Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.542 produits)
- Apoptose(5.816 produits)
- Cycle cellulaire/point de contrôle(4.466 produits)
- Chromatine/Épigénétique(2.252 produits)
- Signalisation du cytosquelette(1.381 produits)
- Altération de l'ADN/réparation de l'ADN(2.830 produits)
- Endocrinologie/Hormones(3.518 produits)
- Enzyme(3.640 produits)
- GPCR/G-Protéine(8.362 produits)
- Immunologie et Inflammation(3.540 produits)
- Virus de la grippe(296 produits)
- Signalisation JAK/STAT(405 produits)
- Signalisation MAPK(1.201 produits)
- Transporteur membranaire/Canal ionique(2.809 produits)
- Métabolisme(9.462 produits)
- Microbiologie/Virologie(7.003 produits)
- Neuroscience(9.942 produits)
- Autres inhibiteurs(37.827 produits)
- Oxydation-Réduction(40 produits)
- Signalisation PI3K/Akt/mTOR(1.399 produits)
- Protéases/Protéasome(1.598 produits)
- Cellules souche et Dérivés(830 produits)
- Tyrosine Kinase/Adaptateurs(2.012 produits)
- Ubiquitination(1.651 produits)
Affichez 16 plus de sous-catégories
66618 produits trouvés pour "Inhibiteurs"
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CAII-IN-1
<p>CAII-IN-1 (3n) is a selective bovine CA-II inhibitor with 10.3 μM IC50, used in carbonic anhydrase disorder studies.</p>Formule :C19H21FN4SCouleur et forme :SolidMasse moléculaire :356.46L 365209
CAS :L 365209 is an oxytocin antagonist.Formule :C40H50N8O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :738.88c-Met/HDAC-IN-2
CAS :<p>Potent dual c-Met/HDAC inhibitor, IC50: HDAC1 5.4 nM, c-Met 18.49 nM; anti-cancer, induces apoptosis, G2/M arrest in HCT-116.</p>Formule :C34H33N5O7Couleur et forme :SolidMasse moléculaire :623.66CDK1-IN-4
<p>CDK1-IN-4 inhibits CDK1 (IC50: 44.52 nM), CDK2/CDK5 less potently, impacts cell cycle, used in cancer studies.</p>Formule :C26H24ClN5SCouleur et forme :SolidMasse moléculaire :474.02α-Glucosidase-IN-15
<p>α-Glucosidase-IN-15 (Compound 14B) exhibits potent inhibitory activity against α-glucosidase, with an IC50 value of 3.34 μM.</p>Formule :C24H24N2SCouleur et forme :SolidMasse moléculaire :372.53Lometrexol hydrate
CAS :<p>Lometrexol hydrate, an antipurine antifolate, inhibits GARFT and purine synthesis, leading to cancer cell apoptosis without causing DNA breaks.</p>Formule :C21H27N5O7Couleur et forme :SolidMasse moléculaire :461.475GSK340
<p>GSK340 is a BET inhibitor.</p>Formule :C26H31N3O2Couleur et forme :SolidMasse moléculaire :417.55Colistin adjuvant-2
<p>Colistin adjuvant-2 is a compound that acts as a potentiation agent for colistin, effectively enhancing its activity against Gram-negative bacteria [1].</p>Formule :C14H7Cl2F3N2OCouleur et forme :SolidMasse moléculaire :347.12Lavendomycin
CAS :<p>Lavendomycin can be extracted from Streptomyces lavendulae and has active against Gram-positive bacteria.</p>Formule :C29H50N10O8Couleur et forme :SolidMasse moléculaire :666.77SBI-581
