Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.542 produits)
- Apoptose(5.816 produits)
- Cycle cellulaire/point de contrôle(4.466 produits)
- Chromatine/Épigénétique(2.252 produits)
- Signalisation du cytosquelette(1.381 produits)
- Altération de l'ADN/réparation de l'ADN(2.830 produits)
- Endocrinologie/Hormones(3.518 produits)
- Enzyme(3.640 produits)
- GPCR/G-Protéine(8.362 produits)
- Immunologie et Inflammation(3.540 produits)
- Virus de la grippe(296 produits)
- Signalisation JAK/STAT(405 produits)
- Signalisation MAPK(1.201 produits)
- Transporteur membranaire/Canal ionique(2.809 produits)
- Métabolisme(9.462 produits)
- Microbiologie/Virologie(7.003 produits)
- Neuroscience(9.942 produits)
- Autres inhibiteurs(37.827 produits)
- Oxydation-Réduction(40 produits)
- Signalisation PI3K/Akt/mTOR(1.399 produits)
- Protéases/Protéasome(1.598 produits)
- Cellules souche et Dérivés(830 produits)
- Tyrosine Kinase/Adaptateurs(2.012 produits)
- Ubiquitination(1.651 produits)
Affichez 16 plus de sous-catégories
66618 produits trouvés pour "Inhibiteurs"
Trier par
Degré de pureté (%)
0
100
|
0
|
50
|
90
|
95
|
100
Tubulin polymerization-IN-35
<p>Tubulin-IN-35 inhibits oxazolylisoindole microtubule formation, targeting VL51 marginal zone lymphoma.</p>Formule :C31H35N3O5Couleur et forme :SolidMasse moléculaire :529.63Casein Kinase II Inhibitor IV Hydrochloride
CAS :<p>Casein Kinase II Inhibitor IV HCl promotes keratinocyte differentiation, potential for skin disorder therapy.</p>Formule :C24H24ClN5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :465.93EGFR-IN-58
<p>EGFR-IN-58 is a potent, selective, ATP-competitive inhibitor of EGFR. EGFR-IN-58 exhibits significant cytotoxicity against melanoma, colon and blood cancers.</p>Formule :C31H30FN7OCouleur et forme :SolidMasse moléculaire :535.61MrgprX2 antagonist-6
<p>MrgprX2 antagonist-6 is a potent antiallergic agent with inhibitory effects on mast cell degranulation.</p>Formule :C24H23F3N6O3Couleur et forme :SolidMasse moléculaire :500.47Dexnebivolol
CAS :<p>Dexnebivolol (R67138), a ß-adrenergic antagonist, is Nebivolol's enantiomer with β1 blocking and vasodilation properties.</p>Formule :C22H25F2NO4Couleur et forme :SolidMasse moléculaire :405.43MsbA-IN-2
<p>MsbA-IN-2 is a potent inhibitor of the lipopolysaccharide transporter MsbA and is able to act on E. coli MsbA (IC50: 2 nM).</p>Formule :C23H19Cl2NO3Couleur et forme :SolidMasse moléculaire :428.31PPO-IN-1
<p>PPO-IN-1 is a potent inhibitor of protoporphyrinogen IX oxidase (PPO) (Ki: 2.5 nM).</p>Formule :C18H10F3N3O4SCouleur et forme :SolidMasse moléculaire :421.35ErSO-DFP
<p>ErSO-DFP activates a-UPR, targets ERα+ cancer cells with high selectivity, and effectively reduces MCF-7 tumours.</p>Formule :C20H17F5N2O2Couleur et forme :SolidMasse moléculaire :412.35CB30865
CAS :CB30865 (ZM 242421) is a selective and highly effective nicotinamide phosphoribosyltransferase (Nampt) inhibitor with potential antitumor activity.Formule :C26H22BrN5O2Degré de pureté :99.04%Couleur et forme :SolidMasse moléculaire :516.39U75302
CAS :<p>U75302 is an antagonist of thymosin beta-4 (TB4) receptor with a Ki value of 159 nM on guinea pig lung membranes.</p>Formule :C22H35NO3Degré de pureté :98%Couleur et forme :Light Yellow OilMasse moléculaire :361.52ACHN-975
CAS :<p>ACHN-975: potent LpxC inhibitor with subnanomolar activity; targets many gram-negative bacteria; MIC ≤1 μg/mL.</p>Formule :C20H23N3O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :369.41Dihydrophaseic acid
CAS :<p>Dihydrophaseic acid 3'-O-b-D-glucopyranoside (D3G) can increase the proliferation and differentiation of osteoblast cells and enhance bone formation, suggests</p>Formule :C15H22O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :282.33AL-6556
CAS :<p>AL-6556 is a prostaglandin DP receptor agonist.</p>Formule :C20H33ClO5Couleur et forme :SolidMasse moléculaire :388.93Taprostene
CAS :<p>Taprostene (CG-4203), a stable Prostacyclin analogue, protects endothelium and myocardium post-ischemia in cats, with minimal hemodynamic impact.</p>Formule :C24H30O5Couleur et forme :SolidMasse moléculaire :398.49Anticancer agent 69
<p>Anticancer agent 69 targets PC3 cells (IC50=26 nM), raises ROS, lowers EGFR, and induces apoptosis.</p>Formule :C19H26N8SCouleur et forme :SolidMasse moléculaire :398.53Silvestrol
CAS :<p>Silvestrol is a eukaryotic translation initiation factor 4A inhibitor. Silvestrol causes autophagy and caspase-mediated apoptosis.</p>Formule :C34H38O13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :654.66LY503430
CAS :<p>LY503430: Oral AMPA enhancer with nootropic, neuroprotective properties, mitigates 6-OHDA/MPTP brain damage.</p>Formule :C20H25FN2O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :392.49EB-0156
<p>EB-0156: potent ER α-glucosidase inhibitor, IC50 of 0.0479/ <0.001 μM, N-substituted valerian, broad-spectrum antiviral potential.</p>Formule :C21H32N6O7Couleur et forme :SolidMasse moléculaire :480.51GLP-1R agonist 8
CAS :<p>GLP-1R agonist 8 is a potent agonist of GLP-1R (EC50 < 2 nM).</p>Formule :C33H32N4O5Couleur et forme :SolidMasse moléculaire :564.63Edotecarin
