Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.834 produits)
- Apoptose(6.315 produits)
- Cycle cellulaire/point de contrôle(4.877 produits)
- Chromatine/Épigénétique(2.613 produits)
- Signalisation du cytosquelette(1.568 produits)
- Altération de l'ADN/réparation de l'ADN(2.871 produits)
- Endocrinologie/Hormones(3.754 produits)
- Enzyme(3.672 produits)
- GPCR/G-Protéine(9.020 produits)
- Immunologie et Inflammation(3.905 produits)
- Virus de la grippe(300 produits)
- Signalisation JAK/STAT(415 produits)
- Signalisation MAPK(1.257 produits)
- Transporteur membranaire/Canal ionique(3.155 produits)
- Métabolisme(10.133 produits)
- Microbiologie/Virologie(7.620 produits)
- Neuroscience(10.473 produits)
- Autres inhibiteurs(35.846 produits)
- Oxydation-Réduction(40 produits)
- Signalisation PI3K/Akt/mTOR(1.429 produits)
- Protéases/Protéasome(1.689 produits)
- Cellules souche et Dérivés(732 produits)
- Tyrosine Kinase/Adaptateurs(1.982 produits)
- Ubiquitination(1.726 produits)
Affichez 16 plus de sous-catégories
66515 produits trouvés pour "Inhibiteurs"
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HER2-IN-8
CAS :HER2-IN-8 is an inhibitor of HER-2 that can be used in the study of cancer and inflammation-related diseases.Formule :C26H25F2N9O3Couleur et forme :SolidMasse moléculaire :549.53AM-6494
CAS :AM-6494 is a potent and orally active BACE1 inhibitor (IC50: 0.4 nM) with in vivo selectivity over BACE2 (IC50: 18.6 nM).Formule :C22H21F2N5O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :473.5Fusarisetin A
CAS :Fusarisetin A, a pentacyclic fungal metabolite, is an acinar morphogenesis inhibitor .Formule :C22H31NO5Couleur et forme :SolidMasse moléculaire :389.49CDK2-IN-8
CDK2-IN-8 is a potent CDK2 inhibitor (IC50= 1.74 μM). CDK2-IN-8 exhibits antiproliferative activity. CDK2-IN-8 can be used for the research of melanoma.Formule :C22H25N5O3Couleur et forme :SolidMasse moléculaire :407.47NBD-14189
CAS :NBD-14189: Potent HIV-1 entry blocker, binds gp120, IC50: 89 nM, strong antiviral (EC50 <200 nM).Formule :C18H16F4N4O2SCouleur et forme :SolidMasse moléculaire :428.40Carazostatin
CAS :Carazostatin is an antioxidant, free radical scavenger, and potent lipid peroxidation inhibitor.Formule :C20H25NODegré de pureté :98%Couleur et forme :Pale Yellow SolidMasse moléculaire :295.42GSK-3036656 free base
CAS :GSK656 (GSK3036656) inhibits Mtb LeuRS with IC50 of 0.20 μM, promising for tuberculosis treatment.Formule :C10H13BClNO4Couleur et forme :SolidMasse moléculaire :257.48BAY-179
CAS :BAY-179 is a potent, selective, species cross-reactive complex I inhibitor for the study of cancer.Formule :C23H21N5OSDegré de pureté :98.29%Couleur et forme :SolidMasse moléculaire :415.51LL-Z 1640-4
CAS :A signal-specific JNK/p38 pathway and TAK 1 inhibitorFormule :C19H24O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :364.39Squalestatin 2
CAS :Squalestatin 2 is an inhibitor of squalene synthase.Formule :C33H44O13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :648.69JAK3-IN-7
CAS :JAK3-IN-7 is a potent and selective JAK3 inhibitor (IC50<0.01 μM) for the treatment of rejection in organ transplantation, graft-versus-host reaction afterFormule :C17H20N6ODegré de pureté :98.81%Couleur et forme :SolidMasse moléculaire :324.38Keap1-Nrf2-IN-1 TFA
Keap1-Nrf2-IN-1 TFA (compound35) is a potent inhibitor (IC50: 43 nM) protecting against acetaminophen liver damage.Formule :C26H25F3N2O9SCouleur et forme :SolidMasse moléculaire :598.54S1P1 agonist 4
