Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.524 produits)
- Apoptose(5.793 produits)
- Cycle cellulaire/point de contrôle(4.452 produits)
- Chromatine/Épigénétique(2.242 produits)
- Signalisation du cytosquelette(1.382 produits)
- Altération de l'ADN/réparation de l'ADN(2.826 produits)
- Endocrinologie/Hormones(3.507 produits)
- Enzyme(3.640 produits)
- GPCR/G-Protéine(8.333 produits)
- Immunologie et Inflammation(3.527 produits)
- Virus de la grippe(296 produits)
- Signalisation JAK/STAT(404 produits)
- Signalisation MAPK(1.203 produits)
- Transporteur membranaire/Canal ionique(2.792 produits)
- Métabolisme(9.449 produits)
- Microbiologie/Virologie(6.981 produits)
- Neuroscience(9.926 produits)
- Autres inhibiteurs(37.921 produits)
- Oxydation-Réduction(41 produits)
- Signalisation PI3K/Akt/mTOR(1.400 produits)
- Protéases/Protéasome(1.597 produits)
- Cellules souche et Dérivés(830 produits)
- Tyrosine Kinase/Adaptateurs(2.015 produits)
- Ubiquitination(1.650 produits)
Affichez 16 plus de sous-catégories
66639 produits trouvés pour "Inhibiteurs"
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PD-L1-IN-1
<p>PD-L1-IN-1, potent PD-L1 inhibitor with 115 nM IC50, suppresses tumors, boosts immune response, and spares healthy cells.</p>Formule :C21H23N5O2Couleur et forme :SolidMasse moléculaire :377.44CK2-IN-3
<p>CK2-IN-3: potent, selective CK2 inhibitor; Kd=12 nM, IC50: 1.51 μM (CK2α), 7.64 μM (CK2α'). For cancer research.</p>Formule :C22H26N4O7Couleur et forme :SolidMasse moléculaire :458.46Antibacterial agent 69
<p>Antibacterial agent 69 is a novel structural antimicrobial modulator that can be used against lethal multidrug-resistant bacterial infections (MIC: 2.978 μM).</p>Formule :C24H19N3O4SCouleur et forme :SolidMasse moléculaire :445.49Sekikaic Acid
CAS :<p>Sekikaic acid, a phenolic lichen metabolite in H. obscurata, has antioxidant and antiviral properties, inhibiting MLL1-CBP.</p>Formule :C22H26O8Couleur et forme :SolidMasse moléculaire :418.44BI-2540
CAS :<p>BI-2540 is a HIV non-nucleoside reverse transcriptase ( NNRT ) inhibitor .</p>Formule :C24H15ClF5NO5Couleur et forme :SolidMasse moléculaire :527.83Elongation factor P-IN-2
<p>Elongation factor P-IN-2, a β-lysine derivative, is a potent EFP inhibitor reducing E. coli growth.</p>Formule :C16H35N3O2Couleur et forme :SolidMasse moléculaire :301.47Tilpisertib fosmecarbil
CAS :<p>Tilpisertib fosmecarbil is a potent inhibitor of serine/threonine kinases with anti-inflammatory properties.</p>Formule :C35H36ClN8O7PCouleur et forme :SolidMasse moléculaire :747.14P2X receptor-1
<p>P2X receptor-1 is a potential inhibitor of P2X receptor for the treatment of pain and inflammation.</p>Formule :C14H14ClN3O3S2Couleur et forme :SolidMasse moléculaire :371.86HIV-1 inhibitor-14
<p>HIV-1 inhibitor-14: potent, broad HIV-1 RT inhibitor. IC50=0.14μM. Effective against wild-type and resistant strains, EC50=5.79-28.3nM.</p>Formule :C29H32N6O4SCouleur et forme :SolidMasse moléculaire :560.67BChE-IN-3
<p>BChE-IN-3: Selective, pseudo-irreversible BChE inhibitor (IC50: 56.9 nM); borderline reversible AChE inhibitor.</p>Formule :C26H41N3O2Couleur et forme :SolidMasse moléculaire :427.62nNOS-IN-25
CAS :<p>nNOS-IN-25 is an effective, selective, and cell-permeable inhibitor of neuronal nitric oxide synthase.</p>Formule :C21H22N4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :330.43Diospyrin
CAS :<p>Diospyrin is a plant product that has significant inhibitory effect on the growth of Leishmania donovani promastigotes.</p>Formule :C22H14O6Couleur et forme :SolidMasse moléculaire :374.34Gimatecan
