Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.523 produits)
- Apoptose(5.792 produits)
- Cycle cellulaire/point de contrôle(4.449 produits)
- Chromatine/Épigénétique(2.238 produits)
- Signalisation du cytosquelette(1.383 produits)
- Altération de l'ADN/réparation de l'ADN(2.825 produits)
- Endocrinologie/Hormones(3.507 produits)
- Enzyme(3.640 produits)
- GPCR/G-Protéine(8.333 produits)
- Immunologie et Inflammation(3.526 produits)
- Virus de la grippe(296 produits)
- Signalisation JAK/STAT(404 produits)
- Signalisation MAPK(1.202 produits)
- Transporteur membranaire/Canal ionique(2.790 produits)
- Métabolisme(9.448 produits)
- Microbiologie/Virologie(6.981 produits)
- Neuroscience(9.926 produits)
- Autres inhibiteurs(37.926 produits)
- Oxydation-Réduction(41 produits)
- Signalisation PI3K/Akt/mTOR(1.400 produits)
- Protéases/Protéasome(1.597 produits)
- Cellules souche et Dérivés(831 produits)
- Tyrosine Kinase/Adaptateurs(2.016 produits)
- Ubiquitination(1.650 produits)
Affichez 16 plus de sous-catégories
66641 produits trouvés pour "Inhibiteurs"
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Pulvomycin
CAS :<p>Pulvomycin is a protein biosynthesis inhibitor preventing ternary complex formation between elongation factor Tu, GTP, and aminoacyl-tRNA.</p>Formule :C47H66O13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :839.032SX 3202
CAS :<p>SX 3202 is an aldose reductase inhibitor being developed for the treatment of diabetic neuropathy.</p>Formule :C17H11BrFN3O4Couleur et forme :SolidMasse moléculaire :420.19WS-898
<p>WS-898 boosts paclitaxel efficacy in resistant cells by inhibiting ABCB1; IC50: SW620/Ad300 - 5.0 nM, KB-C2 - 3.67 nM, HEK293/ABCB1 - 3.68 nM.</p>Formule :C33H25N7OSCouleur et forme :SolidMasse moléculaire :567.66IACS-8779
CAS :<p>IACS-8779 is a potent STING agonist that efficiently stimulates interferon gene activity and exhibits strong systemic antitumor effects.</p>Formule :C21H25N9O10P2S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :689.55COX-2/PI3K-IN-2
<p>COX-2/PI3K-IN-2 (5f): anti-inflammatory & anti-cancer, selectively inhibits COX-2 (Ki=3.02nM), potently blocks PI3K (IC50=2.78nM).</p>Formule :C16H17N5O2Couleur et forme :SolidMasse moléculaire :311.34PDHK-IN-5
<p>PDHK-IN-5, potent PDHK2 (0.006 μM IC50) & PDHK4 (0.0329 μM IC50) inhibitor, may be explored for cancer and diabetes treatment.</p>Formule :C30H31N5O2Couleur et forme :SolidMasse moléculaire :493.6CCT369260
CAS :<p>CCT369260 (compound 1), an orally active inhibitor targeting B-cell lymphoma 6 (BCL6), demonstrates anti-tumor efficacy with an IC50 value of 520 nM [1].</p>Formule :C24H31ClF2N6O2Couleur et forme :SolidMasse moléculaire :508.99GDC-6036-NH
CAS :<p>GDC-6036-NH is a precursor of compound 17a /b, which is a RAS inhibitor that can be used in cancer research.</p>Formule :C26H30ClF4N7ODegré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :568.01TRβ agonist 1
CAS :<p>TRβ Agonist 1, a selective and mutation-sensitive thyroid hormone receptor β (TRβ) agonist, demonstrates an EC50 value of 21 nM.</p>Formule :C29H25FN2O8Couleur et forme :SolidMasse moléculaire :548.52DFBTA
<p>DFBTA inhibits ANO1 with IC50 of 24 nM, effectively treating inflammatory pain orally.</p>Formule :C18H10ClF2NO3SCouleur et forme :SolidMasse moléculaire :393.79HOE-288
