Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.524 produits)
- Apoptose(5.793 produits)
- Cycle cellulaire/point de contrôle(4.452 produits)
- Chromatine/Épigénétique(2.242 produits)
- Signalisation du cytosquelette(1.382 produits)
- Altération de l'ADN/réparation de l'ADN(2.826 produits)
- Endocrinologie/Hormones(3.507 produits)
- Enzyme(3.640 produits)
- GPCR/G-Protéine(8.333 produits)
- Immunologie et Inflammation(3.527 produits)
- Virus de la grippe(296 produits)
- Signalisation JAK/STAT(404 produits)
- Signalisation MAPK(1.203 produits)
- Transporteur membranaire/Canal ionique(2.792 produits)
- Métabolisme(9.449 produits)
- Microbiologie/Virologie(6.981 produits)
- Neuroscience(9.926 produits)
- Autres inhibiteurs(37.921 produits)
- Oxydation-Réduction(41 produits)
- Signalisation PI3K/Akt/mTOR(1.400 produits)
- Protéases/Protéasome(1.597 produits)
- Cellules souche et Dérivés(830 produits)
- Tyrosine Kinase/Adaptateurs(2.015 produits)
- Ubiquitination(1.650 produits)
Affichez 16 plus de sous-catégories
66639 produits trouvés pour "Inhibiteurs"
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Enpp-1-IN-7
<p>Enpp-1-IN-7: potent enpp-1 inhibitor, broad specificity, potential in cancer/infectious disease research. (WO2021203772A1)</p>Formule :C18H19N7O4SCouleur et forme :SolidMasse moléculaire :429.45NS2B/NS3-IN-2
<p>Potent dengue inhibitor NS2B/NS3-IN-2 (IC50: 6 nM, Ki: 0.66 μM) boosts cell viability, non-toxic.</p>Formule :C24H21N3O5SCouleur et forme :SolidMasse moléculaire :463.51PF-00489791
CAS :<p>PF-00489791 (PF4634817) is a long-acting PDE5 inhibitor with hypotensive activity for the study of diabetic nephropathy.</p>Formule :C20H28N8O4SDegré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :476.55Cap-dependent endonuclease-IN-14
CAS :<p>Cap-dependent endonuclease-IN-14 hinders CEN and could treat influenza virus infections. (Patent CN113620948A, compound 1-c).</p>Formule :C30H23FN2O6SCouleur et forme :SolidMasse moléculaire :558.58TGFβ1-IN-1
CAS :<p>TGFβ1-IN-1 is a TGF-β1 inhibitor that inhibits the production of TGF-β1-induced fibrosis markers (α-SMA and fibronectin) and can be used in cancer research.</p>Formule :C22H24N2O3Degré de pureté :99.89% - 99.89%Couleur et forme :SolidMasse moléculaire :364.438PAIR2
CAS :<p>PAIR2 is a selective IRE1α RNase partial antagonist, blocking its ATP site and preventing KIRA from hindering XBP1 splicing.</p>Formule :C27H26F4N6O3SCouleur et forme :SolidMasse moléculaire :590.59Microtubule inhibitor 2
<p>Microtubule inhibitor 2: potent, selective, oral, induces ferroptosis, strong antitumor effect.</p>Formule :C20H23NO7Couleur et forme :SolidMasse moléculaire :389.4MC4355
<p>MC4355 is a dual inhibitor of EZH2 and histone deacetylase (HDAC).</p>Formule :C30H36N4O5Couleur et forme :SolidMasse moléculaire :532.63TrxR-IN-2
<p>TrxR-IN-2 is a potential thioredoxin reductase (TrxR) inhibitor. TrxR-IN-2 has research value in the chemotherapy of drug-resistant hepatocellular carcinoma.</p>Formule :C22H22N4O4Couleur et forme :SolidMasse moléculaire :406.43M-COPA