CAS :Gimatecan (STI481) is a potent topoisomerase I inhibitor. Gimatecan is an orally bioavailable camptothecin analogue with antitumor activity.Formule :C25H25N3O5Degré de pureté :98.47%Couleur et forme :SolidMasse moléculaire :447.48K027
<p>K027 is a potent organophosphate (OP) inhibitor of acetylcholinesterase (AChE) reactivation. k027 can be used to study Alzheimer's disease.</p>Formule :C15H18Br2N4O2Couleur et forme :SolidMasse moléculaire :446.14NLRP3-IN-7
<p>NLRP3-IN-7 (Compound 36) is a selective inhibitor of the NLRP3 inflammasome and is able to assemble the NLRP3 inflammasome.</p>Formule :C18H15ClN2O4S3Couleur et forme :SolidMasse moléculaire :454.97BACE1-IN-5
CAS :<p>BACE1-IN-5 inhibits BACE1 (IC50: 9.1 nM) & Aβ production (IC50: 0.82 nM), enhances hERG inhibition & P-gp efflux.</p>Formule :C18H16F5N5O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :461.41GR 122222X
CAS :<p>GR 122222X is an inhibitor of topoisomerase II.</p>Formule :C26H35N5O11SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :625.65Tofogliflozin
CAS :<p>Tofogliflozin specifically inhibits SGLT2; IC50s are 2.9 nM (human), 14.9 nM (rat), 6.4 nM (mouse).</p>Formule :C22H26O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :386.44Anticancer agent 68
CAS :<p>Compound 12, an anticancer agent, halts G2/M phase, triggers cell death, and activates p53 & PTEN for tumor suppression.</p>Formule :C20H18ClNO5Couleur et forme :SolidMasse moléculaire :387.81STING agonist-7
<p>STING agonist-7 is an agonist of non-nucleotide STING that binds selectively to mouse STING but not human STING [1].</p>Formule :C17H12N4O4Couleur et forme :SolidMasse moléculaire :336.312(S)-HETE
CAS :<p>Enpatoran hydrochloride (M5049 hydrochloride) is a TLR7/8 inhibitor with antiviral activity that is used in the study of autoimmune diseases.</p>Formule :C20H32O3Couleur et forme :SolidMasse moléculaire :320.47Lamivudine, (+/-)-trans-
CAS :<p>Lamivudine, a drug for HIV-1 and HBV, inhibits reverse transcriptase and resembles zalcitabine.</p>Formule :C8H11N3O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :229.26hCAIX/XII-IN-5
<p>Coumarin 9a: Selective inhibitor of hCA IX/XII (Ki 93.3/85.7 nM), blocks cancer cell growth, and induces apoptosis.</p>Formule :C18H13NO3Couleur et forme :SolidMasse moléculaire :291.3DBCO-SS-PEG4-Biotin
<p>DBCO-SS-PEG4-Biotin: cleavable ADC linker with 4-unit PEG, used in ADC synthesis.</p>Formule :C45H62N6O9S3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :927.2CGC 11144
CAS :<p>CGC 11144 is a Polyamine analogue inhibit tumor growth in vitro and in vivo.</p>Formule :C40H100Cl10N10Couleur et forme :SolidMasse moléculaire :1075.82AX15910
<p>AX15910 is a potent inhibitor of BRD4 and ERK5.</p>Formule :C32H38N6O3Couleur et forme :SolidMasse moléculaire :554.7PI3kδ inhibitor 1
CAS :<p>PI3kδ inhibitor 1 is a selective inhibitor of PI3Kδ (IC50 of 3.8 nM).</p>Formule :C28H33FN6O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :504.60Etamicastat
CAS :<p>Etamicastat can be used in the research of cardiovascular diseases.</p>Formule :C14H15F2N3OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :311.35SARS-CoV-2 nsp14-IN-1
<p>SARS-CoV-2 nsp14-IN-1 inhibits Nsp14 Mtase with an IC50 of 0.061 μM, affecting multiple substrates.</p>Formule :C20H20N6O5SCouleur et forme :SolidMasse moléculaire :456.48Sulprostone
CAS :<p>EP3 and EP1 receptor agonist</p>Formule :C23H31NO7SDegré de pureté :98%Couleur et forme :White To Off-White SolidMasse moléculaire :465.56XO/COX/LOX-IN-1
<p>XO/COX/LOX-IN-1 targets XO/COX/LOX, used in research of inflammation, cancer, and metabolic disorders.</p>Formule :C24H20N4O2SCouleur et forme :SolidMasse moléculaire :428.51Cav 3.2 inhibitor 3
