Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.834 produits)
- Apoptose(6.315 produits)
- Cycle cellulaire/point de contrôle(4.877 produits)
- Chromatine/Épigénétique(2.613 produits)
- Signalisation du cytosquelette(1.568 produits)
- Altération de l'ADN/réparation de l'ADN(2.872 produits)
- Endocrinologie/Hormones(3.754 produits)
- Enzyme(3.672 produits)
- GPCR/G-Protéine(9.019 produits)
- Immunologie et Inflammation(3.904 produits)
- Virus de la grippe(300 produits)
- Signalisation JAK/STAT(415 produits)
- Signalisation MAPK(1.257 produits)
- Transporteur membranaire/Canal ionique(3.155 produits)
- Métabolisme(10.136 produits)
- Microbiologie/Virologie(7.620 produits)
- Neuroscience(10.460 produits)
- Autres inhibiteurs(35.848 produits)
- Oxydation-Réduction(40 produits)
- Signalisation PI3K/Akt/mTOR(1.429 produits)
- Protéases/Protéasome(1.691 produits)
- Cellules souche et Dérivés(732 produits)
- Tyrosine Kinase/Adaptateurs(1.982 produits)
- Ubiquitination(1.726 produits)
Affichez 16 plus de sous-catégories
66515 produits trouvés pour "Inhibiteurs"
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AM103
CAS :AM103 is an effective and selective inhibitor of FLAP (IC50 = 4.2 nM).Formule :C36H38N3NaO4SDegré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :631.76Cort108297
CAS :Cort108297: selective GR modulator/antagonist, high GR affinity (Ki: 0.45nM), no other steroid receptor affinity.Formule :C26H25F4N3O3SDegré de pureté :98.36% - 99.94%Couleur et forme :SolidMasse moléculaire :535.55Ref: TM-T15000
1mg260,00€5mg590,00€10mg859,00€25mg1.341,00€50mg1.783,00€100mg2.602,00€1mL*10mM (DMSO)708,00€PF-07258669
CAS :PF-07258669 is a selective melanocortin 4 receptor (MC4) antagonist used in the study of cachexia and loss of appetite.Formule :C25H27FN6O2Degré de pureté :99.9%Couleur et forme :SolidMasse moléculaire :462.52Cap-dependent endonuclease-IN-1
CAS :Cap-dependent endonuclease-IN-1: potent, oral inhibitor with antiviral properties against influenza.Formule :C27H22F2N2O6SDegré de pureté :99.53% - 99.61%Couleur et forme :SolidMasse moléculaire :540.54NRX-252114
CAS :NRX-252114 promotes mutant β-catenin degradation, binding it to E3 ligase SCFβ-TrCP (EC50: 6.5 nM; Kd: 0.4 nM).Formule :C22H12Cl2F3N3O2SDegré de pureté :99.70%Couleur et forme :SolidMasse moléculaire :510.32Enbezotinib
CAS :Enbezotinib is an inhibitor of RET autophosphorylation and can be used in cancer research.Formule :C21H21FN6O3Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :424.43Ref: TM-T62285
1mg77,00€5mg166,00€10mg253,00€25mg414,00€50mg567,00€100mg745,00€1mL*10mM (DMSO)182,00€AZD5462
CAS :AZD5462 is a potent orally available relaxin receptor RXFP1 agonist for the study of heart failure and cancer.Formule :C30H41FN2O6Degré de pureté :98.32% - 99.63%Couleur et forme :SolidMasse moléculaire :544.65BQ-788
CAS :BQ-788 is an ETB receptor antagonist with potential hypertensive activity that inhibits exogenous ET-1-induced elevation of coronary perfusion pressure.Formule :C34H51N5O7Degré de pureté :98.81%Couleur et forme :SolidMasse moléculaire :641.8Ref: TM-T10595
1mg130,00€2mg178,00€5mg313,00€10mg447,00€25mg713,00€50mg964,00€100mg1.305,00€500mg2.592,00€1mL*10mM (DMSO)341,00€Dazostinag disodium
CAS :Dazostinag disodium (TAK-676) is a synthetic novel interferon gene (STING) agonist.Cost-effective and quality-assured.Formule :C21H20F2N8Na2O10P2S2Degré de pureté :98.84% - 99.96%Couleur et forme :SolidMasse moléculaire :754.48SJ6986