<p>SBI-581: oral, potent TAO3 inhibitor, IC50=42nM, alters TKS5α at RAB11+ vesicles, blocks invadopodia, good mouse pharmacokinetics, anti-tumor.</p>Formule :C24H21N3O2Couleur et forme :SolidMasse moléculaire :383.44Antitubercular agent-11
<p>Antitubercular agent-11 (Compound 1e) is an antitubercular agent with a bulkier electron-donating group (Bu-t) that shows the best MIC value of 0.060 μg/mL [1].</p>Formule :C16H15N3O4Couleur et forme :SolidMasse moléculaire :313.31PI3Kα-IN-8
<p>PI3Kα-IN-8 is a selective inhibitor of PI3Kα (IC50: 0.012 μM).</p>Formule :C26H27BrN4O2Couleur et forme :SolidMasse moléculaire :507.42(2R,3S)-Azelaprag
CAS :<p>(2R,3S)-N-(4-(2,6-dimethoxyphenyl)-5-(5-methylpyridin-3-yl)-4H-1,2,4-triazol-3-yl)-3-(5-methylpyrimidin-2-yl)butane-2-sulfonamide is an Apelin receptor agonist</p>Formule :C25H29N7O4SDegré de pureté :97.47% - >99.99%Couleur et forme :SoildMasse moléculaire :523.61(-)-15-Deoxyspergualin
CAS :<p>(-)-15-Deoxyspergualin is a potent antitumor agent that demonstrates significant inhibition against mouse leukemia L-1210.</p>Formule :C17H37N7O3Couleur et forme :SolidMasse moléculaire :387.52CDK5-IN-2
CAS :<p>CDK5-IN-2 (compound 15) is a highly selective CDK5 inhibitor that acts on CDK5/p25 (IC50: 0.2 nM) and CDK2/CycA (IC50: 23 nM).</p>Formule :C29H28FN5OCouleur et forme :SolidMasse moléculaire :481.56T-3861174
CAS :<p>T-3861174 is a prolyl tRNA synthetase (PRS) inhibitor, exhibiting significant in vitro anti-tumor activity with GCN2-ATF4 pathway activation.</p>Formule :C26H25FN6O2Couleur et forme :SolidMasse moléculaire :472.51Antifungal agent 38
<p>Antifungal agent 38, a heterocyclic disulfide, shrinks hyphae and damages cell membranes, causing leakage.</p>Formule :C8H12N2S2Couleur et forme :SolidMasse moléculaire :200.32SARS-CoV-2-IN-23
<p>SARS-CoV-2-IN-23 (compound GRL-0617) is an inhibitor of SARS-COV-2 papain-like protease (PLpro) (IC 50 = 2.3 μM) [1].</p>Formule :C21H22N2OCouleur et forme :SolidMasse moléculaire :318.41KRAS G12C inhibitor 46
CAS :<p>KRAS G12C inhibitor 46 is a potent inhibitor of KRAS G12C.</p>Formule :C32H33F2N7O2Couleur et forme :SolidMasse moléculaire :585.65BRD-9526
CAS :BRD-9526 is a potent and selective inhibitor of Sonic Hedgehog (Shh).Formule :C26H31Cl2N3O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :584.51Ketomethylenebestatin
CAS :<p>Ketomethylenebestatin, a weaker carba-analog of aminopeptidase inhibitor bestatin, is 10x less potent.</p>Formule :C17H25NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :307.38Cacospongionolide B
CAS :<p>Cacospongionolide B from Fasciospongia cavernosa inhibits secretory phospholipase A2, curbing inflammation.</p>Formule :C25H36O4Couleur et forme :SolidMasse moléculaire :400.55BMS 310705
CAS :<p>BMS 310705, an Epothilone B analog, targets ovarian/renal/bladder/lung cancer, inducing apoptosis via mitochondria.</p>Formule :C27H42N2O6SCouleur et forme :SolidMasse moléculaire :522.70Tarloxotinib bromide
CAS :Tarloxotinib bromide (TH-4000) is an irreversible inhibitor of EGFR/HER2.Formule :C24H24Br2ClN9O3Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :681.77SphK2-IN-2