CAS :<p>M-COPA disrupts Golgi, blocks MET & Arf1 activation, and inhibits angiogenesis via VEGFR & NF-kB pathways.</p>Formule :C25H34N2O2Couleur et forme :SolidMasse moléculaire :394.55LLS30
CAS :<p>LLS30 inhibits Gal-1, reduces its binding affinity, and may help treat advanced prostate cancer.</p>Formule :C34H33Cl4N5O3Couleur et forme :SolidMasse moléculaire :701.47YK5
CAS :<p>YK5 is an allosteric inhibitor pocket of Hsp70 and represents a previously unknown chemical tool to investigate cellular mechanisms associated with Hsp70.</p>Formule :C18H24N8O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :432.50KRAS G12D inhibitor 9
CAS :<p>KRAS G12D inhibitor 9 targets RAS protein, key in growth, showing promise against KRAS G12D cancer.</p>Formule :C33H43N7O2Couleur et forme :SolidMasse moléculaire :569.74Antibacterial agent 90
<p>Antibacterial agent 90 (6n), a pleuromutilin derivative, targets Gram-positive pathogens and Mycoplasma pneumoniae.</p>Formule :C30H42N2O6Couleur et forme :SolidMasse moléculaire :526.66MtMetAP1-IN-1
<p>MtMetAP1-IN-1 is an inhibitor of methionine aminopeptidase 1 ( MetAP1 ). MtMetAP1-IN-1 shows antimycobacterial activity.</p>Formule :C15H10BrN5O2SCouleur et forme :SolidMasse moléculaire :404.24HIF-1α-IN-5
<p>HIF-1α-IN-5 is an inhibitor of HIF-1α with an IC 50 value of 24 nM in HEK293T cells that also inhibits the activity of MAO-A.</p>Formule :C16H15N3O2Couleur et forme :SolidMasse moléculaire :281.31NVP-CGM097 sulfate
CAS :<p>NVP-CGM097 sulfate is a potent and selective inhibitor of MDM2 (hMDM2, IC50 of 1.7±0.1 nM).</p>Formule :C38H49ClN4O8SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :757.34Isobetanin
CAS :<p>Isobetanin is a betacyanin that has been shown to enhance vitexin-2-O-xyloside mediated inhibition of proliferation of T24 bladder cancer cells.</p>Formule :C24H26N2O13Couleur et forme :SolidMasse moléculaire :550.47β-N-Acetyl-D-hexosaminidase-IN-1
<p>β-N-Acetyl-D-hexosaminidase-IN-1 is a newly discovered chemical compound that acts as an inhibitor for β-N-acetyl-D-hexosaminidase.</p>Formule :C18H13F2NO2SCouleur et forme :SolidMasse moléculaire :345.36TIY-7
<p>TIY-7 is a selective, orally active inhibitor of the promyosin receptor kinase (TRK) enzyme. TIY-7 exhibited anti-tumour effects in a mouse xenograft model.</p>Couleur et forme :SolidMSX-3 free acid
CAS :<p>MSX-3 free acid is an A2A adenosine receptor antagonist and a prodrug of MSX-2.</p>Formule :C21H23N4O7PCouleur et forme :SolidMasse moléculaire :474.40Ganoderic acid R
CAS :<p>Ganoderic acid R: potent anticancer, induces apoptosis, cytotoxic to MDR and sensitive tumor cells.</p>Formule :C34H50O6Couleur et forme :SolidMasse moléculaire :554.76K027
<p>K027 is a potent organophosphate (OP) inhibitor of acetylcholinesterase (AChE) reactivation. k027 can be used to study Alzheimer's disease.</p>Formule :C15H18Br2N4O2Couleur et forme :SolidMasse moléculaire :446.14LXR agonist 2
<p>LXR agonist 2 is a potent agonist of the LXR (liver X receptor). LXR agonist 2 stabilises NCOA1 (coactivator), which in turn agonises the LXR.</p>Formule :C35H40ClN3O3Couleur et forme :SolidMasse moléculaire :586.16Methyl Streptonigrin
