Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.687 produits)
- Apoptose(6.097 produits)
- Cycle cellulaire/point de contrôle(4.691 produits)
- Chromatine/Épigénétique(2.376 produits)
- Signalisation du cytosquelette(1.472 produits)
- Altération de l'ADN/réparation de l'ADN(2.921 produits)
- Endocrinologie/Hormones(3.611 produits)
- Enzyme(3.655 produits)
- GPCR/G-Protéine(8.755 produits)
- Immunologie et Inflammation(3.765 produits)
- Virus de la grippe(298 produits)
- Signalisation JAK/STAT(407 produits)
- Signalisation MAPK(1.230 produits)
- Transporteur membranaire/Canal ionique(2.947 produits)
- Métabolisme(9.940 produits)
- Microbiologie/Virologie(7.347 produits)
- Neuroscience(10.240 produits)
- Autres inhibiteurs(36.533 produits)
- Oxydation-Réduction(43 produits)
- Signalisation PI3K/Akt/mTOR(1.437 produits)
- Protéases/Protéasome(1.675 produits)
- Cellules souche et Dérivés(830 produits)
- Tyrosine Kinase/Adaptateurs(2.028 produits)
- Ubiquitination(1.682 produits)
Affichez 16 plus de sous-catégories
66582 produits trouvés pour "Inhibiteurs"
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Elamipretide
CAS :<p>Elamipretide (SS-31, MTP-131, Bendavia) is a mitochondria-focused peptide that curbs toxic ROS and stabilizes cardiolipin.</p>Formule :C32H49N9O5Degré de pureté :98.53% - 99.85%Couleur et forme :SolidMasse moléculaire :639.79Ref: TM-TP1095
Produit arrêtéCebranopadol
CAS :<p>Cebranopadol (GRT6005) is an analgesic NOP and opioid receptor agonist with Kis of 0.9 nM, 0.7 nM, 2.6 nM, 18 nM for human NOP, μ-opioid (MOP), κ-opioid (KOP)</p>Formule :C24H27FN2ODegré de pureté :98.32% - 99.78%Couleur et forme :SolidMasse moléculaire :378.48Ref: TM-T5167
Produit arrêtéElamipretide 2TFA
CAS :<p>Elamipretide 2TFA (RX-31 2TFA) is a novel mitochondrion-targeted antioxidant.</p>Formule :C36H51F6N9O9Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :867.84SR17018
CAS :<p>SR17018 is an mu-opioid-receptor (MOR) agonist, binding with GTPγS, with an EC50 of 97 nM.</p>Formule :C19H18Cl3N3ODegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :410.72Danoprevir sodium
CAS :<p>Danoprevir sodium is an NS3/4A protease inhibitor used in the treatment of Hepatitis C</p>Formule :C35H45FN5NaO9SCouleur et forme :SolidMasse moléculaire :753.82Salvianolic acid B
CAS :<p>Salvianolic acid B (Dan Shen Suan B) is a water-soluble antioxidant from Salvia miltiorrhiza extract with antiplatelet aggregation and antithrombotic effects.</p>Formule :C36H30O16Degré de pureté :99.75% - 99.86%Couleur et forme :Yellow SolidMasse moléculaire :718.61p-Toluic Acid
CAS :<p>p-Toluic Acid (4-Methylbenzoic acid) belongs to the class of organic compounds known as benzoic acids. 4-Methylbenzoic acid has been primarily detected in saliva. Within the cell, 4-methylbenzoic acid is primarily located in the cytoplasm.</p>Formule :C8H8O2Degré de pureté :99.44%Couleur et forme :Physical Description White Powder Sublimes (Ntp 1992)Masse moléculaire :136.157-Methoxy-1-tetralone
CAS :<p>7-Methoxy-1-tetralone may have insecticidal activity.</p>Formule :C11H12O2Degré de pureté :99.93%Couleur et forme :White CrystalMasse moléculaire :176.21Ammonium Glycyrrhizinate
CAS :<p>Ammonium Glycyrrhizinate (Glycyram) inhibits the cytopathology and growth of several unrelated DNA/RNA viruses.</p>Formule :C42H62O16·NH3Degré de pureté :98.41%Couleur et forme :SolidMasse moléculaire :839.96Praeruptorin B
CAS :<p>1. Praeruptorin B can inhibit tumor promoter induced phemonenon in vitro.</p>Formule :C24H26O7Degré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :426.46Ref: TM-T6S1423
Produit arrêtéCompound T69202(SC)
CAS :<p>NBQX (FG9202), an AMPA/kainate receptor blocker, counters glutamate toxicity; water-soluble as disodium salt, has anticonvulsant properties.</p>Formule :C12H6N4Na2O6SCouleur et forme :SolidMasse moléculaire :380.2415Sculponeatin O
CAS :<p>Sculponeatin O may have protective effects on the lipid peroxidation-damaged live cells.</p>Formule :C28H40O4Degré de pureté :95.00%Couleur et forme :SolidMasse moléculaire :440.61Pamoic acid
CAS :<p>Pamoic acid is the orphan G protein-coupled receptor GPR35 agonist. Pamoic acid activates ERK and beta-arrestin2 and causes antinociceptive activity.</p>Formule :C23H16O6Degré de pureté :99.99%Couleur et forme :Fine Yellow PowderMasse moléculaire :388.374-Methoxycoumarine
CAS :<p>4-Methoxycoumarine has antitumour effects.</p>Formule :C10H8O3Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :176.17Elamipretide Triacetate
CAS :<p>Elamipretide TriTFA, a tetrapeptide, targets mitochondria, associates with cardiolipin, studied for treating Leber's Optic Neuropathy.</p>Formule :C38H61N9O11Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :819.94Ref: TM-T8644
Produit arrêtéDimethylamine hydrochloride
CAS :<p>Dimethylamine hydrochloride, found in urine, comes from food compound TMAO and NO synthesis inhibitor ADMA, processed by DDAH enzyme.</p>Formule :C2H8ClNDegré de pureté :98% - 99.89%Couleur et forme :White Solid CrystallineMasse moléculaire :81.54Ref: TM-T5309
Produit arrêtéRosmanol
CAS :Rosmanol has antioxidant, anti-inflammatory, CNS effects; induces apoptosis in cancer cells; modulates GABAA receptors.Formule :C20H26O5Degré de pureté :98.82% - 99.79%Couleur et forme :SolidMasse moléculaire :346.42Ref: TM-T7033