CAS :<p>HOE-288 is a converting enzyme (CE) inhibitor.</p>Formule :C27H38N2O5Couleur et forme :SolidMasse moléculaire :470.60FT001
CAS :<p>FT001: Oral BET Bromodomain inhibitor, IC50=0.46μM, suppresses MYC, anti-cancer, effective in vitro/vivo.</p>Formule :C25H29N3O4SDegré de pureté :99.9%Couleur et forme :SolidMasse moléculaire :467.58VHL Ligand 8
CAS :<p>VHL Ligand 8, a VHL ligand essential for synthesizing ARD-266, acts as a highly potent VHL E3 ligase-based androgen receptor (AR) PROTAC degrader.</p>Formule :C23H29N3O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :443.49CS-003 Free base
CAS :<p>CS-003: Triple neurokinin receptor antagonist; Ki=2.3 nM (NK1), 0.54 nM (NK2), 0.74 nM (NK3); treats respiratory diseases.</p>Formule :C34H38Cl2N2O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :673.65HDAC6/HSP90-IN-2
<p>HDAC6/HSP90-IN-2, a cancer research chemical, inhibits HDAC6 & Hsp90 with IC50s of 105.7 & 61 nM.</p>Formule :C19H22N2O5Couleur et forme :SolidMasse moléculaire :358.39Diguanosine 5′-triphosphate lithium
<p>Diguanosine 5′-triphosphate (Gp3G) lithium is a dinucleoside triphosphate and a virus-specific oligonucleotide.Diguanosine 5′-triphosphate lithium is required</p>Formule :C20H27N10O18P3·xLiCouleur et forme :SolidTHR-β agonist 4
CAS :<p>THR-β agonist 4 is a potent agonist of THR-β.</p>Formule :C16H11Cl2F2N5O6SCouleur et forme :SolidMasse moléculaire :510.26BI-207524
CAS :<p>BI-207524 is a novel NS5B Thumb Pocket 1 Inhibitor with Improved Potency for the Potential Treatment of Chronic Hepatitis C Virus Infection.</p>Formule :C35H36ClN5O5Couleur et forme :SolidMasse moléculaire :642.14Axl-IN-3
<p>Axl-IN-3 is a selective, potent and orally active inhibitor of AXL kinase (IC50: 41.5 nM) and has a low inhibitory effect on other kinases.</p>Formule :C24H25ClN6O2Couleur et forme :SolidMasse moléculaire :464.95SARS-CoV-2-IN-24
<p>SARS-CoV-2-IN-24 blocks PLpro, altering its shape and stopping virus replication—useful for SARS-CoV-2 research.</p>Formule :C27H30N4O5Couleur et forme :SolidMasse moléculaire :490.55PAD2-IN-1 hydrochloride
<p>PAD2-IN-1 hydrochloride: potent, selective PAD2 inhibitor; 95x less on PAD4, 79x less on PAD3; benzimidazole derivative.</p>Formule :C25H30ClFN6O3Couleur et forme :SolidMasse moléculaire :5173'-Hydroxy Repaglinide
CAS :<p>'3'-Hydroxy Repaglinide, a CYP2C8 metabolite of Repaglinide, treats type II diabetes.</p>Formule :C27H36N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :468.59HDAC-IN-33
<p>HDAC-IN-33 inhibits HDAC1/2/6 (IC50: 24/46/47 nM), exhibits potent antitumor activity in vitro and in vivo, and activates antitumor immunity.</p>Formule :C21H25N3O3Couleur et forme :SolidMasse moléculaire :367.44SR 33805 oxalate
CAS :<p>Ca2+ channel antagonist</p>Formule :C34H42N2O9SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :654.77BW-10
CAS :<p>BW-10 potently inhibits bombesin evoked release of gastrointestinal hormones in vitro and in vivo.</p>Formule :C57H72N14O8Couleur et forme :SolidMasse moléculaire :1081.27LSD1/2-IN-4
<p>LSD1/2-IN-4, a PCPA derivative, inhibits LSD1 (Ki 0.11 μM) & LSD2 (Ki 130 μM), potentially useful in T-cell leukemia research.</p>Formule :C9H8BrF2NCouleur et forme :SolidMasse moléculaire :248.07MA242