<p>SphK2-IN-2 (21g) is a potent and selective inhibitor of SphK2 (IC50: 0.23 μM).</p>Formule :C21H25ClN10OCouleur et forme :SolidMasse moléculaire :468.94CHF-6366
CAS :<p>CHF-6366: M3 antagonist & β2 agonist (pKi 10.4/11.4), mild Ca channel blocker, used in COPD study.</p>Formule :C42H48N6O8Couleur et forme :SolidMasse moléculaire :764.87Marizomib
CAS :Marizomib is a novel irreversible brain-permeable proteasome inhibitor that inhibits CT-L, CT-T-laspase-like, and trypsin-like 20S proteasomes.Cost-effective and quality-assured.Formule :C15H20ClNO4Degré de pureté :98.03% - 99.41%Couleur et forme :SolidMasse moléculaire :313.78GRPR antagonist-2
<p>GRPR antagonist-2 blocks GRPR, kills some cancer cells, effective on HGC-27 (IC50: 0.77 μM) & Pan02 (IC50: 2.5 μM).</p>Formule :C28H32F3N5O4Couleur et forme :SolidMasse moléculaire :559.58GSK699
CAS :<p>GSK699 is a potent, cell penetrant PCAF/GCN5 PROTAC.</p>Formule :C45H51BrN8O7Couleur et forme :SolidMasse moléculaire :895.84Saprisartan potassium
CAS :<p>Saprisartan potassium is an Angiotensin II Type 1 receptor antagonist and antihypertensive agent.</p>Formule :C25H21BrF3KN4O4SCouleur et forme :SolidMasse moléculaire :649.52VRT-18858
CAS :<p>VRT-18858 is a metabolite of VX-740.</p>Formule :C24H25N5O7Couleur et forme :SolidMasse moléculaire :495.48BTK-IN-10
CAS :<p>BTK-IN-10 is a potent inhibitor of BTK, acting on wild-type BTK (IC50<5 nM) or mutant BTK (C481S) (IC50<5 nM).</p>Formule :C25H24F2N4O2Couleur et forme :SolidMasse moléculaire :450.48MsbA-IN-3
<p>MsbA-IN-3 is a potent and highly selective MsbA inhibitor (IC50: 2 nM). MsbA-IN-3 inhibits Escherichia coli activity (MIC: 35 μM).</p>Formule :C24H22Cl2N2O4SCouleur et forme :SolidMasse moléculaire :505.41FCE-24379
CAS :<p>FCE-24379 is a selective antagonist of vascular serotonin receptors that has been shown to lowers blood pressure in hypertensive rats.</p>Formule :C20H22N4O2Couleur et forme :SolidMasse moléculaire :350.41Dup-714
CAS :<p>Dup-714 is a thrombin inhibitor.</p>Formule :C21H33BN6O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :460.33RWJ-445167
CAS :<p>RWJ-445167 is a thrombin and factor Xa dual inhibitor(Ki of 4.0 nM and 230 nM, respectively), with potent antithrombotic activity.</p>Formule :C18H24N6O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :436.49IRAK4-IN-18
<p>IRAK4-IN-18: Potent IRAK4 inhibitor (IC50: 15 nM), reduces IL23 in cells, prevents rat arthritis.</p>Formule :C24H25FN6O3Couleur et forme :SolidMasse moléculaire :464.49MK-7128
CAS :<p>MK-7128 is a CB1 receptor inverse agonist.</p>Formule :C29H25ClF2N4O2Couleur et forme :SolidMasse moléculaire :534.98AVE-1330A sodium
CAS :<p>AVE-1330A sodium is a beta-Lactamase inhibitor.</p>Formule :C7H10N3NaO6SCouleur et forme :SolidMasse moléculaire :287.23Aeroplysinin 1
CAS :<p>Aeroplysinin I is an antibacterial compound from the sponge. It has cytotoxic activity against colon cancer cells by promoting β-catenin degradation.</p>Formule :C9H9Br2NO3Couleur et forme :SolidMasse moléculaire :338.98(-)-Adenophorine