Produit arrêtéEthyl 4-hydroxyphenylacetate
CAS :<p>Ethyl 4-hydroxyphenylacetate is a selective inhibitor of monoamine oxidase A.</p>Formule :C10H12O3Degré de pureté :99.89%Couleur et forme :Slightly Yellow LiquidMasse moléculaire :180.2Ref: TM-FR12415
Produit arrêtéIGFBP-1 Protein, Rat, Recombinant
<p>IGF-binding proteins prolong the half-life of the IGFs and have been shown to either inhibit or stimulate the growth promoting effects of the IGFs on cell culture. They alter the interaction of IGFs with their cell surface receptors. Promotes cell migration. IGFBP-1 Protein, Rat, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 26.9 kDa and the accession number is P21743.</p>Masse moléculaire :26.9 kDa (predicted)ARGX-112
CAS :<p>Temtokibart is a humanized IgG1 λ2 antibody that specifically targets IL22RA1, and is expressed by cells that are deficient in the glutamine synthetase gene.</p>Couleur et forme :Odour LiquidCOR-001
CAS :<p>Ziltivekimab (COR-001) is a human IL-6 antibody, lowers CRP, and may treat inflammation and heart issues in CKD.</p>Degré de pureté :95%Couleur et forme :Odour LiquidOkadaic acid
CAS :<p>Okadaic acid, a polyether marine toxin, is a highly potent and selective protein phosphatase (PP) inhibitor.</p>Formule :C44H68O13Degré de pureté :98%Couleur et forme :White Crystals Or PowderMasse moléculaire :805Ref: TM-T16381
Produit arrêtéPPARγ-IN-2
CAS :<p>"PPARγ-IN-2 (Compound 5a), a PPARγ inhibitor, exhibits an EC50 of 0.106 μM in inhibiting TG accumulation in 3T3-L1 preadipocytes.</p>Formule :C19H21N5ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :335.4CK176
CAS :CK176 is an HIV-1 inhibitor, 11x more effective than I-XW-053 in human PBMCs.Formule :C21H12IN3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :465.24KP372-1
CAS :<p>KP372-1, an Akt inhibitor, blocks PI3K signaling, arrests cell growth, and triggers apoptosis in head/neck squamous cell carcinoma.</p>Formule :C20H8N12O2Couleur et forme :SolidMasse moléculaire :448.36PS372424 HCl
CAS :<p>PS372424 activates CXCR3, triggers ERK phosphorylation, and inhibits CXCL11's effect on CD45+ cell migration in humanized mice.</p>Formule :C33H45ClN6O4Couleur et forme :SolidMasse moléculaire :625.21GR 218,231
CAS :GR 218,231 is a selective antagonist of D3 dopamine receptor.Formule :C24H33NO3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :415.59PSB-6426
CAS :PSB-6426 is the first potent and selective human nucleoside triphosphate diphosphohydrolase-2 inhibitor.Formule :C22H29N4O10PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :540.46anti-TNBC agent-2
CAS :<p>Anti-TNBC agent-2 (3j), a purine derivative, acts as an anti-triple negative breast cancer (TNBC) therapeutic.</p>Formule :C28H37ClFN7ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :542.09Pazinaclone
CAS :<p>Pazinaclone is a non-benzodiazepine (GABAA) partial agonist with sedative and anxiolytic activity.</p>Formule :C25H23ClN4O4Degré de pureté :97.79% - 99.07%Couleur et forme :SolidMasse moléculaire :478.93Trimetoquinol HCl hydrate
CAS :Trimetoquinol hydrochloride possesses differential and selective beta-adrenergic properties.Formule :C19H26ClNO6Couleur et forme :SolidMasse moléculaire :399.87DprE1-IN-8
CAS :<p>DprE1-IN-8 is a potent inhibitor of DprE1, exhibiting an IC50 of less than 0.75 μM.</p>Formule :C19H12F3N5O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :463.39SB251023
CAS :SB251023 is an agonist of β3-adrenoceptor.Formule :C28H34NO6PCouleur et forme :SolidMasse moléculaire :511.55PKUMDL-LTQ-301
CAS :PKUMDL-LTQ-301 is a potent inhibitor of HipA toxin. PKUMDL-LTQ-301 also inhibits E. coli persistence.Formule :C30H28N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :480.55DPX-3778
CAS :DPX-3778, a triethanolamine salt, boosts tobacco callus growth 4-5x at 0.124-2.48 μM and slows aging with IAA and kinetin.Formule :C16H23ClN4O6Couleur et forme :SolidMasse moléculaire :402.83EGFR-IN-82
CAS :<p>EGFR-IN-82 (Compound 8a) is a potent, orally active inhibitor of EGFR, exhibiting IC50 values of 0.09 nM for EGFR L858R/T790M/C797S and 0.06 nM for EGFR Del19/</p>Formule :C32H41BrN9O2PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :694.6Erythrityl Tetranitrate
CAS :<p>Erythrityl Tetranitrate, a vasodilator similar to nitroglycerin, was first in "sustained release" tablets; may cause "nitro headache."</p>Formule :C4H6N4O12Couleur et forme :SolidMasse moléculaire :302.11Fostedil
CAS :Fostedil enhances heart function, maintains blood flow during partial/total coronary occlusions, and lowers aortic pressure.Formule :C18H20NO3PSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :361.4YM 298198 Hydrochloride
CAS :YM 298198 HCl: non-competitive mGlu1 antagonist, Ki=19 nM. Inactive on mGlu2-7, stronger than CPCCOEt.Formule :C18H22N4OSCouleur et forme :SolidMasse moléculaire :342.46Lp-PLA2-IN-16
CAS :<p>Lp-PLA2-IN-16 (Example 1) is an inhibitor of lipoprotein-associated phospholipase A2 (Lp-PLA2) with potential applications in Alzheimer's disease research [1].</p>Formule :C22H17F5N4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :480.39Anti-NASH agent 1