CAS :<p>Methyl Streptonigrin is an ABCG2 transporter function inhibitor.</p>Formule :C26H24N4O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :520.49L-Moses dihydrochloride
<p>L-Moses (L-45) dihydrochloride is the first, potent, selective p300/CBP-associated factor (PCAF) bromodomain (Brd) inhibitor (Kd: 126 nM).</p>Formule :C21H26Cl2N6Couleur et forme :SolidMasse moléculaire :433.38MRTX849 ethoxypropanoic acid
CAS :<p>MRTX849 is a KRAS G12C ligand and PROTAC linker for creating potent LC-2, degrading KRAS G12C with DC50 of 0.25-0.76 μM.</p>Formule :C37H43ClFN7O5Couleur et forme :SolidMasse moléculaire :720.24Tubulin polymerization-IN-34
<p>"Tubulin-IN-34 inhibits oxazolylisoindole microtubule assembly, selective for VL51 lymphoma."</p>Formule :C31H35N3O6Couleur et forme :SolidMasse moléculaire :545.6312(S)-HETE
CAS :<p>Enpatoran hydrochloride (M5049 hydrochloride) is a TLR7/8 inhibitor with antiviral activity that is used in the study of autoimmune diseases.</p>Formule :C20H32O3Couleur et forme :SolidMasse moléculaire :320.47Karenitecin
CAS :<p>Karenitecin (Cositecan) is an inhibitor of topoisomerase I. It has potent anti-cancer activity.</p>Formule :C25H28N2O4SiDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :448.59I-BET282E
<p>I-BET282E inhibits eight BET bromodomains (pIC50 6.4-7.7) with selectivity for other bromodomain proteins.</p>Formule :C26H34N4O7SCouleur et forme :SolidMasse moléculaire :546.64SG3199
CAS :<p>SG3199, a PBD dimer, binds DNA's minor groove, forms covalent cross-links, and is cytotoxic to various human cancer cells.</p>Formule :C33H36N4O6Couleur et forme :SolidMasse moléculaire :584.66Luffariellolide
CAS :<p>Luffariellolide is a terpene compound obtained from the marine sponge Hyrtios communis that is an HSF-PLA2 inhibitor and a RAR agonist.</p>Formule :C25H38O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :386.57AChE/BChE-IN-1
<p>AChE/BChE-IN-1: dual AChE/BChE inhibitor, IC50 of 1.06 nM/7.3 nM, crosses blood-brain barrier, with antioxidant properties for Alzheimer's research.</p>Formule :C32H35ClN6O3Couleur et forme :SolidMasse moléculaire :587.11(-)-Adenophorine
CAS :<p>(-)-Adenophorine is a moderate alpha-l-fucosidase inhibitor.</p>Formule :C8H17NO4Couleur et forme :SolidMasse moléculaire :191.22HDAC-IN-32
<p>HDAC-IN-32, potent inhibitor: IC50—HDAC1 (5.2 nM), HDAC2 (11 nM), HDAC6 (28 nM). Effective anti-tumor and immunity-boosting traits.</p>Formule :C20H23N3O3Couleur et forme :SolidMasse moléculaire :353.41IRAK4-IN-12
<p>IRAK4-IN-12 (compound 37) is a potent inhibitor of IRAK4 (IC50: 0.015 μM) with cellular pIRAK4 potency (IC50: 0.5 μM).</p>Formule :C24H31FN8OCouleur et forme :SolidMasse moléculaire :466.55MIV-150
CAS :<p>MIV-150 is a nonnucleoside inhibitor of reverse transcriptase (NNRT). MIV-150 also blocking HIV-1 and HIV-2 infections (EC50<1 nM against HIV-1/HIV-2MN).</p>Formule :C19H17FN4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :368.36MK-7128
CAS :<p>MK-7128 is a CB1 receptor inverse agonist.</p>Formule :C29H25ClF2N4O2Couleur et forme :SolidMasse moléculaire :534.98BRD4-BD1/2-IN-2