<p>Cav 3.2 inhibitor 3 is a potent inhibitor of the Cav3.2 T-type Ca2+channel (IC50: 0.1534 μM) and has a low binding affinity for D2 receptors.</p>Formule :C32H37N3O2Couleur et forme :SolidMasse moléculaire :495.66ERα degrader 5
<p>ERα degrader 5 is an orally active, selective estrogen receptor (ER) reducer that acts on ERα (EC50: 1.1 nM). ERα degrader 5 shows anti-tumour effects in vivo.</p>Formule :C29H25F4N3O2SCouleur et forme :SolidMasse moléculaire :555.59RIP1 kinase inhibitor 1
CAS :<p>RIP1 kinase inhibitor 1 is an orally available and brain-penetrating inhibitor of RIP1 kinase with pKi of 9.04.</p>Formule :C24H20ClN5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :461.9YKL-04-085
CAS :<p>YKL-04-085 inhibits viral translation effectively, with strong antiviral action at much lower doses than those affecting host-cell growth.</p>Formule :C30H29N5O2Couleur et forme :SolidMasse moléculaire :491.6HBV-IN-31
CAS :<p>HBV-IN-31: strong cccDNA inhibitor, anti-HBV, IC50=0.13 µM HBsAg, hampers cell growth.</p>Formule :C23H18ClNO6Couleur et forme :SolidMasse moléculaire :439.85L162389
CAS :<p>L162389 is an angiotensin II receptor antagonist with a balanced affinity for AT1 and AT2 receptor and stimulates the conversion of phosphatidylinositol.</p>Formule :C31H38N4O4SDegré de pureté :99.11% - 99.57%Couleur et forme :SolidMasse moléculaire :562.72KIRA9
<p>KIRA9 inhibits IRE1 with a 4.8 μM IC50, blocking ER-stress-induced mRNA decay and apoptosis by fully binding IRE1's ATP site.</p>Formule :C27H27F3N6O3SCouleur et forme :SolidMasse moléculaire :572.6LasR-IN-3
<p>LasR-IN-3 inhibits LasR in Pseudomonas, disrupting its dimer, causing loss of function.</p>Formule :C22H19N3O2Couleur et forme :SolidMasse moléculaire :357.41BRD0418
CAS :<p>BRD0418 acts as an upregulator of TRIB1 expression by leading to reprogramming of hepatic lipoprotein metabolism from adipogenesis to clearance it.</p>Formule :C29H32N2O5Degré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :488.57Tovinontrine
CAS :<p>Tovinontrine (IMR-687) (IMR-687) is a potent and selective inhibitor of phosphodiesterase-9 (PDE9), designed to target sickle cell disease treatment.</p>Formule :C21H26N6O2Degré de pureté :98.14%Couleur et forme :SolidMasse moléculaire :394.47β-Glucuronidase/hCAII-IN-2
<p>β-Glucuronidase/hCAII-IN-2 is a potent inhibitor of β-glucuronidase and hCA II, and their IC50 values were 670.7 μM and 21.77 μM, respectively.</p>Formule :C31H23NO8Couleur et forme :SolidMasse moléculaire :537.52Antibiotic MA 144M1
CAS :<p>Antibiotic MA 144M1, an anthracycline, targets gram-positive bacteria and animal tumors; derived from Streptomyces fermentation or aclacinomycin A conversion.</p>Formule :C42H55NO15Couleur et forme :SolidMasse moléculaire :813.88HBV-IN-19 TFA
CAS :<p>HBV-IN19 TFA suppresses HBsAg, hampers HBV infection, and aids in HBV research.</p>Formule :C26H31F3N2O8Couleur et forme :SolidMasse moléculaire :556.53Lycopodine
CAS :<p>Lycopodine, a bioactive compound derived from Lycopodium clavatum spores, effectively inhibits the proliferation of HeLa cells through the induction of</p>Formule :C16H25NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :247.38PD 140376
CAS :<p>PD 140376: Selective CCK-B/gastrin receptor antagonist radioligand for guinea pig stomach & brain.</p>Formule :C33H40N4O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :572.69SPR7
<p>SPR7 is a potent and selective rhodesain inhibitor (Ki: 0.51 nM). SPR7 exhibited antiparasitic effects against T. b. brucei (EC50: 1.65 μM).</p>Formule :C30H32ClN3O3Couleur et forme :SolidMasse moléculaire :518.05GP-1681
CAS :<p>GP-1681, a G-protein coupled receptor (GPCR) agonist, is used potentially for the treatment of influenza infection.</p>Formule :C24H30NaO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :421.48LY 235959