CAS :<p>Anti-NASH Agent 1 (Compound 3d), derived from Elafibranor, serves as a strong PPAR-α/δ agonist aimed at treating nonalcoholic steatohepatitis (NASH).</p>Formule :C26H33NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :423.54Oxitropium Bromide
CAS :Oxitropium bromide, a mAChR blocker, treats asthma and COPD as an anticholinergic bronchodilator.Formule :C19H26BrNO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :412.32(E)-Crotylbarbital
CAS :<p>(E)-Crotylbarbital, a Crotylbarbital isomer, is a sedative with hypnotic, anticonvulsant properties, aiding sleep and mental stability.</p>Formule :C10H14N2O3Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :210.23Ref: TM-T10002
Produit arrêtéFotemustine
CAS :<p>Fotemustine: antineoplastic, chloroethylates DNA, blocks synthesis, causes cell arrest/apoptosis, lipophilic, crosses blood-brain barrier.</p>Formule :C9H19ClN3O5PCouleur et forme :SolidMasse moléculaire :315.69PL265
CAS :<p>PL265 is a long-acting dual ENKephalinase inhibitor (DENKi) with analgesic potential.</p>Formule :C27H35N2O9PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :562.55Phenazolam
CAS :<p>Phenazolam is an analytical reference standard categorized as a benzodiazepine. [1] This product is intended for research and forensic applications.</p>Formule :C17H12BrClN4Couleur et forme :SolidMasse moléculaire :387.66Mavodelpar free base
CAS :<p>Mavodelpar free acid (REN001 free acid) is an selective agonist of PPARδ.</p>Formule :C31H30FNO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :515.57BChE-IN-17
CAS :<p>BChE-IN-17 (compound 6n) is a potent, selective inhibitor of butyrylcholinesterase (BChE), demonstrating inhibitory half-maximal inhibitory concentrations (</p>Formule :C23H23BrN2O4S2Couleur et forme :SolidMasse moléculaire :535.47HBV-IN-34
CAS :<p>HBV-IN-34 (compound 17i) is a potent inhibitor of HBsAg production, demonstrating remarkable in vitro anti-HBV efficacy with EC50 values of 0.018 μM for HBV DNA</p>Formule :C21H19F2N7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :407.42Dioxifedrine
CAS :Dioxifedrine is a beta-2 -adrenergic agonist with bronchodilator activity.Formule :C10H15NO3Couleur et forme :SolidMasse moléculaire :197.23Cebranopadol ((1α,4α)stereoisomer)
CAS :<p>Cebranopadol ((1α,4α)stereoisomer) is a stereoisomer of cebranopadol which is a potent ORL-1 agonist.</p>Formule :C24H27FN2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :378.48Saxitoxinol
CAS :<p>Saxitoxinol is an analog of saxitoxin, a known voltage-gated sodium channel blocker.</p>Formule :C10H17N7O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :283.29Fosfonet sodium
CAS :Fosfonet sodium is a sodium salt of phosphonoacetic acid, effective against herpesviruses by inhibiting viral DNA polymerase.Formule :C2H4NaO5PCouleur et forme :SolidMasse moléculaire :162.01Neurokinin antagonist 1
CAS :<p>Neurokinin antagonist 1 is a potent is a neuropeptide antagonist that can be used to study neurological disorders.</p>Formule :C38H40N4O3Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :600.75CGP 44532
CAS :CGP 44532 a GABAB receptor agonist.Formule :C4H12NO3PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :153.12Lp-PLA2-IN-12
CAS :<p>Lp-PLA2-IN-12 (compound 19), an Lp-PLA2 inhibitor, is utilized in researching neurodegenerative diseases including Alzheimer's disease (AD), glaucoma, age-</p>Formule :C24H23F2N5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :467.47UBP1112
CAS :group III mGlu receptor antagonistFormule :C10H14NO5PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :259.2CH-100
CAS :CH-100 is a Chinese herbal medicine previously used in the treatment of human hepatitis C.Formule :C14H22ClNO3Couleur et forme :SolidMasse moléculaire :287.78Ceronapril
CAS :Ceronapril (SQ 29852) is an orally active and potent angiotensin-converting enzyme (ACE) inhibitor (IC50 : 36 nM) for the study of dementia and hypertension.Formule :C21H33N2O6PDegré de pureté :97.94%Couleur et forme :SolidMasse moléculaire :440.47Culmerciclib
CAS :<p>Culmerciclib is a cell cycle protein-dependent kinase (CDK) inhibitor that exhibits antitumour effects.</p>Formule :C24H27FN8Couleur et forme :SolidMasse moléculaire :446.52FGFR1 inhibitor-10
CAS :<p>FGFR1 inhibitor-10 (Compound 4i), with an IC50 of 28 nM, effectively inhibits FGFR1 phosphorylation.</p>Formule :C26H30F3N7O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :561.62H 35-25
CAS :H 35-25 is a beta 2-antagonist.Formule :C13H21NOCouleur et forme :SolidMasse moléculaire :207.31KBP-7018
CAS :<p>KBP-7018: potent tyrosine kinase inhibitor targeting c-KIT, RET, PDGFR with IC50s of 10, 7.6, 25nM.</p>Formule :C31H30N4O5Couleur et forme :SolidMasse moléculaire :538.59Radafaxine hydrochloride
CAS :<p>Radafaxine hydrochloride is an inhibitor of DAT and NET transporters, and nAChR family modulator.</p>Formule :C13H19Cl2NO2Degré de pureté :98%Masse moléculaire :292.2anti-TNBC agent-3
CAS :<p>Anti-TNBC agent-3 (compound 3g) is a compound that induces apoptosis and possesses anti-cancer cell proliferation properties.</p>Formule :C29H39F2N7OCouleur et forme :SolidMasse moléculaire :539.66FM-24 HCl
CAS :FM-24 HCl is a long acting beta-adrenergic receptor antagonist.Formule :C19H30ClNO2Couleur et forme :SolidMasse moléculaire :339.9Benzovindiflupyr