CAS :<p>Edotecarin is a potent topoisomerase I inhibitor. It can decrease single-strand DNA cleavage (IC50: 50 nM).</p>Formule :C29H28N4O11Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :608.55KUSC-5037
<p>KUSC-5037 inhibits HIF-1 (IC50 = 1.2 μM) and mitochondrial complex V/FoF1ATP synthase.</p>Formule :C18H17F3N6O2Couleur et forme :SolidMasse moléculaire :406.13651Kahweol Acetate
CAS :<p>Kahweol Acetate, a semi-synthetic coffee bean derivative, inhibits osteoclasts, cancer cells, DNA damage, and oxidative stress.</p>Formule :C22H28O4Couleur et forme :SolidMasse moléculaire :356.46AVE-1330A free acid
CAS :<p>AVE-1330A free acid is a broad-spectrum non-beta-lactam beta-lactamase inhibitor.</p>Formule :C7H11N3O6SCouleur et forme :SolidMasse moléculaire :265.24UCN-01
CAS :<p>inhibitor of Akt, protein kinase C, PDK1 and cyclin-dependent kinases</p>Formule :C28H26N4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :482.53RET-IN-9
CAS :<p>RET-IN-9 is a potent RET kinase inhibitor, potentially useful for studying RET-related diseases, including lung and thyroid cancer.</p>Formule :C26H27N9OCouleur et forme :SolidMasse moléculaire :481.55Adecypenol
CAS :<p>Adecypenol is a unique adenosine deaminase inhibitor. It shows effective inhibitory activity against calf intestinal adenosine deaminase.</p>Formule :C12H16N4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :280.28BAY-7598
CAS :<p>BAY-7598 is a potent, selective, and orally bioavailable MMP12 inhibitor (IC50s: 0.085, 0.67, and 1.1 nM for human/murine/rat MMP12).</p>Formule :C28H31N3O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :505.56Anticancer agent 12
<p>Anticancer agent 12 shows cytotoxic activity in malignant cells with no hepatotoxicity.</p>Formule :C16H17BrN4O2SCouleur et forme :SolidMasse moléculaire :409.3U 75875
CAS :<p>U 75875 is a protease inhibitor.</p>Formule :C45H61N7O7Couleur et forme :SolidMasse moléculaire :812.01SARS-CoV-2-IN-22
CAS :<p>SARS-CoV-2-IN-22 is a SARS-CoV-2 pseudovirus inhibitor (IC50: 16.96 μM).</p>Formule :C27H24N2O3SCouleur et forme :SolidMasse moléculaire :456.56Carbonic anhydrase inhibitor 8
<p>R-13, a carbonic anhydrase inhibitor, has Ki of 60.7 nM (hCA I), 320.7 nM (hCA II), and 2298 nM (hCA IV).</p>Formule :C20H25N3O4SCouleur et forme :SolidMasse moléculaire :403.5ROS1-IN-1
<p>ROS1-IN-1, a potent ROS1 kinase inhibitor, has an IC50 of 0.097 μM.</p>Formule :C17H15ClN6SCouleur et forme :SolidMasse moléculaire :370.86GSK866
CAS :<p>GSK866 is a selective glucocorticoid receptor agonist (SEGRA).</p>Formule :C23H21Cl2F4N5O3Couleur et forme :SolidMasse moléculaire :562.34HIV-1 inhibitor-41
<p>HIV-1 inhibitor-41 (B23): Oral non-nucleoside reverse transcriptase blocker, EC50 of 50 nM (E138K), 20.8 nM (WT), low hERG/CYP impact, non-toxic.</p>Formule :C16H15F2N3OSCouleur et forme :SolidMasse moléculaire :335.37Antiangiogenic agent 3
<p>Antiangiogenic agent 3 blocks HUVEC cell migration, chemotaxis, and lowers Src, cdc42, MAPK gene expression.</p>Formule :C19H20O7Couleur et forme :SolidMasse moléculaire :360.36AChE-IN-24
<p>AChE-IN-24: Strong AChE blocker, crosses blood-brain barrier, IC50=0.053 μM, useful for AD research.</p>Formule :C22H30N2O4S2Couleur et forme :SolidMasse moléculaire :450.61L2H2-6OTD
CAS :<p>L2H2-6OTD is a telomerase inhibitor with G-quadruplex loops; IC50: 15 nM.</p>Formule :C30H30N10O8Couleur et forme :SolidMasse moléculaire :658.62JAK3/BTK-IN-4
CAS :<p>JAK3/BTK-IN-4, a dual inhibitor for JAK3/BTK, shows synergy in autoimmune disease treatment. (Patent WO2021147953A1, compound 003)</p>Formule :C21H25ClN8OCouleur et forme :SolidMasse moléculaire :440.93Ganoderic acid R
CAS :<p>Ganoderic acid R: potent anticancer, induces apoptosis, cytotoxic to MDR and sensitive tumor cells.</p>Formule :C34H50O6Couleur et forme :SolidMasse moléculaire :554.76ent-8-iso-15(S)-Prostaglandin F2α
CAS :<p>Isoprostanes are produced by the non-enzymatic, free radical peroxidation of phospholipid-esterified arachidonic acid.</p>Formule :C20H34O5Couleur et forme :SolidMasse moléculaire :354.48HER2-IN-7
CAS :<p>HER2-IN-7 is a potent HER2 inhibitor with potential for researching ErbB-related diseases, especially cancer.</p>Formule :C28H26F3N7O3Couleur et forme :SolidMasse moléculaire :565.55USP7-IN-10
CAS :<p>USP7-IN-10 is a potent inhibitor of ubiquitin-specific protease 7 (USP7), exhibiting an inhibition concentration half-maximal (IC50) value of 13.39 nM.</p>Formule :C26H29ClN4O3SCouleur et forme :SolidMasse moléculaire :513.05GNE-616
CAS :<p>GNE-616: a potent, stable, oral Nav1.7 inhibitor; Ki: 0.79 nM, Kd: 0.38 nM; for chronic pain.</p>Formule :C24H23F4N5O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :537.53SR121566A
CAS :SR121566A is a novel non-peptide antagonist of Glycoprotein IIb/IIIa (GP IIb-IIIa).Formule :C20H25N5O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :431.51IL-17 modulator 5
CAS :<p>IL-17 modulator 5 is a IL-17 inhibitor, with an IC 50 of 1 nM .</p>Formule :C28H23F6N9O2Couleur et forme :SolidMasse moléculaire :631.53Mesulergine hydrochloride
CAS :<p>5-HT2A and 2C receptor antagonist</p>Formule :C18H27ClN4O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :398.95Aristoforin