CAS :S1P1 agonist 4 exhibits enhanced potency with an EC 50 value of less than 0.05 mg/kg and a predicted human half-life (t1/2) of approximately 5 days, indicatingFormule :C24H31NO3Couleur et forme :SolidMasse moléculaire :381.51AZD-3199 dihydrobromide
CAS :AZD-3199 dihydrobromide is a β2 adrenergic receptor agonist potentially for the treatment of asthma and chronic obstructive.Formule :C32H44Br2N4O4SCouleur et forme :SolidMasse moléculaire :740.59Hydrolyzed Fumonisin B2
CAS :Hydrolyzed Fumonisin B2 (HFB2) is a hydrolysis product of fumonisins (HF), which retains biological activity. It exhibits phytotoxicity.Formule :C22H47NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :389.61Trk-IN-8
Trk-IN-8: TRK inhibitor with IC50 of 0.42 nM (TRKA), 0.89 nM (TRKA-G595R), 1.5 nM (TRKC-G623R).Formule :C18H16F2N6O2Couleur et forme :SolidMasse moléculaire :386.36di-Val-L-dC
CAS :Di-Val-L-dC, a reverse transcriptase inhibitor, is used potentially for treatment of HBV infection.Formule :C19H31N5O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :425.48Notch inhibitor 1
CAS :Notch inhibitor 1 blocks Notch 1/3 (IC50: 7.8/8.5 nM) and aids cancer research.Formule :C26H25F7N4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :574.49AFM-30a hydrochloride
AFM-30a hydrochloride: selective PAD2 inhibitor, EC50 9.5 μM; blocks H3 guanylation, EC50 0.4 μM; used for cancer and autoimmune research.Formule :C24H28ClFN6O3Couleur et forme :SolidMasse moléculaire :502.97B026
CAS :B026: Oral p300/CBP HAT inhibitor, IC50: p300 1.8 nM, CBP 9.5 nM; targets AR+ prostate cancer cells.Formule :C27H23F4N5O4Couleur et forme :SolidMasse moléculaire :557.5(±)-ANAP hydrochloride (1185251-08-4 free base)
(±)-ANAP hydrochloride is the amino acid analog of prodan. It can be used as a fluorescent probes and enhance environmental sensitivity.Formule :C15H17ClN2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :308.76AChE-IN-24
AChE-IN-24: Strong AChE blocker, crosses blood-brain barrier, IC50=0.053 μM, useful for AD research.Formule :C22H30N2O4S2Couleur et forme :SolidMasse moléculaire :450.61AM-3189
CAS :AM-3189: potent, selective GPR40 agonist with low CNS penetration, good pharmacokinetics, and efficacy mirroring AMG 837.Formule :C27H25ClN2O3Couleur et forme :SolidMasse moléculaire :460.95JH295 hydrate
JH295 hydrate: potent, irreversible Nek2 inhibitor (IC50 = 770 nM), selective, doesn't target Cdk1, Aurora B or Plk1.Formule :C18H18N4O3Couleur et forme :SolidMasse moléculaire :338.36HSP90-IN-9
HSP90-IN-9: potent HSP90 inhibitor, dose-dependent fungicide, impedes biofilm/morphology with FLC, reverses FLC resistance.Couleur et forme :SolidDihydro-β-erythroidine hydrobromide
CAS :Dihydro-β-erythroidine hydrobromide(DHβE) is a potent, oral active and competitive antagonist of neuronal nicotinic acetylcholine receptors (nAChRs).Formule :C16H22BrNO3Degré de pureté :98%Couleur et forme :White SolidMasse moléculaire :356.26MCTR3
CAS :MCTR3, derived from DHA via maresin 1 in macrophages, hastens tissue healing and reduces inflammation and eicosanoids post-E. coli infection in mice.Formule :C25H37NO5SCouleur et forme :SolidMasse moléculaire :463.63nAChR antagonist 1
CAS :Compound B15, a potent α7 nAChR antagonist, IC50 = 3.3 μM, promising for research on schizophrenia, Alzheimer's, and inflammation.Formule :C19H22N4O2Couleur et forme :SolidMasse moléculaire :338.4Kalafungin
CAS :Kalafungin inhibits various fungi, yeasts, protozoa, and gram-positive bacteria, less so for gram-negative bacteria.Formule :C16H12O6Couleur et forme :SolidMasse moléculaire :300.26HDAC-IN-9
