Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.847 produits)
- Apoptose(6.334 produits)
- Cycle cellulaire/point de contrôle(4.889 produits)
- Chromatine/Épigénétique(2.616 produits)
- Signalisation du cytosquelette(1.579 produits)
- Altération de l'ADN/réparation de l'ADN(2.869 produits)
- Endocrinologie/Hormones(3.753 produits)
- Enzyme(3.673 produits)
- GPCR/G-Protéine(9.028 produits)
- Immunologie et Inflammation(3.938 produits)
- Virus de la grippe(300 produits)
- Signalisation JAK/STAT(415 produits)
- Signalisation MAPK(1.259 produits)
- Transporteur membranaire/Canal ionique(3.159 produits)
- Métabolisme(10.131 produits)
- Microbiologie/Virologie(7.628 produits)
- Neuroscience(10.544 produits)
- Autres inhibiteurs(35.859 produits)
- Oxydation-Réduction(40 produits)
- Signalisation PI3K/Akt/mTOR(1.435 produits)
- Protéases/Protéasome(1.692 produits)
- Cellules souche et Dérivés(732 produits)
- Tyrosine Kinase/Adaptateurs(1.991 produits)
- Ubiquitination(1.727 produits)
Affichez 16 plus de sous-catégories
66511 produits trouvés pour "Inhibiteurs"
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Moflomycin
CAS :Moflomycin is an anthracycline derivative. It exhibits a higher antileukemic activity compared to other anthracyclines.Formule :C25H25IO10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :612.36Lysyllysyllysine
CAS :Lysyllysyllysine is a cationic moiety. It may be used in the construction of gene delivery vectors and DNA nanoparticles.Formule :C18H38N6O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :402.53TH-6
TH-6, a potent HDAC inhibitor (IC50: HDAC1-0.115, 2-0.135, 3-0.242, 6-0.138, 8-2.120 μM), blocks cell migration, invasion, and has anti-tumor properties.Formule :C22H24FN3O5Couleur et forme :SolidMasse moléculaire :429.44Dyrk1A-IN-1
Dyrk1A-IN-1 is a triple inhibitor of Dyrk1A kinase activity, aggregation of tau and α-syn oligomers, with an IC50 value of 119 nM for Dyrk1A kinase.Formule :C23H20N4O3SCouleur et forme :SolidMasse moléculaire :432.49UK-370106
CAS :UK-370106 is a potent and highly selective inhibitor of MMP-3 with IC50 of 23 nM and MMP-12 with IC50 of 42 nM, and potently inhibits cleavage of [3H]-Formule :C35H44N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :572.73HDAC1-IN-3
HDAC1-IN-3 is a potent inhibitor of Pf HDAC1.Formule :C22H24ClN7O2Couleur et forme :SolidMasse moléculaire :453.92RdRP-IN-4
RdRP-IN-4, an oral arylbenzohydrazide, inhibits influenza A/B by targeting PB1 of RdRP, with EC50s of 53 nM (H1N1) and 20 nM (Flu B), and aids infected mice.Formule :C17H17Br2N3O2Couleur et forme :SolidMasse moléculaire :455.14BAY-850 HCl
BAY-850 is a selective probe targeting Atad2A's bromine domain, displacing acetylated H4 peptides and detaching ATAD2 from chromatin at 1μm.Formule :C38H48Cl5N5O3Couleur et forme :SolidMasse moléculaire :800.08H 218-54
CAS :H 218-54 is a renin inhibitor.Formule :C37H56N2O5SCouleur et forme :SolidMasse moléculaire :640.92Tubulin polymerization-IN-35
Tubulin-IN-35 inhibits oxazolylisoindole microtubule formation, targeting VL51 marginal zone lymphoma.Formule :C31H35N3O5Couleur et forme :SolidMasse moléculaire :529.63L-365260 hemihydrate
L-365260 hemihydrate: selective oral CCK-B/gastrin blocker, Ki=1.9/2.0 nM, competes with guinea pig receptors.Formule :C24H24N4O3Couleur et forme :SolidMasse moléculaire :407.47ONL-1204
CAS :ONL-1204 is a small molecule, CD95 antigen inhibitor (Fas inhibitor) being developed by ONL Therapeutics for the treatment of retinal detachment.Formule :C71H100N18O16Couleur et forme :SolidMasse moléculaire :1461.66VEGFR-2-IN-15
VEGFR-2-IN-15 (Compound 14b) is a potent inhibitor of VEGFR-2. VEGFR-2-IN-15 inhibits the growth of HepG2 cells in the Pre-G1 phase and induces apoptosis.Formule :C23H18ClN3O4SCouleur et forme :SolidMasse moléculaire :467.92Steroid sulfatase/17β-HSD1-IN-4
Steroid sulfatase/17β-HSD1-IN-4 (compound 37) is a potent dual inhibitor of steroid sulfatase ( STS ) and 17β-hydroxysteroid dehydrogenase type 1 ( 17β HSD1 ).Formule :C18H17N3O4S2Couleur et forme :SolidMasse moléculaire :403.48NLRP3/AIM2-IN-1
NLRP3/AIM2-IN-1 is an inhibitor of thermal sepsis (IC50 = 3.136 ± 0.7667 μM).Formule :C15H16BNO4Couleur et forme :SolidMasse moléculaire :285.1BRD4-BD1/2-IN-2
CAS :BRD4-BD1/2-IN-2 inhibits BRD4 BD1/BD2 with IC50 <300 nM/<0.5 nM (WO2021233371A1).Formule :C30H33N5O4Couleur et forme :SolidMasse moléculaire :527.61Exicorilant
CAS :Exicorilant is a selective oral GR antagonist (Ki: 7 nM) that may reduce obesity, glucose intolerance, & dyslipidemia.Formule :C26H23F4N7O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :589.56Glycotriosyl glutamine
CAS :Glycotriosyl glutamine is a nephritogenoside analog.Formule :C23H40N2O18Couleur et forme :SolidMasse moléculaire :632.57LSD1/ER-IN-1
LSD1/ER-IN-1 inhibits ER & LSD1 (IC50: 1.55 μM), and fights MCF-7 breast cancer (IC50: 8.79 μM).Formule :C23H18FNO6SCouleur et forme :SolidMasse moléculaire :455.46Nolpitantium Free Base
CAS :Nolpitantium is a potent, selective NK1 receptor antagonist that inhibits substance P without affecting NK2/NK3 receptors.Formule :C37H45Cl2N2O2Couleur et forme :SolidMasse moléculaire :620.67Allosucrose