CAS :<p>Benzovindiflupyr: a fungicide that inhibits SDH (IC50=5.2nM), halts S. sclerotiorum growth (EC50=0.011μg/ml), and protects crops like eggplants.</p>Formule :C18H15Cl2F2N3OCouleur et forme :SolidMasse moléculaire :398.23Gacyclidine
CAS :Gacyclidine (OTO311), an NMDA receptor blocker, treats tinnitus and injuries in the brain and spinal cord.Formule :C16H25NSDegré de pureté :99.85% - 99.92%Couleur et forme :SolidMasse moléculaire :263.44MEN11467
CAS :MEN11467 is a novel, orally available, potent and selective peptidomimetic tachykinin NK 1 receptor antagonist for the study of acute colon cancer.Formule :C38H40N4O3Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :600.75Glutaminyl Cyclase Inhibitor 4
CAS :Glutaminyl Cyclase Inhibitor 4 is a potent, selective glutaminyl cyclase (QC) inhibitor (IC50: 6.1 nM). It is a potent anti-Alzheimer’s agent.Formule :C22H33N5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :415.53Lp-PLA2-IN-15
CAS :<p>Lp-PLA2-IN-15 (example 2) is an inhibitor of lipoprotein-associated phospholipase A2 (Lp-PLA2) with potential application in Alzheimer's disease research [1].</p>Formule :C22H17F5N4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :480.39Albuterol stearate
CAS :<p>Albuterol stearate, a salt form of Albuterol, is a selective beta2 agonist for treating asthma and COPD, with 29x preference for beta2 over beta1.</p>Formule :C31H57NO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :523.799BET-IN-15
CAS :<p>BET-IN-15 (compound 1) is a potent, orally active inhibitor of BET, demonstrating inhibitory IC50 values of 0.64 nM for BRD4-BD1 and 0.25 nM for BRD4-BD2.</p>Formule :C21H18F2N4O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :444.45CXCR4-IN-1
CAS :<p>CXCR4-IN-1 (Example C5), with an IC50 of 20 nM, is a potent inhibitor of CXCR4, applicable for the research of various conditions such as cancer, HIV, diabetic</p>Formule :C23H32N6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :392.54Bromadoline maleate
CAS :<p>Bromadoline is an opioid analgesic selective for the μ-opioid receptor.</p>Formule :C19H25BrN2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :441.322D(-)-Octopamine CSA salt
CAS :D(-)-Octopamine CSA salt is an agonist of octopamine receptors.Formule :C18H27NO6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :385.48Aminobutane bisphosphonate
CAS :Aminobutane bisphosphonate curbs bone loss; may manage hypercalcemia in cancer.Formule :C4H13NO6P2Couleur et forme :SolidMasse moléculaire :233.1IDX-375
CAS :IDX-375, a HCV NS5B polymerase inhibitor, is used potentially for the treatment of HCV infection.Formule :C29H50N5O7PSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :643.78AMPK activator C2
CAS :AMPK activator C2 is an AMPK allosteric activator.Formule :C7H6NO6PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :231.1SR14150
CAS :<p>SR14150 is a partial agonist of high-affinity NOP receptor.</p>Formule :C21H30N2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :326.48AKOS-22
CAS :<p>AKOS-22: potent VDAC1 inhibitor, Kd=15.4 μM; prevents mitochondrial dysfunction and apoptosis.</p>Formule :C22H21ClF3N3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :467.87ALPK1-IN-1
CAS :<p>ALPK1-IN-1 (A001) strongly inhibits ALPK1, key for innate immunity & NF-κB signaling via TIFA/TRAF.</p>Formule :C25H32N6O2SCouleur et forme :SolidMasse moléculaire :480.63Questiomycin A derivatives 18 TFA
<p>Questiomycin A derivative 18 TFA exhibits antibacterial, anticancer properties and inhibits GRP78.</p>Formule :C16H12F3N3O5Degré de pureté :98.45%Couleur et forme :SoildMasse moléculaire :383.07HPK1-IN-18
CAS :<p>HPK1-IN-18: Potent, specific inhibitor of HPK1, a MAP4K enzyme, for cancer research and treatment.</p>Formule :C24H24N4Couleur et forme :LiquidMasse moléculaire :368.47PAD4-IN-2
CAS :<p>PAD4-IN-2 (compound 5i) is a PAD4 inhibitor with an IC50 value of 1.94 μM, shown to suppress tumor growth in mice through specific inhibition of the PAD4-H3cit-</p>Formule :C20H23BClN7O6Couleur et forme :SolidMasse moléculaire :503.7ALPK1-IN-2
CAS :<p>ALPK1-IN-2 is a potent inhibitor of ALPK1 (α-kinase 1) (IC50: 95 nM). ALPK1-IN-2 inhibits NF-κB (IC50: 1.31 μM).</p>Formule :C20H18F2N4O2SCouleur et forme :SolidMasse moléculaire :416.44MitoE10
CAS :MitoE10 is an effective mitochondrial targeting antioxidant.Formule :C42H55O5PSCouleur et forme :SolidMasse moléculaire :702.92JAK2-IN-9
CAS :<p>Compound A8, known as JAK2-IN-9, is a selective JAK2 inhibitor with an IC50 of 5 nM.</p>Formule :C20H24N6O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :412.51Civorebrutinib
CAS :<p>Civorebrutinib (WS-413) is an inhibitor of Bruton's tyrosine kinase that exhibits antineoplastic activity [1].</p>Formule :C23H22ClN7O2Couleur et forme :SolidMasse moléculaire :463.92Antitumor agent-104
CAS :<p>Antitumor Agent-104 (Compound 9) serves as an antineoplastic by impeding DNA repair mechanisms in tumor cells, primarily through the inhibition of PARP1 enzyme</p>Formule :C31H33FN6O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :556.63MDVN1003
CAS :MDVN1003 inhibits BTK & PI3Kδ in B cells, blocking NHL growth; it kills lymphoma cells, not erythroblasts.Formule :C22H20FN7ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :417.44Estrogen receptor modulator 8