HDAC-IN-9, a dual tubulin/HDAC inhibitor, impedes A549 cell invasion/migration and shows strong anti-tumor/angiogenic effects.Formule :C33H38N2O4Couleur et forme :SolidMasse moléculaire :526.67Mu opioid receptor antagonist 2
Compound 25: potent, selective MOR antagonist, crosses blood-brain barrier (Ki: 0.37 nM, EC50: 0.44 nM), for OUD research.Formule :C25H28N2O4SCouleur et forme :SolidMasse moléculaire :452.57PF-06751979
CAS :PF-06751979 is an inhibitor of β-site amyloid precursor protein cleaving enzyme 1 (BACE1) (IC50 of 7.3 nM in BACE1 binding assay).Formule :C18H19F2N5O3S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :455.5Raloxifene N-Oxide
CAS :Raloxifene N-Oxide is a Raloxifene oxidative degradation product.Formule :C28H27NO5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :489.58PDE4-IN-14
CAS :PDE4-IN-14 (Compound 1) serves as an inhibitor of phosphodiesterase 4 (PDE4), applicable in research concerning diseases associated with PDE4, includingFormule :C19H20F2N4O3SCouleur et forme :SolidMasse moléculaire :422.45HCV-IN-7
CAS :HCV-IN-7: potent oral HCV NS5A inhibitor, pan-genotypic, IC50s 3-47 pM, good pharmacokinetics, favorable liver uptake.Formule :C40H48N8O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :768.92VEGFR-2/DHFR-IN-1
Compound 8b inhibits VEGFR-2/DHFR, combats various bacteria, and fights cancer cells.Formule :C20H18ClNO4Couleur et forme :SolidMasse moléculaire :371.81Falecalcitriol
CAS :Falecalcitriol is an analog of calcitriol. It has a higher potency both in vivo and in vitro systems, which is longer duration of action in vivo.Formule :C27H38F6O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :524.58BRD1991
CAS :BRD1991 is a chemical compound that specifically disrupts the interaction between Beclin 1 and Bcl-2, thereby inducing autophagy.Formule :C33H35Cl2N3O4Couleur et forme :SolidMasse moléculaire :608.55Napsagatran hydrate
CAS :Napsagatran hydrate is a novel and specific inhibitor of thrombin.Formule :C26H36N6O7SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :576.66METTL3-IN-2
CAS :METTL3-IN-2, a potent METTL3 inhibitor, exhibits an IC50 value of 6.1 nM, effectively impairing the proliferation of Caov3 cancer cells.Formule :C25H26N8OCouleur et forme :SolidMasse moléculaire :454.53CB2 receptor antagonist 1
CAS :Compound 29 is a potent, CB2-selective antagonist/reverse agonist. Derivatives 23 & 24 offer antinociception; 24 activates cannabinoid/TRPV1 receptors.Formule :C28H47NO3Couleur et forme :SolidMasse moléculaire :445.68SF0166
CAS :SF0166: potent αvβ3 antagonist, IC50: 0.6 nM. Blocks cell adhesion, IC50: 7.6 pM-76 nM. Reduces neovascularization in mice.Formule :C23H27F2N5O4Couleur et forme :SolidMasse moléculaire :475.49TLR7/8 agonist 7
CAS :TLR7/8 agonist 7 activates immune cells, useful in ISAC synthesis and immunity research.Formule :C26H37N7O2Couleur et forme :SolidMasse moléculaire :479.62Anticancer agent 35
Compound 10, a sulfonylurea, inhibits A549, A431, PACA2 cells with IC50s: 18.1, 4.0, 18.9 μg/mL.Formule :C15H13N3O3S3Couleur et forme :SolidMasse moléculaire :379.48Tubulin inhibitor 16
Tubulin inhibitor 16 is a potent tubulin inhibitor with antiproliferative activity. Tubulin inhibitor 16 exhibits cytotoxicity in HepG2 cells [1].Formule :C16H12FNO2Couleur et forme :SolidMasse moléculaire :269.27BRD0418