CAS :Allosucrose is a biochemical.Formule :C12H22O11Couleur et forme :SolidMasse moléculaire :342.30Monorden diacetate
CAS :Monorden diacetate a Hsp90 Inhibitor. Monorden diacetate is a Promising Lead Compound for the Development of Novel Fungicides.Formule :C22H21ClO8Couleur et forme :SolidMasse moléculaire :448.85Tubulin polymerization-IN-9
CAS :Tubulin-IN-9 inhibits tubulin (IC50: 1.82 μM), halts K562 cells in G2/M, induces apoptosis, and has anti-cancer effects.Formule :C19H19NO5SeCouleur et forme :SolidMasse moléculaire :420.32LLS30
CAS :LLS30 inhibits Gal-1, reduces its binding affinity, and may help treat advanced prostate cancer.Formule :C34H33Cl4N5O3Couleur et forme :SolidMasse moléculaire :701.47TCMDC-136230
TCMDC-136230 is a novel inhibitor of Plasmodium calcium kinetics with minimal inhibition of haemoglobin crystallisation.Formule :C24H34N4O2SCouleur et forme :SolidMasse moléculaire :442.62Top/HDAC-IN-2
Top/HDAC-IN-2 (45b) is a dual inhibitor of Top and HDAC that induces apoptosis and exhibits significant anti-tumour effects.Formule :C30H32N8O4Couleur et forme :SolidMasse moléculaire :568.63ICA-105665
CAS :ICA-105665 is an orally active Kv7.2/7.3/7.5 channel opener, CNS-penetrant with antiseizure effects, and low hepatocyte cytotoxicity.Formule :C19H15F2N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :355.34BRD-9526
CAS :BRD-9526 is a potent and selective inhibitor of Sonic Hedgehog (Shh).Formule :C26H31Cl2N3O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :584.51QPX7728 methoxy acetoxy methy ester
CAS :QPX7728 methoxy acetoxy methy ester is an inhibitor of boronic acid β-lactamase.Formule :C14H14BFO7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :324.07Tubulin inhibitor 13
CAS :Tubulin inhibitor 13 (E27), IC50 16.1 μM, blocks tubulin polymerization, cancer cell migration, and invasion, induces apoptosis.Formule :C25H21N3O4Couleur et forme :SolidMasse moléculaire :427.45AZ0108
CAS :AZ0108, an oral PARP1,2,6 inhibitor, selectively blocks centrosome clustering, is viable for in vivo studies, and doesn't inhibit PARP3/TNKS1.Formule :C24H20F4N6O2Couleur et forme :SolidMasse moléculaire :500.45Protopine hydrochloride
CAS :Protopine inhibits thromboxane, lowers intracellular calcium, and reduces cell adhesion by altering adhesive factors.Formule :C20H20ClNO5Degré de pureté :98%Couleur et forme :Prisms From Alc SolidMasse moléculaire :389.83AMD-7049
CAS :AMD-7049 is a biochemical.Formule :C25H39N5Couleur et forme :SolidMasse moléculaire :409.61FLT3/TrKA-IN-1
FLT3/TrKA-IN-1: Potent dual kinase inhibitor for FLT3 & TrKA, promising for AML research.Formule :C28H30N4O2Couleur et forme :SolidMasse moléculaire :454.56ONO-AE1-259 lysine
CAS :ONO-AE1-259 is a highly selective agonist of prostaglandin e2 receptor (ep2)Formule :C28H49ClN2O6Couleur et forme :SolidMasse moléculaire :545.15GT-055
GT-055 (LCB18-055) is a novel inhibitor of broad-spectrum β-lactamase.Formule :C13H20F3N5O8SCouleur et forme :SolidMasse moléculaire :463.39A 74273
CAS :A 74273, a nonpeptidic and renin inhibitor, may be used to treat cardiovascular diseases due to renin inhibition.Formule :C44H74N4O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :787.08Elongation factor P-IN-1
EFP-IN-1: potent β-lysine derivative, inhibits EFP, slows E. coli growth.Formule :C14H31N3O2Couleur et forme :SolidMasse moléculaire :273.41HER2-IN-7
CAS :HER2-IN-7 is a potent HER2 inhibitor with potential for researching ErbB-related diseases, especially cancer.Formule :C28H26F3N7O3Couleur et forme :SolidMasse moléculaire :565.55MsbA-IN-5
MsbA-IN-5 (compound 40) is a potent and highly selective inhibitor of MsbA (IC50: 2 nM). MsbA-IN-5 can be used in Gram-negative studies.Formule :C23H19Cl2N5OCouleur et forme :SolidMasse moléculaire :452.34HPK1-IN-30
CAS :HPK1-IN-30 is a potent inhibitor of HPK1. HPK1-IN-30 has potential for cancer disease research.Formule :C25H23FN6Couleur et forme :SolidMasse moléculaire :426.49Latrunculin M
CAS :Latrunculin M, a novel marine toxin, disrupts microfilament organization in cultured cells.Formule :C21H33NO5SCouleur et forme :SolidMasse moléculaire :411.55GLS1 Inhibitor-6
GLS1 Inhibitor-6: IC50=68nM, 220x more selective for GLS2, has anti-tumor and pro-apoptosis effects.Formule :C37H52N6O3SCouleur et forme :SolidMasse moléculaire :660.91Antitubulin agent 1
Antitubulin agents-1 disrupts microtubules, ups α-tubulin acetylation, and has anticancer properties.Formule :C21H19N3O3Couleur et forme :SolidMasse moléculaire :361.39BM635 hydrochloride (1493762-74-5 free base)
BM635 hydrochloride is an MmpL3 inhibitor with outstanding anti-mycobacterial activity (MIC50: 0.12 μM against M. tuberculosis H37Rv).Formule :C25H30ClFN2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :428.97Tandutinib (MLN518) HCl
Tandutinib antagonizes FLT3, PDGFR, and c-Kit with an IC50 of ~200 nM.Formule :C31H43ClN6O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :599.16Dicetrorelix pamoate
CAS :Cetrorelix pamoate is a synthetic decapeptide that acts as a GnRH antagonist, inhibiting the release of LH and FSH from the pituitary.Formule :C163H200Cl2N34O34Couleur et forme :SolidMasse moléculaire :3250.49NNTA
CAS :NNTA is a highly selective and potent activator of μ/κ-opioid heteromers.Formule :C31H32N2O4Couleur et forme :SolidMasse moléculaire :496.60Fandosentan