CAS :<p>Aristoforin is a SIRT1 and SIRT2 inhibitor that induces cell cycle arrest, shows potent antitumor effects, and inhibits lymphangiogenesis in vivo.</p>Formule :C37H54O6Couleur et forme :SolidMasse moléculaire :594.82HDAC-IN-27
<p>HDAC-IN-27 is a potent and orally active inhibitor of HDAC Class I (0.43 nM - 3.01 nM for HDAC1-3).</p>Formule :C20H22N4O2Couleur et forme :SolidMasse moléculaire :350.41Efrapeptin F
CAS :<p>Efrapeptin F, from Tolypocladium fungi, inhibits mitochondrial complex V and targets nutrient-deprived tumor cells.</p>Formule :C82H141N18O16Couleur et forme :SolidMasse moléculaire :1635.11Carbonic anhydrase inhibitor 10
<p>CA inhibitor 10 targets MCF-7 cells, IC50: 11.9 μM; potent h CA IX inhibitor, Ki: 6.2 nM. Anti-cancer research.</p>Formule :C14H17N5O3SCouleur et forme :SolidMasse moléculaire :335.38J-104132
CAS :<p>J-104132: potent human ETA/B antagonist; Ki: ETA=0.034nM, ETB=0.104nM; prevents ET-1 effects, ED50 i.v.=0.045mg/kg, p.o.=0.35mg/kg.</p>Formule :C31H33NO7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :531.60Xylarianaphthol-1
CAS :<p>Xylarianaphthol-1 is an activator of p21 promoter in a p53-independent manner.</p>Formule :C16H20BrFN2O2Couleur et forme :SolidMasse moléculaire :371.24ACSS2-IN-1
CAS :<p>ACSS2-IN-1, a potent ACSS2 inhibitor, has IC50 0.01-<1 nM; useful in cancer research.</p>Formule :C27H25ClN6O2Couleur et forme :SolidMasse moléculaire :500.98VEGFR-2-IN-12
<p>VEGFR-2-IN-12 (compound 6g), a 2-oxoquinoxalinyl-1,2,4-triazole, is a potent inhibitor of VEGFR-2 (IC50: 0.037 μM). VEGFR-2-IN-12 has anti-tumour effects.</p>Formule :C22H24N6O3SCouleur et forme :SolidMasse moléculaire :452.53Dehatrine
CAS :<p>Dehatrine: alkaloid from Beilschmiedia madang, inhibits Plasmodium falciparum K1 growth.</p>Formule :C37H38N2O6Couleur et forme :SolidMasse moléculaire :606.71KU-32
CAS :<p>KU-32 is a novel and novobiocin-based Hsp90 inhibitor. It can protect against neuronal cell death.</p>Formule :C20H25NO8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :407.41ICA-105665
CAS :ICA-105665 is an orally active Kv7.2/7.3/7.5 channel opener, CNS-penetrant with antiseizure effects, and low hepatocyte cytotoxicity.Formule :C19H15F2N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :355.34GnRH-R antagonist 1
CAS :<p>Compound 21a: Oral GnRH-R antagonist, IC50=0.57 nM, potent against prostate cancer/prevents LH surges.</p>Formule :C31H28F5N7O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :721.65BRD1991
CAS :<p>BRD1991 is a chemical compound that specifically disrupts the interaction between Beclin 1 and Bcl-2, thereby inducing autophagy.</p>Formule :C33H35Cl2N3O4Couleur et forme :SolidMasse moléculaire :608.55Brostallicin HCl
CAS :<p>Brostallicin, a synthetic MGB, inhibits DNA replication in cancer cells, inducing cell death, effective against MMR-defective tumors.</p>Formule :C30H36BrClN12O5Couleur et forme :SolidMasse moléculaire :760.04Anticancer agent 28
<p>Anticancer agent 28 is 50x more potent than Oridonin, IC50 of 0.09 μM against K562; effective in H22 mouse tumors.</p>Formule :C28H33NO6Couleur et forme :SolidMasse moléculaire :479.56FGFR1 inhibitor-6
<p>FGFR1 inhibitor-6, IC50: 16.31 nM, blocks cell cycle at pro-G1/G2/M and induces apoptosis.</p>Formule :C27H19N5O4S2Couleur et forme :SolidMasse moléculaire :541.6PF-06726304 acetate
CAS :<p>PF-06726304 acetate is a selective inhibitor of EZH2, with robust antitumor growth activity.</p>Formule :C24H25Cl2N3O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :506.38CaMKIIα-IN-1
<p>CaMKIIα-IN-1 (Compound 4d) is an orally active inhibitor of Ca 2+ /calmodulin-dependent protein kinase II α (CaMKIIα) with a Kd of 219 nM for CaMKIIα WT hub.</p>Formule :C14H11ClO4Couleur et forme :SolidMasse moléculaire :278.69Tasidotin hydrochloride
CAS :<p>Tasidotin hydrochloride, a dolastatin 15 analog, inhibits microtubule assembly and dynamics.</p>Formule :C32H59ClN6O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :643.30Salacinol
CAS :<p>Salacinol is a naturally occurring alpha-glucosidase inhibitor isolated from an Ayurvedic traditional medicine Salacia reticulata.</p>Formule :C9H18O9S2Couleur et forme :SolidMasse moléculaire :334.37BRD5631
CAS :BRD5631 is an autophagy enhancer, enhances autophagy through an mTOR-independent pathway.Formule :C30H35N3O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :501.62Rubropunctatin
CAS :<p>Rubropunctatin is a monascus pigment with very potent cancer cell proliferation inhibitory effects.</p>Formule :C21H23NO4Couleur et forme :SolidMasse moléculaire :353.41PI3Kα-IN-8
<p>PI3Kα-IN-8 is a selective inhibitor of PI3Kα (IC50: 0.012 μM).</p>Formule :C26H27BrN4O2Couleur et forme :SolidMasse moléculaire :507.42T-Type calcium channel inhibitor 2
<p>Compound 6g inhibits T-type Ca channels (IC50: Cav3.1-31μM, Cav3.2-83μM), cytotoxic to A549 (IC50: 5μM) & HCT-116 cells (IC50: 6.4μM).</p>Formule :C36H39FN4OSCouleur et forme :SolidMasse moléculaire :594.78Flusoxolol
CAS :<p>Flusoxolol is a beta-adrenoceptor partial agonist.</p>Formule :C22H30FNO4Couleur et forme :SolidMasse moléculaire :391.48KRAS G12D inhibitor 12