CAS :<p>MA242 is a nuclear factor of activated T cells 1 (NFAT1) for Pancreatic Cancer Therapy and dual inhibitor of murine double minute 2 (MDM2).</p>Formule :C26H21ClF3N3O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :579.98Gimatecan
CAS :<p>Gimatecan (STI481) is a potent topoisomerase I inhibitor. Gimatecan is an orally bioavailable camptothecin analogue with antitumor activity.</p>Formule :C25H25N3O5Degré de pureté :98.47%Couleur et forme :SolidMasse moléculaire :447.48MMAF sodium
CAS :<p>MMAF sodium, a potent tubulin inhibitor in ADCs like Vorsetuzumab mafodotin and SGN-CD19A, acts as an antitumor agent.</p>Formule :C39H64N5NaO8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :753.94HER2-IN-11
<p>HER2-IN-11 is a psoralen derivative that induces apoptosis. HER2-IN-11 shows light-activated cytotoxicity and also exhibits anti-breast cancer activity [1].</p>Formule :C17H11NO6Couleur et forme :SolidMasse moléculaire :325.27LY 292728
CAS :<p>LY 292728 is a highly potent antagonist of leukotriene B4 receptor.</p>Formule :C34H29FO9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :600.59ND-654
CAS :<p>ND-654 is an acetyl CoA carboxylase inhibitor.</p>Formule :C29H33N3O8SCouleur et forme :SolidMasse moléculaire :583.65Sucistil
<p>Sucistil is an active biochemical. hemoglobin sucistil (bovine) is an oxygen carrier [1].</p>Formule :C9H15NO4SCouleur et forme :SolidMasse moléculaire :233.28Mt KARI-IN-1
<p>Mt KARI-IN-1 inhibits Mtb KARI with a 3.06 μM Ki, targeting tuberculosis.</p>Formule :C14H11N5O4S2Couleur et forme :SolidMasse moléculaire :377.4FGI-106
CAS :<p>FGI-106 combats Ebola, Rift Valley, Dengue Fever, HCV, and HIV-1; EC50s range from 100-900 nM.</p>Formule :C28H38N6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :458.64NYX-2925
CAS :<p>NYX-2925, an oral NMDAR modulator, enhances Src in mPFC. No CAMKII impact or addictive/sedative effects. Useful for CNS disorder studies.</p>Formule :C14H23N3O4Couleur et forme :SolidMasse moléculaire :297.35MDK-3345
CAS :<p>MDK-3345 is a reversible covalent inhibitor for Mcl-1.</p>Formule :C36H34BN3O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :631.48LXR antagonist 2
<p>LXR antagonist 2 inhibits adipogenesis, downregulates LXR genes, and reduces lipids in hyperlipidemic mice (LXRβ IC50: 0.36μM, LXRα IC50: 2.25μM).</p>Formule :C34H40N2O5SCouleur et forme :SolidMasse moléculaire :588.76HDAC-IN-32
<p>HDAC-IN-32, potent inhibitor: IC50—HDAC1 (5.2 nM), HDAC2 (11 nM), HDAC6 (28 nM). Effective anti-tumor and immunity-boosting traits.</p>Formule :C20H23N3O3Couleur et forme :SolidMasse moléculaire :353.41IMR687
CAS :<p>IMR687: a PDE9 inhibitor that could improve memory in Alzheimer's by slowing cGMP hydrolysis.</p>Formule :C21H26N6O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :394.47microRNA-21-IN-1
CAS :<p>microRNA-21-IN-1: microRNA inhibitor, curbs HeLa/HCT-116 growth (IC50: 5.5/2.8 μM), induces HeLa apoptosis, elevates PTEN/EGR1/SLIT2, for cancer research.</p>Formule :C30H37FN6O3Couleur et forme :SolidMasse moléculaire :548.65GSK-3036656 free base
CAS :<p>GSK656 (GSK3036656) inhibits Mtb LeuRS with IC50 of 0.20 μM, promising for tuberculosis treatment.</p>Formule :C10H13BClNO4Couleur et forme :SolidMasse moléculaire :257.48BRD7929
CAS :<p>BRD7929 is a multistage antimalarial inhibitor for single-dose treatment of malaria in mouse models.</p>Formule :C33H38N4O2Couleur et forme :SolidMasse moléculaire :522.68Idraparinux Na
