19H20N2O3Couleur et forme :SolidMasse moléculaire :324.37SK&F 108361
CAS :<p>SK&F 108361 is a symmetric diol that binds HIV-1 protease symmetrically.</p>Formule :C24H48N6O6Couleur et forme :SolidMasse moléculaire :516.67Cenicriviroc Sulfone
CAS :<p>Cenicriviroc Sulfone, a Cenicriviroc derivative, inhibits CCR2/CCR5 to block HIV entry into cells.</p>Formule :C41H52N4O5SCouleur et forme :SolidMasse moléculaire :712.94BACE1-IN-2
CAS :<p>BACE1-IN-2 is a BACE1 inhibitor (IC50: 22 nM).</p>Formule :C19H15F4N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :421.35CD73-IN-7
CAS :<p>CD73-IN-7: potent inhibitor of CD73, blocks adenosine production to treat tumors.</p>Formule :C13H11ClN4O2Couleur et forme :SolidMasse moléculaire :290.7Streptonigrin (racemate)
CAS :<p>Streptonigrin: aminoquinone antibiotic; antitumor, antibacterial; blocks β-Catenin/Tcf, cytotoxic; alters hamster chromosomes; (-)-isomer, CAS#3930-19-6.</p>Formule :C25H22N4O8Couleur et forme :SolidMasse moléculaire :506.46Dihydrophaseic acid
CAS :<p>Dihydrophaseic acid 3'-O-b-D-glucopyranoside (D3G) can increase the proliferation and differentiation of osteoblast cells and enhance bone formation, suggests</p>Formule :C15H22O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :282.33Silvestrol
CAS :<p>Silvestrol is a eukaryotic translation initiation factor 4A inhibitor. Silvestrol causes autophagy and caspase-mediated apoptosis.</p>Formule :C34H38O13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :654.66Anticancer agent 65
CAS :<p>Anticancer agent 65: Effective on A549 cells, IC50 1.07 μM, halts S phase, triggers apoptosis, elevates p53/p21, causes ROS and MMP collapse.</p>Formule :C36H63NO5Couleur et forme :SolidMasse moléculaire :589.89BRD-7880
CAS :<p>BRD-7880 is a potent and highly specific inhibitor of aurora kinases B and C.</p>Formule :C32H38N4O7Couleur et forme :SolidMasse moléculaire :590.67CDK/HDAC-IN-1
<p>CDK/HDAC-IN-1 inhibits CDK2/4/6 & HDAC6 with IC50s: 60.9, 276, 27.2, and 128.6 nM respectively.</p>Formule :C20H18N4O4Couleur et forme :SolidMasse moléculaire :378.38Antitrypanosomal agent 5
<p>Antitrypanosal agent 5 is a selective anti-trypanosomal agent that acts on T. brucei (IC50: 1 nM) and HEK293 cells (IC50: 483.3 μM).</p>Formule :C30H30N6O4SCouleur et forme :SolidMasse moléculaire :570.66Y1 receptor antagonist 1
CAS :<p>Y1 receptor antagonist 1 is an antagonist of neuropeptide Y1 receptor.</p>Formule :C28H33N5O3Degré de pureté :98.17%Couleur et forme :SolidMasse moléculaire :487.59Tuvatidine
CAS :<p>Tuvatidine is a histamine 2 receptor antagonist.</p>Formule :C10H17N9O2S3Couleur et forme :SolidMasse moléculaire :391.5RXR antagonist 2
<p>RXR antagonist 2 is a potent antagonist of RXR (Ki: 0.391 μM, Kd: 0.281 μM). RXR antagonist 2 has shown research potential for RXR-related diseases.</p>Formule :C29H35F3N2O3Couleur et forme :SolidMasse moléculaire :516.6Estrogen receptor antagonist 6
CAS :<p>Estrogen receptor antagonist 6 is a potent blocker of estrogen signaling, regulating various biological effects. (Compound 166)</p>Formule :C25H31F3N2O3Couleur et forme :SolidMasse moléculaire :464.52TP3011
CAS :<p>TP3011 is a potent topoisomerase I inhibitor equipotent as SN38 and is an active metabolite of CH-0793076.</p>Formule :C26H26N4O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :474.51MAO-B-IN-6