<p>KRAS G12D inhibitor 12 targets Ras protein for cancer research. (Patent WO2021108683A1, Compound 134)</p>Formule :C23H21ClFN5O3Couleur et forme :SolidMasse moléculaire :469.9Tofogliflozin
CAS :Tofogliflozin specifically inhibits SGLT2; IC50s are 2.9 nM (human), 14.9 nM (rat), 6.4 nM (mouse).Formule :C22H26O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :386.44KRAS inhibitor-21
CAS :<p>KRAS inhibitor-21 (22b) is a KRAS G12C inhibitor (IC50<0.01 μM) that can be used in cancer research.</p>Formule :C33H41N5O3Couleur et forme :SolidMasse moléculaire :555.71Fradafiban
CAS :<p>Fradafiban binds to the human platelet GP IIb/IIIa complex with a Kd value of 148 nM. Fradafiban is a non-polypeptide platelet glycoprotein IIb/IIIa antagonist.</p>Formule :C20H21N3O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :367.40S1PR1 agonist 1
CAS :<p>S1PR1 agonist 1 is a potent agonist of S1PR1. S1PR1 agonist 1 has potential in autoimmune diseases.</p>Formule :C29H30N4O4Couleur et forme :SolidMasse moléculaire :498.57NMDA receptor antagonist-3
<p>NMDA antagonist-3: recovery rate 40% at 100 μM, low toxicity in SH-SY5Y, human stem cells.</p>Formule :C13H19N3O6Couleur et forme :SolidMasse moléculaire :313.31Disulergine
CAS :<p>Disulergine is a dopamine receptor agonist. It also prolactin release-inhibiting 8 alpha-amino-ergoline.</p>Formule :C17H24N4O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :348.46ATR-IN-14
CAS :<p>ATR-IN-14: potent ATR kinase inhibitor; 98.03% inhibition at 25 nM; IC50 of 64 nM in LoVo cells.</p>Formule :C20H20FN7OCouleur et forme :SolidMasse moléculaire :393.42OP-5244
CAS :<p>OP-5244 has comparable potency to bisphosphonic acid series and targets CD73.</p>Formule :C19H29ClN5O9PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :537.89Antitumor agent-65
CAS :<p>Antitumor agent-65 (Compound 5) is an analogue/derivative of (-)-cleistenolide. Antitumor agent-65 has potential in cancer research.</p>Formule :C18H17NO10Couleur et forme :SolidMasse moléculaire :407.33Cap-dependent endonuclease-IN-2
<p>Cap-dependent endonuclease-IN-2 strongly blocks influenza A virus RNA polymerase; it's a CEN inhibitor.</p>Formule :C30H24FN3O7SCouleur et forme :SolidMasse moléculaire :589.5915-keto-Prostaglandin E2
CAS :<p>15-keto-Prostaglandin E2, an endogenous metabolite, inhibits STAT3 activation through binding to Cys259 and regulates breast cancer cell growth and progression.</p>Formule :C20H30O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :350.45CXCR7 modulator 2
CAS :CXCR7 modulator 2 is a 7-type C-X-C chemokine receptor (CXCR7) modulator with a Ki of 13 nM.Formule :C29H42N6O3Couleur et forme :SolidMasse moléculaire :522.68Azotomycin
CAS :Azotomycin is an antagonist of L-glutamine and may be used as an immunosuppressant.Formule :C17H23N7O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :453.41DS69910557
<p>DS69910557: potent hPTHR1 antagonist, IC50 0.08 μM, oral, for hyperparathyroidism & osteoporosis research.</p>Formule :C32H33Cl2FN4O3Couleur et forme :SolidMasse moléculaire :611.53Piperazinomycin
CAS :<p>Piperazinomycin is an antifungal antibiotic, showing inhibitory activity against fungi and yeasts, especially against Trichophyton.</p>Formule :C18H20N2O2Couleur et forme :SolidMasse moléculaire :296.36(S)-Purvalanol B
CAS :<p>(S)-Purvalanol B is the S enantiomer of Purvalanol B. Purvalanol B is an inhibitor of cyclin-dependent kinase(CDK) .</p>Formule :C20H25ClN6O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :432.9APJ receptor agonist 3
CAS :<p>APJ receptor agonist 3 is a highly effective and orally administerable agonist of the APJ receptor, demonstrating a potent EC50 value of 0.027 nM.</p>Formule :C26H29ClN4O5Couleur et forme :SolidMasse moléculaire :512.98Dyrk1A-IN-2
<p>Dyrk1A-IN-2 is a DYRK1A inhibitor (EC50: 37 nM). dyrk1A-IN-2 exhibits efficient promotion of human β-cell replication, as well as low cytotoxicity.</p>Formule :C27H32N6O4Couleur et forme :SolidMasse moléculaire :504.58D4R antagonist-1
<p>Potent, selective D4R antagonist; IC50 = 6.87 µM; potential in Parkinson’s disease research.</p>Formule :C21H25F2NO2Couleur et forme :SolidMasse moléculaire :361.43CLK1/4-IN-1
<p>CLK1/4-IN-1 inhibits Clk1/4 (IC50: 9.7/6.6 nM), curbing T24 cell growth (GI50: 1.1 μM). Potential cancer research tool.</p>Formule :C18H14ClNO4SCouleur et forme :SolidMasse moléculaire :375.83SB-612111
CAS :<p>SB-612111: potent ORL-1 antagonist, Ki=0.33 nM; μ-, κ-, δ-receptor Ki=57.6, 160.5, 2109 nM; blocks nociceptin's pain effect.</p>Formule :C24H29Cl2NOCouleur et forme :SolidMasse moléculaire :418.40Antioxidant agent-8
<p>Antioxidant agent-8, an oral Aβ 1-42 inhibitor, reduces fibril aggregation & promotes disaggregation; it's neuroprotective & BBB permeable.</p>Formule :C13H12O5Couleur et forme :SolidMasse moléculaire :248.23Fabimycin
CAS :<p>Fabimycin, a FabI inhibitor, combats drug-resistant gram-negative bacterial infections effectively.</p>Formule :C23H25ClN4O3Couleur et forme :SolidMasse moléculaire :440.92APN/AKT-IN-1
<p>APN/AKT-IN-1, a dual APN (IC50=0.21μM) & AKT (IC50=0.27μM) inhibitor, hinders GSK3β phosphorylation.</p>Formule :C18H27N7O3Couleur et forme :SolidMasse moléculaire :389.45ERK2 IN-1