CAS :<p>Idraparinux Na is an Antithrombotic, Indirect, Selective, Synthetic Factor Xa Inhibitor</p>Formule :C38H55Na9O49S7Couleur et forme :SolidMasse moléculaire :1727.14PARP-1-IN-1
<p>PARP-1-IN-1: Selective, oral PARP-1 inhibitor with 0.96 nM IC50; well-tolerated and effective in single-dose MDA-MB-436 model.</p>Formule :C23H25FN4OCouleur et forme :SolidMasse moléculaire :392.47CDK4/6-IN-3
CAS :<p>CDK4/6-IN-3 is a brain-penetrant CDK4/CDK6 inhibitor (Kis: <0.3 nM and 2.2 nM) used for the treatment of glioblastoma. It inhibits CDK1 with a Ki of 110 nM.</p>Formule :C25H31FN8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :462.5716(S)-Iloprost
CAS :<p>Iloprost, a potent prostacyclin analog, binds to human IP & EP1 receptors with high affinity; inhibits platelet aggregation effectively.</p>Formule :C22H32O4Couleur et forme :SolidMasse moléculaire :360.49TGFβ1-IN-1
CAS :<p>TGFβ1-IN-1 is a TGF-β1 inhibitor that inhibits the production of TGF-β1-induced fibrosis markers (α-SMA and fibronectin) and can be used in cancer research.</p>Formule :C22H24N2O3Degré de pureté :99.89% - 99.89%Couleur et forme :SolidMasse moléculaire :364.438Luffolide
CAS :<p>Luffolide, a Luffariella sponge metabolite, shares manoalide's anti-inflammatory traits and fully inhibits PLA2's cleavage of phosphatidylcholine.</p>Formule :C27H40O6Couleur et forme :SolidMasse moléculaire :460.60GR 122222X
CAS :<p>GR 122222X is an inhibitor of topoisomerase II.</p>Formule :C26H35N5O11SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :625.65PCSK9-IN-17
CAS :<p>PCSK9-IN-17 is a PCSK9 inhibitor utilized in the research of cholesterol metabolism.</p>Formule :C16H19N5OSCouleur et forme :SolidMasse moléculaire :329.42Tofogliflozin
CAS :<p>Tofogliflozin specifically inhibits SGLT2; IC50s are 2.9 nM (human), 14.9 nM (rat), 6.4 nM (mouse).</p>Formule :C22H26O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :386.44Oncopterin
CAS :<p>Oncopterin is found in urine from patients with solid and blood cancers.</p>Formule :C12H18N6O3Couleur et forme :SolidMasse moléculaire :294.31SCO-792
<p>SCO-792: potent, reversible oral enteropeptidase inhibitor, with slow in vitro dissociation and in vivo protein digestion blocking.</p>Formule :C22H22N4O8·xH2OCouleur et forme :SolidKI696
CAS :<p>KI696 is a high-affinity probe that potently inhibits the interaction of Keap1 and NRF2.</p>Formule :C28H30N4O6SDegré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :550.63Elacytarabine
CAS :<p>Elacytarabine (M7594 0037), a lipid-conjugated derivative of the nucleoside analog cytarabine, is an antineoplastic drug. It has cytotoxicity in solid tumors.</p>Formule :C27H45N3O6Degré de pureté :97.69%Couleur et forme :SolidMasse moléculaire :507.66Treprostinil diethanolamine
CAS :<p>Treprostinil diethanolamine (UT-15C) is a potent agonist of EP2, DP1 and IP, with values of 3.6, 4.4, 32.1, 212, 826, 2505 and 4680 nM for EP2, DP1, IP, EP1,</p>Formule :C27H45NO7Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :495.65Obicetrapib
CAS :<p>Obicetrapib (AMG-899) is an inhibitor of cholesteryl ester transfer protein.</p>Formule :C32H31F9N4O5Degré de pureté :99.26% - >99.99%Couleur et forme :SolidMasse moléculaire :722.6SYM2206