<p>MAO-B-IN-6 is a selective, potent, orally active MAO-B inhibitor (IC50: 0.019 μM). MAO-B-IN-6 is superior to Safinamide both in vitro and in vivo.</p>Couleur et forme :SolidCOX-2-IN-7
<p>COX-2-IN-7: potent, orally active COX-2 inhibitor with higher selectivity than Celecoxib, IC50 6.585 uM, anti-inflammatory, low ulcer risk.</p>Formule :C15H13N3O2S2Couleur et forme :SolidMasse moléculaire :331.41Burapitant
CAS :<p>Burapitant (SSR 240600) is a novel non-peptide tachykinin neurokinin 1 (NK) receptor antagonist with anti-coke oven and antidepressant activity.</p>Formule :C31H35Cl2F6N3O3Degré de pureté :>99.99% - >99.99%Couleur et forme :SolidMasse moléculaire :682.52KRAS G12D inhibitor 1
CAS :<p>KRAS G12D inhibitor 1 (example 243) is an inhibitor of KRAS G12D with an IC 50 of 0.8 nM for KRAS G12D-mediated ERK phosphorylation [1].</p>Formule :C33H32F2N6O2Couleur et forme :SolidMasse moléculaire :582.64P-gp modulator 3
<p>P-gp modulator 3 (Compound 37) is a potent, competitive, metabotropic P-glycoprotein (P-gp) modulator.</p>Formule :C31H37N3O5Couleur et forme :SolidMasse moléculaire :531.64ERα degrader 5
<p>ERα degrader 5 is an orally active, selective estrogen receptor (ER) reducer that acts on ERα (EC50: 1.1 nM). ERα degrader 5 shows anti-tumour effects in vivo.</p>Formule :C29H25F4N3O2SCouleur et forme :SolidMasse moléculaire :555.59Dyrk1A/α-synuclein-IN-1
<p>Dyrk1A/α-synuclein-IN-1 (Compound b1) is a dual inhibitor of Dyrk1A (IC50: 177 nM) and α-synuclein aggregation (IC50: 10.5 μM).</p>Formule :C20H21N5O3SCouleur et forme :SolidMasse moléculaire :411.48Saussureamine C
CAS :<p>Saussureamine C is an inhibitor of H274Y and N294S mutants.</p>Formule :C19H26N2O5Couleur et forme :SolidMasse moléculaire :362.42Tubulin inhibitor 19
<p>Tubulin inhibitor 19 (9b), a potent indole chalcone, strongly blocks tubulin, valuable in cancer studies.</p>Formule :C21H23NO5Couleur et forme :SolidMasse moléculaire :369.41BAY-364
CAS :<p>BAY-364 (BAY-299N) functions as an inhibitor targeting the second bromine domain in TAF1, demonstrating inhibitory effects on TAF1 in Kasumi-1 cells, CD34+</p>Formule :C23H19N3O4Couleur et forme :SolidMasse moléculaire :401.41XIAP/cIAP1 antagonist-1
<p>Potent oral XIAP/cIAP1 inhibitor with EC50s: XIAP 5.1 nM, cIAP1 0.32 nM; curbs tumor growth in vivo.</p>Couleur et forme :SolidBGC-638
CAS :<p>BGC-638, an analogue of BGC-945, is a thymidylate synthase inhibitor specifically transported into α-folate receptor (α-FR)–overexpressing tumors.</p>Formule :C32H33N5O9Couleur et forme :SolidMasse moléculaire :631.63AChE-IN-24
<p>AChE-IN-24: Strong AChE blocker, crosses blood-brain barrier, IC50=0.053 μM, useful for AD research.</p>Formule :C22H30N2O4S2Couleur et forme :SolidMasse moléculaire :450.61Odiparcil
CAS :<p>Odiparcil is an orally active beta-d-thioxyloside analog.</p>Formule :C15H16O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :324.35Antibacterial agent 76
<p>Antibacterial agent 76 (compound 9) is a potent antibacterial agent.</p>Formule :C23H27N3O2SCouleur et forme :SolidMasse moléculaire :409.54(2S,4S)-Sacubitril
CAS :<p>(2S,4S)-Sacubitril (Sacubitril Impurity C) is a stereoisomer derived from Sacubitril which is a potent NEP inhibitor.</p>Formule :C24H29NO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :411.49ZK118182 isopropyl ester