CAS :<p>BRD4-BD1/2-IN-2 inhibits BRD4 BD1/BD2 with IC50 <300 nM/<0.5 nM (WO2021233371A1).</p>Formule :C30H33N5O4Couleur et forme :SolidMasse moléculaire :527.61Disulergine
CAS :<p>Disulergine is a dopamine receptor agonist. It also prolactin release-inhibiting 8 alpha-amino-ergoline.</p>Formule :C17H24N4O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :348.46p38-α MAPK-IN-5
CAS :<p>p38-α MAPK-IN-5: potent p38α inhibitor, IC50s: 0.1 nM (α), 0.2 nM (β), 944 nM (γ), 4100 nM (δ); anti-inflammatory, promising for asthma/COPD research.</p>Formule :C37H49N11O2Couleur et forme :SolidMasse moléculaire :679.86c-Met-IN-2
CAS :<p>c-Met-IN-2 is a selective and orally available c-Met inhibitor (IC50: 0.6 nM) with antitumor activity.</p>Formule :C24H21FN10ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :484.49HDAC2-IN-1
<p>HDAC2-IN-1 is an oral HDAC2 inhibitor (IC50: 0.5 μM), crosses the blood-brain barrier, and inhibits HDAC1 and HDAC8.</p>Formule :C22H23ClN4OSCouleur et forme :SolidMasse moléculaire :426.96Mal-PEG4-VA-PBD
CAS :<p>Mal-PEG4-VA-PBD is a drug-linker conjugate for Antibody-Drug Conjugates (ADCs), comprising the antitumor antibiotic Pyrrolobenzodiazepine (PBD), connected</p>Formule :C68H79N9O17Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1294.41MI-1851
CAS :<p>MI-1851 is a potent peptidomimetic inhibitor. MI-1851could prevent proteolytic processing of the S protein from SARSCoV-2 by endogenous furin in HEK293 cells.</p>Formule :C34H53N15O6Couleur et forme :SolidMasse moléculaire :767.88(±)-J 113397
CAS :<p>(±)-J-113397 is a potent and selective non-peptidyl ORL1 receptor antagonist (K(i): cloned human ORL1=1.8 nM).</p>Formule :C24H37N3O2Couleur et forme :SolidMasse moléculaire :399.57SARS-CoV-2-IN-6
<p>SARS-CoV-2-IN-6 is an inhibitor of SARS-CoV-2 3CLpro with the IC 50 value of 73 nM.</p>Formule :C17H13ClN2O2Couleur et forme :SolidMasse moléculaire :312.75Anti-inflammatory agent 16
<p>Compound 14 is a peptidomimetic that significantly lowers TNFα, NO, CD40, and CD86, showcasing strong anti-inflammatory effects.</p>Formule :C21H23N5O3Couleur et forme :SolidMasse moléculaire :393.44PD-L1-IN-1
<p>PD-L1-IN-1, potent PD-L1 inhibitor with 115 nM IC50, suppresses tumors, boosts immune response, and spares healthy cells.</p>Formule :C21H23N5O2Couleur et forme :SolidMasse moléculaire :377.44hAChE/Aβ1-42-IN-1
CAS :<p>Compound 16 (hAChE/Aβ1-42-IN-1) is a potent inhibitor targeting both hAChE and Aβ1-42 aggregation, demonstrating considerable safety in hepG2 cell lines and</p>Formule :C20H24N6OCouleur et forme :SolidMasse moléculaire :364.44DI-404
CAS :<p>DI-404: Potent DCN1-UBC12 inhibitor, selectivity blocks cullin 3 neddylation, Kd=6.9 nM.</p>Formule :C35H45ClN6O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :713.29VDR agonist 1
CAS :<p>Compound 28 is a nonsteroidal VDR agonist with 690 nM potency, inducing cell cycle arrest and apoptosis in MCF-7 cells.</p>Formule :C32H51N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :509.77Cav 3.2 inhibitor 1