CAS :<p>SYM2206 is a low affinity non-competitive AMPA receptor antagonist with an IC50 value of 1.6 μM.SYM2206 exhibits anticancer activity by blocking Nav1.6-mediated</p>Formule :C20H22N4O3Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :366.41Aleglitazar
CAS :<p>Aleglitazar (R1439) (R1439) is a potent dual PPARα/γ agonist, with IC50s of 38 nM and 19 nM for human PPARa and PPARγ, respectively.</p>Formule :C24H23NO5SDegré de pureté :99.03%Couleur et forme :SolidMasse moléculaire :437.51IDX184
CAS :<p>IDX184 is a potent, orally active, targeted HCV polymerase inhibitor and nucleoside polymerase.IDX184 effectively inhibits HCV polymerase (IC50=0.31 μM, Ki=52.3</p>Formule :C25H35N6O9PSDegré de pureté :97.15%Couleur et forme :SolidMasse moléculaire :626.62CCF0058981
CAS :<p>CCF0058981: noncovalent inhibitor for SARS-CoV-2 & -1 proteases; IC50s: 68 nM (SC2) & 19 nM (SC1). Potential COVID-19 research use.</p>Formule :C24H19ClN6ODegré de pureté :98.94%Couleur et forme :SoildMasse moléculaire :442.9Odevixibat
CAS :<p>Odevixibat (A4250) is a selective oral inhibitor for ileal bile acid transport, potentially treating primary biliary cirrhosis.</p>Formule :C37H48N4O8S2Degré de pureté :99.53% - 99.83%Couleur et forme :SolidMasse moléculaire :740.93EZM0414
CAS :<p>EZM0414 is a potent, selective, orally bioavailable inhibitor of SETD2 with IC50 of 18 nM in SETD2 biochemical assay and IC50 of 34 nM in a cellular assay.</p>Formule :C22H29FN4O2Degré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :400.49NRX-103095
CAS :<p>NRX-103095 increases β-catenin binding to SCFβ-TrCP E3 ligase; EC50 is 163 nM for pSer33/Ser37 affinity boost.</p>Formule :C22H16Cl2F3N3O3SDegré de pureté :99.58% - 99.95%Couleur et forme :SolidMasse moléculaire :530.35USP15-IN-1
CAS :<p>USP15-IN-1 is a potent USP15 inhibitor (IC50 is 3.76 μM).</p>Formule :C22H23N3O3Degré de pureté :99.509% - 99.81%Couleur et forme :SolidMasse moléculaire :377.44Cbl-b-IN-3
CAS :<p>Cbl-b-IN-3 is a potent inhibitor of casitas b lineage lymphoma proto-oncogene-b (Cbl-b) (ic50 < 1 nM).Cost-effective and quality-assured.</p>Formule :C30H34F3N5ODegré de pureté :99%Couleur et forme :SolidMasse moléculaire :537.62AZD5462
CAS :<p>AZD5462 is a potent orally available relaxin receptor RXFP1 agonist for the study of heart failure and cancer.</p>Formule :C30H41FN2O6Degré de pureté :98.32% - 99.63%Couleur et forme :SolidMasse moléculaire :544.65Pocenbrodib
CAS :<p>Pocenbrodib (FT-7051) is a potent inhibitor of the bromodomain of the CBP/p300 family with potential antitumour activity and is palatable for cancer research.</p>Formule :C28H32FN3O6Degré de pureté :98.48% - 99.54%Couleur et forme :SolidMasse moléculaire :525.57DRF-1042
CAS :<p>DRF-1042 is a camptothecin analog with anticancer and insecticidal activity and is used to study solid tumors such as prostate and colon cancer.</p>Formule :C22H20N2O6Degré de pureté :98.34%Couleur et forme :SolidMasse moléculaire :408.4Aldometanib
CAS :<p>Aldometanib (LXY-05-029) is an oral aldolase inhibitor that maintains metabolic balance by blocking FBP and activating lysosomal AMPK.</p>Formule :C27H43Cl2IN2Degré de pureté :99.32% - 99.55%Couleur et forme :SolidMasse moléculaire :593.46Dazostinag disodium
CAS :<p>Dazostinag disodium (TAK-676) is a synthetic novel interferon gene (STING) agonist.Cost-effective and quality-assured.</p>Formule :C21H20F2N8Na2O10P2S2Degré de pureté :98.84% - 99.96%Couleur et forme :SolidMasse moléculaire :754.48Darizmetinib