CAS :<p>(-)-Adenophorine is a moderate alpha-l-fucosidase inhibitor.</p>Formule :C8H17NO4Couleur et forme :SolidMasse moléculaire :191.22QPX7728 bis-acetoxy methyl ester
CAS :<p>QPX7728 bis-acetoxy methyl ester is an inhibitor of boronic acid β-lactamase.</p>Formule :C15H14BFO8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :352.08OPC-167832
CAS :<p>OPC-167832: oral dprE1 inhibitor, IC50 0.258 μM, anti-tuberculosis, for Mycobacterium tuberculosis research.</p>Formule :C21H20ClF3N2O4Couleur et forme :SolidMasse moléculaire :456.84AL 8810
CAS :<p>AL-8810 is an 11β-fluoro analog of PGF 2α with selective antagonist effects at the PGF 2α receptor (FP receptor) [1].</p>Formule :C24H31FO4Couleur et forme :SolidMasse moléculaire :402.5PEN-866
CAS :<p>PEN-866, a conjugate of HSP90i and SN-38, may control early NSCLC tumor growth.</p>Formule :C49H49N7O9Couleur et forme :SolidMasse moléculaire :879.95Antitumor agent-42
<p>Antitumor agent-42 inhibits microtubule multimerisation and NO release, exhibiting anti-angiogenic, colony-forming and apoptosis-inducing effects.</p>Formule :C24H19BrN2O8SCouleur et forme :SolidMasse moléculaire :575.39Topoisomerase I inhibitor 8
CAS :<p>Topoisomerase I inhibitor 8, a hexacyclic analogue of camptothecin, is also a potent inhibitor of topoisomerase I and is toxic to tumour cells.</p>Formule :C24H21FN2O4Couleur et forme :SolidMasse moléculaire :420.43Teoprolol
CAS :<p>Teoprolol is a blocker of β-adrenergic receptor.</p>Formule :C23H30N6O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :454.52Pegcantratinib
CAS :<p>Pegcantratinib is a tropomyosin receptor kinase inhibitor for treatment for inherited CYLD defective skin tumours.</p>Formule :C32H28N4O7Couleur et forme :SolidMasse moléculaire :580.59CDK7-IN-18
CAS :<p>CDK7-IN-18: potent, pyrimidine-based CDK7 inhibitor with cancer research potential.</p>Formule :C22H24F3N7OSCouleur et forme :SolidMasse moléculaire :491.53Tacrolimus anhydrous 8-epimer
CAS :<p>Tacrolimus anhydrous 8-epimer, an immunosuppressive l-pipecolic acid macrolide, blocks T cell growth by hindering IL-2.</p>Formule :C44H69NO12Couleur et forme :SolidMasse moléculaire :804.02SAR-114137
CAS :<p>SAR-114137 is a histone sphingomyelin kinase inhibitor used in the study of molluscum arteriosum and peripheral neuropathic pain.</p>Formule :C25H34N4O7SDegré de pureté :99.09% - 99.91%Couleur et forme :SolidMasse moléculaire :534.63Zurletrectinib
CAS :<p>Zurletrectinib is a tyrosine kinase inhibitor with potential as an antineoplastic agent.</p>Formule :C19H19F2N7O2Couleur et forme :SolidMasse moléculaire :415.4AS2575959
CAS :<p>AS2575959 is a novel GPR40 agonist, exhibiting glucose metabolism improvement and synergistic effect with sitagliptin on insulin and incretin secretion.</p>Formule :C32H35NaO7Couleur et forme :SolidMasse moléculaire :554.6148(3S,4R)-Tofacitinib