CAS :BRD0418 acts as an upregulator of TRIB1 expression by leading to reprogramming of hepatic lipoprotein metabolism from adipogenesis to clearance it.Formule :C29H32N2O5Degré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :488.57C108297
CAS :C108297: glucocorticoid modulator, combats diet obesity/inflammation, reduces appetite/lipid storage, boosts fat burn.Formule :C30H36FN3O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :553.69FLT3/ITD-IN-1
FLT3/ITD-IN-1 inhibits FLT3-ITD with IC50s: 38.2 nM (FLT3) and 144.1 nM (ITD), and fights acute myeloid leukemia.Formule :C19H22N6O2Couleur et forme :SolidMasse moléculaire :366.42Prohibitin ligand 1
Compound 22i, a prohibitin ligand, protects the heart at nanomolar levels by inducing STAT3 phosphorylation.Formule :C20H22N2OCouleur et forme :SolidMasse moléculaire :306.4Anticancer agent 12
Anticancer agent 12 shows cytotoxic activity in malignant cells with no hepatotoxicity.Formule :C16H17BrN4O2SCouleur et forme :SolidMasse moléculaire :409.3PD 113271
CAS :PD 113,271 is an analog of the fermentation products fostriecin with antitumor activity in vitro and in vivo.Formule :C19H27O10PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :446.39BW 443C
CAS :BW 443C is a selective agonist of mu-opioid receptor.Formule :C33H46N10O10Couleur et forme :SolidMasse moléculaire :742.791FTI-2148
CAS :FTI-2148 blocks RAS-related FT-1 & GGT-1; IC50: 1.4 nM & 1.7 μM.Formule :C24H28N4O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :452.57SM-433 hydrochloride
SM-433 hydrochloride, a Smac mimetic & IAP inhibitor, binds XIAP BIR3; potent IC50 <1 μM. (Patent WO2008128171A2)Formule :C32H44ClN5O4Couleur et forme :SolidMasse moléculaire :598.18(±)-ANAP hydrochloride
CAS :'(±)-ANAP hydrochloride, an unnatural amino acid analog of prodan, serves as a fluorescent probe with enhanced environmental sensitivity.'Formule :C15H17ClN2O3Couleur et forme :SolidMasse moléculaire :308.76Basroparib
CAS :Basroparib is an inhibitor of ribose polymerase (PARP) and has shown antitumour effects.Formule :C18H21F2N7O3Couleur et forme :SolidMasse moléculaire :421.4CREB-IN-1 TFA
CREB-IN-1 TFA: Potent oral CREB inhibitor, IC50 of 0.18 μM, suppresses breast cancer cell growth.Couleur et forme :SolidCilengitide hydrochloride
CAS :Cilengitide hydrochloride is a salt that may combat cancer by blocking specific integrins, disrupting cell interactions and angiogenesis.Formule :C27H41ClN8O7Couleur et forme :SolidMasse moléculaire :625.12AZD2353
CAS :AZD2353 is a potent inhibitor of diacylglycerol acetyl transferase 1 (DGAT1).Formule :C22H19ClFN3O3Couleur et forme :SolidMasse moléculaire :427.86MMG-11 quarterhydrate
MMG-11 quarterhydrate, a potent hTLR2 antagonist, inhibits TLR2/1 and TLR2/6 with IC50s of 1.7μM and 5.7μM; low toxicity.Formule :C15H16O8Couleur et forme :SolidMasse moléculaire :310.78G-4120
CAS :G-4120 is a biochemical that has been shown to have a dose-dependent complete inhibition of arterial and venous thrombosis.Formule :C26H36N8O11SCouleur et forme :SolidMasse moléculaire :668.68Cortistatin A
CAS :Cortistatin A is a potent and selective mediator-associated kinase CDK8 and its paralogue CDK19 inhibitor.Formule :C30H36N2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :472.62Vindeburnol
CAS :Vindeburnol is a cerebral vasodilator vincamine analog that bears neuroprotective properties.Formule :C17H20N2OCouleur et forme :SolidMasse moléculaire :268.35Lp-PLA2-IN-6
CAS :Lp-PLA2-IN-6: Potent tetracyclic inhibitor of rhLp-PLA2, with pIC50 of 10.0, and potential in neurodegenerative research.Formule :C25H21F5N4O3Couleur et forme :SolidMasse moléculaire :520.45P-gp inhibitor 2