CAS :<p>Estrogen Receptor Modulator 8 (compound 4) is an orally active inhibitor targeting Estrogen Receptor/ERR α with potent efficacy (IC50 = 0.437 nM in MCF-7 cells</p>Formule :C25H24F4N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :460.46BET-IN-14
CAS :<p>BET-IN-14 is a pan BET inhibitor with an IC50 of 5.35 nM, demonstrating oral activity and anticancer properties [1].</p>Formule :C30H37N7O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :527.66Mal-cyclohexane-Gly-Gly-Phe-Gly-Exatecan
CAS :<p>Mal-cyclohexane-Gly-Gly-Phe-Gly-Exatecan is a linker molecule employed in the synthesis of antibody-drug conjugates (ADCs), demonstrating potent antitumor</p>Formule :C55H60FN9O13Couleur et forme :SolidMasse moléculaire :1074.12BCR-ABL-IN-8
CAS :<p>BCR-ABL-IN-8 (compound 26f) is a BCR-ABL inhibitor featuring a trimethoxy group [1].</p>Formule :C30H33N7O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :571.63Bumetanide sodium
CAS :Bumetanide sodium, a potent diuretic, blocks NKCC1 (IC50: 0.68 μM) and NKCC2 (IC50: 4.0 μM).Formule :C17H19N2NaO5SCouleur et forme :SolidMasse moléculaire :386.4Antitumor photosensitizer-2
CAS :<p>Compound 11, also known as Antitumor Photosensitizer-2, is a potent photosensitizer with remarkable photodynamic anti-tumor properties and minimal skin photo-</p>Formule :C40H47N5O7Couleur et forme :SolidMasse moléculaire :709.83PI3Kδ-IN-13
CAS :<p>PI3Kδ-IN-13 (compound 89), with an IC50 value of 2.6 nM, is an inhibitor of PI3Kδ, applicable for researching diseases involving cell proliferation, including</p>Formule :C27H39N7O4S2Couleur et forme :SolidMasse moléculaire :589.77Antibacterial agent 160
CAS :<p>Antibacterial Agent 160 is a potent antibacterial agent that rapidly eradicates bacteria and inhibits the formation of bacterial biofilms.</p>Formule :C29H27ClFN3O6Couleur et forme :SolidMasse moléculaire :567.99Py-MAA-Val-Cit-PAB-MMAE
CAS :<p>Py-MAA-Val-Cit-PAB-MMAE (AAJ8D6-PY-Val-Cit-MMAE) serves as an ADC linker for Zapadcine-3a, a broad-spectrum anti-TRAILR2 ADC with antineoplastic properties.</p>Formule :C72H111N13O16SCouleur et forme :SolidMasse moléculaire :1446.79FAP-IN-2
CAS :<p>FAP-IN-2 is a 99mTc-labeled, isonitrile-containing derivative of a fibroblast activation protein (FAPI) inhibitor suitable for tumor imaging [1].</p>Formule :C24H28F2N6O3Couleur et forme :SolidMasse moléculaire :486.51IDO/Tubulin-IN-2
CAS :<p>IDO/Tubulin-IN-2 inhibits TDO/tubulin, effective on U87, HepG2, A549, HCT-116, LO2 cancer cells; IC50 values 0.036-1.04 μM, boosts antitumor action.</p>Formule :C48H40N6O10Couleur et forme :SolidMasse moléculaire :860.87BTK-IN-25
CAS :<p>BTK-IN-25 (compound 71) is a potent BTK inhibitor, demonstrating an IC50 of 0.77 nM against BTK(C481S) and achieving an IC50 of 1 nM in DOHH2 cells [1].</p>Formule :C28H27F2N3O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :523.53SHP2-IN-14
CAS :<p>SHP2-IN-14 (compound 27) is a potent, orally active allosteric inhibitor of SHP2, displaying strong anti-tumor activity with an IC50 of 7 nM.</p>Formule :C22H20Cl2N8OCouleur et forme :SolidMasse moléculaire :483.35EST73502
CAS :<p>EST73502 is a compound that functions as a dual agonist for the μ-opioid receptor (MOR) and an antagonist for the σ1 receptor (σ1R). It is selective, orally active, and possesses the ability to penetrate the blood-brain barrier (BBB). The compound exhibits a Ki value of 64 nM for the MOR and 118 nM for the σ1R. Additionally, EST73502 demonstrates antinociceptive activity [1].</p>Formule :C19H26F2N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :352.426JDB175
CAS :<p>JDB175, a selective BTK inhibitor with oral bioavailability, demonstrates excellent penetration through the blood-brain barrier.</p>Formule :C26H21F3N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :478.47Davelizomib
CAS :<p>Davelizomib is a proteasome inhibitor that exhibits antineoplastic activity [1].</p>Formule :C21H26BF2N3O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :481.25TrkB-IN-1
CAS :<p>TrkB-IN-1 is a potent, orally active agonist of the TrkB receptor, with favorable pharmacokinetic (PK) properties.</p>Formule :C19H16N2O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :368.34L 689037
CAS :L 689037 is an inhibitor of leukotriene biosynthesis.Formule :C36H37ClN2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :597.14APG-2449
CAS :<p>APG-2449 is an orally active inhibitor targeting ALK, ROS1, and FAK, demonstrating antitumor efficacy in mouse models of non-small cell lung cancer (NSCLC) [1].</p>Formule :C33H42ClN5O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :640.24CIAC001
CAS :<p>CIAC001, a pyruvate kinase PKM2 inhibitor, exhibits anti-neuroinflammatory properties.</p>Formule :C20H25N3O2Couleur et forme :SolidMasse moléculaire :339.43YK-029A
CAS :<p>YK-029A, an orally active EGFR mutant inhibitor, targets both EGFR T790M and EGFRex20ins mutations.</p>Formule :C27H32N8O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :500.6I-BET282
CAS :<p>BET-IN-1 is a bromodomain inhibitor extracted from patent WO/2013024104A1 (example 2, plC50: 6.0 - 7.0).</p>Formule :C25H30N4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :450.53JAK1-IN-10