CAS :<p>LY 235959 is a NMDA receptor antagonist.</p>Formule :C11H20NO5PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :277.25CDK2-IN-9
<p>CDK2-IN-9: potent CDK2 inhibitor (IC50: 0.63 μM), anti-proliferative, arrests S/G2M cell cycle, induces apoptosis, promising for melanoma study.</p>Formule :C21H16ClN3O4SCouleur et forme :SolidMasse moléculaire :441.89AK-295
CAS :<p>AK 295, also known as CX 295, is a dipeptide inhibitor of alpha-ketoamide calpain.</p>Formule :C26H40N4O6Couleur et forme :SolidMasse moléculaire :504.62J-104871
CAS :<p>J-104871 (UNII-6137X5QNJF) is an FTase inhibitor that inhibits tumor growth in nude mice transplanted with activated H-ras-transformed NIH3T3 cells.</p>Formule :C38H32N2O12Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :708.67BRD-7880
CAS :<p>BRD-7880 is a potent and highly specific inhibitor of aurora kinases B and C.</p>Formule :C32H38N4O7Couleur et forme :SolidMasse moléculaire :590.67MK2-IN-4
CAS :<p>MK2-IN-4 is a MAPKAPK2 (MK2) inhibitor (IC50: 45 nM). MK2-IN-4 can be used in cancer, inflammation and immunology studies.</p>Formule :C25H24N4O2Couleur et forme :SolidMasse moléculaire :412.48Cenicriviroc Sulfone
CAS :<p>Cenicriviroc Sulfone, a Cenicriviroc derivative, inhibits CCR2/CCR5 to block HIV entry into cells.</p>Formule :C41H52N4O5SCouleur et forme :SolidMasse moléculaire :712.94Eprociclovir Na
CAS :<p>Eprociclovir Na (A-5021) is 15x stronger than acyclovir at inhibiting herpesviruses, showing promise for EHV1 and herpetic keratitis treatment.</p>Formule :C11H14N5NaO3Couleur et forme :SolidMasse moléculaire :287.25MtTMPK-IN-8
<p>MtTMPK-IN-8 inhibits MtbTMPK, has low cytotoxicity, shows 0.78-9.4 μM activity against Mycobacterium, useful for tuberculosis research.</p>Formule :C24H24N6O7Couleur et forme :SolidMasse moléculaire :508.48HPK1-IN-3
<p>HPK1-IN-3: Selective HPK1 inhibitor, ATP-competitive, IC50=0.25nM; boosts IL-2 in PBMCs, EC50=108nM.</p>Formule :C23H22F4N6O2Couleur et forme :SolidMasse moléculaire :490.45BI 224436
CAS :<p>BI 224436 is an inhibitor of HIV-1 noncatalytic site integrase. With EC50 values of less than 15 nM against different HIV-1 laboratory strains.</p>Formule :C27H26N2O4Couleur et forme :SolidMasse moléculaire :442.51(S)-Purvalanol B
CAS :<p>(S)-Purvalanol B is the S enantiomer of Purvalanol B. Purvalanol B is an inhibitor of cyclin-dependent kinase(CDK) .</p>Formule :C20H25ClN6O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :432.9FTI 276 TFA
CAS :<p>FTI 276 TFA targets plasmodium falciparum & humans, inhibits PFT with IC50s: 0.9 nM (parasite) & 0.5 nM (human).</p>Formule :C23H28F3N3O5S2Couleur et forme :SolidMasse moléculaire :547.61Iloprost
CAS :<p>Iloprost (Ciloprost) is an inhibitor of platelet aggregation and vasodilatation used in the study of cardiovascular disease.</p>Formule :C22H32O4Couleur et forme :Colorless OilMasse moléculaire :360.49DSP-1053 benzenesulfonate
CAS :<p>DSP-1053: Benzylpiperidine-based, potent SERT inhibitor (Ki=1.02nM), partial 5-HT1A receptor agonist (Ki=5.05nM), antidepressant.</p>Formule :C32H38BrNO7SCouleur et forme :SolidMasse moléculaire :660.62AAA-10 formic
<p>AAA-10 formic is an orally active inhibitor of intestinal bacterial bile salt hydrolase (BSH) against B.</p>Formule :C26H43FO7SCouleur et forme :SolidMasse moléculaire :518.68Plasma kallikrein-IN-2
<p>Plasma kallikrein-IN-2: PKal inhibitor, IC50=0.1 nM. Used in angioedema, diabetic eye disease research.</p>Formule :C28H24ClF3N8O3Couleur et forme :SolidMasse moléculaire :612.99P-gp modulator 1