CAS :<p>ZK118182 isopropyl ester is a PG analog with potent DP-agonist activity (EC50 = 16.5 nM) and high affinity for the DP receptor (Ki = 74 nM).</p>Formule :C23H37ClO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :428.99AD012
<p>AD012, a dual cACE/NEP inhibitor, leverages lenopril-tryptophan for potential anti-hypertensive and cardioprotective benefits.</p>Formule :C25H32N2O6Couleur et forme :SolidMasse moléculaire :456.53Tofogliflozin
CAS :Tofogliflozin specifically inhibits SGLT2; IC50s are 2.9 nM (human), 14.9 nM (rat), 6.4 nM (mouse).Formule :C22H26O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :386.44GR 122222X
CAS :<p>GR 122222X is an inhibitor of topoisomerase II.</p>Formule :C26H35N5O11SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :625.65PROTAC CDK12/13 Degrader-1
<p>PROTAC CDK12/13 Degrader-1 (7f) selectively degrades CDK12/13 at nanomolar potency, targeting breast cancer.</p>Couleur et forme :SolidK20
<p>K20 selectively inhibits KRas G12C (IC50: 1.16 nM), shows anticancer activity in H358 cells (IC50: 0.78 μM), and induces apoptosis via Erk dephosphorylation.</p>Formule :C24H20Cl2F4N4O2Couleur et forme :SolidMasse moléculaire :543.34Gimatecan
CAS :Gimatecan (STI481) is a potent topoisomerase I inhibitor. Gimatecan is an orally bioavailable camptothecin analogue with antitumor activity.Formule :C25H25N3O5Degré de pureté :98.47%Couleur et forme :SolidMasse moléculaire :447.48CB30865
CAS :CB30865 (ZM 242421) is a selective and highly effective nicotinamide phosphoribosyltransferase (Nampt) inhibitor with potential antitumor activity.Formule :C26H22BrN5O2Degré de pureté :99.04%Couleur et forme :SolidMasse moléculaire :516.39ChemR23-IN-3
<p>ChemR23-IN-3 is a potent thiazole-based ChemR23 inhibitor with an IC 80 value of 12 nM.</p>Formule :C31H33N5O5S2Couleur et forme :SolidMasse moléculaire :619.75HIF-1α-IN-5
<p>HIF-1α-IN-5 is an inhibitor of HIF-1α with an IC 50 value of 24 nM in HEK293T cells that also inhibits the activity of MAO-A.</p>Formule :C16H15N3O2Couleur et forme :SolidMasse moléculaire :281.31Alkannin
CAS :<p>Alkannin: potent, tumor-specific PKM2 inhibitor; non-inhibitory to PKM1/PKL; potential anticancer agent.</p>Formule :C16H16O5Couleur et forme :SolidMasse moléculaire :288.3NU5455
CAS :<p>NU5455 is a potent DNA-PKcs inhibitor, oral, boosts doxorubicin in liver tumors, amplifies topoisomerase inhibitors, no adverse effects.</p>Formule :C34H33N3O5SCouleur et forme :SolidMasse moléculaire :595.71FR 900452
CAS :<p>FR 900452 is a platelet activating factor antagonist from fermentatiion products of Streptomyces phaeofaciens.</p>Formule :C22H25N3O3SCouleur et forme :SolidMasse moléculaire :411.52MRS2179 tetrasodium hydrate
<p>MRS2179 blocks turkey P2Y1 receptor (Kb 102 nM, pA2 6.99), affects platelet aggregation, and has varying IC50s on P2 receptors.</p>Formule :C11H15N5Na4O10P2Couleur et forme :SolidMasse moléculaire :576.21JAK3 covalent inhibitor-1
CAS :<p>JAK3 Covalent Inhibitor-1 is a compound characterized by its potent and selective inhibition of Janus kinase 3 (JAK3), possessing an IC50 of 11 nM and</p>Formule :C22H17FN6O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :448.47MRS2279 diammonium
CAS :<p>MRS2279 diammonium, a P2Y1 antagonist with K i 2.5 nM, IC 50 51.6 nM, blocks ADP-induced platelet aggregation, pK b 8.05.</p>Formule :C13H24ClN7O8P2Couleur et forme :SolidMasse moléculaire :503.77AKR1C3-IN-7