CAS :SJ6986 is a potent, selective and orally active GSPT1/2 degrader. SJ6986 degrades GSPT1 with a DC 50 of 2.1 nM (D max 99%) [1].Formule :C20H14F3N3O7SDegré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :497.4Ref: TM-T41257
5mg52,00€10mg86,00€25mg140,00€50mg245,00€100mg378,00€500mg898,00€1mL*10mM (DMSO)59,00€VX-984
CAS :VX-984 (M9831) is an oral DNA-PK inhibitor, crossing the blood-brain barrier, targeting GBM and NSC-LC.Formule :C23H21D2N7ODegré de pureté :97.65% - 99.98%Couleur et forme :SolidMasse moléculaire :415.49Ref: TM-T11067
1mg117,00€5mg248,00€10mg369,00€25mg575,00€50mg863,00€100mg1.305,00€200mg1.755,00€1mL*10mM (DMSO)271,00€SB-224289 hydrochloride
CAS :SB-224289 hydrochloride (SB-224289A) is a selective antagonist of 5-HT1B receptor, with anxiolytic effect.Formule :C32H33ClN4O3Degré de pureté :98.99% - 99.96%Couleur et forme :SolidMasse moléculaire :557.08Darizmetinib
CAS :Darizmetinib (HRX215) is an MKK4 inhibitor.Formule :C21H17F2N5O3SDegré de pureté :98.03% - 99.57%Couleur et forme :SolidMasse moléculaire :457.45Ref: TM-T72956
1mg69,00€2mg89,00€5mg147,00€10mg224,00€25mg324,00€50mg400,00€100mg587,00€1mL*10mM (DMSO)148,00€DN02
DN02: a potent, selective BRD8(1) bromodomain probe; Ki=32 nM; 30x more affine than BRD8(2).Formule :C22H24FN3O3Degré de pureté :98.22% - 99.74%Couleur et forme :SolidMasse moléculaire :397.44FABPs ligand 6
CAS :FABPs ligand 6 (MF6) is an inhibitor of FABP5 and FABP7.Formule :C28H27FN2O3Degré de pureté :97.45%Couleur et forme :SolidMasse moléculaire :458.52PREP inhibitor-1
CAS :PREP inhibitor-1 is a prolyl oligopeptidase (PREP) inhibitor for the study of Alzheimer's disease.Formule :C22H28N4O2Degré de pureté :98.78%Couleur et forme :SoildMasse moléculaire :380.48Glycosyltransferase-IN-1
Glycosyltransferase-IN-1 is a glycosyltransferase inhibitor with bacteriostatic activity, inhibiting MSSA, MRSA, Bacillus subtilis, and Enterobacteriaceae.Formule :C19H21N5ODegré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :335.4JTK-109
CAS :JTK-109 is an inhibitor of hepatitis C virus NS5B RNA-dependent RNA polymerase inhibitor and inhibits G1b and G3a subgenomic replicons and recombinant enzymes.Formule :C37H33ClFN3O4Degré de pureté :98.48% - 99.68%Couleur et forme :SolidMasse moléculaire :638.13Ref: TM-T27696
1mg296,00€5mg718,00€10mg982,00€25mg1.485,00€50mg2.008,00€100mg2.637,00€1mL*10mM (DMSO)1.108,00€Dersimelagon
CAS :Dersimelagon (MT-7117) is an orally active, selective melanocortin 1 receptor (MC1R) agonist.Cost-effective and quality-assured.Formule :C36H45F4N3O5Degré de pureté :97.35% - 98.23%Couleur et forme :SolidMasse moléculaire :675.75MAO-B-IN-17
CAS :MAO-B-IN-17 is a selective and potent monoamine oxidase B (MAO-B) inhibitor (IC50: 5.08 μM) for the study of central nervous system disorders like Parkinson's.Formule :C17H17F2NO2Degré de pureté :99.41%Couleur et forme :SoildMasse moléculaire :305.32Aldometanib
CAS :Aldometanib (LXY-05-029) is an oral aldolase inhibitor that maintains metabolic balance by blocking FBP and activating lysosomal AMPK.Formule :C27H43Cl2IN2Degré de pureté :99.32% - 99.55%Couleur et forme :SolidMasse moléculaire :593.46BODIPY FL prazosin
CAS :BODIPY FL prazosin is an α1-adrenergic antagonist that inhibits α1a-AR and α1b-AR.
