Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.542 produits)
- Apoptose(5.816 produits)
- Cycle cellulaire/point de contrôle(4.466 produits)
- Chromatine/Épigénétique(2.252 produits)
- Signalisation du cytosquelette(1.381 produits)
- Altération de l'ADN/réparation de l'ADN(2.830 produits)
- Endocrinologie/Hormones(3.518 produits)
- Enzyme(3.640 produits)
- GPCR/G-Protéine(8.362 produits)
- Immunologie et Inflammation(3.540 produits)
- Virus de la grippe(296 produits)
- Signalisation JAK/STAT(405 produits)
- Signalisation MAPK(1.201 produits)
- Transporteur membranaire/Canal ionique(2.809 produits)
- Métabolisme(9.462 produits)
- Microbiologie/Virologie(7.003 produits)
- Neuroscience(9.942 produits)
- Autres inhibiteurs(37.827 produits)
- Oxydation-Réduction(40 produits)
- Signalisation PI3K/Akt/mTOR(1.399 produits)
- Protéases/Protéasome(1.598 produits)
- Cellules souche et Dérivés(830 produits)
- Tyrosine Kinase/Adaptateurs(2.012 produits)
- Ubiquitination(1.651 produits)
Affichez 16 plus de sous-catégories
66618 produits trouvés pour "Inhibiteurs"
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DFBTA
<p>DFBTA inhibits ANO1 with IC50 of 24 nM, effectively treating inflammatory pain orally.</p>Formule :C18H10ClF2NO3SCouleur et forme :SolidMasse moléculaire :393.79ZIKV-IN-5
<p>ZIKV-IN-5 is an acid-stable, low cytotoxic anti-ZIKV agent with an EC50 value of 0.71 μM. ZIKV-IN-5 showed effective inhibition of ZIKV NS5 MTase activity.</p>Formule :C36H45NO4SiCouleur et forme :SolidMasse moléculaire :583.83Lp-PLA2-IN-10
<p>Lp-PLA2-IN-10, a potent Lp-PLA2 inhibitor, may research neurodegenerative and cardiovascular diseases.</p>Formule :C21H15F5N4O4Couleur et forme :SolidMasse moléculaire :482.36Falecalcitriol
CAS :<p>Falecalcitriol is an analog of calcitriol. It has a higher potency both in vivo and in vitro systems, which is longer duration of action in vivo.</p>Formule :C27H38F6O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :524.58RDN2150
CAS :<p>RDN2150 (Compound 25), a ZAP-70 inhibitor with an IC50 of 14.6 nM, covalently binds to the C346 residue of ZAP-70, suppressing the expression of CD25 and CD69</p>Formule :C28H29ClN8O4Couleur et forme :SolidMasse moléculaire :577.03FGFR4-IN-4
CAS :<p>FGFR4-IN-4 is a FGFR4 inhibitor with anti-tumor activity.</p>Formule :C28H32Cl2N6O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :603.5T-2513 hydrochloride
CAS :<p>T-2513 hydrochloride: selective topoisomerase I inhibitor, binds DNA complex, halts DNA/RNA synthesis, causes cell death.</p>Formule :C25H28ClN3O5Couleur et forme :SolidMasse moléculaire :485.96MtMetAP1-IN-1
<p>MtMetAP1-IN-1 is an inhibitor of methionine aminopeptidase 1 ( MetAP1 ). MtMetAP1-IN-1 shows antimycobacterial activity.</p>Formule :C15H10BrN5O2SCouleur et forme :SolidMasse moléculaire :404.24HOE-288
CAS :<p>HOE-288 is a converting enzyme (CE) inhibitor.</p>Formule :C27H38N2O5Couleur et forme :SolidMasse moléculaire :470.60Dopamine D3 receptor antagonist-1
<p>Dopamine D3 receptor antagonist-1 is a dopamine D3 receptor selective or multi-targeting ligand with a Ki value of 1.58 nM that has demonstrated therapeutic</p>Formule :C31H35Cl2N3O3Couleur et forme :SolidMasse moléculaire :568.53MA242 free base
CAS :<p>MA242 free base is a dual MDM2/NFAT1 inhibitor that triggers apoptosis in pancreatic cancer cells.</p>Formule :C24H20ClN3O3SCouleur et forme :SolidMasse moléculaire :465.95SSR 146977
CAS :<p>NK3 receptor antagonist</p>Formule :C35H42Cl2N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :621.64Sucistil
<p>Sucistil is an active biochemical. hemoglobin sucistil (bovine) is an oxygen carrier [1].</p>Formule :C9H15NO4SCouleur et forme :SolidMasse moléculaire :233.28Oncopterin
CAS :<p>Oncopterin is found in urine from patients with solid and blood cancers.</p>Formule :C12H18N6O3Couleur et forme :SolidMasse moléculaire :294.31CCR1 antagonist 11 hydrochloride
<p>Oral CCR1 antagonist A1B1 targets h/m/rCCR1 (IC50: 0.03/0.58/0.32 μM), potential for treating inflammatory diseases.</p>Couleur et forme :SolidADP-2341
<p>ADP-2341 is a soluble analog of FiVe1.</p>Formule :C24H29Cl2N5O3Couleur et forme :SolidMasse moléculaire :506.43CXCR2 antagonist 4
<p>CXCR2 antagonist 4 inhibits CXCR2 (IC50: 0.13 μM) and CXCL8-induced calcium rise (IC50: 27 μM), promising for cancer research.</p>Formule :C15H14F2N4OS2Couleur et forme :SolidMasse moléculaire :368.42NNTA
CAS :<p>NNTA is a highly selective and potent activator of μ/κ-opioid heteromers.</p>Formule :C31H32N2O4Couleur et forme :SolidMasse moléculaire :496.60GnRH-R antagonist 1
CAS :<p>Compound 21a: Oral GnRH-R antagonist, IC50=0.57 nM, potent against prostate cancer/prevents LH surges.</p>Formule :C31H28F5N7O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :721.65Thiolactomycin
CAS :<p>Thiolactomycin is a novel reversible dual inhibitor of D-amino acid oxidase (DAO) and D-Aspartate oxidase (DDO).</p>Formule :C11H14O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :210.29CDK1-IN-3
<p>CDK1-IN-3 is a selective inhibitor targeting CDK1 (36.8 nM), CDK2 (305.17 nM), CDK5 (369.37 nM); used in cancer research.</p>Formule :C28H25ClF3N5O2Couleur et forme :SolidMasse moléculaire :555.98HIV-1 inhibitor-8