CAS :(3S,4R)-Tofacitinib is an less active enantiomer of Tofacitinib. Tofacitinib is a JAK3 inhibitor(IC50 : 1 nM).Formule :C16H20N6ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :312.37GDC-0927 Racemate
CAS :<p>GDC-0927 Racemate is a degrader of estrogen receptor, is used in the research of ER-related diseases, potently inhibits ER-α activity, with an IC50 of 0.2 nM.</p>Formule :C28H28FNO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :461.52TP-030-1
CAS :<p>TP-030-1, RIPK1 inhibitor: K(i) hRIPK1 at 3.9nM, IC50 mRIPK1 at 4.2μM; targets inflammation, neurodegeneration research.</p>Formule :C23H22N4O3Couleur et forme :SolidMasse moléculaire :402.45Anti-Aβ agent 1A
<p>Anti-Aβ agent 1A is a potent anti-amyloid-β agent.</p>Formule :C35H49NO4Couleur et forme :SolidMasse moléculaire :547.77GW-597901 cinnamate
CAS :<p>GW-597901 cinnamate is a long-acting beta(2)-agonist.</p>Formule :C34H46N2O8SCouleur et forme :SolidMasse moléculaire :642.80AQX-435
CAS :<p>AQX-435 activates SHIP1, inhibits PI3K in BCR signaling, induces apoptosis in B cells, and slows lymphoma growth.</p>Formule :C27H34N2O4Couleur et forme :SolidMasse moléculaire :450.57AMG-222 tosylate
CAS :<p>AMG-222 tosylate is a DPP-IV inhibitor in clinical development for type II diabetes.</p>Formule :C39H47N9O6SCouleur et forme :SolidMasse moléculaire :769.91Carbodine
CAS :<p>Carbodine is an antiviral targeting CTP synthetase, effective against influenza A0/PR-8/34 and A2/Aichi/2/68.</p>Formule :C10H15N3O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :241.24Suloctidil HCl
CAS :<p>Suloctidil HCl is a peripheral vascular dilator.</p>Formule :C20H36ClNOSCouleur et forme :SolidMasse moléculaire :374.02PDE4B/7A-IN-2
CAS :<p>5-HT1A/5-HT7 antagonist; 5-HT1A Ki=8 nM, 5-HT7 Ki=451 nM; PDE4B IC50=80.4 μM, PDE7A IC50=151.3 μM; stronger than escitalopram.</p>Formule :C25H35N3O2Couleur et forme :SolidMasse moléculaire :409.56DIDS
CAS :<p>DIDS inhibits anion exchangers reversibly then irreversibly and blocks RAD51.</p>Formule :C16H10N2O6S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :454.52COX-2-IN-12
<p>COX-2-IN-12: Potent, selective COX-2 inhibitor, IC50=19.98μM, safe anti-inflammatory with low acute toxicity.</p>Formule :C17H19NO3Couleur et forme :SolidMasse moléculaire :285.34LLS30
CAS :<p>LLS30 inhibits Gal-1, reduces its binding affinity, and may help treat advanced prostate cancer.</p>Formule :C34H33Cl4N5O3Couleur et forme :SolidMasse moléculaire :701.47Laulimalide
CAS :<p>Microtubule stabilizer; halts cancer cell growth (IC50: 3-30 nM); arrests cells in prometaphase; prevents bipolar spindle formation.</p>Formule :C30H42O7Couleur et forme :SolidMasse moléculaire :514.65Anticancer agent 80
<p>Anticancer agent 80 (Compound 3c) is an anticancer agent that exhibits a significant dark toxic effect on T47-D (IC50: 10.14 μM).</p>Formule :C19H12BrNO5Couleur et forme :SolidMasse moléculaire :414.21AM-6494
CAS :<p>AM-6494 is a potent and orally active BACE1 inhibitor (IC50: 0.4 nM) with in vivo selectivity over BACE2 (IC50: 18.6 nM).</p>Formule :C22H21F2N5O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :473.5AK-295