Formule :C28H32BF2N7O3Degré de pureté :97.27%Couleur et forme :SolidMasse moléculaire :563.41Zelasudil
CAS :Zelasudil (RXC007) is a Rho-related (ROCK) kinase inhibitor for the study of idiopathic pulmonary fibrosis and inflammation.Formule :C22H21F2N7ODegré de pureté :99.15%Couleur et forme :SolidMasse moléculaire :437.445Ref: TM-T69665
1mg92,00€5mg168,00€10mg248,00€25mg421,00€50mg587,00€100mg820,00€1mL*10mM (DMSO)170,00€INCB054329
CAS :INCB054329 is a BET inhibitor targeting BRD2/3/4 and BRDT with IC50s ranging from 1-119 nM.Formule :C19H16N4O3Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :348.36STK-15
CAS :STK-15 is a candidate for use as a fatty acid binding protein 5 (FABP5) inhibitor.Formule :C34H29NO5Degré de pureté :98.05%Couleur et forme :SolidMasse moléculaire :531.6Gepotidacin mesylate dihydrate
CAS :Gepotidacin mesylate dihydrate (GSK2140944 mesylate dihydrate) is an antibiotic and an inhibitor of bacterial type II topoisomerase.Formule :C25H36N6O8SDegré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :580.65AChE-IN-26
CAS :AChE-IN-26 (compound 4a) is an AChE (acetylcholinesterase) inhibitor (IC50: 0.42 μM).
Formule :C21H21BrN2O3Degré de pureté :99.24% - 99.85%Couleur et forme :SoildMasse moléculaire :429.31SDZ 220-040
CAS :SDZ 220-040 是一种选择性哺乳动物 NMDA 受体拮抗剂，可诱导根系生长的部分无重力模式 。Formule :C16H16Cl2NO6PDegré de pureté :98.13%Couleur et forme :SolidMasse moléculaire :420.18D75-4590
CAS :D75-4590, a β-1,6-Glucan synthetase inhibitor, combats fungal infections by targeting cell walls.Formule :C21H27N5Degré de pureté :98.56% - 98.85%Couleur et forme :SolidMasse moléculaire :349.47Ref: TM-T61194
5mg39,00€10mg62,00€25mg122,00€50mg187,00€100mg269,00€200mg358,00€1mL*10mM (DMSO)46,00€CCF0058981
CAS :CCF0058981: noncovalent inhibitor for SARS-CoV-2 & -1 proteases; IC50s: 68 nM (SC2) & 19 nM (SC1). Potential COVID-19 research use.
Formule :C24H19ClN6ODegré de pureté :98.94%Couleur et forme :SoildMasse moléculaire :442.9Ref: TM-T60095
1mg46,00€2mg60,00€5mg92,00€10mg160,00€25mg324,00€50mg449,00€100mg562,00€500mgÀ demanderBAY-3827
CAS :BAY-3827 is an AMPK inhibitor with antiproliferative activity and antitumor activity. BAY-3827 inhibits the phosphorylation of acetyl CoA carboxylase 1.Formule :C27H25FN6ODegré de pureté :99.90%Couleur et forme :SolidMasse moléculaire :468.53Ref: TM-T73350
1mg52,00€5mg113,00€10mg177,00€25mg334,00€50mg560,00€100mg792,00€500mg1.575,00€1mL*10mM (DMSO)117,00€BE1218
CAS :BE1218 is a liver X receptor (LXR) inverse agonist active on LXRα and LXRβ with an IC50 of 9 nM and 7 nM, respectively.