CAS :<p>Darizmetinib (HRX215) is an MKK4 inhibitor.</p>Formule :C21H17F2N5O3SDegré de pureté :98.03% - 99.57%Couleur et forme :SolidMasse moléculaire :457.45Vofopitant
CAS :<p>Vofopitant (GR 205171) is a potent NK1 receptor antagonist with anxiolytic and antiemetic activity for the study of post-traumatic stress disorder (PTSD).</p>Formule :C21H23F3N6ODegré de pureté :97.86%Couleur et forme :SolidMasse moléculaire :432.44GSK3368715 dihydrochloride
CAS :<p>GSK3368715 dihydrochloride (EPZ019997 dihydrochloride) is a PRMTs inhibitor , with anticancer activity, for the study of advanced solid tumors.</p>Formule :C20H40Cl2N4O2Degré de pureté :99.66% - 99.66%Couleur et forme :SolidMasse moléculaire :439.46BMS453
CAS :<p>BMS453 (BMS-189453), a synthetic retinoid, is a potent and selective agonist of RARβ and a potent testicular toxin.</p>Formule :C27H24O2Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :380.48Rupintrivir
CAS :<p>Rupintrivirvr (AG7088) is a mimetic peptide inhibitor of rhinovirus (HRV) 3C cysteine protease with antiviral activity for the study of viral infections.</p>Formule :C31H39FN4O7Degré de pureté :97.72% - 99.35%Couleur et forme :SolidMasse moléculaire :598.66Eravacycline dihydrochloride
CAS :<p>Eravacycline dihydrochloride (TP-434-046) is a potent and broad-spectrum antibacterial agent against six E. coli (MICs: 0.125-0.25 mg/L).</p>Formule :C27H33Cl2FN4O8Degré de pureté :94.59% - 95%Couleur et forme :SolidMasse moléculaire :631.48Cap-dependent endonuclease-IN-1
CAS :<p>Cap-dependent endonuclease-IN-1: potent, oral inhibitor with antiviral properties against influenza.</p>Formule :C27H22F2N2O6SDegré de pureté :98.88% - 99.09%Couleur et forme :SolidMasse moléculaire :540.54NDI-034858
CAS :<p>NDI-034858 (TAK-279) is a tyrosine kinase 2 (TYK2) inhibitor (Kd<200 pM) that targets the JH2 structural domain of Tyk2 for the treatment of autoimmune diseases</p>Formule :C23H24N8O3Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :460.49BCL6-IN-3
CAS :<p>BCL6-IN-3: potent BCL6 inhibitor, 70 nM GI50 in SU-DHL4, affects cell functions, antitumor.</p>Formule :C24H31ClF2N6O2Degré de pureté :98.17%Couleur et forme :SolidMasse moléculaire :508.99Umibecestat
CAS :<p>Umibecestat inhibits human and mouse BACE-1 (IC50: 11 nM & 10 nM), potentially for Alzheimer's research.</p>Formule :C19H15ClF7N5O2Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :513.8Vofopitant dihydrochloride
CAS :<p>Vofopitant dihydrochloride (GR 205171A) is a tachykinin NK1 receptor antagonist and a potential compound for the treatment of pathologic vomiting.</p>Formule :C21H25Cl2F3N6ODegré de pureté :98.99%Couleur et forme :SolidMasse moléculaire :505.36Gepotidacin mesylate dihydrate
CAS :<p>Gepotidacin mesylate dihydrate (GSK2140944 mesylate dihydrate) is an antibiotic and an inhibitor of bacterial type II topoisomerase.</p>Formule :C25H36N6O8SDegré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :580.65PF-07258669
CAS :<p>PF-07258669 is a selective melanocortin 4 receptor (MC4) antagonist used in the study of cachexia and loss of appetite.</p>Formule :C25H27FN6O2Degré de pureté :99.9%Couleur et forme :SolidMasse moléculaire :462.52ZD 7155 hydrochloride