CAS :<p>ERK2 IN-1 is a selective ERK2 inhibitor with an IC50 of 7 nM.</p>Formule :C36H34FN7O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :647.76CDK8-IN-5
CAS :<p>CDK8-IN-5: potent CDK8 inhibitor, IC50=72 nM, boosts IL-10 by 43%, may aid inflammatory bowel disease research.</p>Formule :C26H22N2O4Couleur et forme :SolidMasse moléculaire :426.46VEGFR-2-IN-16
<p>VEGFR-2-IN-16 (Compound 15b) is a potent inhibitor of VEGFR-2 (IC50: 86.36 nM) that exhibits antitumour effects.</p>Formule :C21H13Cl2N3O2Couleur et forme :SolidMasse moléculaire :410.25GSK864
CAS :<p>GSK864 is an inhibitor of isocitrate dehydrogenase 1 (IDH1) mutant. GSK864 inhibits IDH1 mutants R132C, R132H, and R132G (IC50: 8.8, 15.2, and 16.6 nM).</p>Formule :C30H31FN6O4Degré de pureté :97.07%Couleur et forme :SolidMasse moléculaire :558.6Henagliflozin
CAS :<p>Henagliflozin (SHR3824): an oral, selective SGLT2 inhibitor, weak on SGLT1.</p>Formule :C22H24ClFO7Couleur et forme :SolidMasse moléculaire :454.87Thiolactomycin
CAS :<p>Thiolactomycin is a novel reversible dual inhibitor of D-amino acid oxidase (DAO) and D-Aspartate oxidase (DDO).</p>Formule :C11H14O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :210.29Dicetrorelix pamoate
CAS :<p>Cetrorelix pamoate is a synthetic decapeptide that acts as a GnRH antagonist, inhibiting the release of LH and FSH from the pituitary.</p>Formule :C163H200Cl2N34O34Couleur et forme :SolidMasse moléculaire :3250.49PARP-1-IN-1
<p>PARP-1-IN-1: Selective, oral PARP-1 inhibitor with 0.96 nM IC50; well-tolerated and effective in single-dose MDA-MB-436 model.</p>Formule :C23H25FN4OCouleur et forme :SolidMasse moléculaire :392.47Pyridoxatin
CAS :<p>Pyridoxatin: fungal metabolite; blocks TBARS production, prevents AAPH-induced hemolysis, and acts against C. albicans.</p>Formule :C15H21NO3Couleur et forme :SolidMasse moléculaire :263.33Nrf2 activator-6
CAS :<p>Nrf2 activator-6, a tetrahydroisoquinoline, inhibits Kelch-Nrf2 at 5 nM IC50 (WO2021214470A1).</p>Formule :C31H37ClFN5O5Couleur et forme :SolidMasse moléculaire :614.11Antitrypanosomal agent 5
<p>Antitrypanosal agent 5 is a selective anti-trypanosomal agent that acts on T. brucei (IC50: 1 nM) and HEK293 cells (IC50: 483.3 μM).</p>Formule :C30H30N6O4SCouleur et forme :SolidMasse moléculaire :570.66HCV-IN-38
<p>Potent oral HCV inhibitor HCV-IN-38 has 15 nM EC50, 431 SI, high efficacy, and low toxicity.</p>Formule :C22H24ClF3N4O4Couleur et forme :SolidMasse moléculaire :500.9COX-1/2-IN-2
<p>COX-1/2-IN-2, a potent dual inhibitor, has IC50s: COX-1 at 9.7μM & COX-2 at 4.6μM.</p>Formule :C15H10ClIN2OCouleur et forme :SolidMasse moléculaire :396.61GSK3368715
CAS :<p>GSK3368715 is an orally active, reversible, and S-adenosyl-L-methionine (SAM) uncompetitive type I protein arginine methyltransferases (PRMTs) inhibitor (IC50s</p>Formule :C20H38N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :366.54MtTMPK-IN-2
CAS :<p>MtTMPK-IN-2 inhibits M. tuberculosis TMPK (IC50: 1.1 μM), Mtb H37Rv (MIC: 12.5 μM), and is cytotoxic in MRC-5 cells (EC50: 6.1 μM).</p>Formule :C23H24ClN3O3Couleur et forme :SolidMasse moléculaire :425.91AN-12-H5
CAS :<p>AN-12-H5 is an anti-enteroviral compound that targets the replication process of PV and EV71 viruses.</p>Formule :C24H23N3O4S3Couleur et forme :SolidMasse moléculaire :513.65TA-316
CAS :<p>Agent induces megakaryocytes/platelets from stem cells to treat thrombopenia.</p>Formule :C28H25BrN4O5S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :641.56COX-2-IN-13
<p>COX-2-IN-13 is a potent, selective COX-2 inhibitor with 0.98 μM IC50; shows strong anti-inflammatory properties and low acute toxicity.</p>Formule :C19H18N2O5SCouleur et forme :SolidMasse moléculaire :386.42TD-0212
CAS :TD-0212: Oral dual antagonist for AT1 (pKi 8.9) & NEP inhibitor (pIC50 9.2).Formule :C28H34FN3O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :527.65GSK945237
CAS :<p>GSK945237 is a type IIA topoisomerase inhibitor, effective on Gram-positive and negative bacteria, with favorable pharmacokinetics and in vivo efficacy.</p>Formule :C24H26FN5O3Couleur et forme :SolidMasse moléculaire :451.49α-Glucosidase-IN-12
<p>α-Glucosidase-IN-12 is a potent inhibitor of α-glucosidase (IC50: 10.20 μM).</p>Formule :C25H30N4O4S2Couleur et forme :SolidMasse moléculaire :514.66PDHK-IN-5
<p>PDHK-IN-5, potent PDHK2 (0.006 μM IC50) & PDHK4 (0.0329 μM IC50) inhibitor, may be explored for cancer and diabetes treatment.</p>Formule :C30H31N5O2Couleur et forme :SolidMasse moléculaire :493.6L 734217
CAS :<p>L 734217 is an antagonist of the fibrinogen receptor.</p>Formule :C18H31N3O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :353.46Anticancer agent 35
<p>Compound 10, a sulfonylurea, inhibits A549, A431, PACA2 cells with IC50s: 18.1, 4.0, 18.9 μg/mL.</p>Formule :C15H13N3O3S3Couleur et forme :SolidMasse moléculaire :379.48FAK-IN-6
<p>FAK-IN-6: Potent FAK inhibitor (IC50=1.415 nM), anti-cancer, for pancreatic studies.</p>Formule :C25H31ClN5O6PSCouleur et forme :SolidMasse moléculaire :596.04Antibacterial agent 63
CAS :<p>Aztreonam-siderophore conjugate 63 is an antibacterial agent that exhibits efficacy against Gram-negative bacteria through the linkage of aztreonam to a</p>Formule :C35H43N9O14S2Couleur et forme :SolidMasse moléculaire :877.9NYX-2925