Formule :C30H30FNO4S2Degré de pureté :99.7%Couleur et forme :SoildMasse moléculaire :551.69BLU2864
CAS :BLU2864: oral PRKACA inhibitor, IC50=0.3 nM, potential in cancer/poly. kidney disease research.Formule :C24H19F3N4O2Degré de pureté :97.58% - 99.92%Couleur et forme :SoildMasse moléculaire :452.43SY-5609
CAS :SY-5609 (CDK7-IN-3) is a selective non-covalent CDK7 inhibitor, with weak inhibitory activity against CDK2, CDK9 and CDK12.Cost-effective and quality-assured.Formule :C23H26F3N6OPDegré de pureté :99.34% - >99.99%Couleur et forme :SolidMasse moléculaire :490.46Ref: TM-T36038
1mg139,00€2mg200,00€5mg343,00€10mg553,00€25mgÀ demander50mgÀ demander1mL*10mM (DMSO)373,00€LLY-283
CAS :LLY-283, PRMT5 inhibitor, IC50 22 nM, Kd 6 nM, oral, selective, with antitumor effects.Formule :C17H18N4O4Degré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :342.35Moiramide B
CAS :Moiramide B is an acetyl coenzyme A carboxylase inhibitor with antimicrobial activity, strongly inhibiting Gram-positive bacteria.Formule :C25H31N3O5Degré de pureté :98.53% - 99.90%Couleur et forme :SolidMasse moléculaire :453.53(+)-Tetrabenazine
CAS :(+)-Tetrabenazine ((3R,11bR)-Tetrabenazine) is a reversible vesicular monoamine transporter 2 (VMAT-2) inhibitor, inhibits transport by VMAT2 with 10-foldFormule :C19H27NO3Degré de pureté :98.69%Couleur et forme :SolidMasse moléculaire :317.42IDX184
CAS :IDX184 is a potent, orally active, targeted HCV polymerase inhibitor and nucleoside polymerase.IDX184 effectively inhibits HCV polymerase (IC50=0.31 μM, Ki=52.3Formule :C25H35N6O9PSDegré de pureté :97.15%Couleur et forme :SolidMasse moléculaire :626.62Zotizalkib
CAS :TPX-0131: potent, selective, CNS-ready, oral ALK inhibitor (WT IC50: 1.4nM, G1202R/L1196M IC50: 0.3nM) with robust antitumor effects.Formule :C21H20F3N5O3Degré de pureté :98.7%Couleur et forme :SolidMasse moléculaire :447.41Ref: TM-T9414
1mg114,00€5mg268,00€10mg439,00€25mg879,00€50mg1.395,00€100mg1.873,00€1mL*10mM (DMSO)303,00€AZD 3147
CAS :AZD 3147 inhibits mTORC1 (40.7 nM), mTORC2 (5.75 nM), and PI3Kα/β/δ/γ (912/5495/9333/6310 nM IC50s).
Formule :C24H31N5O4S2Degré de pureté :99.99%Couleur et forme :SolidMasse moléculaire :517.66BDZ-g
CAS :BDZ-g: potent, selective AMPA receptor antagonist; useful for researching neurological disorders.Formule :C21H21N5O2SDegré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :407.49JNJ-6204
CAS :JNJ-6204 is a deuterated compound that efficiently inhibits CSNK1D and CSNK1E.Formule :C19H11D6FN6ODegré de pureté :97.42% - 99.87%Couleur et forme :SolidMasse moléculaire :370.41ARN19702
CAS :ARN19702: orally active, brain-penetrant, selective NAAA inhibitor, IC50 230 nM, broad analgesic profile.Formule :C21H22FN3O3S2Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :447.55Ref: TM-T9528
1mg52,00€5mg113,00€10mg177,00€25mg350,00€50mg560,00€100mg880,00€200mg1.189,00€500mg1.765,00€1mL*10mM (DMSO)124,00€Sinefungin
CAS :Sinefungin (Adenosyl-Ornithine) is an effective inhibitor of virion mRNA(guanine-7-)-methyltransferase, mRNA(nucleoside-2'-)-methyltransferase, and viralFormule :C15H23N7O5Degré de pureté :98% - 98.12%Couleur et forme :SolidMasse moléculaire :381.39BRD0639
CAS :BRD0639 is a first-in-class PRMT5-substrate interaction inhibitor for PBM-dependent PRMT5 activity studies.Formule :C21H22ClN5O4SDegré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :475.95BAY-8400