CAS :Fandosentan is an endothelin receptor antagonist.Formule :C25H18F3NO6SCouleur et forme :SolidMasse moléculaire :517.47DNA Gyrase-IN-1
DNA Gyrase-IN-1: potent, selective promoter inhibitor. IC50: 2.6 μM, inhibits Mtb, MIC: 0.49 μM. Useful for tuberculosis research.Formule :C24H24FN7O6Couleur et forme :SolidMasse moléculaire :525.49Anticancer agent 44
Anticancer agent 44 induces apoptosis, is selective, cytotoxic to cancer cells, and minimally toxic to human lymphocytes.Formule :C22H13Cl2N3O5S2Couleur et forme :SolidMasse moléculaire :534.39HSP90-IN-11
HSP90-IN-11: potent HSP90 inhibitor, akin to AUY-922; hinders CRC/NSCLC cell proliferation; degrades EGFR, Akt proteins.Formule :C27H30FN3O6Couleur et forme :SolidMasse moléculaire :511.54Lafadofensine (D-(-)-Mandelic acid)
Lafadofensine D-(-)-Mandelic acid is a monoamines reuptake inhibitor with adequate effects when administered short-term.Formule :C32H32F2N2O6Couleur et forme :SolidMasse moléculaire :578.6Aurora/LIM kinase-IN-1
Aurora/LIM kinase-IN-1 (Compound F114) is a dual inhibitor targeting aurora and lim kinases, potentially useful in GBM cancer treatment efforts.Formule :C16H20N6OCouleur et forme :SolidMasse moléculaire :312.37Sulprostone
CAS :EP3 and EP1 receptor agonistFormule :C23H31NO7SDegré de pureté :98%Couleur et forme :White To Off-White SolidMasse moléculaire :465.56Abarelix acetate
CAS :Abarelix acetate: synthetic GnRHR antagonist, spikes histamine, lowers LH and testosterone temporarily, used in advanced prostate cancer.Formule :C72H95ClN14O14·xC2H4O2Couleur et forme :SolidMasse moléculaire :1476.14Antitubercular agent-13
Compound 3d: antitubercular, MIC 0.007 μg/mL vs MTB H37Rv, 1.851 μg/mL vs MDR-MTB 16833, metabolically unstable.Formule :C18H18N4O5Couleur et forme :SolidMasse moléculaire :370.36D4R antagonist-1
Potent, selective D4R antagonist; IC50 = 6.87 µM; potential in Parkinson’s disease research.Formule :C21H25F2NO2Couleur et forme :SolidMasse moléculaire :361.43DNA-PK-IN-2
CAS :DNA-PK-IN-2 is an inhibitor of the DNA-PK enzyme complex, useful in cancer research.Formule :C20H23N5O3Couleur et forme :SolidMasse moléculaire :381.43MDL-28050
CAS :MDL-28050 is a synthetic analog of hirudin 55-65 C-terminal fragment and a peptide inhibitor.Formule :C61H88N10O23Couleur et forme :SolidMasse moléculaire :1329.4Anti-ToCV agent 1
Anti-ToCV agent 1 can be used as a potential anti-ToCV drug.Formule :C22H19FN2O5SCouleur et forme :SolidMasse moléculaire :442.46RET-IN-9
CAS :RET-IN-9 is a potent RET kinase inhibitor, potentially useful for studying RET-related diseases, including lung and thyroid cancer.Formule :C26H27N9OCouleur et forme :SolidMasse moléculaire :481.55ATM Inhibitor-4
ATM Inhibitor -4: selective, potent (IC50: 0.32 nM), inhibits PI3K family, stable, stops mTOR at 1 μM.Formule :C26H29FN6O3Couleur et forme :SolidMasse moléculaire :492.55CXCR7 modulator 2
CAS :CXCR7 modulator 2 is a 7-type C-X-C chemokine receptor (CXCR7) modulator with a Ki of 13 nM.Formule :C29H42N6O3Couleur et forme :SolidMasse moléculaire :522.68DG013A
CAS :DG013A inhibits ERAP1 & ERAP2 (IC50: 33 nM & 11 nM) to research autoimmune diseases & cancer.Formule :C27H37N4O4PCouleur et forme :SolidMasse moléculaire :512.58MRL-494
MRL-494, a small-molecule BamA inhibitor, resists efflux and outer membrane permeability, with antibacterial properties.Formule :C26H35FN16O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :622.66CD73-IN-12
CD73-IN-12, a compound from CN114437038A, shows strong anti-tumor activity by effectively inhibiting CD73 enzyme.Formule :C17H14F2N4O2Couleur et forme :SolidMasse moléculaire :344.32Vimirogant hydrochloride
Vimirogant (VTP-43742) HCl: Oral, selective RORγt inhibitor (IC50: 17 nM, Ki: 3.5 nM), >1000x selectivity over RORα/β, targets Th17, not Th1/2/Treg.Formule :C27H36ClF3N4O3SCouleur et forme :SolidMasse moléculaire :588.21487MtTMPK-IN-2
CAS :MtTMPK-IN-2 inhibits M. tuberculosis TMPK (IC50: 1.1 μM), Mtb H37Rv (MIC: 12.5 μM), and is cytotoxic in MRC-5 cells (EC50: 6.1 μM).Formule :C23H24ClN3O3Couleur et forme :SolidMasse moléculaire :425.91Symplostatin 1
CAS :Symplostatin 1 is a dolastatin 10 analog from the marine cyanobacterium Symploca hydnoides.Formule :C43H70N6O6SCouleur et forme :SolidMasse moléculaire :799.12rel-MDM2/4-p53-IN-3
rel-MDM2/4-p53-IN-3 inhibits MDM2/4-p53 PPI, IC50: MDM2 18.5nM, MDM4 14.8nM, targets cancer research.Formule :C25H24Cl2FN3O3Couleur et forme :SolidMasse moléculaire :504.38UK 356618
CAS :UK 356618 is a potent and selective inhibitor of matrix metalloprotease-3 (IC50: 5.9 nM).Formule :C34H43N3O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :557.72TNP-470
CAS :TNP-470 is a methionine aminopeptidase-2 inhibitor. TNP-470 is also an angiogenesis inhibitor.Formule :C19H28ClNO6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :401.88iNOs-IN-1
iNOs-IN-1 (YPW) is a strong iNOS inhibitor with dose-dependent anti-inflammatory properties, reducing IL-6, iNOS, and NO levels.Formule :C25H30N4O5Couleur et forme :SolidMasse moléculaire :466.539(S)-HEPE
CAS :9(S)-HEPE is a monohydroxy fatty acid derived from EPA. The biological activity of 9(S)-HEPE has not been documented.Formule :C20H30O3Couleur et forme :SolidMasse moléculaire :318.45LRRK2-IN-3