CAS :<p>P-gp modulator 1 is a high affinity and orally available P-glycoprotein (Pgp) modulator</p>Formule :C41H72N2O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :689.02YM 202074
CAS :<p>metabotropic glutamate receptor type 1 (mGlu1) antagonist</p>Formule :C56H72N8O16S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1177.34Anticancer agent 29
<p>Compound E/Z-6f, anticancer, IC50: CDK2 (0.054 μM), CDK1 (0.127 μM), CDK4 (0.129 μM), CDK6 (0.396 μM).</p>Formule :C22H15ClFNOCouleur et forme :SolidMasse moléculaire :363.81KRas G12C inhibitor 2
CAS :<p>KRas G12C inhibitor 2 is a compound that inhibits KRas G12C.</p>Formule :C32H37N7O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :567.68Mu opioid receptor antagonist 4
<p>Compound 31: Potent, selective MOR antagonist; crosses blood-brain barrier; Ki & EC50: 0.38 nM; useful for OUD research.</p>Formule :C25H28N2O4SCouleur et forme :SolidMasse moléculaire :452.57Topo I/COX-2-IN-1
<p>Topo I/COX-2-IN-1: potent dual inhibitor; IC50 0.24μM (COX-2), 4.42μM (Topo I); anti-cancer; induces apoptosis, halts migration.</p>Formule :C21H18ClFN2O3Couleur et forme :SolidMasse moléculaire :400.83Cbl-b-IN-1
CAS :<p>Cbl-b-IN-1 is a potent Cbl-b inhibitor (IC50 <100 nM) with potential anticancer activity for the study of intestinal inflammation.</p>Formule :C29H34N6O2Degré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :498.631I-BET282E
<p>I-BET282E inhibits eight BET bromodomains (pIC50 6.4-7.7) with selectivity for other bromodomain proteins.</p>Formule :C26H34N4O7SCouleur et forme :SolidMasse moléculaire :546.64D4R antagonis-2
<p>Potent D4R antagonist-2: selective, IC50=6.52 μM, good in vitro PK and brain penetration, potential for Parkinson's research.</p>Formule :C21H23ClF2N2O2Couleur et forme :SolidMasse moléculaire :408.87TS010
<p>TS010 is a highly potent inhibitor of GLO-I, with an IC50 value of 0.57 μM. It holds significant promise for advancements in cancer research [1].</p>Formule :C16H12N4O4SCouleur et forme :SolidMasse moléculaire :356.36VEGFR-2-IN-10
<p>VEGFR-2-IN-10 has enhanced antiangiogenic potency against VEGFR2 phosphorylation induced by VEGF with an IC50 value of 0.7 μM and no cytotoxic effects.</p>Formule :C20H21N3O2Couleur et forme :SolidMasse moléculaire :335.4COX-2-IN-9
<p>COX-2-IN-9: potent oral COX-2 blocker, selective over Celecoxib, IC50 10.17 μM, less ulcers, strong anti-inflammatory.</p>Formule :C25H23N5O4S2Couleur et forme :SolidMasse moléculaire :521.61Zaragozic acid C
CAS :<p>Zaragozic acid C is an effective inhibitor of squalene synthase.</p>Formule :C40H50O14Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :754.82DGY-08-097
CAS :<p>DGY-08-097: potent HCV NS3 degrader, low resistance risk, strong inhibition in cells, DC50 of 50nM at 4h.</p>Formule :C60H76N10O14Couleur et forme :SolidMasse moléculaire :1161.3CBR Agonist-2
<p>CBR Agonist-2: CB1 receptor agonist, EC50 - 960 nM, Ki - 970 nM, useful for hCB1R-related disease research.</p>Formule :C27H27FN4OCouleur et forme :SolidMasse moléculaire :442.53Antiviral agent 6
<p>Antiviral agent 6 showed excellent anti-TSWV effects in vivo (EC50: 188 mg/L).</p>Formule :C23H27BrN2O3S2Couleur et forme :SolidMasse moléculaire :523.51Hymenidin
CAS :<p>Hymenidin, isolated from the Okinawan sponge Hymeniacidon sp., is a 5-hydroxytryptaminergic receptor antagonist and voltage-gated potassium channel inhibitor.</p>Formule :C11H12BrN5ODegré de pureté :96.85% - 99.52%Couleur et forme :SolidMasse moléculaire :310.15PptT-IN-2
<p>PptT-IN-2 inhibits PptT enzyme crucial in tuberculosis, with 2.5 μM IC50, showing potential in TB research.</p>Formule :C22H29N5O2Couleur et forme :SolidMasse moléculaire :395.5Cap-dependent endonuclease-IN-10