<p>HIV-1 inhibitor-8: potent oral NNRTI, low toxicity, IC50: 0.081 μM, effective on multiple strains, EC50: 4.44-54.5 nM.</p>Formule :C25H21N5OSCouleur et forme :SolidMasse moléculaire :439.53Pyridoxatin
CAS :<p>Pyridoxatin: fungal metabolite; blocks TBARS production, prevents AAPH-induced hemolysis, and acts against C. albicans.</p>Formule :C15H21NO3Couleur et forme :SolidMasse moléculaire :263.33PAD2-IN-1 hydrochloride
<p>PAD2-IN-1 hydrochloride: potent, selective PAD2 inhibitor; 95x less on PAD4, 79x less on PAD3; benzimidazole derivative.</p>Formule :C25H30ClFN6O3Couleur et forme :SolidMasse moléculaire :517GR-112000
CAS :<p>GR-112000 is a peptide-based tachykinin NK2 receptor antagonist.</p>Formule :C30H36N6O3Couleur et forme :SolidMasse moléculaire :528.65VEGFR-2-IN-12
<p>VEGFR-2-IN-12 (compound 6g), a 2-oxoquinoxalinyl-1,2,4-triazole, is a potent inhibitor of VEGFR-2 (IC50: 0.037 μM). VEGFR-2-IN-12 has anti-tumour effects.</p>Formule :C22H24N6O3SCouleur et forme :SolidMasse moléculaire :452.53Ledene
CAS :<p>Ledene (Viridiflorene) is an essential oil produced by viridiflorene synthase.</p>Formule :C15H24Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :204.35PIM1-IN-3
<p>PIM1-IN-3 (HL8) selectively blocks PIM1, induces Colo320 cell apoptosis, and may be researched for cancer.</p>Formule :C27H25BrN6OCouleur et forme :SolidMasse moléculaire :529.43KCL-440
CAS :<p>RS 57639 is a bioactive chemical.</p>Formule :C18H18N2O2Couleur et forme :SolidMasse moléculaire :294.35EB-0176
<p>EB-0176: A valerian derivative; broad-spectrum antiviral; potent ER α-glucosidase I/II inhibitor; IC50s: 0.6439/0.0011 μM.</p>Formule :C23H33N5O7Couleur et forme :SolidMasse moléculaire :491.54LSD1/ER-IN-1
<p>LSD1/ER-IN-1 inhibits ER & LSD1 (IC50: 1.55 μM), and fights MCF-7 breast cancer (IC50: 8.79 μM).</p>Formule :C23H18FNO6SCouleur et forme :SolidMasse moléculaire :455.46Zaragozic acid C
CAS :<p>Zaragozic acid C is an effective inhibitor of squalene synthase.</p>Formule :C40H50O14Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :754.82Gln-AMS TFA
<p>Gln-AMS (TFA) is a type Ia amido-tRNA synthetase (AARS) inhibitor with a Ki value of 1.32 μM for glutaminyl-tRNA synthetase.</p>Formule :C17H23F3N8O10SCouleur et forme :SolidMasse moléculaire :588.47RAD51-IN-8
<p>RAD51-IN-8 inhibits RAD51-BRCA2 interaction and H4A4 with EC50 of 19 μM; a micromolar PPI inhibitor.</p>Formule :C16H14Cl2FN3O2Couleur et forme :SolidMasse moléculaire :370.21OP-5244 sodium
<p>OP-5244 sodium: potent oral CD73 inhibitor (IC50: 0.25 nM), potential in cancer research by hindering adenosine, reversing immunosuppression.</p>Formule :C19H28ClN5NaO9PCouleur et forme :SolidMasse moléculaire :559.87IL-17 modulator 5
CAS :<p>IL-17 modulator 5 is a IL-17 inhibitor, with an IC 50 of 1 nM .</p>Formule :C28H23F6N9O2Couleur et forme :SolidMasse moléculaire :631.53VDR agonist 1
CAS :<p>Compound 28 is a nonsteroidal VDR agonist with 690 nM potency, inducing cell cycle arrest and apoptosis in MCF-7 cells.</p>Formule :C32H51N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :509.77Anticancer agent 62
CAS :<p>Anticancer agent 62 inhibits HepG2, Bel-7402, MCF-7 growth with IC50: 0.019, 0.060, 0.016 μM respectively, and halts tumors.</p>Formule :C20H19ClN3Na2O8PSCouleur et forme :SolidMasse moléculaire :573.85GL0388
<p>GL0388, a Bax activator, induces apoptosis, hinders breast cancer growth, and has IC50 of 0.299-1.57 μM.</p>Formule :C21H17FN2OCouleur et forme :SolidMasse moléculaire :332.37SCP1-IN-1
CAS :<p>SCP1-IN-1 (SH T-62) is a potent inhibitor of SCP1, promoting REST degradation and potentially aiding glioblastoma research.</p>Formule :C20H19F3N2O7S2Degré de pureté :99.53%Couleur et forme :SoildMasse moléculaire :520.5Karenitecin
CAS :<p>Karenitecin (Cositecan) is an inhibitor of topoisomerase I. It has potent anti-cancer activity.</p>Formule :C25H28N2O4SiDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :448.59Sinulatumolin E
CAS :<p>Sinulatumolin E, a terpenoid, inhibits TNF-α (IC 50: 3.6 μM); has anti-inflammatory properties.</p>Formule :C15H22O2Couleur et forme :SolidMasse moléculaire :234.33PPO-IN-1
<p>PPO-IN-1 is a potent inhibitor of protoporphyrinogen IX oxidase (PPO) (Ki: 2.5 nM).</p>Formule :C18H10F3N3O4SCouleur et forme :SolidMasse moléculaire :421.35AP5 sodium
CAS :<p>AP5 sodium: potent oral GPR40 agonist, enhances ligands, may aid type II diabetes research.</p>Formule :C28H27FNNaO4Couleur et forme :SolidMasse moléculaire :483.515BRD4-BD1/2-IN-2
CAS :<p>BRD4-BD1/2-IN-2 inhibits BRD4 BD1/BD2 with IC50 <300 nM/<0.5 nM (WO2021233371A1).</p>Formule :C30H33N5O4Couleur et forme :SolidMasse moléculaire :527.61CDK7/12-IN-1
CAS :<p>CDK7/12-IN-1 is a selective CDK7 (IC50: 3 nM) and CDK12 (IC50: 277 nM) inhibitor, effective against tumor growth.</p>Formule :C25H34N8OCouleur et forme :SolidMasse moléculaire :462.59Kallikrein-IN-1
CAS :<p>Kallikrein-IN-1 (Formula A) is an inhibitor of the kinin-releasing enzyme Kallikrein.</p>Formule :C28H26FN5O4Couleur et forme :SolidMasse moléculaire :515.54FGFR1 inhibitor-6