CAS :<p>NYX-2925, an oral NMDAR modulator, enhances Src in mPFC. No CAMKII impact or addictive/sedative effects. Useful for CNS disorder studies.</p>Formule :C14H23N3O4Couleur et forme :SolidMasse moléculaire :297.35FTO-IN-4
CAS :<p>FTO-IN-4 is a potent and selective inhibitor of adiposity and obesity-associated protein (FTO).</p>Formule :C22H16Cl2N6O6Couleur et forme :SolidMasse moléculaire :531.31AFM-30a hydrochloride
<p>AFM-30a hydrochloride: selective PAD2 inhibitor, EC50 9.5 μM; blocks H3 guanylation, EC50 0.4 μM; used for cancer and autoimmune research.</p>Formule :C24H28ClFN6O3Couleur et forme :SolidMasse moléculaire :502.97WEHI-9625
CAS :<p>WEHI-9625 is a tricyclic sulfone small molecule apoptosis inhibitor (EC50: 69 nM).</p>Formule :C34H27NO5S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :593.71eIF4A3-IN-4
<p>eIF4A3-IN-4 is a novel inhibitor of eIF4A (IC50: 8.6 μM).</p>Formule :C24H20N2O5Couleur et forme :SolidMasse moléculaire :416.43CI-988
CAS :<p>CCK2 (CCK-B) receptor antagonist</p>Formule :C35H42N4O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :614.73PDE4-IN-12
<p>PDE4-IN-12 is a potent and safe PDE4 ubiquitous inhibitor that acts on PDE4 (IC50: 3.5 nM, SI: 2.71) and PDE7 (IC50: 15 nM, SI: 4.27).</p>Formule :C34H35NO6Couleur et forme :SolidMasse moléculaire :553.64Taranabant
CAS :<p>Taranabant: potent CB1 receptor inverse agonist; inhibits agonists with 0.13 nM Ki in vitro.</p>Formule :C27H25ClF3N3O2Degré de pureté :99.06% - 99.06%Couleur et forme :SolidMasse moléculaire :515.96BXL0124
CAS :<p>BXL0124 is a gemini vitamin D analog which targets CD44-STAT3 signaling and inhibits breast cancer invasion.</p>Formule :C32H44F6O4Couleur et forme :SolidMasse moléculaire :606.68G108
CAS :<p>G108 is an inhibitor of human cGAS and is used in the study of autoimmune diseases associated with human cGAS.</p>Formule :C16H14Cl2N4O2Degré de pureté :99.13% - 99.75%Couleur et forme :SolidMasse moléculaire :365.21MRK003
CAS :<p>MRK003, a γ-secretase inhibitor, induces apoptosis, halts cell growth in myeloma/NHL, and affects notch signaling and PI3K/Akt pathway.</p>Formule :C25H31F6N3O2SCouleur et forme :SolidMasse moléculaire :551.59Freselestat
CAS :<p>Freselestat (ONO-6818) inhibits neutrophil elastase, reduces interleukin 8, C5B-9, and inflammation in cardiopulmonary bypass.</p>Formule :C23H28N6O4Couleur et forme :SolidMasse moléculaire :452.51MCTR3
CAS :<p>MCTR3, derived from DHA via maresin 1 in macrophages, hastens tissue healing and reduces inflammation and eicosanoids post-E. coli infection in mice.</p>Formule :C25H37NO5SCouleur et forme :SolidMasse moléculaire :463.63Dinalbuphine sebacate
CAS :<p>Dinalbuphine sebacate: long-acting nalbuphine prodrug, μ-opioid partial agonist/antagonist, κ-opioid high-efficacy agonist.</p>Formule :C52H68N2O10Couleur et forme :SolidMasse moléculaire :881.1HDAC1-IN-3
<p>HDAC1-IN-3 is a potent inhibitor of Pf HDAC1.</p>Formule :C22H24ClN7O2Couleur et forme :SolidMasse moléculaire :453.92LpxC-IN-10
CAS :<p>LpxC-IN-10 is a selective LpxC inhibitor with an MIC of 0.5 μg/mL against E. coli and K. pneumoniae and is capable of being used to study bacterial infections.</p>Formule :C30H31N5O3Couleur et forme :SolidMasse moléculaire :509.6E7090 succinate
CAS :<p>E7090 succinate inhibits FGFR1, FGFR2, and FGFR3 with IC50: 0.71, 0.50, 1.2 nM; less so FGFR4 at 120 nM.</p>Formule :C76H92N10O24Couleur et forme :SolidMasse moléculaire :1529.60ATR-IN-11
<p>ATR-IN-11, a potent ATR kinase inhibitor, shows promise as a lead for DNA damage response-targeted cancer drugs.</p>Formule :C25H30N6O2Couleur et forme :SolidMasse moléculaire :446.544α-PDD
CAS :<p>4alpha-PDD activates transient receptor potential vanilloid 4 (TRPV4) channels and is inactive for signaling through PKC.</p>Formule :C40H64O8Couleur et forme :SolidMasse moléculaire :672.93HIV-1 inhibitor-8
<p>HIV-1 inhibitor-8: potent oral NNRTI, low toxicity, IC50: 0.081 μM, effective on multiple strains, EC50: 4.44-54.5 nM.</p>Formule :C25H21N5OSCouleur et forme :SolidMasse moléculaire :439.53ONO-9780307
CAS :<p>ONO-9780307 is a specific antagonist of LPA1 (lysophosphatidic acid receptor 1) (IC50: 2.7 nM).</p>Formule :C30H35NO7Couleur et forme :SolidMasse moléculaire :521.6DFBTA
<p>DFBTA inhibits ANO1 with IC50 of 24 nM, effectively treating inflammatory pain orally.</p>Formule :C18H10ClF2NO3SCouleur et forme :SolidMasse moléculaire :393.79HIV-IN-3
<p>HIV-IN-3 (Compound 22a) is a potent inhibitor of HIV (IC50: 1.5 μM). HIV-IN-3 has potential for the study of HIV-related diseases.</p>Formule :C21H32ClN7O3Couleur et forme :SolidMasse moléculaire :465.98CCT369260
CAS :<p>CCT369260 (compound 1), an orally active inhibitor targeting B-cell lymphoma 6 (BCL6), demonstrates anti-tumor efficacy with an IC50 value of 520 nM [1].</p>Formule :C24H31ClF2N6O2Couleur et forme :SolidMasse moléculaire :508.99Napsagatran hydrate
CAS :Napsagatran hydrate is a novel and specific inhibitor of thrombin.Formule :C26H36N6O7SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :576.66CD73-IN-12