CAS :LRRK2-IN-3: potent, selective oral LRRK2 blocker, BBB-penetrant, IC50 of 0.6 nM in hPBMCs, for Parkinson's research.Formule :C25H29ClF2N6O2Couleur et forme :SolidMasse moléculaire :518.99HIF-1α-IN-5
HIF-1α-IN-5 is an inhibitor of HIF-1α with an IC 50 value of 24 nM in HEK293T cells that also inhibits the activity of MAO-A.Formule :C16H15N3O2Couleur et forme :SolidMasse moléculaire :281.31Finafloxacin
CAS :Finafloxacin is a pH-activated fluoroquinolone, most effective at pH 5.0-6.0, targeting bacterial topoisomerases, used for UTIs and H. pylori infections.Formule :C20H19FN4O4Couleur et forme :SolidMasse moléculaire :398.39AFP-07 free acid
CAS :AFP 07 free acid is a 7,7-difluoroprostacyclin derivative. It also acts as a selective and highly potent agonist for the IP receptor.Formule :C22H30F2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :412.47BW-10
CAS :BW-10 potently inhibits bombesin evoked release of gastrointestinal hormones in vitro and in vivo.Formule :C57H72N14O8Couleur et forme :SolidMasse moléculaire :1081.27AChE-IN-8
AChE-IN-8 (Compound 19), potent acetylcholinesterase blocker; IC50 = 1.95 μM; potential Alzheimer's treatment.Formule :C20H22N4O2SCouleur et forme :SolidMasse moléculaire :382.48AKR1C3-IN-7
AKR1C3-IN-7 (Compound 13) is an effective and selective AKR1C3 inhibitor (IC50=0.19 μM). AKR1C3-IN-7 has antitumor activity.Formule :C24H20N2O4Couleur et forme :SolidMasse moléculaire :400.43PARP-1-IN-1
PARP-1-IN-1: Selective, oral PARP-1 inhibitor with 0.96 nM IC50; well-tolerated and effective in single-dose MDA-MB-436 model.Formule :C23H25FN4OCouleur et forme :SolidMasse moléculaire :392.47Lp-PLA2-IN-10
Lp-PLA2-IN-10, a potent Lp-PLA2 inhibitor, may research neurodegenerative and cardiovascular diseases.Formule :C21H15F5N4O4Couleur et forme :SolidMasse moléculaire :482.36VHL Ligand 8
CAS :VHL Ligand 8, a VHL ligand essential for synthesizing ARD-266, acts as a highly potent VHL E3 ligase-based androgen receptor (AR) PROTAC degrader.Formule :C23H29N3O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :443.49EP-7041 HCl
CAS :EP-7041 is a novel, potent, and selective Factor XIa inhibitor.Formule :C19H27ClN4O4Couleur et forme :SolidMasse moléculaire :410.89Antibiotic LL Z1640-2
CAS :Antibiotic LL Z1640-2 is an inhibitor against the TAK1 activity.Formule :C19H22O7Couleur et forme :SolidMasse moléculaire :362.38MRS2279 diammonium
CAS :MRS2279 diammonium, a P2Y1 antagonist with K i 2.5 nM, IC 50 51.6 nM, blocks ADP-induced platelet aggregation, pK b 8.05.Formule :C13H24ClN7O8P2Couleur et forme :SolidMasse moléculaire :503.77Fumarranol
CAS :Fumarranol inhibits angiogenesis and malaria growth by targeting PfMAP2.Formule :C16H24O4Couleur et forme :SolidMasse moléculaire :280.36PI3K-IN-35
CAS :PI3K-IN-35 (6l) selectively inhibits PI3K-α, β, δ (IC50: 13.98, 7.22, 10.94 μM), blocks G2/M phase, induces apoptosis, and is useful in leukemia research.Formule :C25H23N7O2Couleur et forme :SolidMasse moléculaire :453.5CDK/HDAC-IN-1
CDK/HDAC-IN-1 inhibits CDK2/4/6 & HDAC6 with IC50s: 60.9, 276, 27.2, and 128.6 nM respectively.Formule :C20H18N4O4Couleur et forme :SolidMasse moléculaire :378.38Anticancer agent 65
CAS :Anticancer agent 65: Effective on A549 cells, IC50 1.07 μM, halts S phase, triggers apoptosis, elevates p53/p21, causes ROS and MMP collapse.Formule :C36H63NO5Couleur et forme :SolidMasse moléculaire :589.89FPDT
FPDT combats glioblastoma by inhibiting the AKT pathway; IC50: >100 μM (astrocytes), 45-68 μM (GBM cells).Formule :C16H12FNO2SCouleur et forme :SolidMasse moléculaire :301.34Brostallicin HCl
CAS :Brostallicin, a synthetic MGB, inhibits DNA replication in cancer cells, inducing cell death, effective against MMR-defective tumors.Formule :C30H36BrClN12O5Couleur et forme :SolidMasse moléculaire :760.0417β-HSD1-IN-1
17β-HSD1-IN-1 (Compound 1) can be used in the non-small cell lung cancer (NSCLC) research.Formule :C21H21NO3Couleur et forme :SolidMasse moléculaire :335.4Urease-IN-2
Urease-IN-2 is a non-competitive inhibitor of urease (IC50: 0.94 μM, Ki: 1.6 μM) that non-competitively inhibits Jack bean urease (JBU).Formule :C26H25N5O5S3Couleur et forme :SolidMasse moléculaire :583.7Antioxidant agent-8
Antioxidant agent-8, an oral Aβ 1-42 inhibitor, reduces fibril aggregation & promotes disaggregation; it's neuroprotective & BBB permeable.Formule :C13H12O5Couleur et forme :SolidMasse moléculaire :248.23Carbacyclin
CAS :Carbacyclin, a PGI2 analog, is a prostacyclin (PGI2) receptor agonist and vasodilator with potent inhibitory platelet aggregation.Formule :C21H34O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :350.49FNC-TP trisodium
FNC-TP trisodium, active intracellular FNC form, inhibits NRTI, fights HIV, HBV, and HCV.Formule :C9H11FN6Na3O13P3Couleur et forme :SolidMasse moléculaire :592.11LDHA-IN-5
CAS :LDHA-IN-5 is a novel and potent inhibitor targeting both glycolate oxidase (GO) and lactate dehydrogenase A (LDHA), designed for the treatment of primaryFormule :C27H22FN7O6S3Couleur et forme :SolidMasse moléculaire :655.7MLKL-IN-6
MLKL-IN-6 (compound P28) is a mixed lineage kinase inhibitor that specifically targets the Mixed Lineage Kinase domain-like (MLKL) protein.