<p>FGFR1 inhibitor-6, IC50: 16.31 nM, blocks cell cycle at pro-G1/G2/M and induces apoptosis.</p>Formule :C27H19N5O4S2Couleur et forme :SolidMasse moléculaire :541.6AFM-30a hydrochloride
<p>AFM-30a hydrochloride: selective PAD2 inhibitor, EC50 9.5 μM; blocks H3 guanylation, EC50 0.4 μM; used for cancer and autoimmune research.</p>Formule :C24H28ClFN6O3Couleur et forme :SolidMasse moléculaire :502.97GID4 Ligand 1
<p>GID4 Ligand 1: cell-permeable, selective binder, IC50 5.4 μM, Kd 5.6 μM, binds in cells with EC50 558 nM, useful for PROTAC synthesis.</p>Formule :C28H34N4O5SCouleur et forme :SolidMasse moléculaire :538.66TAK-828F
CAS :<p>TAK-828F: potent, selective RORγt inverse agonist. Oral. IC50=1.9 nM; reporter gene IC50=6.1 nM.</p>Formule :C28H32FN3O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :509.57Estrogen receptor antagonist 4
CAS :<p>Estrogen receptor antagonist 4 blocks ER, impacting cell growth and cancer research potential.</p>Formule :C23H29BF4N4O2Couleur et forme :SolidMasse moléculaire :480.31α-Glucosidase-IN-17
CAS :<p>α-Glucosidase-IN-17 (Compound 12B) is a potent and orally active inhibitor of α-glucosidase, demonstrating antidiabetic activity with an inhibitory</p>Formule :C30H27NO2SCouleur et forme :SolidMasse moléculaire :465.61Diospyrin
CAS :<p>Diospyrin is a plant product that has significant inhibitory effect on the growth of Leishmania donovani promastigotes.</p>Formule :C22H14O6Couleur et forme :SolidMasse moléculaire :374.34Etamicastat
CAS :<p>Etamicastat can be used in the research of cardiovascular diseases.</p>Formule :C14H15F2N3OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :311.35Calphostin A
CAS :<p>Calphostins, from Cladosporium fungus, inhibit PKC; calphostin C is most potent, used as a biochemical tool.</p>Formule :C44H38O12Couleur et forme :SolidMasse moléculaire :758.77Bilanafos
CAS :<p>Bilanafos is an agent of Anti-Bacterial.</p>Formule :C11H22N3O6PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :323.28SSTR4 agonist 4
CAS :<p>SSTR4 agonist 4, potent in pain research, shows promise in rodent pain models, with potential for Alzheimer's due to hippocampus activity.</p>Formule :C19H26N4OCouleur et forme :SolidMasse moléculaire :326.44PD-1/PD-L1-IN-30
CAS :<p>PD-1/PD-L1-IN-30: Cancer research inhibitor with 0.018 μM IC50.</p>Formule :C29H28F3NO5Couleur et forme :SolidMasse moléculaire :527.53HDAC/Top-IN-1
CAS :<p>HDAC/Top-IN-1, an oral HDAC/Top inhibitor, targets HDAC1-3,6,8 with low IC50s; blocks S-phase & induces apoptosis in HEL cells.</p>Formule :C29H25FN4O4Couleur et forme :SolidMasse moléculaire :512.53NR1H4 activator 1
CAS :NR1H4 activator 1 is a potent and selective agonist of Famesoid X Receptor (FXR).Formule :C34H53NO7SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :619.85Antibacterial agent 78
<p>Antibacterial agent 78 (compound 30) is an antibacterial agent with improved cytotoxicity profile[1].</p>Formule :C16H23N3S2Couleur et forme :SolidMasse moléculaire :321.5Antitumor agent-72
CAS :<p>Antitumor agent-72 (compound 6w) is a potent anticancer agent that exhibits its anticancer activity by inducing apoptosis via caspase-3 activation and PARP</p>Formule :C25H20ClNO6Couleur et forme :SolidMasse moléculaire :465.88RMG8-8
<p>RMG8-8 shows the excellent efficacy against C. neoformans (1.56 μg/mL).</p>Formule :C41H78N8O5Couleur et forme :SolidMasse moléculaire :763.11Nipradolol
CAS :<p>Nipradolol blocks alpha-1-adrenergic receptors, lowers IOP in rabbits, and reduces NA-induced muscle contraction and dog artery vasodilation.</p>Formule :C15H22N2O6Couleur et forme :SolidMasse moléculaire :326.35CXCR2 antagonist 7
<p>CXCR2 antagonist 7 is a powerful blocker with IC50s: 0.044 μM for binding, 0.66 μM for calcium mobilization.</p>Formule :C14H14F2N6OSCouleur et forme :SolidMasse moléculaire :352.36Homomoschatoline
CAS :Homomoschatoline is an antibacterial isolated from Artabotrys crassifolius.Formule :C19H15NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :321.33EGFR/HER2-IN-7
<p>EGFR/HER2-IN-7: Potent, selective dual inhibitor for MCF-7 cancer; IC50: EGFR 0.18μM, HER2 0.146μM, DHFR 0.907μM.</p>Formule :C19H21N3O2SCouleur et forme :SolidMasse moléculaire :355.45Adiaft
CAS :<p>Adiaftis a bioactive chemical.</p>Formule :C10H11IN2O4Couleur et forme :SolidMasse moléculaire :350.1122-HDHA
CAS :<p>22-HDHA is an oxidation product of docosahexaenoic acid .</p>Formule :C22H32O3Couleur et forme :SolidMasse moléculaire :344.49CI-988
CAS :<p>CCK2 (CCK-B) receptor antagonist</p>Formule :C35H42N4O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :614.73Asimicin
CAS :<p>Asimicin is a effective complex I inhibitor.</p>Formule :C37H66O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :622.92Prohibitin ligand 1
<p>Compound 22i, a prohibitin ligand, protects the heart at nanomolar levels by inducing STAT3 phosphorylation.</p>Formule :C20H22N2OCouleur et forme :SolidMasse moléculaire :306.4MsbA-IN-5
<p>MsbA-IN-5 (compound 40) is a potent and highly selective inhibitor of MsbA (IC50: 2 nM). MsbA-IN-5 can be used in Gram-negative studies.</p>Formule :C23H19Cl2N5OCouleur et forme :SolidMasse moléculaire :452.34Enantiomer of Sofosbuvir