BAY-8400 is an orally active, potent and selective DNA-dependent protein kinase ( DNA-PK ) inhibitor ( IC 50 =81 nM) which shows synergistic efficacy inFormule :C21H17F2N5ODegré de pureté :99.53%Couleur et forme :SolidMasse moléculaire :393.39Ref: TM-T9498
1mg80,00€5mg147,00€10mg215,00€25mg439,00€50mg750,00€100mg1.009,00€1mL*10mM (DMSO)161,00€CK2 inhibitor 2
CAS :CK2 Inhibitor 2, characterized as a potent, selective, and orally active inhibitor of CK2, demonstrates an impressive IC50 value of 0.66 nM.Formule :C21H17ClN4O2Degré de pureté :99.02%Couleur et forme :SolidMasse moléculaire :392.84Ref: TM-T35557
1mg62,00€5mg138,00€10mg215,00€25mg425,00€50mg637,00€100mg853,00€200mg1.153,00€1mL*10mM (DMSO)152,00€XMD-17-51 Trifluoroacetate
CAS :XMD-17-51 Trifluoroacetate is a pyrimido-diazepinone compound that regulates protein kinases.Formule :C23H25F3N8O3Degré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :518.49JAK2-IN-7
CAS :JAK2-IN-7 selectively inhibits JAK2 (IC50: 3 nM), shows 14-fold selectivity over JAK1/3, FLT3, induces G0/G1 arrest, apoptosis, and has antitumor effects.Formule :C26H33N7ODegré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :459.59Ref: TM-T35900
1mg138,00€5mg334,00€10mg597,00€25mg1.234,00€50mg1.648,00€100mg2.232,00€1mL*10mM (DMSO)339,00€LY3143921 hydrate
CAS :LY3143921 ((S)-Example 2) hydrate is an orally active CDC7 kinase inhibitor with broad in vitro anticancer activity [1].Formule :C16H14FN5O2Degré de pureté :98.43%Couleur et forme :SolidMasse moléculaire :327.3110-Methoxycamptothecin
CAS :10-Methoxycamptothecin is a natural bioactive derivative of camptothecin (CPT) isolated from Camptotheca acuminata and possesses high anti-cancer properties.Formule :C21H18N2O5Degré de pureté :98.36%Couleur et forme :SolidMasse moléculaire :378.38(E/Z)-GSK5182
CAS :GSK5182 is a racemic mix of (E/Z) isomers, a selective ERRγ inverse agonist (IC50: 79 nM), and induces ROS in liver cancer.Formule :C27H31NO3Degré de pureté :97.58%Couleur et forme :SolidMasse moléculaire :417.54Ref: TM-T7709
1mg77,00€5mg167,00€10mg260,00€25mg477,00€50mg707,00€100mg1.063,00€1mL*10mM (DMSO)177,00€TGFβRI-IN-3
CAS :TGFβRI-IN-3 inhibits TGFβR1 with an IC 50 of 0.79 nM with 2000-fold selectivity against MAP4K4.Formule :C28H23N3O2SDegré de pureté :99.85%Couleur et forme :SoildMasse moléculaire :465.57Ref: TM-T9523
1mg84,00€5mg177,00€10mg281,00€25mg552,00€50mg859,00€100mg1.234,00€500mg2.457,00€1mL*10mM (DMSO)177,00€Rolapitant hydrochloride
CAS :Rolapitant HCl is a potent NK1 antagonist, non-CYP3A4 interactive, with anti-emetic effects and a Ki of 0.66 nM.Formule :C25H27ClF6N2O2Degré de pureté :98.35% - 99.79%Couleur et forme :SolidMasse moléculaire :536.94Ref: TM-T3724
1mg153,00€5mg365,00€10mg520,00€25mg780,00€50mg1.054,00€100mg1.425,00€200mg1.882,00€1mL*10mM (DMSO)439,00€PD 151746
CAS :PD151746: calpain inhibitor, Ki μ-calpain=0.26μM, Ki m-calpain=5.33μM; reduces oxLDL cytotoxicity.Formule :C11H8FNO2SDegré de pureté :98.63% - ≥95%Couleur et forme :SolidMasse moléculaire :237.25Gemcitabine elaidate hydrochloride
CAS :CP-4126, a lipophilic pro-drug of Gemcitabine, converts to active form by esterases, allowing oral administration with dose-dependent effects.