<p>Cav 3.2 inhibitor 1 targets T-type calcium channels, weakly binds D2 receptors, and aids physical and visceral pain research.</p>Formule :C32H39N3OCouleur et forme :SolidMasse moléculaire :481.6716(R)-Iloprost
CAS :<p>Iloprost, a potent prostacyclin analog, binds IP & EP1 receptors (Ki 11 nM), contains 16(S/R) isomers, and inhibits platelets (IC50 65 nM).</p>Formule :C22H32O4Couleur et forme :SolidMasse moléculaire :360.49Aurora A inhibitor 1
CAS :<p>Aurora A inhibitor 1: potent, selective, targets cancer-linked Aurora A overexpression, potential for cancer research. (WO2021147974A1, 49)</p>Formule :C25H28ClF2N5O2Couleur et forme :SolidMasse moléculaire :503.97GKA50 quarterhydrate
<p>GKA50 quarterhydrate: glucokinase activator, EC50 of 33 nM, boosts insulin, cuts glucose in rats.</p>Formule :C26H30N2O7Couleur et forme :SolidMasse moléculaire :469.01IACS-8779 disodium
CAS :<p>IACS-8779 disodium: potent STING agonist, strong systemic anti-tumor effects, effective in melanoma model.</p>Formule :C21H23N9Na2O10P2S2Couleur et forme :SolidMasse moléculaire :733.52ONO-AE1-329
CAS :<p>ONO-AE1-329 is a novel agonist of the prostaglandin PGE2 receptor EP4.</p>Formule :C22H30O6S2Couleur et forme :SolidMasse moléculaire :454.6(S)-ZG197
<p>(S)-ZG197 is a compound that acts as a highly selective activator of the Staphylococcus aureus Caseinolytic Protease P (Sa ClpP), demonstrating efficacy at a</p>Formule :C28H35F3N4O3Couleur et forme :SolidMasse moléculaire :532.6GGTI-2154 hydrochloride
CAS :<p>GGTI-2154 hydrochloride: selective GGTase I inhibitor, IC50 21 nM, used in cancer research.</p>Formule :C24H29ClN4O3Couleur et forme :SolidMasse moléculaire :456.97Flusoxolol
CAS :<p>Flusoxolol is a beta-adrenoceptor partial agonist.</p>Formule :C22H30FNO4Couleur et forme :SolidMasse moléculaire :391.48HDAC-IN-27
<p>HDAC-IN-27 is a potent and orally active inhibitor of HDAC Class I (0.43 nM - 3.01 nM for HDAC1-3).</p>Formule :C20H22N4O2Couleur et forme :SolidMasse moléculaire :350.41β-Glucuronidase/hCAII-IN-1
CAS :<p>β-Glucuronidase/hCAII-IN-2 (Compound 12e) is a compound that effectively inhibits both β-glucuronidase and human Carbonic Anhydrase II (hCA II), exhibiting IC50</p>Formule :C30H21NO9Couleur et forme :SolidMasse moléculaire :539.49PPARγ phosphorylation inhibitor 1
<p>PPARγ phosphorylation inhibitor 1 (Compound 10) is a potent PPARγ binding agent (IC50: 24 nM) with antidiabetic effects.</p>Formule :C22H14Cl2N2O4Couleur et forme :SolidMasse moléculaire :441.26Vimirogant
CAS :<p>Vimirogant is a RORγ inhibitor (Ki: <100 nM).</p>Formule :C27H35F3N4O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :552.65RhlR antagonist 1
<p>RhlR antagonist 1: IC50 of 26 μM, selective for RhlR, inhibits P. aeruginosa biofilm and virulence factors.</p>Formule :C12H10F2OCouleur et forme :SolidMasse moléculaire :208.2AMG-315
CAS :<p>AMG-315: Chiral AEA analogue, potent CB1 agonist (Ki 7.8 nM, EC50 0.6 nM), stable against hydrolyzing/oxidative enzymes.</p>Formule :C24H41NO2Couleur et forme :SolidMasse moléculaire :375.59BET-IN-1
<p>BET-IN-1 is a potent inhibitor of BET, exhibiting good brain permeability and a reasonable metabolic stability.</p>Formule :C23H24ClFN4O3SCouleur et forme :SolidMasse moléculaire :490.98M-525