CAS :Potent P-gp inhibitor 2 reverses Doxorubicin resistance in colorectal carcinoma cells with IC50 of 0.22 µM.Formule :C29H26N2O6Couleur et forme :SolidMasse moléculaire :498.53Dyrk1A-IN-1
Dyrk1A-IN-1 is a triple inhibitor of Dyrk1A kinase activity, aggregation of tau and α-syn oligomers, with an IC50 value of 119 nM for Dyrk1A kinase.Formule :C23H20N4O3SCouleur et forme :SolidMasse moléculaire :432.49Tezampanel hydrate
CAS :Tezampanel is used for the treatment of migraine, neuropathic pain.Formule :C13H23N5O3Couleur et forme :SolidMasse moléculaire :297.35Antitumor agent-78
Antitumor agent-78 blocks GPx-4, raises COX2, triggers apoptosis, halts EMT, and stifles cancer cell growth and migration.Couleur et forme :Soild(S)-MALT1-IN-5
CAS :(S)-MALT1-IN-5: Potent MALT1 protease inhibitor, may help in abnormal T/B-cell signalling and MALT1-linked diseases.Formule :C17H17ClF2N6O3Couleur et forme :SolidMasse moléculaire :426.80(RS)-AMPA hydrobromide
CAS :AMPAR agonistFormule :C7H11BrN2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :267.08KRAS G12D inhibitor 1
CAS :KRAS G12D inhibitor 1 (example 243) is an inhibitor of KRAS G12D with an IC 50 of 0.8 nM for KRAS G12D-mediated ERK phosphorylation [1].Formule :C33H32F2N6O2Couleur et forme :SolidMasse moléculaire :582.6420-HEDE
CAS :20-HEDE (WIT 002) is a 20-hydroxyeicosatetraenoic acid (20-HETE) antagonist.Formule :C20H36O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :324.50KRAS inhibitor-8
CAS :KRAS inhibitor-8 is a potent KRAS G12C inhibitor.Formule :C26H24ClF4N5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :565.95hCAII-IN-4
CAS :hCAII-IN-4 (Compound 12j) is a potent inhibitor of human carbonic anhydrase II (hCA II), exhibiting an inhibitory concentration (IC50) of 7.78 μM.Formule :C31H23NO9Couleur et forme :SolidMasse moléculaire :553.52(Z)-Lanoconazole
(Z)-Lanoconazole, an imidazole antifungal for dermatophytosis and onychomycosis, inhibits fungal ergosterol production.Formule :C14H10ClN3S2Couleur et forme :SolidMasse moléculaire :319.83SML-10-70-1
CAS :SML-10-70-1 is a Novel Active Site Inhibitor of Oncogenic K-Ras G12C.Formule :C25H42ClN7O13P2Couleur et forme :SolidMasse moléculaire :746.04FTO-IN-1 TFA
FTO-IN-1 TFA: FTO enzyme inhibitor, anti-obesity, IC50 < 1μM, potential cancer research tool.Formule :C20H17Cl2F3N4O4Couleur et forme :SolidMasse moléculaire :505.27Bafilomycin C1
CAS :vacuolar H+-ATPases (V-ATPases) inhibitorFormule :C39H60O12Degré de pureté :98%Couleur et forme :Light Tan SolidMasse moléculaire :720.89Antiallergic agent-1
Antiallergic agent-1, an Src family kinase inhibitor, is a new and valuable lead compound with potential as an anti-allergic agent.Formule :C27H19F6N5OCouleur et forme :SolidMasse moléculaire :543.46XIAP/cIAP1 antagonist-1
Potent oral XIAP/cIAP1 inhibitor with EC50s: XIAP 5.1 nM, cIAP1 0.32 nM; curbs tumor growth in vivo.Couleur et forme :SolidNLRP3/AIM2-IN-1
NLRP3/AIM2-IN-1 is an inhibitor of thermal sepsis (IC50 = 3.136 ± 0.7667 μM).Formule :C15H16BNO4Couleur et forme :SolidMasse moléculaire :285.1PptT-IN-1
PptT-IN-1, a potent PptT inhibitor (IC50: 2.8 μM), shows promise for tuberculosis research.Formule :C18H29N5O2Couleur et forme :SolidMasse moléculaire :347.46Isoleucyl tRNA synthetase-IN-1
CAS :Isoleucyl tRNA synthetase-IN-1 is a selective and potent inhibitor (Ki: 88 nM) that targets isoleucyl tRNA synthetase (IleRS).Formule :C23H35N5O7SCouleur et forme :SolidMasse moléculaire :525.62Homodestcardin