CAS :<p>AK 295, also known as CX 295, is a dipeptide inhibitor of alpha-ketoamide calpain.</p>Formule :C26H40N4O6Couleur et forme :SolidMasse moléculaire :504.62Mu opioid receptor antagonist 4
<p>Compound 31: Potent, selective MOR antagonist; crosses blood-brain barrier; Ki & EC50: 0.38 nM; useful for OUD research.</p>Formule :C25H28N2O4SCouleur et forme :SolidMasse moléculaire :452.57BMS-248360
CAS :<p>BMS-248360: Oral dual hAT1/hETA antagonist with Kis of 10nM & 1.9nM, respectively; treats hypertension.</p>Formule :C36H45N5O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :659.84Y1 receptor antagonist 1
CAS :<p>Y1 receptor antagonist 1 is an antagonist of neuropeptide Y1 receptor.</p>Formule :C28H33N5O3Degré de pureté :98.17%Couleur et forme :SolidMasse moléculaire :487.59A25822B
CAS :<p>A25822B is an antifungal agent.</p>Formule :C28H45NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :411.66SS-RJW100
<p>SS-RJW100 is an enantiomer of RJW100 targeting LRH-1, SF-1, enhances Tif2 interaction, and disrupts LRH-1 networks with lowered stability.</p>Formule :C28H34OCouleur et forme :SolidMasse moléculaire :386.57AP5
CAS :<p>AP5: GPR40 agonist, positive allosteric modulator; rat hIP1 EC50: 0.49 nM.</p>Formule :C28H28FNO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :461.52AL-GDa62
<p>AL-GDa62, a gastric cancer treatment lead, has EC50 of 3.2 μM (MCF10A-WT) and 2 μM (MCF10A-CDH1 -/-).</p>Formule :C24H28FN3OCouleur et forme :SolidMasse moléculaire :393.5CAII-IN-2
<p>CAII-IN-2 (3g): potent, selective CA-II inhibitor; IC50-12.1 μM for bovine CA-II; valuable in CA-related disorder research.</p>Formule :C18H19BrN4SCouleur et forme :SolidMasse moléculaire :403.34CREB-IN-1 TFA
<p>CREB-IN-1 TFA: Potent oral CREB inhibitor, IC50 of 0.18 μM, suppresses breast cancer cell growth.</p>Couleur et forme :SolidCOX-2-IN-6
CAS :<p>COX-2-IN-6: Potent, selective COX-2 inhibitor; oral; IC50 0.84μM, Ki 69nM; blocks PGE2 synthesis; prevents colorectal cancer.</p>Formule :C20H27NO6SDegré de pureté :99.29% - 99.69%Couleur et forme :SoildMasse moléculaire :409.5L 156903
CAS :<p>L 156903 is a bioactive chemical. It also inhibits the binding of neurotensin to brain tissue.</p>Formule :C35H41N7O5SCouleur et forme :SolidMasse moléculaire :671.81Cilazaprilat
CAS :<p>Cilazaprilat is the active metabolite of cilazapril, a pyridazine angiotensin-converting enzyme (ACE) inhibitor with antihypertensive activity.</p>Formule :C20H27N3O5Couleur et forme :SolidMasse moléculaire :389.45Falecalcitriol
CAS :<p>Falecalcitriol is an analog of calcitriol. It has a higher potency both in vivo and in vitro systems, which is longer duration of action in vivo.</p>Formule :C27H38F6O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :524.58BXL0124
CAS :<p>BXL0124 is a gemini vitamin D analog which targets CD44-STAT3 signaling and inhibits breast cancer invasion.</p>Formule :C32H44F6O4Couleur et forme :SolidMasse moléculaire :606.68Chitin synthase inhibitor 7