<p>AKR1C3-IN-7 (Compound 13) is an effective and selective AKR1C3 inhibitor (IC50=0.19 μM). AKR1C3-IN-7 has antitumor activity.</p>Formule :C24H20N2O4Couleur et forme :SolidMasse moléculaire :400.43YKL-05-093
CAS :<p>YKL-05-093 is a alt inducible kinase (SIK) inhibitor. YKL-05-093 increases bone formation and bone mass.</p>Formule :C35H40N6O4Couleur et forme :SolidMasse moléculaire :608.73Aniline-MPB-amino-C3-PBD
CAS :<p>Aniline-MPB-amino-C3-PBD is a cytotoxic agent comprised of the non-alkylating group. It is a sequence-selective DNA minor-groove binding agent.</p>Formule :C42H46N8O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :758.86GSK1820795A
CAS :<p>GSK1820795A: Telmisartan analog, selective hGPR132a antagonist, blocks yeast activation by N-acylamides, angiotensin II antagonist, partial PPARγ agonist.</p>Formule :C35H34N8Couleur et forme :SolidMasse moléculaire :566.7EGFR/HER2-IN-5
<p>EGFR/HER2-IN-5: Irreversible, oral dual EGFR inhibitor, IC50 0.6 nM, targets L858R/T790M mutations, anti-tumor in vivo for lung cancer study.</p>Couleur et forme :SolidK203
<p>K203 is a potent tabun-inhibited AChE reactivator and is an important antidote to organophosphorus poisoning.</p>Formule :C16H18Br2N4O2Couleur et forme :SolidMasse moléculaire :458.15Menin-MLL inhibitor 4
CAS :Menin-MLL inhibitor 4 has antitumor activity.Menin-MLL inhibitor 4 is an inhibitor of Menin- MLL (mixed-lineage leukemia protein) interaction .Formule :C32H38FN7O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :587.69SLC4011540
<p>SLC4011540 is a potent and selective SphK1/2 dual inhibitor with Ki value of 120 nM and 90 nM respectively.</p>Formule :C24H23ClF3N7OSCouleur et forme :SolidMasse moléculaire :550Anticancer agent 16
<p>Anticancer agent 16 showed good cytotoxic effects on HCT-116 cell line (IC50: 8.55 μM), NCI-H460 cell line (IC50: 5.41 μM) and SKOV3 cell line (IC50: 6.4 μM).</p>Formule :C27H33N5O6Couleur et forme :SolidMasse moléculaire :523.58MK-2748
CAS :<p>MK-2748 is an inhibitor of NS3 protease, hepatitis C virus.</p>Formule :C42H56N6O10SCouleur et forme :SolidMasse moléculaire :836.99FGFR4-IN-4
CAS :<p>FGFR4-IN-4 is a FGFR4 inhibitor with anti-tumor activity.</p>Formule :C28H32Cl2N6O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :603.5Freselestat quarterhydrate
<p>ONO-6818 quarterhydrate: oral neutrophil elastase inhibitor, Ki 12.2 nM; >100x less effective on other proteases; strong anti-inflammatory.</p>Formule :C23H30N6O5Couleur et forme :SolidMasse moléculaire :457.03CDK9-IN-11
CAS :<p>CDK9-IN-11 is a potent CDK9 inhibitor that is the ligand for the PROTAC CDK9 Degrader-1 [1].</p>Formule :C20H25N3O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :371.43Teslexivir
CAS :Teslexivir is a topical antiviral agent that is an effective and selective inhibitor of the interaction between two essential viral proteins, E1 and E2.Formule :C35H36BrN3O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :642.58Faldaprevir sodium
CAS :<p>Faldaprevir sodium: HCV treatment, inhibits NS3/NS4A protease, P-glycoprotein, CYP3A4, UGT1A1.</p>Formule :C40H48BrN6NaO9SCouleur et forme :SolidMasse moléculaire :891.81ATR-IN-12
<p>ATR-IN-12, a potent ATR kinase inhibitor with IC50 of 0.007 μM, shows promise for drug development.</p>Formule :C22H27N5O3SCouleur et forme :SolidMasse moléculaire :441.55TCMDC-135051 TFA (2413716-15-9 free base)