Formule :C27H44ClF2N3O5Degré de pureté :98.50% - 99.6%Couleur et forme :SolidMasse moléculaire :564.11Durlobactam sodium salt
CAS :Durlobactam sodium salt (ETX2514) have an IC50 values of 4, 14 and 190 nM against class A KPC-2, class C AmpC and class D OXA-24.Cost-effective and quality-assured.Formule :C8H10N3NaO6SDegré de pureté :97.01% - 99.03%Couleur et forme :SolidMasse moléculaire :299.23FGI-106 tetrahydrochloride
CAS :FGI-106 tetrahydrochloride demonstrates potent inhibitory activity across a broad spectrum of viruses, including those causing hemorrhagic fevers such as EbolaFormule :C28H42Cl4N6Degré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :604.48Ref: TM-T11281L
1mg82,00€5mg161,00€10mg245,00€25mg406,00€50mg572,00€100mg772,00€200mg1.035,00€1mL*10mM (DMSO)207,00€Rineterkib
CAS :Rineterkib (ERK-IN-1) is an inhibitor of RAF and ERK1/2 activating mutations in the MAPK pathway.Formule :C26H27BrF3N5O2Degré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :578.42Ref: TM-T11224
1mg87,00€5mg170,00€10mg318,00€25mg538,00€50mg765,00€100mg1.035,00€1mL*10mM (DMSO)224,00€SR 11302
CAS :SR 11302 is an inhibitor of activator protein-1 (AP-1).Formule :C26H32O2Degré de pureté :98.65%Couleur et forme :SolidMasse moléculaire :376.53Ref: TM-T23384
1mg93,00€5mg137,00€10mg205,00€25mg356,00€50mg587,00€100mg888,00€1mL*10mM (DMSO)150,00€LSZ-102
CAS :LSZ-102 is an effective and selective degrader of estrogen receptor (IC50 = 0.2 nM) and can be used in studies about ERα positive breast cancer.Formule :C25H17F3O4SDegré de pureté :98.56%Couleur et forme :SolidMasse moléculaire :470.46Sebetralstat
CAS :Sebetralstat (KVD900) is an inhibitor of plasma kallikrein and can be used in studies about metabolic diseases.
Formule :C26H26FN5O4Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :491.51INCB086550
CAS :INCB086550 (PD-1/PD-L1-IN-8) (example 24) is a PD-1/PD-L1 inhibitor, with an IC50 <= 10 nM.Formule :C41H39N7O4Degré de pureté :98.49%Couleur et forme :SolidMasse moléculaire :693.79FX-11
CAS :FX-11: potent LDHA inhibitor (Ki 8 μM), activates PKM2, reduces ATP, induces oxidative stress/ROS, cell death, shows antitumor effects.Formule :C22H22O4Degré de pureté :98.95% - 98.95%Couleur et forme :SolidMasse moléculaire :350.41Clorophene
CAS :Clorophene (Clorofene) is an antimicrobial agent and can be used in personal care products.Formule :C13H11ClODegré de pureté :99.87%Couleur et forme :White To Light Tan Or Pink Flakes Phenolic Odor (Ntp 1992)Masse moléculaire :218.68GAS6 Protein, Human, Recombinant (His)
GAS6 (Growth arrest-specific protein 6) is also known as AXL receptor tyrosine kinase ligand, AXLLG, is a multimodular protein that is up-regulated by a wide variety of cell types in response to growth arrest. Gas6 binds and induces signaling through the receptor tyrosine kinases Axl, Dtk, and Mer whose signaling is implicated in cell growth and survival, cell adhesion and cell migration. GAS6/AXL signaling plays a role in various processes such as endothelial cell survival during acidification by preventing apoptosis, optimal cytokine signaling during human natural killer cell development, hepatic regeneration, gonadotropin-releasing hormone neuron survival and migration, platelet activation, or regulation of thrombotic responses. GAS6 Protein, Human, Recombinant (His) is expressed in HEK293 cells.
Degré de pureté :＞99.90%Couleur et forme :SoildMasse moléculaire :72.7 KDa (Predicted), 80-90 KDa (Reducing conditions)TCblR Protein, Human, Recombinant (His)
TCblR Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with C-6xHis tag. The predicted molecular weight is 32-58 KDa and the accession number is Q9NPF0.
Couleur et forme :SolidMasse moléculaire :32-58 KDa (reducing condition)TEM1/CD248 Protein, Mouse, Recombinant (His)
TEM1/CD248 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with C-His tag. The predicted molecular weight is 73.6 kDa and the accession number is Q91V98.
Couleur et forme :SolidMasse moléculaire :73.6 kDa (predicted). Due to glycosylation, the protein migrates to 75-140 kDa based on Tris-Bis PAGE result.EGFR-IN-7
CAS :EGFR-IN-7 (TQB3804) is a selective and potent EGFR kinase inhibitor.
Formule :C32H41BrN9O2PDegré de pureté :95.32% - 99.64%Couleur et forme :SolidMasse moléculaire :694.64-Ethoxycoumarin
CAS :4-Ethoxycoumarin has antimicrobial activity.