CAS :<p>JAK1-IN-10 (compound 9), a cyano-substituted cyclic hydrazine derivative, functions as a potent and selective inhibitor of JAK1 [1].</p>Formule :C15H17N7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :295.34Syk-IN-8
CAS :<p>Syk-IN-8 (compound 19q) functions as a Syk inhibitor with demonstrated antiproliferative effects on a variety of hematological tumor cells.</p>Formule :C23H26N10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :442.52Omeprazole acid
CAS :Omeprazole treats GERD, ulcers, Zollinger-Ellison syndrome, prevents GI bleeding; it's a proton pump inhibitor.Formule :C34H32N6Na2O10S2Couleur et forme :SolidMasse moléculaire :794.76I5B2
CAS :<p>I5B2 is a novel phosphorus-containing angiotensin I converting enzyme inhibitor. Angiotensin I converting enzyme is produced by Actinomadura sp.</p>Formule :C23H32N3O7PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :493.49Belfosdil
CAS :Belfosdil is a blocker of antihypertensive calcium channel.Formule :C27H50O7P2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :548.63Cap-dependent endonuclease-IN-9
CAS :<p>Cap-dependent endonuclease-IN-9, a strong influenza inhibitor, shows low toxicity, good pharmacokinetics, and dynamic action.</p>Formule :C29H22F2N4O7SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :608.57CGP 56999A
CAS :CGP 56999A is a GABA(B) receptor antagonist; it boosts BDNF and reduces dopamine loss in rat striatum.Formule :C19H30NO5PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :383.42Antitumor photosensitizer-1
CAS :<p>Antitumor Photosensitizer-1 (Compound 8) is a potent photosensitizer with remarkable photodynamic anti-tumor properties and minimal skin photo-toxicity,</p>Formule :C42H51N5O6Couleur et forme :SolidMasse moléculaire :721.88FLT3-IN-19
CAS :<p>FLT3-IN-19 (Comp 50) is a potent, selective inhibitor of FLT3, demonstrating an IC50 value of 0.213 nM, and is applicable in research pertaining to acute</p>Formule :C22H26N8OCouleur et forme :SolidMasse moléculaire :418.49IDO1-IN-22
CAS :<p>IDO1-IN-22 (Compound 3) is an inhibitor of IDO1, demonstrating potent activity with biochemical hIDO1 IC50 of 67.4 nM and HeLa hIDO1 IC50 of 17.6 nM.</p>Formule :C12H12BrFN6O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :387.16URAT1 inhibitor 5
CAS :<p>URAT1 Inhibitor 5 (compound 16) serves as a powerful inhibitor of URAT1 and is utilized in hyperuricemia research [1].</p>Formule :C18H14BrN3O2SCouleur et forme :SolidMasse moléculaire :416.29LT-540-717
CAS :<p>LT-540-717 (compound 32), a potent FLT3 inhibitor (IC50=0.62 nM), exhibits antiproliferative activity and effectively inhibits various acquired FLT3 mutations,</p>Formule :C24H24N8O2Couleur et forme :SolidMasse moléculaire :456.5JAK1-IN-11
CAS :<p>JAK1-IN-11 (compound 11) serves as a potent inhibitor of Janus kinases, exhibiting nanomolar inhibitory concentrations with IC50 values of 0.02 nM (JAK1) and 0.</p>Formule :C26H36N6O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :528.67STAT3-IN-18
CAS :<p>STAT3-IN-18 (compound SPP), a platinum (IV) complex featuring an axial ligand from sandalwood, suppresses the JAK2-STAT3 pathway in breast cancer (BC) cells and</p>Formule :C18H24Cl2N2O6PtDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :630.38DDO-2213
CAS :<p>DDO-2213 is a potent, orally active inhibitor of the WDR5-MLL1 interaction, demonstrating an IC50 of 29 nM and a Kd of 72.9 nM against WDR5.</p>Formule :C24H27ClFN7OCouleur et forme :SolidMasse moléculaire :483.97BTK-IN-27
CAS :<p>BTK-IN-27 (example 8), a potent BTK inhibitor with an IC50 of 0.2 nM, demonstrates anti-proliferative effects in TMD8 cells with an IC50 of less than 5 nM.</p>Formule :C31H35N7O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :537.66URAT1&XO inhibitor 1
CAS :<p>URAT1&XO Inhibitor 1 (compound 29) serves as a dual inhibitor with IC50 values of approximately 10 μM for URAT1 and 1.01 μM for Xanthine Oxidase.</p>Formule :C20H13N5O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :403.41And1-IN-1
CAS :<p>And1-IN-1, also known as compound III, is a potent inhibitor of And1 [1].</p>Formule :C15H11BCl2O2Couleur et forme :SolidMasse moléculaire :304.96Tibremciclib
CAS :<p>Tibremciclib is a cyclin-dependent kinase 4 (CDK4) inhibitor that exhibits antineoplastic properties [1].</p>Formule :C28H32F2N8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :518.6HPK1-IN-38
CAS :<p>HPK1-IN-38 (compound 15) is an inhibitor of MAP4K1/HPK1, suitable for research into disorders related to HPK1 [1].</p>Formule :C29H29N5O3Couleur et forme :SolidMasse moléculaire :495.57FOXM1-IN-2
CAS :<p>FOXM1-IN-2, a FOXM1 inhibitor, exhibits antineoplastic activity [1].</p>Formule :C48H47F4N7O12SCouleur et forme :SolidMasse moléculaire :1021.99Insecticidal agent 6
CAS :<p>Compound Im (Insecticidal agent 6) is a potent inhibitor of insect ryanodine receptors (RyRs), exhibiting an EC50 of 0.6308 µM against S.</p>Formule :C19H14BrCl2N5O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :527.16MDL-811
CAS :<p>MDL-811, an allosteric activator of SIRT6, markedly enhances the deacetylation of histone H3 at lysine residues 9, 18, and 56 (H3K9Ac, H3K18Ac, and H3K56Ac),</p>Formule :C25H25BrCl2FN3O5S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :681.42JAK-IN-27