Formule :C20H18N4O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :394.383'-Hydroxy Repaglinide
CAS :'3'-Hydroxy Repaglinide, a CYP2C8 metabolite of Repaglinide, treats type II diabetes.Formule :C27H36N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :468.59M826
M826, a non-peptide, potent, selective, and reversible caspase-3 inhibitor, exhibits an IC50 of 0.005 μM and demonstrates strong anti-apoptotic activity inFormule :C28H45N7O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :575.7Salvinorin A Propionate
CAS :Salvinorin A propionate: partial KOR agonist, Ki=32.6 nM, EC50=4.7 nM; ignores μ/δ/ORL-1, non-opioid receptors; less potent analgesic vs. salvinorin A.Formule :C24H30O8Couleur et forme :SolidMasse moléculaire :446.49Oberadilol
CAS :Oberadilol is a pyridazinone derivative with vasodilatory and beta-adrenergic blocking activities and type III phosphodiesterase inhibitory actionFormule :C25H30ClN5O3Couleur et forme :SolidMasse moléculaire :483.99Pefcalcitol
CAS :Pefcalcitol is a novel antipsoriatic prodrug candidate containing a 16-en-22-oxa-vitamin D3 structure.Formule :C26H34F5NO4Couleur et forme :SolidMasse moléculaire :519.54BMS-751324
CAS :BMS-751324: p38α MAPK inhibitor with carbamyl-methyl, esters, phosphate from HPA. Reduces rat arthritis swelling and TNFα.Formule :C32H35N6O10PCouleur et forme :SolidMasse moléculaire :694.63cis-4-Br-2,5-F2-PCPA
cis-4-Br-2,5-F2-PCPA (S1024) blocks LSD1/LSD2 (Ki: 94 nM/8.4 μM), hinders cancer stem cell growth, raises H3K4me2 in CCRF-CEM cells.Formule :C9H8BrF2NCouleur et forme :SolidMasse moléculaire :248.07Antitrypanosomal agent 5
Antitrypanosal agent 5 is a selective anti-trypanosomal agent that acts on T. brucei (IC50: 1 nM) and HEK293 cells (IC50: 483.3 μM).Formule :C30H30N6O4SCouleur et forme :SolidMasse moléculaire :570.66Galectin-3-IN-2
Galectin-3-IN-2 inhibits galactose lectin-3 (Gal-3) with an 8.3 μM IC50, impacting cancer-related metabolism.Formule :C24H30FN3O10SCouleur et forme :SolidMasse moléculaire :571.57PF-00489791
CAS :PF-00489791 (PF4634817) is a long-acting PDE5 inhibitor with hypotensive activity for the study of diabetic nephropathy.Formule :C20H28N8O4SDegré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :476.55Gln-AMS TFA
Gln-AMS (TFA) is a type Ia amido-tRNA synthetase (AARS) inhibitor with a Ki value of 1.32 μM for glutaminyl-tRNA synthetase.Formule :C17H23F3N8O10SCouleur et forme :SolidMasse moléculaire :588.47ZM514
ZM514 inhibits CD73 (hCD73 IC50: 1.39 μM, mCD73 IC50: 14.65 μM) with low cytotoxicity, suitable for cancer research.Formule :C36H57NO4Couleur et forme :SolidMasse moléculaire :567.84FAK-IN-6
FAK-IN-6: Potent FAK inhibitor (IC50=1.415 nM), anti-cancer, for pancreatic studies.Formule :C25H31ClN5O6PSCouleur et forme :SolidMasse moléculaire :596.04Pan-Trk-IN-3
Pan-Trk-IN-3: potent Trk inhibitor (IC50: 2-26 nM), effective against drug-resistant mutants, induces apoptosis, anti-tumor effects.Formule :C29H31ClN8O3Couleur et forme :SolidMasse moléculaire :575.06YCW-E11
CAS :YCW-E11 is an antiapoptotic Bcl-2 family proteins inhibitor.Formule :C25H21Cl2N3O6S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :594.49Lavendomycin
CAS :Lavendomycin can be extracted from Streptomyces lavendulae and has active against Gram-positive bacteria.Formule :C29H50N10O8Couleur et forme :SolidMasse moléculaire :666.77MAO-B-IN-5
CAS :MAO-B-IN-5: potent, selective oral MAO-B inhibitor, IC50=0.204μM, potential for Parkinson's research.