Formule :C11H10O3Degré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :190.2(-)-Isopulegol
CAS :Isopulegol has antioxidant, and neuroactive properties. It also has gastroprotective effects induced by isopulegol appear to be mediated, at least in part, by endogenous prostaglandins, K+ATP channel opening and antioxidant proprieties related to GSH increased.
Formule :C10H18ODegré de pureté :99.89%Couleur et forme :LiquidMasse moléculaire :154.25α-Terpineol
CAS :Terpineol possesses antifungal activity against Trichophyton mentagrophytes, it also exhibits strong antimicrobial activity against periodontopathic and cariogenic bacteria. α-Terpineol (Terpineol) shows anticonvulsant, and anti-inflammatory activities, it inhibits the gene expression of the IL-6 receptor.
Formule :C10H18ODegré de pureté :97.55%Couleur et forme :Colorless LiquidMasse moléculaire :154.252'-Hydroxy-4'-methylacetophenone
CAS :2'-Hydroxy-4'-methylacetophenone, a phenolic compound isolated from Angelicae koreana roots possesses acaricidal property. 2'-Hydroxy-4'-methylacetophenone has acaricidal activity, it could be used in the preparation of 4'-methyl-2'-[(p-tolylsulfonyl) oxy] acetophenone.
Formule :C9H10O2Degré de pureté :99.88%Couleur et forme :Black LiquidMasse moléculaire :150.17Anisylacetone
CAS :Anisylacetone (Anisylacetone) is an effective lure for the male melon fly.
Formule :C11H14O2Degré de pureté :99.74%Couleur et forme :LiquidMasse moléculaire :178.23Relacorilant
CAS :Relacorilant is an oral glucocorticoid receptor antagonist with Ki of 7.2 nM, potential for treating Cushing's syndrome.
Formule :C27H22F4N6O3SDegré de pureté :98.53% - 99%Couleur et forme :SolidMasse moléculaire :586.56Ref: TM-T16727
Produit arrêté3-Acetylcoumarin
CAS :3-Acetylcoumarin as a practical ligand for copper-catalyzed CN coupling reactions at room temperature. It has neuroprotective and acaricidal properties.
Formule :C11H8O3Degré de pureté :99.41%Couleur et forme :Yellow Crystalline PowderMasse moléculaire :188.183-Methoxyphenylacetic acid
CAS :3-Methoxyphenylacetic acid belongs to the class of organic compounds known as anisoles. 3-Methoxyphenylacetic acid is slightly soluble (in water) and a weakly acidic compound (based on its pKa).3-Methoxyphenylacetic acid (m-Methoxyphenylacetic acid), a m-hydroxyphenylacetic acid (m-OHPAA) derivative, is a phytotoxin in Rhizoctonia solani. 3-Methoxyphenylacetic acid is used to develop a toxin-mediated bioassay for resistance to rhizoctonia root rot
Formule :C9H10O3Degré de pureté :98.61%Couleur et forme :White SolidMasse moléculaire :166.17PRGL493
CAS :PRGL493 blocks ACSL4, halts PC3/MDA-MB-231 cancer cell spread, and inhibits MA-10 tumor progesterone. Effective in mouse PC3 tumor model at 0.25 mg/kg.Formule :C25H21N7O2Degré de pureté :98.80% - 99.11%Couleur et forme :SolidMasse moléculaire :451.48PD-1/PD-L1-IN 5 TFA
CAS :PD-1/PD-L1-IN 5 is an inhibitor of PD-1/PD-L1 protein/protein interaction (IC50 of ≤100 nM).
Formule :C22H18N4O3S·xC2HF3O2Degré de pureté :98%Couleur et forme :SolidCAY10736
CAS :CAY10736: Anticancer agent, blocks cell growth & migration in various cancers, effective in mouse models.
Formule :C41H59N3O3SCouleur et forme :SoildMasse moléculaire :673.99Sel-green
CAS :Sel-green: a probe for quantifying Sec in thioredoxin reductase and imaging Sec in live HepG2 cells.Formule :C19H18N4O8SCouleur et forme :SolidMasse moléculaire :462.43TSPP tetrasodium
CAS :TSPP tetrasodium, a photosensitizer, has demonstrated significant efficacy in the in vivo regression of cancer and microbial infections (Ex: 413 nm, Em: 640 nmFormule :C44H26N4Na4O12S4Couleur et forme :SolidMasse moléculaire :1022.92Fungicide5
CAS :Fungicide5 is a fungicide candidate targeting succinate dehydrogenase ( K i = 0.095 μM).