Inactive enantiomer of Sofosbuvir, used for chronic hepatitis C; lacks reported biological activity.Formule :C22H29FN3O9PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :529.455-Ph-IAA-AM
<p>5-Ph-IAA-AM, eggshell-permeable analog of 5-Ph-IAA, boosts protein degradation in embryos, useful for studying proteins in C. elegans.</p>Formule :C19H17NO4Couleur et forme :SolidMasse moléculaire :323.34E 5090
CAS :E5090 is a novel orally active inhibitor of IL-1 generation. It also has anti-inflammatory properties.Formule :C19H20O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :328.36R-96544 hydrochloride
CAS :<p>5-HT2 receptor antagonist</p>Formule :C22H29NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :355.47SMCypI C31
<p>SMCypIC31, a non-peptide cyclophilin inhibitor, blocks PPIase at 0.1 μM IC50 and fights various HCV genotypes (EC50: 1.20-7.76 μM).</p>Formule :C27H30N4O2SCouleur et forme :SolidMasse moléculaire :474.62Anti-MRSA agent 3
CAS :<p>Anti-MRSA agent 3 targets MRSA with 0.098 μg/ml MIC, low toxicity, binds DNA, and disrupts cell walls/membranes.</p>Formule :C29H18BrN3O2Couleur et forme :SolidMasse moléculaire :520.386BChE-IN-5
<p>BChE-IN-5: potent, selective BChE inhibitor (IC50: 2.8 nM), more effective on hBChE, potential in Alzheimer's research.</p>Formule :C30H42N4OCouleur et forme :SolidMasse moléculaire :474.68N'-(2-Fluorophenyl)pyrazine-2-carbohydrazide
<p>N'-(2-Fluorophenyl)pyrazine-2-carbohydrazide is a Ole1p desaturase inhibitor as well as antifungal agent [1].</p>Formule :C11H9FN4OCouleur et forme :SolidMasse moléculaire :232.21Rostratin A
CAS :<p>Rostratin A, a disulfide from Exserohilum rostratum, is cytotoxic to HCT-116 cells with an IC50 of 8.5 μg/mL.</p>Formule :C18H24N2O6S2Couleur et forme :SolidMasse moléculaire :428.52TLR7/8 antagonist 1
<p>Compound 16c, an imidazoquinoline, is a TLR7/8 agonist; IC50: 3.91 μM (TLR7), 2.19 μM (TLR8); targets TLR-2050 for disease treatment.</p>Formule :C24H27N5O2Couleur et forme :SolidMasse moléculaire :417.5Amrubicin HCl
CAS :<p>Amrubicin (SM-5887), an anthracycline, treats lung cancer by inhibiting DNA replication and topoisomerase II, with less cardiac toxicity.</p>Formule :C25H25NO9Couleur et forme :SolidMasse moléculaire :483.47Equisetin
CAS :<p>Equisetin: a QSI from Fusarium equiseti, curbs P. aeruginosa virulence, fights Gram-positive bacteria & HIV-1 integrase; not antibacterial to Gram-negative.</p>Formule :C22H31NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :373.49Integrase-LEDGF/p75 allosteric inhibitor 1
CAS :<p>Oral HIV-1 allosteric integrase inhibitor, blocks DNA integration, antiviral, potent against NL432 (EC50: 3.9 nM).</p>Formule :C33H41NO6SCouleur et forme :SolidMasse moléculaire :579.75AK-295
CAS :<p>AK 295, also known as CX 295, is a dipeptide inhibitor of alpha-ketoamide calpain.</p>Formule :C26H40N4O6Couleur et forme :SolidMasse moléculaire :504.62TTT 3002
CAS :<p>TTT 3002: oral FLT3 inhibitor for AML research, blocks D835 mutations, potent at 0.2 nM IC50.</p>Formule :C27H23N5O3Couleur et forme :SolidMasse moléculaire :465.50BRL-42715
CAS :<p>BRL-42715 is an effective inhibitor of bacterial beta-lactamases.</p>Formule :C10H7N4NaO3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :286.24PNU-140457
CAS :<p>PNU-140457 is a bio-active chemical.</p>Formule :C14H14FN5O3Couleur et forme :SolidMasse moléculaire :319.29Cicaprost
CAS :<p>Cicaprost (ZK 96480) is an IP agonist with artery relaxing effects; EC50 is 5.8 nM.</p>Formule :C22H30O5Couleur et forme :SolidMasse moléculaire :374.47VU6005806
CAS :<p>VU6005806 is a potent M4 PAM with EC50s: 94 nM (human), 28 nM (rat), 87 nM (dog), 68 nM (cyno); studied for neuropsychiatric disorders.</p>Formule :C17H16F3N7O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :439.41GAT564
<p>GAT564, an allosteric CB1R modulator, shows EC50s of 87 nM (cAMP) & 320 nM (β-arrestin2) and lowers IOP effectively in glaucoma mice.</p>Formule :C20H16N2O2SCouleur et forme :SolidMasse moléculaire :348.42DYRKs-IN-1 hydrochloride
CAS :DYRKs-IN-1 HCl inhibits DYRK1A (5 nM IC50) & DYRK1B (8 nM IC50) with antitumor properties.Formule :C30H31Cl2N7O4Couleur et forme :SolidMasse moléculaire :624.52MS8815
CAS :<p>MS8815 is a selective EZH2 PROTAC degrader with IC50 of 8.6 nM, used in triple-negative breast cancer research.</p>Formule :C65H87N9O8SCouleur et forme :SolidMasse moléculaire :1154.51TP-6076
CAS :<p>TP-6076 is a fluorocycline antibiotic, inhibiting bacterial protein synthesis, exhibiting great antimicrobial activity against carbapenem-resistant A.</p>Formule :C28H32F3N3O7Couleur et forme :SolidMasse moléculaire :579.56Cilobamine mesylate
CAS :<p>Cilobamine mesylate is a drug which acts as a norepinephrine-dopamine reuptake inhibitor (NDRI) and has stimulant and antidepressant effects.</p>Formule :C18H27Cl2NO4SCouleur et forme :SolidMasse moléculaire :424.38(2S,3R)-LP99
CAS :(2S,3R)-LP99 is a less active enantiomer of LP99.Formule :C26H30ClN3O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :516.05Anticancer agent 142
CAS :<p>Compound 142 (also known as Compound 235) is a PTPN inhibitor with potential applications in cancer research [1].</p>Formule :C13H14BrF2N2O7PS2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :523.26BTK-IN-8