CAS :<p>Cap-dependent endonuclease-IN-10, with low toxicity & good stability, effectively inhibits flu viruses and shows promise against A, B, C types.</p>Formule :C25H18F2N4O5SCouleur et forme :SolidMasse moléculaire :524.50Neuraminidase-IN-7
<p>Neuraminidase-IN-7, a thiophene, inhibits neuraminidase (IC50 0.03 μM), showing promise for flu research.</p>Formule :C21H20N2O6SCouleur et forme :SolidMasse moléculaire :428.46Alkyne-probe 1
<p>Alkyne-probe 1 is usually used as an Alkyne-labeled fluorescent or chemical probe.</p>Formule :C14H23N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :293.36HIF-1α-IN-5
<p>HIF-1α-IN-5 is an inhibitor of HIF-1α with an IC 50 value of 24 nM in HEK293T cells that also inhibits the activity of MAO-A.</p>Formule :C16H15N3O2Couleur et forme :SolidMasse moléculaire :281.31VEGFR-2-IN-18
<p>VEGFR-2-IN-18 is a potent VEGFR-2 inhibitor with a 60 nM IC50, promoting cell apoptosis and anticancer effects.</p>Formule :C20H13ClN4O2Couleur et forme :SolidMasse moléculaire :376.8AS-1940477 hydrobromide
CAS :<p>AS-1940477 hydrobromide is a p38 mitogen-activated protein kinase (MAPK) inhibitor.</p>Formule :C24H23BrFN5O2Couleur et forme :SolidMasse moléculaire :512.38SB-423557
CAS :<p>SB-423557 is an orally active antagonist of calcium-sensing receptor (CaR) with IC50 of 520 nM</p>Formule :C28H36N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :464.60Deleobuvir
CAS :<p>Deleobuvir(BI207127) is an inhibitor of non-nucleoside hepatitis C virus NS5B polymerase for the treatment of hepatitis C.</p>Formule :C34H33BrN6O3Couleur et forme :SolidMasse moléculaire :653.57HPK1-IN-14
CAS :<p>HPK1-IN-14 is a potent inhibitor of HPK1. HPK1-IN-14 has potential for the study of HPK1-related diseases.</p>Formule :C24H23FN6O2Couleur et forme :SolidMasse moléculaire :446.48K252d
CAS :<p>K252d: indolocarbazole alkaloid in Nocardiopsis; inhibits PKC in rat brain and bovine heart phosphodiesterase.</p>Formule :C26H23N3O5Couleur et forme :SolidMasse moléculaire :457.48CFT8634
CAS :<p>CFT8634 degrades BRD9, for synovial sarcoma and SMARCB1 tumor research, from patent WO2021178920A1.</p>Formule :C37H45F3N6O5Couleur et forme :SolidMasse moléculaire :710.79Anticancer agent 80
<p>Anticancer agent 80 (Compound 3c) is an anticancer agent that exhibits a significant dark toxic effect on T47-D (IC50: 10.14 μM).</p>Formule :C19H12BrNO5Couleur et forme :SolidMasse moléculaire :414.21Freselestat
CAS :<p>Freselestat (ONO-6818) inhibits neutrophil elastase, reduces interleukin 8, C5B-9, and inflammation in cardiopulmonary bypass.</p>Formule :C23H28N6O4Couleur et forme :SolidMasse moléculaire :452.51AMG-222 tosylate
CAS :<p>AMG-222 tosylate is a DPP-IV inhibitor in clinical development for type II diabetes.</p>Formule :C39H47N9O6SCouleur et forme :SolidMasse moléculaire :769.91GW-597901 cinnamate
CAS :<p>GW-597901 cinnamate is a long-acting beta(2)-agonist.</p>Formule :C34H46N2O8SCouleur et forme :SolidMasse moléculaire :642.80DNA crosslinker 4 dihydrochloride
CAS :<p>DNA Crosslinker 4 binds DNA's minor groove, inhibits NCI-H460, A2780, MCF-7 cancer cells, and is used in cancer research.</p>Formule :C16H24Cl2N8OCouleur et forme :SolidMasse moléculaire :415.32Anti-Aβ agent 1A
<p>Anti-Aβ agent 1A is a potent anti-amyloid-β agent.</p>Formule :C35H49NO4Couleur et forme :SolidMasse moléculaire :547.77IRAK4-IN-14
CAS :<p>IRAK4-IN-14 is a selective, potent, orally active IRAK4 inhibitor (IC50: 0.003 μM) with favorable PK parameters in rats and mice. effect.</p>Formule :C25H28FN9OCouleur et forme :SolidMasse moléculaire :489.55Pyruvate Carboxylase-IN-2
CAS :<p>Pyruvate Carboxylase-IN-2, erianin analog, inhibits PC with IC50s of 0.065/0.097 μM in lysate/cell assays, targets HCC.</p>Formule :C21H22O8Couleur et forme :SolidMasse moléculaire :402.39L5-DA