Formule :C20H13F8N3O2Couleur et forme :SolidMasse moléculaire :479.33Antiviral agent 8
CAS :Antiviral agent 8, surpassing lead compounds crocin-1 and crocin-2, has been identified as a potent and promising candidate with enhanced antiviral activities.
Formule :C36H38F2O4Couleur et forme :SolidMasse moléculaire :572.693AI3-10714
CAS :AI3-10714 is a biochemical.Formule :C14H6F17NO2SCouleur et forme :SolidMasse moléculaire :575.24MCA17-1
CAS :MCA17-1 exhibits superior bioactivity compared to the positive control, obeticholic acid (OCA), in the treatment of liver fibrosis.
Formule :C14H15NO5Couleur et forme :SolidMasse moléculaire :277.276PEG2-bis(phosphonic acid)
CAS :PEG2-bis(phosphonic acid) is a PEG Linker.Formule :C6H16O8P2Couleur et forme :SolidMasse moléculaire :278.13TLQP-21 TFA
TLQP-21 TFA is a VGF-derived peptide, C3aR1 agonist (mouse EC50: 10.3μM; human EC50: 68.8μM), that raises intracellular Ca2+ for nociception research.
Degré de pureté :98%Couleur et forme :LiquidPLK1-IN-6
PLK1-IN-6: potent, selective PLK1 inhibitor, IC50 = 0.45 nM, hinders cancer cell growth.
Formule :C28H37N9O3Couleur et forme :SolidMasse moléculaire :547.65Phosalacine
CAS :Phosalacine, isolated from Kitasatosporia phosalacinea, is a new herbicidal antibiotic that contains phosphinothricin.Formule :C14H28N3O6PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :365.367PROTAC eEF2K degrader-1
CAS :PROTAC eEF2K degrader-1 (11l) targets eEF2K, induces apoptosis in MDA-MB-231 cells, and degrades eEF2K.
Formule :C31H33N9O11Couleur et forme :SolidMasse moléculaire :707.65MRS2802
CAS :MRS2802 is a P2Y14 receptor agonist, its EC50 value for P2Y14 receptor is 63 nM.Formule :C10H14F2N2O11P2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :438.169H-L-Photo-lysine hydrochloride
H-L-Photo-lysine HCl is a diazirine lysine for site-specific protein incorporation and in vivo cross-linking.Formule :C11H21ClN4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :308.76C12 NBD Sphingomyelin
CAS :C12 NBD sphingomyelin, a fluorescent sphingomyelin derivative, serves as a sphingomyelinase substrate (Ex=470 nm, Em=525 nm).Formule :C41H73N6O9PCouleur et forme :SolidMasse moléculaire :825.03PROTAC MDM2 Degrader-2
CAS :PROTAC MDM2 Degrader-2: A potent MDM2-targeting compound with PROTAC tech for E3 ligase-mediated degradation.
Formule :C70H76Cl4N10O12Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1391.22Firefly Luciferase circRNA
Firefly Luciferase circRNA, originally isolated from Photinus pyralis (Firefly), expresses a luciferase protein and serves as an optimal marker for monitoring
Couleur et forme :Odour SolidApratoxin A
CAS :Apratoxin A is a potent cytotoxin isolated from the marine cyanobacterium Lyngbya majuscula Harvey ex Gomont.Formule :C45H69N5O8SCouleur et forme :SolidMasse moléculaire :840.13Antitubercular agent-10
CAS :Antitubercular agent-10 shows potent antitubercular activity with a MIC value of 30 nM.
Formule :C19H15N5O6S2Couleur et forme :SolidMasse moléculaire :473.48SIAIS117
CAS :SIAIS117: A Brigatinib-VHL-1 ALK PROTAC; degrades ALK G1202R, inhibits SR/H2228 cells, may fight small cell lung cancer.
Formule :C57H76ClN10O7PSCouleur et forme :SolidMasse moléculaire :1111.77Spiratisanin A
CAS :Spiratisanin A is a natural product from Spiraea japonica.
Formule :C29H40O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :436.63