<p>CD73-IN-12, a compound from CN114437038A, shows strong anti-tumor activity by effectively inhibiting CD73 enzyme.</p>Formule :C17H14F2N4O2Couleur et forme :SolidMasse moléculaire :344.32DGY-08-097
CAS :<p>DGY-08-097: potent HCV NS3 degrader, low resistance risk, strong inhibition in cells, DC50 of 50nM at 4h.</p>Formule :C60H76N10O14Couleur et forme :SolidMasse moléculaire :1161.3LAF-153
CAS :<p>LAF-153 is a reversible Methionine Aminopeptidase‑2 (MetAP-2) Inhibitor.</p>Formule :C18H32N2O7Couleur et forme :SolidMasse moléculaire :388.46HDAC2-IN-1
<p>HDAC2-IN-1 is an oral HDAC2 inhibitor (IC50: 0.5 μM), crosses the blood-brain barrier, and inhibits HDAC1 and HDAC8.</p>Formule :C22H23ClN4OSCouleur et forme :SolidMasse moléculaire :426.96BTK-IN-16
CAS :<p>BTK-IN-16 is a potential inhibitor of wild-type BTK and C481S mutants.BTK-IN-16 can be used to study various autoimmune diseases and cancers caused by BTK.</p>Formule :C15H14N4O2Degré de pureté :99.04%Couleur et forme :SoildMasse moléculaire :282.3STA 2
CAS :<p>STA 2 is an analogue of TXA2, a thromboxane receptor in the colonic epithelium.</p>Formule :C21H34O3SCouleur et forme :SolidMasse moléculaire :366.56TAK-637
CAS :<p>TAK-637 is a tachykinin 1 (NK1) receptor antagonist.</p>Formule :C30H25F6N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :573.53Cemdomespib
CAS :<p>Cemdomespib (KU-596) is a potent Hsp90 modulator with neuroprotective effects and can improve diabetic neuropathy.</p>Formule :C24H30FNO6Couleur et forme :SolidMasse moléculaire :447.5HIF-2α-IN-7
CAS :<p>HIF-2α-IN-7 is a hypoxia inducible factor 2α (HIF-2α) inhibitor.</p>Formule :C18H9F6NO2Couleur et forme :SolidMasse moléculaire :385.26TAK-828F
CAS :<p>TAK-828F: potent, selective RORγt inverse agonist. Oral. IC50=1.9 nM; reporter gene IC50=6.1 nM.</p>Formule :C28H32FN3O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :509.57Human carbonic anhydrase II-IN-1
<p>Compound S-13: Potent hCA II inhibitor, Kis 4.4, 9.2, 480.2, 14.7 nM for hCA II, I, IV, IX. Used in glaucoma research.</p>Formule :C20H25N3O4SCouleur et forme :SolidMasse moléculaire :403.5(S)-Seco-Duocarmycin SA
CAS :<p>(S)-Seco-Duocarmycin SA is a DNA alkylating agent and antibiotic with potent antitumor activity that can be used to synthesize ADC compounds.</p>Formule :C25H24ClN3O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :513.93VEGFR-2-IN-25
CAS :<p>VEGFR-2-IN-25 (compound 5d) is a potent inhibitor of VEGFR-2 (IC50: 12.1 nM).</p>Formule :C24H22N6O2Couleur et forme :SolidMasse moléculaire :426.47GABAA receptor agonist 1
<p>Compound 3e, a potent GABAA agonist, targets GABA sites and has potential anti-depressive effects in mice.</p>Formule :C20H30O3Couleur et forme :SolidMasse moléculaire :318.45Leualacin
CAS :<p>Leualacin is a novel calcium blocker from Hapsidospora irregularis.</p>Formule :C31H47N3O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :573.72Annonin VI
CAS :<p>Annonin VI is a natural inhibitor of NADH:ubiquinone oxidoreductase.</p>Formule :C37H66O7Couleur et forme :SolidMasse moléculaire :622.92O4
CAS :<p>O4 is a novel stabilizer of amyloid- fibrils. O4 used for accelerating the formation of end-stage mature fibrils.</p>Formule :C24H15NO7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :429.38MS117
<p>MS117 is a first-in-class and cell-active irreversible covalent inhibitor of protein arginine methyltransferase 6 (PRMT6) (IC50 = 18 nM) [1].</p>Formule :C17H22N4OCouleur et forme :SolidMasse moléculaire :298.38Hypothemycin
CAS :<p>Hypothemycin, a fungal polyketide, inhibits multiple kinases (VEGFR, MEK, FLT-3, PDGFR, ERK) with Kis ranging from 10 nM to 2.4 μM.</p>Formule :C19H22O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :378.37CK2-IN-3
<p>CK2-IN-3: potent, selective CK2 inhibitor; Kd=12 nM, IC50: 1.51 μM (CK2α), 7.64 μM (CK2α'). For cancer research.</p>Formule :C22H26N4O7Couleur et forme :SolidMasse moléculaire :458.46SP4206
CAS :SP4206 is an interaction inhibitor of IL-2/IL-2Rα (IL-2 and IL-2Rα with Kd of 70 nM and 10 nM,respectively)Formule :C30H37Cl2N7O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :662.56SGLT1/2-IN-1
CAS :<p>SGLT1/2-IN-1 is a dual SGLT1/SGLT2 inhibitor.</p>Formule :C25H28O8Couleur et forme :SolidMasse moléculaire :456.48CDK1-IN-3
<p>CDK1-IN-3 is a selective inhibitor targeting CDK1 (36.8 nM), CDK2 (305.17 nM), CDK5 (369.37 nM); used in cancer research.</p>Formule :C28H25ClF3N5O2Couleur et forme :SolidMasse moléculaire :555.98PSMA-1007
CAS :<p>PSMA-1007 is a novel Glu-Ureido-type prostate-specific membrane antigen (PSMA) inhibitor.</p>Formule :C49H55FN8O16Couleur et forme :SolidMasse moléculaire :1030.01GGTI298
CAS :<p>GGTI298 is a potent GGTase I inhibitor; IC50 3μM for Rap1A, >20μM for Ha-Ras.</p>Formule :C27H33N3O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :479.63UTPγS trisodium salt
CAS :<p>P2Y2 and P2Y4 receptor agonist</p>Formule :C9H12N2Na3O14P3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :566.15Antitumor agent-37
<p>Antitumor agent-37: strong anti-growth, anti-spread, induces DNA damage, apoptosis via Bcl-2/Bax/caspase3, boosts immune response.</p>Formule :C16H18Cl2N2O4PtCouleur et forme :SolidMasse moléculaire :568.32LMD-A