Formule :C19H21FN2O2Degré de pureté :97.68%Couleur et forme :SolidMasse moléculaire :328.38MY-875
MY-875 inhibits microtubule formation, binds like colchicine (IC50: 0.92 μM), activates Hippo pathway, and induces apoptosis with anticancer properties.Formule :C21H25NO6Couleur et forme :SolidMasse moléculaire :387.43SJG-136
CAS :SJG-136 is a DNA cross-linking agent (XL50: 45 nM for pBR322 DNA).Formule :C31H32N4O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :556.61c-Myc inhibitor 4
Potent oral c-Myc inhibitor 4 reduces the proto-oncogene linked to tumor development.Formule :C26H33FN6O3Couleur et forme :SolidMasse moléculaire :496.58Heparastatin
CAS :Heparastatin is an inhibitor of heparanase.Formule :C8H11F3N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :272.18EGFR-IN-62
EGFR-IN-62: IC50 of 10-242 nM for various EGFR mutations, blocks A549/H1975 cell cycle, induces apoptosis, and inhibits cell motility and proliferation.Formule :C30H33N9O2Couleur et forme :SolidMasse moléculaire :551.64MF-592
CAS :MF-592: EP4 receptor antagonist, hEP4 IC50 3 nM, hWB IC50 78 nM, great oral PK, rat arthritis ED50 0.1 mg/kg/day, promising for development.Formule :C34H33Cl2N3O6SCouleur et forme :SolidMasse moléculaire :682.61di-Val-L-dC
CAS :Di-Val-L-dC, a reverse transcriptase inhibitor, is used potentially for treatment of HBV infection.Formule :C19H31N5O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :425.48Mesulergine hydrochloride
CAS :5-HT2A and 2C receptor antagonistFormule :C18H27ClN4O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :398.95Tacrolimus anhydrous 8-epimer
CAS :Tacrolimus anhydrous 8-epimer, an immunosuppressive l-pipecolic acid macrolide, blocks T cell growth by hindering IL-2.Formule :C44H69NO12Couleur et forme :SolidMasse moléculaire :804.02KCL-440
CAS :RS 57639 is a bioactive chemical.Formule :C18H18N2O2Couleur et forme :SolidMasse moléculaire :294.35GSK-3β inhibitor 6
GSK-3β inhibitor 6 is a highly potent inhibitor of GSK-3β, with an IC50 value of 24.4 μM.Formule :C20H17BrN4Couleur et forme :SolidMasse moléculaire :393.28GPBAR1-IN-3
CAS :GPBAR1-IN-3 (Compound 14) is both a selective agonist for GPBAR1, with an EC50 value of 0.17 μM, and an antagonist for CysLT1R [1].Formule :C21H23NO2Couleur et forme :SolidMasse moléculaire :321.41Tamitinol
CAS :Tamitinol is a neurotropic drug. It has been found to help symptoms of obsessive rumination in conjunction with maprotiline.Formule :C12H20N2OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :240.37Ganoderic acid R
CAS :Ganoderic acid R: potent anticancer, induces apoptosis, cytotoxic to MDR and sensitive tumor cells.Formule :C34H50O6Couleur et forme :SolidMasse moléculaire :554.76Elongation factor P-IN-2
Elongation factor P-IN-2, a β-lysine derivative, is a potent EFP inhibitor reducing E. coli growth.Formule :C16H35N3O2Couleur et forme :SolidMasse moléculaire :301.47INCB-9471 dihydrochloride
CAS :INCB-9471 HCl: a potent CCR5 antagonist, blocks monocyte migration & HIV-1.Formule :C30H42Cl2F3N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :632.59Antiangiogenic agent 3
Antiangiogenic agent 3 blocks HUVEC cell migration, chemotaxis, and lowers Src, cdc42, MAPK gene expression.Formule :C19H20O7Couleur et forme :SolidMasse moléculaire :360.36G092
G092 is a potent inhibitor of MsbA. MsbA is an ABC transporter protein. G092 has potential for antibacterial drug research.Formule :C23H20Cl2N2O3Couleur et forme :SolidMasse moléculaire :443.32Pim-1 kinase inhibitor 3
CAS :Pim-1 kinase inhibitor 3 (Compound H5) is a potent inhibitor of Pim-1 kinase, demonstrating an inhibitory concentration (IC50) of 35.13 nM [1].Formule :C20H25N3O2Couleur et forme :SolidMasse moléculaire :339.43hCAII-IN-3
hCAII-IN-3 inhibits key hCA isoforms with Ki: hCA I (403.8 nM), hCA II (5.1 nM), hCA IX (10.2 nM), hCA XII (5.2 nM); shows anticancer potential.Formule :C17H21N3O3SCouleur et forme :SolidMasse moléculaire :347.43CTX-712
CAS :CTX-712 is a potent inhibitor of cdc2-like kinase ( CLK ). CTX-712 inhibits inhibits cancer survival and cancer cell growth.Formule :C19H17FN8O2Couleur et forme :SolidMasse moléculaire :408.39BRD0418
CAS :BRD0418 acts as an upregulator of TRIB1 expression by leading to reprogramming of hepatic lipoprotein metabolism from adipogenesis to clearance it.Formule :C29H32N2O5Degré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :488.57AXKO-0046
AXKO-0046 is an indole derivative and small-molecule LDHB selective inhibitor.Formule :C25H33N3Couleur et forme :SolidMasse moléculaire :375.55(rel)-Myrislignan
CAS :(rel)-Myrislignan, a lignan compound with a relative configuration, has been isolated from Myristica fragrans Houtt.Formule :C21H26O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :374.43NB-533
CAS :NB-533 is a macrocyclic peptidic BACE-1 inhibitor.Formule :C33H55N3O4Couleur et forme :SolidMasse moléculaire :557.81DRX-065
CAS :DRX-065, a deuterated R-enantiomer of pioglitazone, treats NASH without PPARγ weight gain issues.Formule :C19H20N2O3SCouleur et forme :SolidMasse moléculaire :357.45CP-608039
CAS :CP-608039 is a selective adenosine A3 receptor agonist for both human A3 and human A1 receptors.Formule :C23H25ClN8O5Couleur et forme :SolidMasse moléculaire :528.95VEGFR-IN-3
CAS :VEGFR-IN-3 inhibits cancer cell growth (OVCAR-4, MDA-MB-468) with IC50s: 0.29, 0.35μM. Used in cancer research.Formule :C27H28N2O6Couleur et forme :SolidMasse moléculaire :476.52ATM Inhibitor-3