<p>Compound 9c, a chitin synthase inhibitor, has an IC50 of 0.37 nM and is useful for studying fungal infections.</p>Formule :C24H25N3O5Couleur et forme :SolidMasse moléculaire :435.47AZD-4121
CAS :<p>AZD-4121 is an oral cholesterol absorption inhibitor targeting NPC1L1 for the treatment of dyslipidaemia.</p>Formule :C36H39F2N3O7SCouleur et forme :SolidMasse moléculaire :695.77IRE1α kinase-IN-5
<p>IRE1α kinase-IN-5 (compound 7) is a potent inhibitor of IRE1α (Ki: 98 nM) and is an ATP-competitive ligand for IRE1α.</p>Formule :C28H30N6O3SCouleur et forme :SolidMasse moléculaire :530.64GS-9822
CAS :<p>GS-9822 is a new LEDGIN inhibitor targeting LEDGF/p75 to alter HIV integration, showing a block-and-lock effect in cells.</p>Formule :C36H39ClN4O4SCouleur et forme :SolidMasse moléculaire :659.24Kolavenic acid analog
CAS :<p>KAA, an anticancer compound, inhibits centrosome clustering and targets HSET+ yeast and cancer cells.</p>Formule :C25H38O4Couleur et forme :SolidMasse moléculaire :402.57Steroid sulfatase/17β-HSD1-IN-3
<p>Steroid sulfatase/17β-HSD1-IN-3 (compound 19) is a dual inhibitor of steroid sulfatase (STS) and 17β-hydroxysteroid dehydrogenase type 1 (17β HSD1).</p>Formule :C19H17ClN2O5SCouleur et forme :SolidMasse moléculaire :420.87BI-44370
CAS :<p>BI-44370, a CGRP (calcitonin gene-related peptide) receptor antagonist, can be used to treat migraines and other chronic pain.</p>Formule :C35H47N5O6Couleur et forme :SolidMasse moléculaire :633.78CDK4/6-IN-10
<p>CDK4/6-IN-10: Oral CDK4 (IC50: 22 nM) & CDK6 (IC50: 10 nM) inhibitor with anti-cancer potential for MM research.</p>Couleur et forme :SolidMEIS-IN-3
<p>MEIS-IN-3 is a potent inhibitor of MEIS.</p>Formule :C25H26N2O4Couleur et forme :SolidMasse moléculaire :418.48DH376
CAS :<p>DH376 inhibits DAGLα in a time and dose dependent manner in mouse brain. DH376 shows picomolar activity.</p>Formule :C31H28F2N4O3Couleur et forme :SolidMasse moléculaire :542.58Antibacterial agent 63
CAS :<p>Aztreonam-siderophore conjugate 63 is an antibacterial agent that exhibits efficacy against Gram-negative bacteria through the linkage of aztreonam to a</p>Formule :C35H43N9O14S2Couleur et forme :SolidMasse moléculaire :877.9MtTMPK-IN-2
CAS :<p>MtTMPK-IN-2 inhibits M. tuberculosis TMPK (IC50: 1.1 μM), Mtb H37Rv (MIC: 12.5 μM), and is cytotoxic in MRC-5 cells (EC50: 6.1 μM).</p>Formule :C23H24ClN3O3Couleur et forme :SolidMasse moléculaire :425.91GNE-203
CAS :<p>GNE-203 is a Met inhibitor.</p>Formule :C30H29Cl2F3N8O3Couleur et forme :SolidMasse moléculaire :677.50Anticancer agent 64
CAS :<p>Anticancer agent 64 (5m) induces apoptosis, has IC50 2.4μM in CCRF-CEM, activates caspases, cleaves PARP, affects mitochondria.</p>Formule :C31H46N2O2SCouleur et forme :SolidMasse moléculaire :510.77NS2B/NS3-IN-3
CAS :<p>NS2B/NS3-IN-3 (Compd 66) is an inhibitor of Flavivirus NS2B-NS3 protease [1] .</p>Formule :C19H21N3O2Couleur et forme :SolidMasse moléculaire :323.39