<p>L5-DA, a G-quadruplex ligand, stabilizes G4s in HeLa cells, induces apoptosis, and is cytotoxic with an IC50 of 4.3 μM.</p>Formule :C32H34N6O2Couleur et forme :SolidMasse moléculaire :534.65BMS-824
CAS :<p>BMS-824: potent HCV NS5A inhibitor, IC50 ~5 nM, therapeutic index >10,000, specific to HCV.</p>Formule :C27H25F3N4O5Couleur et forme :SolidMasse moléculaire :542.51Antifungal agent 13
CAS :<p>Antifungal agent 13 demonstrates significant antifungal activity against Sclerotinia sclerotiorum, achieving an EC50 of 1.25 mg/L.</p>Formule :C21H16ClF3N4OCouleur et forme :SolidMasse moléculaire :432.83COX-2/NO-IN-1
<p>COX-2/NO-IN-1: oral iNOS & NO blocker (IC50=3.52μM), COX-2 supressor, anti-inflammatory, protects kidneys.</p>Formule :C15H15NO3Couleur et forme :SolidMasse moléculaire :257.28SML-10-70-1
CAS :<p>SML-10-70-1 is a Novel Active Site Inhibitor of Oncogenic K-Ras G12C.</p>Formule :C25H42ClN7O13P2Couleur et forme :SolidMasse moléculaire :746.04Enantiomer of Sofosbuvir
<p>Inactive enantiomer of Sofosbuvir, used for chronic hepatitis C; lacks reported biological activity.</p>Formule :C22H29FN3O9PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :529.45α-Glucosidase-IN-14
<p>α-Glucosidase-IN-14 is a potent inhibitor of α-glucosidase (IC50: 5.22 μM).</p>Formule :C24H27N5O4S2Couleur et forme :SolidMasse moléculaire :513.63CRV431
CAS :<p>CRV431 is a novel Pan-Cyclophilin Inhibitor, potently inhibiting all cyclophilin isoforms tested - A, B, D, and G (IC50 values ranged from 1-7 nM).</p>Formule :C67H122N12O13Couleur et forme :SolidMasse moléculaire :1303.76DNA crosslinker 3 dihydrochloride
CAS :<p>Compound 1: a DNA minor groove binder with 1.4°C ΔTm; useful in cancer research.</p>Formule :C15H22Cl2N8OCouleur et forme :SolidMasse moléculaire :401.29MsbA-IN-3
<p>MsbA-IN-3 is a potent and highly selective MsbA inhibitor (IC50: 2 nM). MsbA-IN-3 inhibits Escherichia coli activity (MIC: 35 μM).</p>Formule :C24H22Cl2N2O4SCouleur et forme :SolidMasse moléculaire :505.41Imolamine hydrochloride
CAS :<p>Imolamine hydrochloride is a blood platelet aggregation antagonist.</p>Formule :C14H21ClN4OCouleur et forme :SolidMasse moléculaire :296.80Foroxymithine
CAS :<p>Foroxymithine is an inhibitor of angiotensin-converting enzyme.</p>Formule :C22H37N7O11Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :575.57MtTMPK-IN-3
CAS :<p>MtTMPK-IN-3 inhibits Mycobacterium tuberculosis kinase with IC50 0.12μM, MIC 12.5μM on Mtb, cytotoxic EC50 12.5μM on MRC-5 cells.</p>Formule :C23H23Cl2N3O3Couleur et forme :SolidMasse moléculaire :460.35MtDTBS-IN-1
<p>MtDTBS-IN-1 is a notably potent binder (K_D = 57 nM) and inhibitor (K_i = 5 μM) of MtDTBS.</p>Formule :C16H16N4O5Couleur et forme :SolidMasse moléculaire :344.32CB2 receptor antagonist 1
CAS :<p>Compound 29 is a potent, CB2-selective antagonist/reverse agonist. Derivatives 23 & 24 offer antinociception; 24 activates cannabinoid/TRPV1 receptors.</p>Formule :C28H47NO3Couleur et forme :SolidMasse moléculaire :445.68Mimocine
CAS :<p>Mimosine, a plant amino acid, is known to act as a normoxic inducer of hypoxia-inducible factor (HIF).</p>Formule :C15H14N2O5Couleur et forme :SolidMasse moléculaire :302.28PDE4-IN-5
<p>PDE4-IN-5: potent PDE4 inhibitor, IC50 = 3.1 nM, superb skin penetration, anti-psoriasis effect.</p>Formule :C21H28N2O3Couleur et forme :SolidMasse moléculaire :356.46GID4 Ligand 2
<p>GID4 Ligand 2 (compound 67) is a selective binder for GID4 with IC50 of 18.9 μM and Kd of 17 μM. GID4 Ligand 2 can be used for the synthesis of PROTACs [1].</p>Formule :C15H16N2Couleur et forme :SolidMasse moléculaire :224.3Fonadelpar