<p>BTK-IN-8: potent, selective covalent BTK inhibitor; IC50=0.22 nM, Kd=0.91 nM; effective in blood CD69 cells (IC50=0.029 μM).</p>Formule :C26H36N6O3Couleur et forme :SolidMasse moléculaire :480.6FW 34569
CAS :<p>FW 34569, an enkephalin analog, boosts growth hormones and prolactin, reduces cortisol and LH; FSH stable.</p>Formule :C30H43N5O7SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :617.76AL-GDa62
<p>AL-GDa62, a gastric cancer treatment lead, has EC50 of 3.2 μM (MCF10A-WT) and 2 μM (MCF10A-CDH1 -/-).</p>Formule :C24H28FN3OCouleur et forme :SolidMasse moléculaire :393.54-Bromo A23187
CAS :<p>4-Bromo A23187 is a halogenated analog of the calcium ionophore A-23187. 4-Bromo A23187 is a calcium modulator and induces apoptosis in different cells.</p>Formule :C29H36BrN3O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :602.52HbF inducer-1
<p>HbF inducer-1 is a fetal hemoglobin inducer which is orally bioavailable.</p>Formule :C18H19N3O3Couleur et forme :SolidMasse moléculaire :325.36Vibegron
CAS :<p>Vibegron (MK-4618) is an effective and selective Beta 3 adrenergic receptor agonist, used to treat overactive bladder (OAB).</p>Formule :C26H28N4O3Couleur et forme :SolidMasse moléculaire :444.53IACS-8779
CAS :<p>IACS-8779 is a potent STING agonist that efficiently stimulates interferon gene activity and exhibits strong systemic antitumor effects.</p>Formule :C21H25N9O10P2S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :689.55Antifungal agent 38
<p>Antifungal agent 38, a heterocyclic disulfide, shrinks hyphae and damages cell membranes, causing leakage.</p>Formule :C8H12N2S2Couleur et forme :SolidMasse moléculaire :200.32RET-IN-9
CAS :<p>RET-IN-9 is a potent RET kinase inhibitor, potentially useful for studying RET-related diseases, including lung and thyroid cancer.</p>Formule :C26H27N9OCouleur et forme :SolidMasse moléculaire :481.55Ph-Ph+
<p>Ph-Ph+ is a dimerized phenanthroline derivative with antitumor, antibacterial, and antifungal effects.</p>Formule :C24H17N4Couleur et forme :SolidMasse moléculaire :361.42Detajmium
CAS :Detajmium is an anti-arrhythmia compound. It is an Na(+)-channel-blocking drug with an extremely long recovery from use-dependent sodium channel block.Formule :C27H42N3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :456.64Emtricitabine triphosphate
CAS :<p>Emtricitabine triphosphate is an active metabolite of Emtricitabine, a drug for HIV/HBV that inhibits reverse transcriptase.</p>Formule :C8H13FN3O12P3SCouleur et forme :SolidMasse moléculaire :487.19MEN-10354
CAS :<p>MEN-10354 is a less potent and less selective NK-2 tachykinin receptor antagonist compared to the linear analog, R 396.</p>Formule :C37H46N8O9Couleur et forme :SolidMasse moléculaire :746.81Topoisomerase I/II inhibitor 2
<p>Compound 1a inhibits Topoisomerase I/II, shrinks mouse liver tumors, IC50: 6.83/9.82 μM for LM9/Huh7 cells.</p>Formule :C19H16N2O4Couleur et forme :SolidMasse moléculaire :336.34Hypothemycin
CAS :<p>Hypothemycin, a fungal polyketide, inhibits multiple kinases (VEGFR, MEK, FLT-3, PDGFR, ERK) with Kis ranging from 10 nM to 2.4 μM.</p>Formule :C19H22O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :378.37AKT-IN-11
<p>AKT-IN-11 is one of the most potent antibacterial agents against human hepatocellular carcinoma Bel-7402 cell line (IC50: 1.15 μM).</p>Formule :C27H27ClF3NO4Couleur et forme :SolidMasse moléculaire :521.963-IN-PP1
CAS :<p>3-IN-PP1: PKD inhibitor (IC50: 94-108 nM for PKD1/2/3), broad anticancer agent for research.</p>Formule :C17H18N6Couleur et forme :SolidMasse moléculaire :306.36L 156903
CAS :<p>L 156903 is a bioactive chemical. It also inhibits the binding of neurotensin to brain tissue.</p>Formule :C35H41N7O5SCouleur et forme :SolidMasse moléculaire :671.81Carboxylesterase-IN-3
CAS :<p>Carboxylesterase-IN-3 is a potent inhibitor of Carboxylesterase Notum (IC50 ≤ 10 nM).Carboxylesterase-IN-3 has the potential to study cancer diseases.</p>Formule :C11H6Cl2N4OSDegré de pureté :97.49% - 98.47%Couleur et forme :SolidMasse moléculaire :313.16L-Sepiapterin
CAS :<p>L-Sepiapterin aids in making BH4, a coenzyme essential for eNOS, enhancing artery function and angiogenesis, while suppressing ovarian cancer cell growth.</p>Formule :C9H11N5O3Couleur et forme :SolidMasse moléculaire :237.22Dual AChE-MAO B-IN-1
<p>Dual AChE-MAO B-IN-1: orally active CNS-permeable, safe, stable neuroprotective agent; AChE IC50=550 nM, MAO-B IC50=8.2 nM.</p>Formule :C23H25F2NO4Couleur et forme :SolidMasse moléculaire :417.45AD012
<p>AD012, a dual cACE/NEP inhibitor, leverages lenopril-tryptophan for potential anti-hypertensive and cardioprotective benefits.</p>Formule :C25H32N2O6Couleur et forme :SolidMasse moléculaire :456.53SARS-CoV-2-IN-8
<p>SARS-CoV-2-IN-8 is a major protease inhibitor of SARS-CoV-2 (IC50: 0.75 μM).</p>Formule :C35H38N6O3Couleur et forme :SolidMasse moléculaire :590.71Lapaquistat
CAS :<p>Lapaquistat: active TAK-475 metabolite; reduces cholesterol synthesis and statin myotoxicity.</p>Formule :C31H39ClN2O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :603.1ZLWT-37