CAS :<p>ZD 7155 hydrochloride is an angiotensin II receptor type 1 (AT1 receptor) antagonist.</p>Formule :C26H27ClN6ODegré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :474.98BDZ-g
CAS :<p>BDZ-g: potent, selective AMPA receptor antagonist; useful for researching neurological disorders.</p>Formule :C21H21N5O2SDegré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :407.49JTK-109
CAS :<p>JTK-109 is an inhibitor of hepatitis C virus NS5B RNA-dependent RNA polymerase inhibitor and inhibits G1b and G3a subgenomic replicons and recombinant enzymes.</p>Formule :C37H33ClFN3O4Degré de pureté :98.48% - 99.68%Couleur et forme :SolidMasse moléculaire :638.13FABPs ligand 6
CAS :<p>FABPs ligand 6 (MF6) is an inhibitor of FABP5 and FABP7.</p>Formule :C28H27FN2O3Degré de pureté :97.45%Couleur et forme :SolidMasse moléculaire :458.52STK-15
CAS :<p>STK-15 is a candidate for use as a fatty acid binding protein 5 (FABP5) inhibitor.</p>Formule :C34H29NO5Degré de pureté :98.05%Couleur et forme :SolidMasse moléculaire :531.6Dersimelagon
CAS :<p>Dersimelagon (MT-7117) is an orally active, selective melanocortin 1 receptor (MC1R) agonist.Cost-effective and quality-assured.</p>Formule :C36H45F4N3O5Degré de pureté :97.35% - 98.23%Couleur et forme :SolidMasse moléculaire :675.75Suzetrigine
CAS :<p>Suzetrigine (VX-548) is an oral NaV1.8 inhibitor with analgesic properties for acute pain research.</p>Formule :C21H20F5N3O4Degré de pureté :98.08% - 99.27%Couleur et forme :SolidMasse moléculaire :473.39Glycosyltransferase-IN-1
<p>Glycosyltransferase-IN-1 is a glycosyltransferase inhibitor with bacteriostatic activity, inhibiting MSSA, MRSA, Bacillus subtilis, and Enterobacteriaceae.</p>Formule :C19H21N5ODegré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :335.4VX-984
CAS :<p>VX-984 (M9831) is an oral DNA-PK inhibitor, crossing the blood-brain barrier, targeting GBM and NSC-LC.</p>Formule :C23H21D2N7ODegré de pureté :97.65% - 99.98%Couleur et forme :SolidMasse moléculaire :415.49ALOX15-IN-2
CAS :<p>ALOX15-IN-2: Potent ALOX15 inhibitor. IC50: 1.55 μM for LA; 2.79 μM for AA. Stops linoleic/arachidonic acid oxidation.</p>Formule :C23H29N3O4SDegré de pureté :98.10%Couleur et forme :SolidMasse moléculaire :443.56KU-60019
CAS :<p>KU-60019 is a specific inhibitor of ATM kinase (IC50: 6.3 nM).</p>Formule :C30H33N3O5SDegré de pureté :98.05% - 98.50%Couleur et forme :SolidMasse moléculaire :547.67MAO-B-IN-17
CAS :<p>MAO-B-IN-17 is a selective and potent monoamine oxidase B (MAO-B) inhibitor (IC50: 5.08 μM) for the study of central nervous system disorders like Parkinson's.</p>Formule :C17H17F2NO2Degré de pureté :99.41%Couleur et forme :SoildMasse moléculaire :305.32DRB18
CAS :<p>DRB18 inhibits GLUT proteins, altering glucose metabolism and inducing cancer cell death by G1/S arrest and oxidative stress.</p>Formule :C22H23ClN2O2Degré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :382.88ELOVL1-IN-2
CAS :<p>ELOVL1-IN-2 weakly inhibits ELOVL1 enzyme (IC50: 21 μM) and shows moderate potency in HEK293 cells (IC50: 6.7 μM).</p>Formule :C18H15FN2ODegré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :294.32LSN3318839
CAS :<p>LSN3318839 is a potent and orally available glucagon-like peptide-1 receptor (GLP-1R) modulator.LSN3318839 enhances GLP-1R G-protein-coupled signaling and can</p>Formule :C26H23Cl2N3O2Degré de pureté :99.21%Couleur et forme :SolidMasse moléculaire :480.39