CAS :<p>JAK-IN-27, also known as compound 1, is an orally active, potent inhibitor of the JAKS family kinases, displaying inhibitory concentrations (IC50s) of 3.0 nM</p>Formule :C20H21F2N7ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :413.42diMal-O-CH2COOH
CAS :<p>DiMal-O-CH2COOH is a cleavable linker utilized in antibody-drug conjugates (ADCs).</p>Formule :C13H12N2O7Couleur et forme :SolidMasse moléculaire :308.24AEF0117
CAS :<p>AEF0117 is a signaling inhibitor of CB1-SSi that inhibits cannabinoid self-administration and can be used to study cannabis withdrawal.</p>Formule :C29H40O3Degré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :436.63Ref: TM-T79909
Produit arrêtéBi-Mc-VC-PAB-MMAE
CAS :<p>Bi-Mc-VC-PAB-MMAE is an agent-linker conjugate for antibody-drug conjugates (ADCs), featuring the linker (Fmoc-Val-Cit-PAB) and the potent tubulin inhibitor (</p>Formule :C71H104N12O18Couleur et forme :SolidMasse moléculaire :1413.66(αR)-Cyclopropaneacetamide-Exatecan
CAS :<p>(αR)-Cyclopropaneacetamide-Exatecan (compound 2-A), an Exenotecan derivative, serves as a cytotoxic agent that effectively inhibits the proliferation of U87MG</p>Formule :C29H28FN3O6Couleur et forme :SolidMasse moléculaire :533.55VISTA-IN-2
CAS :<p>VISTA-IN-2 (Compound 1) is a V-domain Ig suppressor of T-cell activation (VISTA) inhibitor that promotes the degradation of VISTA in cells via autophagy,</p>Formule :C23H23N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :357.45S1P1 agonist 6
CAS :<p>Compound I (S1P1 agonist 6) is an S1P1 agonist that mitigates autoimmune activity by inhibiting lymphocyte trafficking and has potential as an immunosuppressive</p>Formule :C25H26F3NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :445.47DPP
CAS :<p>DPP, a Platinum(IV) complex with a pterostilbene-derived axial ligand, inhibits the JAK2-STAT3 pathway in breast cancer (BC) cells, demonstrating</p>Formule :C36H40Cl2N2O10PtDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :926.7LFS-1107
CAS :<p>LFS-1107, a reversible CRM1 inhibitor (Kd: 12.5 pM), selectively targets and eliminates ENKTL cells, offering potential for cancer research applications [1].</p>Formule :C12H11N5OS2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :305.38MOR agonist-1
CAS :<p>MOR Agonist-1 is a μ-opioid receptor (MOR) agonist noted for its potent analgesic properties and is utilized in research concerning pain and associated</p>Formule :C22H26ClFN2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :404.91Antibacterial agent 157
CAS :<p>Compound B12 (Antibacterial agent 157) is a fungicidal agent that can impact protein synthesis in Botrytis cinerea.</p>Formule :C26H23BrF4N2O3Couleur et forme :SolidMasse moléculaire :567.37BBDDL2059
CAS :<p>BBDDL2059 is a selective covalent inhibitor targeting EZH2, exhibiting an IC50 of 1.5 nM against the EZH2-Y641F mutant.</p>Formule :C27H36N4O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :512.66ALPK1-IN-3
CAS :<p>ALPK1-IN-3,serves as an ALPK1 inhibitor that dampens proinflammatory gene expression in the kidney and enhances survival in animal models of sepsis-induced</p>Formule :C20H16F2N4OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :398.43Immune cell migration-IN-1
CAS :<p>Immune cell migration-IN-1 (compound 2) serves as a potent inhibitor of immune cell migration, with potential research applications for mitigating conditions</p>Formule :C30H25ClN4O6SCouleur et forme :SolidMasse moléculaire :605.06Yhhu6669
CAS :<p>Yhhu6669 is an anti-HBV agent that suppresses viral DNA and replication by promoting DNA-free capsid assembly, effectively reducing HBV DNA and HBcAg levels in</p>Formule :C29H28ClFN6O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :563.02RIOK2-IN-2
CAS :<p>RIOK2-IN-2 (8) functions as an inhibitor of RIOK2, exhibiting IC50 values of 3.02 μM in MKN-1 cells and 5.34 μM in MOLT4 cells [1].</p>Formule :C27H23F3N6O2Couleur et forme :SolidMasse moléculaire :520.51Azilsartan mepixetil potassium
CAS :<p>Azilsartan medoxomil potassium (QR-01019K), an angiotensin II receptor antagonist, exhibits a potent and sustained antihypertensive effect, along with a more</p>Formule :C36H33KN6O8Couleur et forme :SolidMasse moléculaire :716.78ROCK2-IN-6
CAS :<p>ROCK2-IN-6 (Comp A) is a selective inhibitor of ROCK2, applicable in the study and treatment of ROCK-mediated, autoimmune, and inflammatory diseases [1].</p>Formule :C26H21F2N7ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :485.49Canlitinib
CAS :<p>Canlitinib, a tyrosine kinase inhibitor, holds potential for cancer research.</p>Formule :C33H31F2N3O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :619.61CYY292
CAS :<p>CYY292 is a chemical compound acting as an inhibitor of PDGFRα, PDGFRβ, FGFR1, -2, and -3, with respective IC50 values of 5.35, 4.6, 28, 28, and 78 nM.</p>Formule :C24H28N8OCouleur et forme :SolidMasse moléculaire :444.53Mal-VC-PAB-PNP-CDN-A
CAS :<p>Mal-VC-PAB-PNP-CDN-A is a conjugate comprised of an agent and a linker, utilized in antibody-drug conjugates (ADC) [1] [2].</p>Formule :C51H67N17O20P2Couleur et forme :SolidMasse moléculaire :1300.13Mc-Alanyl-Alanyl-Asparagine-PAB-MMAE