<p>ZLWT-37: Oral CDK inhibitor, CDK9 IC50=0.002 µM, CDK2 IC50=0.054 µM; halts HCT116 cells at G2/M, induces apoptosis.</p>Formule :C26H30ClN5OCouleur et forme :SolidMasse moléculaire :464Fonsartan free acid
CAS :<p>Fonsartan: Angiotensin receptor blocker, halts angiotensin II effects on rat vascular cells.</p>Formule :C26H32N4O5S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :544.69microRNA-21-IN-1
CAS :<p>microRNA-21-IN-1: microRNA inhibitor, curbs HeLa/HCT-116 growth (IC50: 5.5/2.8 μM), induces HeLa apoptosis, elevates PTEN/EGR1/SLIT2, for cancer research.</p>Formule :C30H37FN6O3Couleur et forme :SolidMasse moléculaire :548.65BMT-052
CAS :<p>BMT-052 is a potent and selective Pan-genotypic HCV NS5B Polymerase Inhibitor (EC50 = 7 nM).</p>Formule :C30H17D9F4N6O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :635.61ERK1/2 inhibitor 6
CAS :<p>ERK1/2 inhibitor 6 - potent cancer/inflammation treatment from WO2021063335A1.</p>Formule :C27H29ClFN7O5Couleur et forme :SolidMasse moléculaire :586.01p38 MAPK-IN-3
<p>Compound 2c is a potent p38α MAPK inhibitor with antitumor effects, enhancing apoptosis and ROS.</p>Formule :C22H17BrO2Couleur et forme :SolidMasse moléculaire :393.27GLS-1-IN-1
<p>GLS-1-IN-1 (compound 1d) is a GLS-1 inhibitor that inhibits Hep G2, MCF 7 and MCF 10A cells.</p>Formule :C26H25FN4OSCouleur et forme :SolidMasse moléculaire :460.57ZD6021
CAS :<p>ZD6021 is an antagonist of neurokinin 1 receptor.</p>Formule :C35H35Cl2N3O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :632.64Menin-MLL inhibitor 26
CAS :<p>Menin-MLL inhibitor 26: Active reference, inhibits cell growth, used in leukemia research.</p>Formule :C27H29F3N6O3SCouleur et forme :SolidMasse moléculaire :574.62A 74273
CAS :<p>A 74273, a nonpeptidic and renin inhibitor, may be used to treat cardiovascular diseases due to renin inhibition.</p>Formule :C44H74N4O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :787.08Dinordrin
CAS :Dinordrin is an implantation inhibitor and hormone.Formule :C27H36O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :424.57Polvitolimod
CAS :<p>Polvitolimod is a TLR7 agonist used to treat infectious disease and cancer.</p>Formule :C13H14FN5O4Couleur et forme :SolidMasse moléculaire :323.28MK-8318
CAS :<p>MK-8318 is an effective and selective antagonist of the CRTh2 receptor (Ki: 5.0 nM).</p>Formule :C27H26F4N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :534.5STING agonist-20
CAS :<p>STING agonist-20: potent, aids in XMT-2056 synthesis, used as a cancer vaccine adjuvant.</p>Formule :C36H39N11O8Couleur et forme :SolidMasse moléculaire :753.76LT-850-166
<p>LT-850-166 is a potent inhibitor of FLT3 and has shown efficacy in overcoming a wide range of FLT3 mutations.</p>Formule :C30H29Cl2N7OCouleur et forme :SolidMasse moléculaire :574.5Combretastatin A1 phosphate
CAS :<p>Combretastatin A1 phosphate: potent anti-angiogenic and tumor vascular disruptor, with research potential in pancreatic neuroendocrine tumors.</p>Formule :C18H22O12P2Couleur et forme :SolidMasse moléculaire :492.31eIF4A3-IN-6
CAS :<p>eIF4A3-IN-6 is a potent eIF4A inhibitor, potentially used for treating eIF4A-related diseases like cancer. (US20170145026A1)</p>Formule :C26H25N3O5Couleur et forme :SolidMasse moléculaire :459.49Anti-inflammatory agent 13
<p>Pentacyclic triterpene, Anti-inflammatory 13 inhibits DAMP/PAMP inflammation models.</p>Formule :C30H48O4Couleur et forme :SolidMasse moléculaire :472.7USP7-IN-10
CAS :<p>USP7-IN-10 is a potent inhibitor of ubiquitin-specific protease 7 (USP7), exhibiting an inhibition concentration half-maximal (IC50) value of 13.39 nM.</p>Formule :C26H29ClN4O3SCouleur et forme :SolidMasse moléculaire :513.05NUCC-555
CAS :<p>NUCC-555 is a first-in-class antagonist of activin. It opens a completely new approach to inhibiting the activity of TGF-beta receptor superfamily members.</p>Formule :C25H25N5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :443.5Pyripyropene A
CAS :<p>Pyripyropene A is a potent and selective inhibitor of sterol O-acyltransferase 2 (SOAT2)/acyl-coenzyme A:cholesterol acyltransferase 2 (ACAT2)(IC50 of 0.07 μM).</p>Formule :C31H37NO10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :583.63TAI-95
CAS :<p>TAI-95 is an inhibitor of highly expressed cancer protein 1 (Hec1).</p>Formule :C24H23N5O3S2Couleur et forme :SolidMasse moléculaire :493.60Macropa-NCS
CAS :<p>Macropa-NCS is a macropa bifunctional analog with antitumor activity and can be used to study prostate cancer.</p>Formule :C27H35N5O8SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :589.66Anticancer agent 53
CAS :<p>Anticancer agent 53 exhibits potent in vitro cytotoxicity, triggers apoptosis, halts S/G2/M cycle, and has antitumor effects without toxicity.</p>Formule :C31H25FN4O6SCouleur et forme :SolidMasse moléculaire :600.62LY503430
CAS :<p>LY503430: Oral AMPA enhancer with nootropic, neuroprotective properties, mitigates 6-OHDA/MPTP brain damage.</p>Formule :C20H25FN2O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :392.49M-89 MLL inhibitor