ATM Inhibitor-3 selectively inhibits ATM (IC50: 0.71 nM), targets PI3K kinase family, and is metabolically stable.Formule :C25H29FN6O3Couleur et forme :SolidMasse moléculaire :480.53NS2B/NS3-IN-2
Potent dengue inhibitor NS2B/NS3-IN-2 (IC50: 6 nM, Ki: 0.66 μM) boosts cell viability, non-toxic.Formule :C24H21N3O5SCouleur et forme :SolidMasse moléculaire :463.51Antifungal agent 16
Antifungal agent 16 has antimicrobial activity comparable to that of ciprofloxacin and has higher antifungal activity than fluconazole.Formule :C27H21N5O2SCouleur et forme :SolidMasse moléculaire :479.55SAR-114137
CAS :SAR-114137 is a histone sphingomyelin kinase inhibitor used in the study of molluscum arteriosum and peripheral neuropathic pain.Formule :C25H34N4O7SDegré de pureté :99.09% - 99.91%Couleur et forme :SolidMasse moléculaire :534.63AMG-369
CAS :AMG-369 (AMG 247) is an S1P1/S1P5 dual agonist that delays the development of experimental autoimmune encephalomyelitis in rats.Formule :C26H22FN3O2SDegré de pureté :98.04% - 98.92%Couleur et forme :SolidMasse moléculaire :459.54AZD 2066 hydrate
AZD 2066 hydrate is a selective, orally active, and brain-penetrant antagonist of mGluR5. It exhibits antinociceptive effects [1].Formule :C19H18ClN5O3Couleur et forme :SolidMasse moléculaire :386.33hCA XII/II/IX-IN-1
hCA XII/II/IX-IN-1 inhibits hCA I/II/IX/XII (IC50: 2.6, 0.004, 0.005, 0.001 μM) with anticancer properties.Formule :C25H34N4O7SCouleur et forme :SolidMasse moléculaire :534.63Mepixetil
Mepixetil is a potent angiotensin II receptor antagonist[1].Formule :C12H18N2O3Couleur et forme :SolidMasse moléculaire :238.28FW 34569
CAS :FW 34569, an enkephalin analog, boosts growth hormones and prolactin, reduces cortisol and LH; FSH stable.Formule :C30H43N5O7SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :617.76Cav 3.2 inhibitor 3
Cav 3.2 inhibitor 3 is a potent inhibitor of the Cav3.2 T-type Ca2+channel (IC50: 0.1534 μM) and has a low binding affinity for D2 receptors.Formule :C32H37N3O2Couleur et forme :SolidMasse moléculaire :495.66PF-06648671
CAS :PF-06648671 is a γ-secretase modulator for the treatment of neurodegenerative and/or neurological disorders.Formule :C25H23ClF4N4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :538.92Autophagy-IN-1
Autophagy-IN-1 blocks autophagy in cancer cells, hinders tumor growth in mice, and aids in studying colorectal cancer.Formule :C23H25NO7Couleur et forme :SolidMasse moléculaire :427.45D6808
D6808: selective c-Met inhibitor, IC50=2.9 nM, induces apoptosis and cell cycle arrest, for NSCLC/gastric cancer research.Formule :C30H25F3N6O2Couleur et forme :SolidMasse moléculaire :558.55FY-56
FY-56: potent, selective LSD1/KDM1A inhibitor (IC50=42nM); differentiates MOLM-13/MV4-11 cells; promising for AML research.Formule :C23H19FN2O3Couleur et forme :SolidMasse moléculaire :390.4120S Proteasome-IN-4
CAS :20S Proteasome-IN-4: brain-penetrant, parasite-specific, oral, inhibits T.b. brucei proteasome (IC50: 6.3nM), for HAT research.Formule :C20H18ClF2N3O3Couleur et forme :SolidMasse moléculaire :421.83M1069
M1069 is an oral A2A/A2B receptor antagonist, 100x more selective over A1/A3, with antitumor properties by blocking adenosine's immunosuppressive effects.Formule :C25H30N4O8SCouleur et forme :SolidMasse moléculaire :546.59(-)-Mesembrine
CAS :Mesembrine is a serotonin reuptake inhibitor and is also a weak inhibitor of the enzyme phosphodiesterase 4 (PDE4).Formule :C17H23NO3Couleur et forme :SolidMasse moléculaire :289.37PD 136450
CAS :PD-136,450: partial stomach secretory agonist, full pancreas agonist in rats; potential acid-reducing drug, adjuvant for gastrin-sensitive tumors.Formule :C35H40N4O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :612.72NDM-1 inhibitor-3
NDM-1 inhibitor-3 is a New Delhi Metallo-β-lactamase-1 (NDM-1) inhibitor (Ki : 4 μM) widely found in nature and is associated with antibiotic resistance.Formule :C16H12O4Degré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :268.26CRM1 degrader 1
CRM1 degrader 1 (1l) is a low-toxic CRM1 degrader that induces apoptosis in gastric carcinoma and selectively inhibits the proliferation of gastric cancer[1].Formule :C16H20O3Couleur et forme :SolidMasse moléculaire :260.33Sdz 210-096
CAS :Sdz 210-096: a 14 beta-benzyl morphinan, mu/kappa opiate receptor antagonist, stimulates LH secretion in rats.Formule :C27H31NO2Couleur et forme :SolidMasse moléculaire :401.54NVP-CFC218
CAS :NVP-CFC218 is a novel potent and selective p53-HDM2 inhibitor.Formule :C37H45ClN4O4Couleur et forme :SolidMasse moléculaire :645.23Musettamycin
CAS :Musettamycin triggers erythroid differentiation in blood cells, acts like anthracycline antibiotics, but only inhibits gram-positive bacteria.Formule :C36H45NO14Couleur et forme :SolidMasse moléculaire :715.74IACS-8779 disodium
CAS :IACS-8779 disodium: potent STING agonist, strong systemic anti-tumor effects, effective in melanoma model.Formule :C21H23N9Na2O10P2S2Couleur et forme :SolidMasse moléculaire :733.52S1P1 agonist 4
CAS :S1P1 agonist 4 exhibits enhanced potency with an EC 50 value of less than 0.05 mg/kg and a predicted human half-life (t1/2) of approximately 5 days, indicatingFormule :C24H31NO3Couleur et forme :SolidMasse moléculaire :381.51(Rac)-OSMI-1
(Rac)-OSMI-1, a racemate, inhibits OGT (IC50: 2.7 μM) affecting O-GlcNAcylation without changing surface glycans.Formule :C28H25N3O6S2Couleur et forme :SolidMasse moléculaire :563.64KU 59403