CAS :<p>M-525, a potent first-in-class menin-MLL inhibitor, binds at 3 nM IC50 and curbs MLL leukemia cell growth & gene expression.</p>Formule :C39H51FN6O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :734.92GSK-3β inhibitor 7
<p>GSK-3β inhibitor 7 is a GSK-3β inhibitor (IC50: 5.25 μM).</p>Formule :C27H23BrN4O2SCouleur et forme :SolidMasse moléculaire :547.47PD-149163
CAS :<p>PD-149163: brain-penetrating, selective NTR1 agonist; shows pro-cognitive, anti-psychotic, anxiolytic effects.</p>Formule :C42H71N9O6Couleur et forme :SolidMasse moléculaire :798.07GDC-6036-NH
CAS :<p>GDC-6036-NH is a precursor of compound 17a /b, which is a RAS inhibitor that can be used in cancer research.</p>Formule :C26H30ClF4N7ODegré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :568.01Anticancer agent 54
<p>Anticancer agent 54 blocks cell cycle in G0/G1, induces apoptosis, and fights cancer via DNA embedding and ROS.</p>Formule :C33H36N6Couleur et forme :SolidMasse moléculaire :516.68AEP-IN-1
<p>APE-IN-1, a potent AEP inhibitor (IC50: 89 nM), aids Alzheimer's diagnosis and drug research.</p>Formule :C18H27N3O3Couleur et forme :SolidMasse moléculaire :333.43VEGFR-2-IN-26
CAS :<p>VEGFR-2-IN-26 inhibits VEGFR-2 (IC50: 15.5 nM), combating various cancers' cell growth.</p>Formule :C24H19F3N6O2Couleur et forme :SolidMasse moléculaire :480.44ABD957
CAS :<p>ABD957: covalent ABHD17 depalmitoylases inhibitor, IC50 0.21µM for ABHD17B, blocks N-Ras, halts NRAS-mutant AML cell growth.</p>Formule :C27H36F3N7O5SCouleur et forme :SolidMasse moléculaire :627.68NA 0346
CAS :<p>NA 0346 is a derivative of SF 2370 that shows long lasting antihypertensive action as well as potent protein kinases inhibitory activity.</p>Formule :C26H22N4O3Couleur et forme :SolidMasse moléculaire :438.48CDK1-IN-5
<p>CDK1-IN-5 is a selective inhibitor for CDK1 (IC50: 42.19 nM), CDK2, CDK5, halting cancer cell growth.</p>Formule :C27H26ClN5OSCouleur et forme :SolidMasse moléculaire :504.05Tubulin inhibitor 16
<p>Tubulin inhibitor 16 is a potent tubulin inhibitor with antiproliferative activity. Tubulin inhibitor 16 exhibits cytotoxicity in HepG2 cells [1].</p>Formule :C16H12FNO2Couleur et forme :SolidMasse moléculaire :269.27SB-612111
CAS :<p>SB-612111: potent ORL-1 antagonist, Ki=0.33 nM; μ-, κ-, δ-receptor Ki=57.6, 160.5, 2109 nM; blocks nociceptin's pain effect.</p>Formule :C24H29Cl2NOCouleur et forme :SolidMasse moléculaire :418.40SBI-581
<p>SBI-581: oral, potent TAO3 inhibitor, IC50=42nM, alters TKS5α at RAB11+ vesicles, blocks invadopodia, good mouse pharmacokinetics, anti-tumor.</p>Formule :C24H21N3O2Couleur et forme :SolidMasse moléculaire :383.44RO5101576
CAS :<p>RO5101576 is a potent antagonist of LTB4 receptor.</p>Formule :C36H38O8SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :630.75QCA570
CAS :<p>QCA570 is an effective BET degrader based on PROTAC (IC50: 10 nM for BRD4 BD1 Protein).</p>Formule :C39H33N7O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :695.79AMXI-5001 hydrochloride