<p>TCMDC-135051 TFA is a highly selective and potent inhibitor of protein kinase PfCLK3.</p>Formule :C31H34F3N3O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :585.61FTO-IN-1 TFA
<p>FTO-IN-1 TFA: FTO enzyme inhibitor, anti-obesity, IC50 < 1μM, potential cancer research tool.</p>Formule :C20H17Cl2F3N4O4Couleur et forme :SolidMasse moléculaire :505.27M826
<p>M826, a non-peptide, potent, selective, and reversible caspase-3 inhibitor, exhibits an IC50 of 0.005 μM and demonstrates strong anti-apoptotic activity in</p>Formule :C28H45N7O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :575.7G092
<p>G092 is a potent inhibitor of MsbA. MsbA is an ABC transporter protein. G092 has potential for antibacterial drug research.</p>Formule :C23H20Cl2N2O3Couleur et forme :SolidMasse moléculaire :443.32MRGPRX1 agonist 3
<p>Compound 1f, a potent MRGPRX1 agonist, has an EC50 of 0.22 μM, useful for neuropathic pain studies.</p>Formule :C14H11FN2OSCouleur et forme :SolidMasse moléculaire :274.31DMGF
CAS :<p>DMGF, a biflavonoid from Taxus, induces apoptosis, autophagy, and inhibits B16F10 cell motility and MMP-2 expression, hindering melanoma metastasis.</p>Formule :C32H22O10Couleur et forme :SolidMasse moléculaire :566.51DNDI-8219
CAS :<p>DNDI-8219 is an antitubercular agent. It has potent antileishmanial effects.</p>Formule :C13H10F3N3O5Couleur et forme :SolidMasse moléculaire :345.23Nurr1 agonist 1
<p>Nurr1 agonist 1 is an inverse agonist tool for the neuroprotective transcription factor Nurr1 which is an appealing target to treat neurodegenerative diseases.</p>Formule :C16H14N2O2Couleur et forme :SolidMasse moléculaire :266.29Casuarinin
CAS :<p>Casuarinin, an ellagitannin found in pomegranates and certain Casuarina/Stachyurus plants, is a carbonic anhydrase inhibitor and astringent.</p>Formule :C41H28O26Couleur et forme :SolidMasse moléculaire :936.65FY-56
<p>FY-56: potent, selective LSD1/KDM1A inhibitor (IC50=42nM); differentiates MOLM-13/MV4-11 cells; promising for AML research.</p>Formule :C23H19FN2O3Couleur et forme :SolidMasse moléculaire :390.41hDHODH-IN-10
<p>hDHODH-IN-10: selective oral inhibitor of hDHODH (IC50: 10.9 nM); blocks cancer cell growth, aids cancer research.</p>Formule :C21H15ClF4N2O4Couleur et forme :SolidMasse moléculaire :470.8Multi-kinase-IN-1
CAS :<p>Multi-kinase-IN-1, a powerful kinase inhibitor, exhibits antitumor properties by inducing cell apoptosis.</p>Formule :C35H36F2N6O6SCouleur et forme :SolidMasse moléculaire :706.76Lamivudine, (+/-)-trans-
CAS :<p>Lamivudine, a drug for HIV-1 and HBV, inhibits reverse transcriptase and resembles zalcitabine.</p>Formule :C8H11N3O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :229.26L 691816
CAS :<p>L 691816 is an effective inhibitor of the 5-LO reaction.</p>Formule :C36H35ClN6OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :635.22PARP10/15-IN-3
<p>Compound 8a, a dual PARP10 & PARP15 inhibitor, has IC50s: PARP10 at 0.14μM & PARP15 at 0.40μM; it's cell-permeable & anti-apoptotic.</p>Formule :C12H12N2O3Couleur et forme :SolidMasse moléculaire :232.24Antibacterial agent 66
<p>Compound 6q, a trifluoromethylpyridine oxadiazole, targets Xanthomonas oryzae with EC50 of 7.2 μg/mL.</p>Formule :C17H10ClF6N3O2SCouleur et forme :SolidMasse moléculaire :469.79SARS-CoV-2-IN-24