CAS :KU 59403 is an effective ATM inhibitor (IC50: 3 nM, 9.1 μM, and 10 μM for ATM, DNA-PK, and PI3K, respectively).Formule :C29H32N4O4S2Degré de pureté :99.10%Couleur et forme :SolidMasse moléculaire :564.72SK&F 108361
CAS :SK&F 108361 is a symmetric diol that binds HIV-1 protease symmetrically.Formule :C24H48N6O6Couleur et forme :SolidMasse moléculaire :516.67Rimegepant sulfate hydrate
CAS :Rimegepant (BMS-927711/BHV-3000): oral CGRP blocker for migraines, effective without vasoconstriction, beats placebo, well-tolerated.Formule :C56H64F4N12O13SCouleur et forme :SolidMasse moléculaire :1221.2526TRPV1 antagonist 3
TRPV1 antagonist 3 (7q) strongly blocks TRPV1 at 2.66 nM IC50, is selective, 60% bioavailable, and crosses the blood-brain barrier.Formule :C23H25N3OSCouleur et forme :SolidMasse moléculaire :391.53JAK3/BTK-IN-3
CAS :JAK3/BTK-IN-3: strong dual JAK3/BTK suppressor, promising for autoimmune disease research.Formule :C22H28N8OCouleur et forme :SolidMasse moléculaire :420.51Netupitant metabolite Monohydroxy Netupitant
CAS :Monohydroxy Netupitant is a highly selective antagonist of NK1 receptor, and is Netupitant metabolite.Formule :C30H32F6N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :594.59Topoisomerase II inhibitor 5
Topoisomerase II inhibitor 5 (Compound E24) is a DNAtopoisomerase II inhibitor with anticancer effects.Formule :C26H27N5O4Couleur et forme :SolidMasse moléculaire :473.52Indoluidin E
Indoluidin E selectively inhibits DHODH and has an inhibitory effect on cancer cell growth.Formule :C28H30N4O2Couleur et forme :SolidMasse moléculaire :454.56SCO-792
SCO-792: potent, reversible oral enteropeptidase inhibitor, with slow in vitro dissociation and in vivo protein digestion blocking.Formule :C22H22N4O8·xH2OCouleur et forme :SolidMetoquizine
CAS :Metoquizine is an anticholinergic compound. It is a muscarinic acetylcholine receptor antagonist that has been used to treat ulcers.Formule :C22H27N5ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :377.48DS-9300
CAS :DS-9300, an orally administered potent and selective inhibitor of EP300/CBP HAT, exhibits a significant inhibitory activity with an IC50 value of 28 nM.Formule :C25H26F3N5O3Couleur et forme :SolidMasse moléculaire :501.50Lp-PLA2-IN-6
CAS :Lp-PLA2-IN-6: Potent tetracyclic inhibitor of rhLp-PLA2, with pIC50 of 10.0, and potential in neurodegenerative research.Formule :C25H21F5N4O3Couleur et forme :SolidMasse moléculaire :520.45FT3967385
FT3967385: New USP30 inhibitor boosts mitochondrial ubiquitylation via PINK1-PARKIN.Formule :C21H19N5O2Couleur et forme :SolidMasse moléculaire :373.41Cilengitide hydrochloride
CAS :Cilengitide hydrochloride is a salt that may combat cancer by blocking specific integrins, disrupting cell interactions and angiogenesis.Formule :C27H41ClN8O7Couleur et forme :SolidMasse moléculaire :625.12Verrucarin A
CAS :Verrucarin A, a mycotoxin from Myrothecium verrucaria, inhibits protein synthesis, leukemia growth, and triggers apoptosis.Formule :C27H34O9Couleur et forme :SolidMasse moléculaire :502.55ML-SI1
CAS :ML-SI1, a racemic mixture of diastereoisomers, is a TRPML inhibitor and acts on TRPML1 (IC50: 15 μM).Formule :C23H26Cl2N2O3Couleur et forme :SolidMasse moléculaire :449.37ADP-2341
ADP-2341 is a soluble analog of FiVe1.Formule :C24H29Cl2N5O3Couleur et forme :SolidMasse moléculaire :506.43SHP2-IN-9
SHP2-IN-9: Potent SHP2 inhibitor, IC50=1.174 μM, 85x SHP1 selectivity, crosses blood-brain barrier, hampers cancer growth.Formule :C20H20FN3O2SCouleur et forme :SolidMasse moléculaire :385.46DAD dichloride
DAD dichloride is a 3rd-gen photoelectric switch, blocks K+ channels, and helps in visual function research.Formule :C26H42Cl2N6OCouleur et forme :SolidMasse moléculaire :525.56Trk-IN-8
Trk-IN-8: TRK inhibitor with IC50 of 0.42 nM (TRKA), 0.89 nM (TRKA-G595R), 1.5 nM (TRKC-G623R).Formule :C18H16F2N6O2Couleur et forme :SolidMasse moléculaire :386.36Vindeburnol
CAS :Vindeburnol is a cerebral vasodilator vincamine analog that bears neuroprotective properties.Formule :C17H20N2OCouleur et forme :SolidMasse moléculaire :268.35hDHODH-IN-10
hDHODH-IN-10: selective oral inhibitor of hDHODH (IC50: 10.9 nM); blocks cancer cell growth, aids cancer research.Formule :C21H15ClF4N2O4Couleur et forme :SolidMasse moléculaire :470.8Quinagolide hydrochloride
CAS :Quinagolide hydrochloride is a selective agonist of dopamine D2 receptor.Formule :C20H34ClN3O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :432.02CAII-IN-3
CAII-IN-3, a thiosemicarbazone, potently inhibits CA-II with an IC50 of 13.4 μM.Formule :C18H18F2N4SCouleur et forme :SolidMasse moléculaire :360.42Anticancer agent 12
Anticancer agent 12 shows cytotoxic activity in malignant cells with no hepatotoxicity.Formule :C16H17BrN4O2SCouleur et forme :SolidMasse moléculaire :409.3IMP-321
CAS :IMP-321 is a soluble dimeric recombinant form of LAG-3 and first-in-class antigen presenting cell activator.Formule :C56H78N18O14SCouleur et forme :SolidMasse moléculaire :1259.4Olanzapine/Samidorphan
CAS :Olanzapine/Samidorphan, a tablet blending olanzapine and samidorphan, targets schizophrenia and bipolar I, curbing weight gain.Formule :C38H46N6O4SCouleur et forme :SolidMasse moléculaire :682.88METTL3-IN-2
CAS :METTL3-IN-2, a potent METTL3 inhibitor, exhibits an IC50 value of 6.1 nM, effectively impairing the proliferation of Caov3 cancer cells.Formule :C25H26N8OCouleur et forme :SolidMasse moléculaire :454.53