<p>AMXI-5001 hydrochloride, an oral inhibitor of PARP1/2 and microtubules, shows greater potency and selective anti-cancer effects.</p>Formule :C25H21ClFN5O3Couleur et forme :SolidMasse moléculaire :493.92PIKfyve-IN-1
<p>PIKfyve-IN-1: potent, cell-active inhibitor for PIKfyve research, IC50=6.9 nM.</p>Formule :C20H21N5Couleur et forme :SolidMasse moléculaire :331.41Colistin adjuvant-1
<p>Colistin adjuvant-1, inhibits NF-κB (IC50: 0.209 μM), boosts mucin against gram-negative bacteria.</p>Formule :C16H7F9N2OCouleur et forme :SolidMasse moléculaire :414.23VEGFR-2-IN-17
<p>VEGFR-2-IN-17 (15a) is a potent VEGFR-2 inhibitor with an IC50 of 67.25 nM, showing significant antitumor effects.</p>Formule :C21H14ClN3O2Couleur et forme :SolidMasse moléculaire :375.81SK&F 108361
CAS :<p>SK&F 108361 is a symmetric diol that binds HIV-1 protease symmetrically.</p>Formule :C24H48N6O6Couleur et forme :SolidMasse moléculaire :516.67iMDK quarterhydrate
<p>iMDK quarterhydrate, PI3K inhibitor, blocks MDK growth; suppresses NSCLC safely with MEK inhibitor.</p>Formule :C21H15FN2O3SCouleur et forme :SolidMasse moléculaire :380.91MrgprX2 antagonist-6
<p>MrgprX2 antagonist-6 is a potent antiallergic agent with inhibitory effects on mast cell degranulation.</p>Formule :C24H23F3N6O3Couleur et forme :SolidMasse moléculaire :500.47CYP2C9/CYP2C19-IN-1
<p>CYP2C9/CYP2C19-IN-1 is a potent inhibitor of CYP2C9/CYP2C19 without liver toxicity or genotoxicity and can be used to study Zika virus (ZIKV) infection.</p>Formule :C27H28N2O6SCouleur et forme :SolidMasse moléculaire :508.594,5'-Dimethylangelicin-NHS
<p>NHS-modified coumarin, 4,5'-Dimethylangelicin-NHS, shows photochemical activity & photosensitivity.</p>Formule :C21H19NO7SCouleur et forme :SolidMasse moléculaire :429.44OncoFAP
CAS :<p>OncoFAP is an ultra-high affinity fibroblast activating protein (FAP) ligand with potential tumour targeting.</p>Formule :C21H19F2N5O5Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :459.40MAP855
CAS :<p>MAP855: potent, selective, oral MEK1/2 inhibitor; IC50=3 nM, pERKEC50=5 nM; effective on wild-type/mutant MEK1/2.</p>Formule :C28H23ClF2N6O3Couleur et forme :SolidMasse moléculaire :564.97Antioxidant agent-8
<p>Antioxidant agent-8, an oral Aβ 1-42 inhibitor, reduces fibril aggregation & promotes disaggregation; it's neuroprotective & BBB permeable.</p>Formule :C13H12O5Couleur et forme :SolidMasse moléculaire :248.23FAK-IN-6
<p>FAK-IN-6: Potent FAK inhibitor (IC50=1.415 nM), anti-cancer, for pancreatic studies.</p>Formule :C25H31ClN5O6PSCouleur et forme :SolidMasse moléculaire :596.04Cimpuciclib tosylate
CAS :<p>Cimpuciclib tosylate, a selective CDK4 inhibitor (IC50: 0.49 nM), exhibits anti-tumor activity.</p>Formule :C37H43FN8O4SCouleur et forme :SolidMasse moléculaire :714.85RSK4-IN-1
CAS :<p>RSK4-IN-1 is a compound exhibiting potent inhibition of RSK4, demonstrated by an IC50 value of 9.5 nM.</p>Formule :C19H20F2N4O3Couleur et forme :SolidMasse moléculaire :390.38SH498
CAS :<p>SH498 is a novel Bmi-1-mediated anti-tumor agent with significant anti-proliferative effects.</p>Formule :C27H25F3N2O4Couleur et forme :SolidMasse moléculaire :498.49