<p>SARS-CoV-2-IN-24 blocks PLpro, altering its shape and stopping virus replication—useful for SARS-CoV-2 research.</p>Formule :C27H30N4O5Couleur et forme :SolidMasse moléculaire :490.55Zanapezil fumarate
CAS :<p>Zanapezil is an acetylcholinesterase (AChE) inhibitor. Zanapezil increases choline acetyltransferase activity in cultured rat septal cholinergic neurons.</p>Formule :C29H36N2O5Couleur et forme :SolidMasse moléculaire :492.61PF-06462894
CAS :PF-06462894: morpholinopyrimidone, mGlu5 antagonist (Ki=6nM), no immune activation in mouse model.Formule :C18H23N3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :329.39Colistin adjuvant-1
<p>Colistin adjuvant-1, inhibits NF-κB (IC50: 0.209 μM), boosts mucin against gram-negative bacteria.</p>Formule :C16H7F9N2OCouleur et forme :SolidMasse moléculaire :414.23RET-IN-10
CAS :<p>RET-IN-10: Potent RET inhibitor, may treat congenital megacolon and tumors (Patent WO2021135938A1, compound 18).</p>Formule :C29H28N8OSCouleur et forme :SolidMasse moléculaire :536.65AGN-204396
CAS :AGN-204396 is an antagonist that selectively blocks the activity of prostamides (prostaglandin-ethanolamides).Formule :C32H44FN3O4Couleur et forme :SolidMasse moléculaire :553.71Chitin synthase inhibitor 8
<p>Chitin synthase inhibitor 8 is a chitin synthase (CHS) inhibitor with broad-spectrum antifungal effects that can be used in studies related to fungal infections</p>Formule :C23H23N3O5Couleur et forme :SolidMasse moléculaire :421.45Nnc 09-0026
CAS :<p>Nnc 09-0026 is a neuronal calcium channel blocker</p>Formule :C25H35Cl2F3N2OCouleur et forme :SolidMasse moléculaire :507.46BPN-15606 besylate
<p>BPN-15606 besylate is a potent oral γ-secretase regulator reducing Aβ42 and Aβ40 with good pharmacokinetics. IC50: 7 nM (Aβ42), 17 nM (Aβ40).</p>Formule :C29H29FN6O4SCouleur et forme :SolidMasse moléculaire :576.6416(S)-Iloprost
CAS :<p>Iloprost, a potent prostacyclin analog, binds to human IP & EP1 receptors with high affinity; inhibits platelet aggregation effectively.</p>Formule :C22H32O4Couleur et forme :SolidMasse moléculaire :360.49JTE 151A
CAS :<p>JTE-151 is a novel RORγ inverse agonist.</p>Formule :C26H30ClN3O5Couleur et forme :SolidMasse moléculaire :499.99CK156
CAS :<p>CK156 inhibits DAPK with high selectivity; IC50: 182 nM (DRAK1), 34 μM (CK2a1), 39 μM (CK2a2); key in autoimmune/inflammation research.</p>Formule :C21H25N5O3Couleur et forme :SolidMasse moléculaire :395.45CY208-243 Mandelate
CAS :<p>CY208-243 is a D1 agonist boosting memory in T-maze, enhances adenylate cyclase (EC50=125nM), and alters monkey electroretinogram.</p>Formule :C27H26N2O3Couleur et forme :SolidMasse moléculaire :426.52Cav 3.2 inhibitor 1
<p>Cav 3.2 inhibitor 1 targets T-type calcium channels, weakly binds D2 receptors, and aids physical and visceral pain research.</p>Formule :C32H39N3OCouleur et forme :SolidMasse moléculaire :481.67Anti-inflammatory agent 10
<p>Tilomisole-derived benzimidazole-thiazole, orally active, favors COX-2 inhibition over COX-1.</p>Formule :C17H13BrN4O3S2Couleur et forme :SolidMasse moléculaire :465.34Pibrozelesin
CAS :<p>Pibrozelesin, a water-soluble duocarmycin B2 derivative, binds AT-rich DNA, blocking replication and inducing cell death.</p>Formule :C32H36BrN5O8Couleur et forme :SolidMasse moléculaire :698.56