CAS :Homodestcardin: cyclic depsipeptide from T. roseum with immunosuppressant properties; inhibits mouse T cell proliferation.Formule :C32H55N5O7Couleur et forme :SolidMasse moléculaire :621.81Tenellin
CAS :Tenellin is a fungal metabolite that inhibits Mg2+-, Ca2+-, and Na+/K+-ATPase activities in erythrocytes. Tenellin is cytotoxic to Sf9 and Sf21 insect cells.Formule :C21H23NO5Couleur et forme :SolidMasse moléculaire :369.41Anti-inflammatory agent 13
Pentacyclic triterpene, Anti-inflammatory 13 inhibits DAMP/PAMP inflammation models.Formule :C30H48O4Couleur et forme :SolidMasse moléculaire :472.7Gusperimus
CAS :Gusperimus was synthesized by chemical modification of spergualin and in combination with cyclosporine A to prevent diabetes in susceptible NOD mice.Formule :C17H37N7O3Couleur et forme :SolidMasse moléculaire :387.52HDAC-IN-32
HDAC-IN-32, potent inhibitor: IC50—HDAC1 (5.2 nM), HDAC2 (11 nM), HDAC6 (28 nM). Effective anti-tumor and immunity-boosting traits.Formule :C20H23N3O3Couleur et forme :SolidMasse moléculaire :353.41MCTR2
CAS :MCTR2, synthesized from DHA in macrophages, aids in tissue repair and reduces inflammation by promoting eicosanoid PGD2 and PGF2α decrease.Formule :C27H40N2O6SCouleur et forme :SolidMasse moléculaire :520.68GSK065
CAS :GSK065 is a potent inhibitor of kynurenine-3-monooxygenase (KMO).Formule :C17H15ClN2O4Couleur et forme :SolidMasse moléculaire :346.77E6201
CAS :E6201, a dual kinase inhibitor, blocks MEK1/FLT3 and has anti-tumor/psoriasis effects with low IC50s: ERK2 (5.2 nM), JNK (91 nM), p38 MAPK (19 nM).Formule :C21H27NO6Couleur et forme :SolidMasse moléculaire :389.44Carboxylesterase-IN-3
CAS :Carboxylesterase-IN-3 is a potent inhibitor of Carboxylesterase Notum (IC50 ≤ 10 nM).Carboxylesterase-IN-3 has the potential to study cancer diseases.
Formule :C11H6Cl2N4OSDegré de pureté :97.49% - 98.47%Couleur et forme :SolidMasse moléculaire :313.16MDK-3345
CAS :MDK-3345 is a reversible covalent inhibitor for Mcl-1.Formule :C36H34BN3O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :631.48Geissoschizoline
CAS :Geissoschizoline inhibits human AChE/BChE (IC50: 20.40/10.21 µM) and has anti-inflammatory properties.Formule :C19H26N2OCouleur et forme :SolidMasse moléculaire :298.42Autophagy-IN-1
Autophagy-IN-1 blocks autophagy in cancer cells, hinders tumor growth in mice, and aids in studying colorectal cancer.Formule :C23H25NO7Couleur et forme :SolidMasse moléculaire :427.45MALT1-IN-5
CAS :MALT1-IN-5 is a potent inhibitor of the MALT1 protease and can be used in cancer research.Formule :C17H17ClF2N6O3Couleur et forme :SolidMasse moléculaire :426.80BTK-IN-15
BTK-IN-15: Oral BTK inhibitor, IC50 0.7 nM, induces cancer cell apoptosis, selective with anti-tumor effects.Formule :C28H24FN5O2Couleur et forme :SolidMasse moléculaire :481.52DC41SMe
CAS :DC41SMe, a DC1 derivative and CC-1065 analogue, targets cancer with 18-25 pM IC50 against Ramos, Namalwa, HL60/s cells.Formule :C38H36ClN5O4S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :726.31Cathepsin C-IN-3
Cathepsin C-IN-3 is a potent inhibitor of histone C (IC50: 61.79 nM) and also inhibits THP-1 cells (IC50: 101.5 nM) and U937 cells (IC50: 86.5 nM).Formule :C28H21F3N6OSCouleur et forme :SolidMasse moléculaire :546.57G108
CAS :G108 is an inhibitor of human cGAS and is used in the study of autoimmune diseases associated with human cGAS.Formule :C16H14Cl2N4O2Degré de pureté :99.13% - 99.75%Couleur et forme :SolidMasse moléculaire :365.21