CAS :<p>M-89, a potent Menin-MLL blocker: Kd 1.4 nM, IC50 25 nM for MV4;11 cells, 55 nM for MOLM-13, >100x selective over HL-60.</p>Formule :C37H47N5O4SCouleur et forme :SolidMasse moléculaire :657.87RET-IN-10
CAS :<p>RET-IN-10: Potent RET inhibitor, may treat congenital megacolon and tumors (Patent WO2021135938A1, compound 18).</p>Formule :C29H28N8OSCouleur et forme :SolidMasse moléculaire :536.65TA-316
CAS :<p>Agent induces megakaryocytes/platelets from stem cells to treat thrombopenia.</p>Formule :C28H25BrN4O5S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :641.56AChE-IN-10
<p>AChE-IN-10 (24r) inhibits AChE (IC50=2.4 nM), reducing amyloid buildup, tau phosphorylation, and promotes neuron health.</p>Formule :C23H27F2NO4SCouleur et forme :SolidMasse moléculaire :451.53Sekdel sequence
CAS :Sekdel sequence, as a signal, leads to retention of at least two proteins in the endoplasmic reticulum of animal cells.Formule :C29H49N7O14Couleur et forme :SolidMasse moléculaire :719.74Pol I-IN-1
<p>Pol I-IN-1 is a powerful inhibitor of RNA polymerase I (Pol I), specifically targeting the large catalytic subunit RPA194, demonstrating an inhibition</p>Formule :C23H22N4O2Couleur et forme :SolidMasse moléculaire :386.45USP7-IN-6
CAS :<p>USP7-IN-6 is a potent inhibitor of ubiquitin-specific protease 7 (USP7, IC50: 6.8 nM).</p>Formule :C41H43N7O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :729.89(S)-Purvalanol B
CAS :<p>(S)-Purvalanol B is the S enantiomer of Purvalanol B. Purvalanol B is an inhibitor of cyclin-dependent kinase(CDK) .</p>Formule :C20H25ClN6O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :432.9Namitecan
CAS :Namitecan is an effective inhibitor of topoisomerase I. It has antitumor property.Formule :C23H22N4O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :434.44Latrunculin M
CAS :<p>Latrunculin M, a novel marine toxin, disrupts microfilament organization in cultured cells.</p>Formule :C21H33NO5SCouleur et forme :SolidMasse moléculaire :411.55Carbonic anhydrase inhibitor 5
<p>Potent hCA inhibitor: targets hCA II, IX & XII with IC50s of 42.9, 47.6, & 6.7 nM respectively.</p>Formule :C24H20ClN3O3SCouleur et forme :SolidMasse moléculaire :465.95CV 5975
CAS :<p>CV 5975 is a nonsulfhydryl ACE inhibitor that was investigated for use in hypertension and heart failure.</p>Formule :C22H31N3O5SCouleur et forme :SolidMasse moléculaire :449.56Steroid sulfatase/17β-HSD1-IN-3
<p>Steroid sulfatase/17β-HSD1-IN-3 (compound 19) is a dual inhibitor of steroid sulfatase (STS) and 17β-hydroxysteroid dehydrogenase type 1 (17β HSD1).</p>Formule :C19H17ClN2O5SCouleur et forme :SolidMasse moléculaire :420.87YW3-56
CAS :<p>YW3-56 is a potent peptidylarginine deiminase (PAD) inhibitor, with an IC50 of 1-5 μM for PAD4.</p>Formule :C27H32ClN5O2Couleur et forme :SolidMasse moléculaire :494.03WIN 66306
CAS :<p>WIN 66306: Cyclic heptapeptide, blocks NK1/NK2 receptors, inhibits substance P-triggered contractions in guinea pig ileum.</p>Formule :C41H52N8O9Couleur et forme :SolidMasse moléculaire :800.9Mesulergine
CAS :<p>Mesulergine is metabolized into dopaminergic agonists.</p>Formule :C18H26N4O2SCouleur et forme :SolidMasse moléculaire :362.49Chitin synthase inhibitor 8
<p>Chitin synthase inhibitor 8 is a chitin synthase (CHS) inhibitor with broad-spectrum antifungal effects that can be used in studies related to fungal infections</p>Formule :C23H23N3O5Couleur et forme :SolidMasse moléculaire :421.45IRE1α kinase-IN-5
<p>IRE1α kinase-IN-5 (compound 7) is a potent inhibitor of IRE1α (Ki: 98 nM) and is an ATP-competitive ligand for IRE1α.</p>Formule :C28H30N6O3SCouleur et forme :SolidMasse moléculaire :530.64Salvinorin A Propionate
CAS :<p>Salvinorin A propionate: partial KOR agonist, Ki=32.6 nM, EC50=4.7 nM; ignores μ/δ/ORL-1, non-opioid receptors; less potent analgesic vs. salvinorin A.</p>Formule :C24H30O8Couleur et forme :SolidMasse moléculaire :446.49Chitin synthase inhibitor 7
<p>Compound 9c, a chitin synthase inhibitor, has an IC50 of 0.37 nM and is useful for studying fungal infections.</p>Formule :C24H25N3O5Couleur et forme :SolidMasse moléculaire :435.47Cilazaprilat
CAS :<p>Cilazaprilat is the active metabolite of cilazapril, a pyridazine angiotensin-converting enzyme (ACE) inhibitor with antihypertensive activity.</p>Formule :C20H27N3O5Couleur et forme :SolidMasse moléculaire :389.4516,16-Dimethyl prostaglandin E2
CAS :<p>16,16-Dimethyl prostaglandin E2 regulates hematopoietic stem cells via EP2/EP4 and Wnt, taken orally.</p>Formule :C22H36O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :380.52SHR902275
CAS :<p>SHR902275: potent RAF inhibitor, hits RAS mutations, oral use. cRAF IC50=1.6 nM, bRAFwt IC50=10 nM, bRAFV600E IC50=5.7 nM, hinders cell growth.</p>Formule :C26H23F3N4O4Couleur et forme :SolidMasse moléculaire :512.48BPN-15606 besylate
<p>BPN-15606 besylate is a potent oral γ-secretase regulator reducing Aβ42 and Aβ40 with good pharmacokinetics. IC50: 7 nM (Aβ42), 17 nM (Aβ40).</p>Formule :C29H29FN6O4SCouleur et forme :SolidMasse moléculaire :576.64ChE/Aβ1-42-IN-1
<p>ChE/Aβ1-42-IN-1 (compound 28) is a potent aggregation inhibitor of ChE and Aβ 1-42 with excellent BBB permeability.</p>Formule :C19H24N2O3Couleur et forme :SolidMasse moléculaire :328.41P300 bromodomain-IN-1