CAS :<p>Compound S6, Mc-Alanyl-Alanyl-Asparagine-PAB-MMAE, is a potent anticancer agent specifically activated by the tumor microenvironment; it demonstrates efficacy</p>Formule :C67H101N11O16Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1316.58DiaFluo
CAS :<p>DiaFluo is a probe for protein S-sulfinylation from cells.</p>Formule :C32H32N4O9SCouleur et forme :SolidMasse moléculaire :648.69Anti-MI/R injury agent 1
CAS :<p>Anti-MI/R injury agent 1 (compound 18), derived from Panaxatriol, represents an orally administered, potent agent against myocardial ischemia/reperfusion (MI/R</p>Formule :C32H49NO6Couleur et forme :SolidMasse moléculaire :543.73ATR-IN-24
CAS :<p>ATR-IN-24 (Compound 1) is an ATR inhibitor with demonstrated anticancer activity [1].</p>Formule :C23H26N6O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :418.49VMAT2-IN-2 tosylate
CAS :<p>VMAT2-IN-2 tosylate is a potent inhibitor of VMAT2 and is applicable in the research of tardive dyskinesia [1].</p>Formule :C27H36F3NO6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :559.64Xilmenolone
CAS :<p>Xilmenolone acts as a positive allosteric modulator of the GABA_A receptor [1].</p>Formule :C26H37N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :423.59LM2I
CAS :<p>LM2I, a derivative of Spinosyn A (SPA), serves both as an argininosuccinate synthase (ASS1) enzyme activator and a tumor inhibitor through direct interaction</p>Formule :C47H77N3O11Couleur et forme :SolidMasse moléculaire :860.13S-72
CAS :<p>S-72 acts as a microtubule polymerization inhibitor, effective in cell-free assays at concentrations of 1, 3, and 10 µM.</p>Formule :C20H22N4O3SCouleur et forme :SolidMasse moléculaire :398.50Igermetostat
CAS :<p>Igermetostat, an EZH2 inhibitor, is utilized both in vivo and in vitro for cancer research [1].</p>Formule :C32H46N4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :550.73SARS-CoV-2-IN-68
CAS :<p>SARS-CoV-2-IN-68 (compound 6C) is a covalent inhibitor of both SARS-CoV-2 PLpro and Mpro, exhibiting potent antiviral properties by targeting the Zn-finger</p>Formule :C14H12N2OSeDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :303.22Sakura 6
CAS :<p>Sakura 6, a synthetic serotonin transporter (SERT)-binding peptide, enhances the interaction between SERT and neuronal nitric oxide synthase.</p>Formule :C31H45N5O7Couleur et forme :SolidMasse moléculaire :599.73Lerzeparib
CAS :<p>Lerzeparib is a PARP (ADP-ribose polymerase) inhibitor that exhibits antineoplastic activity [1].</p>Formule :C21H20FN3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :365.4HBV-IN-38
CAS :<p>HBV-IN-38 (Example 193), an HBV DNA inhibitor with an EC50 value of ≤100 nM, serves as a research tool for investigating viral infections [1].</p>Formule :C18H16F3N5O4S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :487.48JAK-IN-34
CAS :<p>JAK-IN-34 (compound 11n) is a potent inhibitor of Janus kinases (JAKs), demonstrating IC50 values of 0.40 nM for JAK1, 0.83 nM for JAK2, 2.10 nM for JAK3,</p>Formule :C27H26N6ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :450.53Tauro-Obeticholic Acid sodium
CAS :<p>Tauro-obeticholic acid, a farnesoid X receptor (FXR) agonist and semisynthetic derivative of chenodeoxycholic acid, is an active metabolite of obeticholic acid.</p>Formule :C28H48NO6S·NaCouleur et forme :SolidMasse moléculaire :549.74PHI-101
CAS :<p>PHI-101 is a checkpoint kinase 2 (Chk2) inhibitor that can be used for the study of refractory acute myeloid leukemia (AML) and ovarian cancer.</p>Formule :C19H19FN4O2SDegré de pureté :99.4%Couleur et forme :SolidMasse moléculaire :386.44hDHODH-IN-8
<p>hDHODH-IN-8 is a potent human dihydroorotic dehydrogenase (hDHODH) inhibitor (IC50: 16 nM) that exhibits potent antiproliferative effects and has good water solubility, with potential for oncology studies, especially in lymphoma.</p>Formule :C21H15F6N3O4Degré de pureté :98%Masse moléculaire :487.35Ifetroban sodium
CAS :<p>Ifetroban sodium (BMS-180291), oral TXA2/PGH2 antagonist for researching heart, stroke, BP, thrombosis.</p>Formule :C25H31N2NaO5Couleur et forme :SolidMasse moléculaire :462.522DG026
CAS :DG026 selectively inhibits IRAP, reducing its cross-presentation in dendritic cells without affecting ERAP1.Formule :C35H40N3O4PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :597.68Dimethandrolone Undecanoate
CAS :Dimethandrolone Undecanoate (DMAU) is a novel orally available androgen with progestational activity and is a potential male contraceptive compound.Formule :C31H50O3Degré de pureté :99.65% - >99.99%Couleur et forme :SolidMasse moléculaire :470.73ROCK-IN-6
CAS :<p>ROCK-IN-6, a selective ROCK2 inhibitor, exhibits potent inhibition with an IC50 of 2.19 nM and holds promise for research into glaucoma and retinal diseases [1</p>Formule :C19H19N5O8SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :477.45BPH-628
CAS :<p>BPH-628 is a bioactive chemical.</p>Formule :C20H20O7P2Couleur et forme :SolidMasse moléculaire :434.32Ifetroban
CAS :<p>Ifetroban is a potent and selective TxA2/PGH2 receptor antagonist.</p>Formule :C25H32N2O5Couleur et forme :SolidMasse moléculaire :440.53ALS-I-41
CAS :ALS-I-41 is a novel, potent and selective antagonist of oxytocin receptor.Formule :C30H38FN3O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :587.7Cortivazol
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