CAS :<p>LMD-A, also known as CCR8 antagonist LMD-A, is a CCR8 antagonist.</p>Formule :C27H32N4O4SCouleur et forme :SolidMasse moléculaire :508.63CDK9-IN-11
CAS :<p>CDK9-IN-11 is a potent CDK9 inhibitor that is the ligand for the PROTAC CDK9 Degrader-1 [1].</p>Formule :C20H25N3O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :371.43VVD-118313
CAS :<p>VVD-118313 (5a) is a potent JAK1 inhibitor targeting allosteric cysteine, blocking cytokine signaling for cancer research.</p>Formule :C19H22Cl2N2O3SCouleur et forme :SolidMasse moléculaire :429.36Antibacterial agent 81
CAS :<p>Antibacterial agent 81 blocks DNA transcription, targets S. aureus (MIC 12.5μM) & M. smegmatis (MIC 7.8μM). Used in infection research.</p>Formule :C33H28N2O8Couleur et forme :SolidMasse moléculaire :580.58SB-423557
CAS :SB-423557 is an orally active antagonist of calcium-sensing receptor (CaR) with IC50 of 520 nMFormule :C28H36N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :464.60Tetrahydrouridine dihydrate
<p>THU dihydrate, a potent CDA inhibitor, outperforms cytidine by blocking the enzyme's active site.</p>Formule :C9H20N2O8Couleur et forme :SolidMasse moléculaire :284.26Osanetant HCl
CAS :<p>Osanetant HCl is the (R)-enantiomer; neurokinin-3 receptor antagonist</p>Formule :C35H42Cl3N3O2Couleur et forme :SolidMasse moléculaire :643.09SJG-136
CAS :SJG-136 is a DNA cross-linking agent (XL50: 45 nM for pBR322 DNA).Formule :C31H32N4O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :556.61BAY-364
CAS :<p>BAY-364 (BAY-299N) functions as an inhibitor targeting the second bromine domain in TAF1, demonstrating inhibitory effects on TAF1 in Kasumi-1 cells, CD34+</p>Formule :C23H19N3O4Couleur et forme :SolidMasse moléculaire :401.41BAY-899
CAS :<p>BAY-899, oral LH-R antagonist, IC50: 185 nM (hLH), 46 nM (rLH), lowers sex hormones in vivo.</p>Formule :C25H19F2N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :459.45Substituted piperidines-1
CAS :<p>Substituted piperidines-1 can promote the release of growth hormone in humans and animals.</p>Formule :C29H39N7O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :517.67AChE/BACE1/GSK3β-IN-1
<p>AChE/BACE1/GSK3β-IN-1 is an orally active, blood-brain barrier-transparent, moderately bioavailable triple inhibitor of AChE/BACE1/GSK3β.</p>Formule :C26H27FN2O4Couleur et forme :SolidMasse moléculaire :450.5GSK065
CAS :<p>GSK065 is a potent inhibitor of kynurenine-3-monooxygenase (KMO).</p>Formule :C17H15ClN2O4Couleur et forme :SolidMasse moléculaire :346.77MB725
CAS :<p>MB725 is a strong and selective inducer of viability reduction in several cancer cell lines containing the oncogenic p53-Y220C mutation.</p>Formule :C18H21IN4O2SCouleur et forme :SolidMasse moléculaire :484.35Hypoglycemic agent 1
CAS :<p>Hypoglycemic agent 1 has an action for lowering blood sugar. It acts as a therapeutic and/or prophylactic agent for diabetes.</p>Formule :C25H24FN5O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :477.49Antitumor agent-78
<p>Antitumor agent-78 blocks GPx-4, raises COX2, triggers apoptosis, halts EMT, and stifles cancer cell growth and migration.</p>Couleur et forme :SoildNikkomycin Z
CAS :Nikkomycin Z (Nikkomycin Z from Streptomyces tendae) is a competitive chitin synthase inhibitor.It inhibitor of the growth of filamentous fungi, insects,Formule :C20H25N5O10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :495.44Kri 1314
CAS :Kri 1314 is a cyclohexyl-norstatine-containing dipeptide renin inhibitor which has potential for the treatment of hypertension.Formule :C38H51N5O7Couleur et forme :SolidMasse moléculaire :689.84YCW-E11
CAS :<p>YCW-E11 is an antiapoptotic Bcl-2 family proteins inhibitor.</p>Formule :C25H21Cl2N3O6S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :594.49KMH-233
CAS :<p>KMH-233 effectively blocks LAT1, inhibiting L-leucine uptake and cell growth, boosting betastatin and cisplatin efficacy at 25 μM.</p>Formule :C32H25N7O5Couleur et forme :SolidMasse moléculaire :587.58Antifungal agent 27
<p>Antifungal agent 27 shows moderate action against MRSA, weak against C. albicans, with MICs of 8 μg/mL and 32 μg/mL, respectively.</p>Formule :C18H23N5OSCouleur et forme :SolidMasse moléculaire :357.47A1-Phytoprostane-I
CAS :<p>A1-Phytoprostane-I: cyclopentenone from α-linolenic acid in plants, induces gene expression & increases phytoalexin synthesis.</p>Formule :C18H28O4Couleur et forme :SolidMasse moléculaire :308.41ONO-AE1-329
CAS :<p>ONO-AE1-329 is a novel agonist of the prostaglandin PGE2 receptor EP4.</p>Formule :C22H30O6S2Couleur et forme :SolidMasse moléculaire :454.6Glycotriosyl glutamine
CAS :<p>Glycotriosyl glutamine is a nephritogenoside analog.</p>Formule :C23H40N2O18Couleur et forme :SolidMasse moléculaire :632.57NS2B/NS3-IN-3
CAS :<p>NS2B/NS3-IN-3 (Compd 66) is an inhibitor of Flavivirus NS2B-NS3 protease [1] .</p>Formule :C19H21N3O2Couleur et forme :SolidMasse moléculaire :323.39Samuraciclib
CAS :<p>Samuraciclib (CT7001) is an oral CDK7 inhibitor with 41 nM IC50, notable for its high selectivity and potency against breast cancer cells.</p>Formule :C22H30N6OCouleur et forme :SolidMasse moléculaire :394.51