<p>P300 bromodomain-IN-1 blocks c-Myc, induces G1/G0 arrest, apoptosis. Potent EP300 inhibitor (IC50: 49 nM).</p>Formule :C29H31ClN4O4Couleur et forme :SolidMasse moléculaire :535.03AZD0424
CAS :<p>AZD0424: oral Src/Abl kinase inhibitor; potential anticancer; induces apoptosis, cell cycle arrest in lymphoma.</p>Formule :C25H29ClN6O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :528.99Kahweol Acetate
CAS :<p>Kahweol Acetate, a semi-synthetic coffee bean derivative, inhibits osteoclasts, cancer cells, DNA damage, and oxidative stress.</p>Formule :C22H28O4Couleur et forme :SolidMasse moléculaire :356.46JTE 151A
CAS :<p>JTE-151 is a novel RORγ inverse agonist.</p>Formule :C26H30ClN3O5Couleur et forme :SolidMasse moléculaire :499.99Estrogen receptor antagonist 6
CAS :<p>Estrogen receptor antagonist 6 is a potent blocker of estrogen signaling, regulating various biological effects. (Compound 166)</p>Formule :C25H31F3N2O3Couleur et forme :SolidMasse moléculaire :464.52LRRK2-IN-4
CAS :<p>LRRK2-IN-4: Potent, selective LRRK2 inhibitor, oral, BBB-penetrating, IC50=2.6 nM, potential for Parkinson's.</p>Formule :C25H29ClF2N6O2Couleur et forme :SolidMasse moléculaire :518.99ACHN-975 TFA
CAS :<p>ACHN-975 TFA is a selective LpxC inhibitor with a subnanomolar inhibitory. It is against a wide range of gram-negative bacterias with low MIC values (≤1 μg/mL).</p>Formule :C22H24F3N3O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :483.4377AMG-222 tosylate
CAS :<p>AMG-222 tosylate is a DPP-IV inhibitor in clinical development for type II diabetes.</p>Formule :C39H47N9O6SCouleur et forme :SolidMasse moléculaire :769.91GW-597901 cinnamate
CAS :<p>GW-597901 cinnamate is a long-acting beta(2)-agonist.</p>Formule :C34H46N2O8SCouleur et forme :SolidMasse moléculaire :642.80Anti-Aβ agent 1A
<p>Anti-Aβ agent 1A is a potent anti-amyloid-β agent.</p>Formule :C35H49NO4Couleur et forme :SolidMasse moléculaire :547.77Tasidotin hydrochloride
CAS :<p>Tasidotin hydrochloride, a dolastatin 15 analog, inhibits microtubule assembly and dynamics.</p>Formule :C32H59ClN6O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :643.30Vulolisib
CAS :<p>Vulolisib inhibits PI3K (α: IC50 0.2nM, β: 168nM, γ: 90nM, δ: 49nM), taken orally with anti-cancer properties.</p>Formule :C18H19F2N5O3SCouleur et forme :SolidMasse moléculaire :423.44ERRγ agonist-1
<p>ERRγ agonist-1 can be used in neuropsychological disorders research.</p>Formule :C17H21N5OCouleur et forme :SolidMasse moléculaire :311.38ZK824859 hydrochloride
<p>ZK824859 hydrochloride: oral uPA inhibitor with IC50 of 79 nM (uPA), 1580 nM (tPA), 1330 nM (fibrin).</p>Formule :C23H23ClF2N2O4Couleur et forme :SolidMasse moléculaire :464.89MY-875
<p>MY-875 inhibits microtubule formation, binds like colchicine (IC50: 0.92 μM), activates Hippo pathway, and induces apoptosis with anticancer properties.</p>Formule :C21H25NO6Couleur et forme :SolidMasse moléculaire :387.43Tovinontrine
CAS :<p>Tovinontrine (IMR-687) (IMR-687) is a potent and selective inhibitor of phosphodiesterase-9 (PDE9), designed to target sickle cell disease treatment.</p>Formule :C21H26N6O2Degré de pureté :98.14%Couleur et forme :SolidMasse moléculaire :394.47LH secretion antagonist 1
CAS :<p>LH secretion antagonist 1 is an antagonist of luteinizing hormone secretion with analgesic activity.</p>Formule :C18H24ClNO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :321.84Org-31710
CAS :<p>Org-31710 is a progesterone receptor antagonist potentially for contraception.</p>Formule :C30H39NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :445.64CVT-5440
CAS :<p>CVT-5440 is a selective, high-affinity (2B) adenosine receptor antagonist with good selectivity.</p>Formule :C27H28N6O5Couleur et forme :SolidMasse moléculaire :516.55TMC353121
CAS :TMC353121 is an effective inhibitor of respiratory syncytial virus fusion (pEC50: 9.9).Formule :C32H42N6O3Degré de pureté :≥98%Couleur et forme :SolidMasse moléculaire :558.71HBV-IN-12
CAS :<p>HBV-IN-12: strong HBsAg & HBV DNA inhibitor; EC50 0.001-0.05 μM & 0.001-0.02 μM respectively. (WO2021204252A1)</p>Formule :C23H27NO8Couleur et forme :SolidMasse moléculaire :445.46FtsZ-IN-4
<p>FtsZ-IN-4 is an oral FtsZ inhibitor with strong antibacterial effects and good drug traits, low toxicity (CC50 >20μg/mL).</p>Formule :C21H16ClF2NO2Couleur et forme :SolidMasse moléculaire :387.815(S),6(S)-DiHETE
CAS :<p>5(S),6(S)-DiHETE: a 5,6-dihydroxy acid from LTA4 hydrolysis, lacks leukotriene activity.</p>Formule :C20H32O4Couleur et forme :SolidMasse moléculaire :336.47DNA-PK-IN-2
CAS :<p>DNA-PK-IN-2 is an inhibitor of the DNA-PK enzyme complex, useful in cancer research.</p>Formule :C20H23N5O3Couleur et forme :SolidMasse moléculaire :381.43Dehydrocrenatidine
CAS :<p>Dehydrocrenatidine (Kumujian G) is an inhibitor of JAK and induces cell apoptosis.</p>Formule :C15H14N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :254.28PptT-IN-1
<p>PptT-IN-1, a potent PptT inhibitor (IC50: 2.8 μM), shows promise for tuberculosis research.</p>Formule :C18H29N5O2Couleur et forme :SolidMasse moléculaire :347.46