CAS :<p>Fonadelpar is an agonist of PPARδ. It also is used in the research of neuroparalytic keratopathy.</p>Formule :C25H23F3N2O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :504.52LY309887
CAS :<p>LY309887 is a potent inhibitor of glycinamide ribonucleotide formyltransferase (Ki: 6.5 nM). It also has antitumor activity.</p>Formule :C19H23N5O6SCouleur et forme :SolidMasse moléculaire :449.48Utrophin modulator 1
<p>UM1 upregulates utrophin, has EC50 of 0.11 μM, useful in DMD research.</p>Formule :C22H18N6OCouleur et forme :SolidMasse moléculaire :382.42CVT-5440
CAS :<p>CVT-5440 is a selective, high-affinity (2B) adenosine receptor antagonist with good selectivity.</p>Formule :C27H28N6O5Couleur et forme :SolidMasse moléculaire :516.55KDOAM-25 trihydrochloride (2230731-99-2 free base)
<p>KDOAM-25 trihydrochloride, a selective KDM5 inhibitor (IC50: 19-71 nM), boosts H3K4 methylation and hinders MM1S cell growth.</p>Formule :C15H28Cl3N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :416.77GPR84 antagonist 3
CAS :<p>Potent GPR84 antagonist 3 (compound 42), pIC50 8.28, inhibits GTPγS, with good pharmacokinetics.</p>Formule :C29H27N5OCouleur et forme :SolidMasse moléculaire :461.56PTP1B-IN-19
<p>PTP1B-IN-19, a benzimidazole, selectively inhibits protein tyrosine phosphatase 1B with a Ki of 23.3 μM, potential for type 2 diabetes research.</p>Formule :C26H19N3O4SCouleur et forme :SolidMasse moléculaire :469.51CXCR2 antagonist 4
<p>CXCR2 antagonist 4 inhibits CXCR2 (IC50: 0.13 μM) and CXCL8-induced calcium rise (IC50: 27 μM), promising for cancer research.</p>Formule :C15H14F2N4OS2Couleur et forme :SolidMasse moléculaire :368.42DS-9300
CAS :<p>DS-9300, an orally administered potent and selective inhibitor of EP300/CBP HAT, exhibits a significant inhibitory activity with an IC50 value of 28 nM.</p>Formule :C25H26F3N5O3Couleur et forme :SolidMasse moléculaire :501.50CDK8-IN-5
CAS :<p>CDK8-IN-5: potent CDK8 inhibitor, IC50=72 nM, boosts IL-10 by 43%, may aid inflammatory bowel disease research.</p>Formule :C26H22N2O4Couleur et forme :SolidMasse moléculaire :426.46NS2B/NS3-IN-4
CAS :<p>Compound 34e inhibits DENV2/ZIKV proteases; IC50: 0.69 µM (DENV2), 1.04 µM (ZIKV).</p>Formule :C15H11NO4Couleur et forme :SolidMasse moléculaire :269.25GSK-3β inhibitor 7
<p>GSK-3β inhibitor 7 is a GSK-3β inhibitor (IC50: 5.25 μM).</p>Formule :C27H23BrN4O2SCouleur et forme :SolidMasse moléculaire :547.47WEHI-539
CAS :<p>WEHI-539 is a selective Bcl-XL inhibitor (IC50: 1.1 nM).</p>Formule :C31H29N5O3S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :583.72BMS 310705
CAS :<p>BMS 310705, an Epothilone B analog, targets ovarian/renal/bladder/lung cancer, inducing apoptosis via mitochondria.</p>Formule :C27H42N2O6SCouleur et forme :SolidMasse moléculaire :522.70KT2-962
CAS :<p>KT2-962 is a TXA2/prostaglandin endoperoxide receptor antagonist.</p>Formule :C23H27ClNNaO5S2Couleur et forme :SolidMasse moléculaire :520.04PF-06462894
CAS :PF-06462894: morpholinopyrimidone, mGlu5 antagonist (Ki=6nM), no immune activation in mouse model.Formule :C18H23N3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :329.39T-3861174
CAS :<p>T-3861174 is a prolyl tRNA synthetase (PRS) inhibitor, exhibiting significant in vitro anti-tumor activity with GCN2-ATF4 pathway activation.</p>Formule :C26H25FN6O2Couleur et forme :SolidMasse moléculaire :472.51Turoctocog alfa
CAS :<p>Turoctocog alfa: recombinant FVIII from CHO cells for hemophilia A study.</p>Couleur et forme :SolidAMD-7049
CAS :<p>AMD-7049 is a biochemical.</p>Formule :C25H39N5Couleur et forme :SolidMasse moléculaire :409.6116(S)-Iloprost
CAS :<p>Iloprost, a potent prostacyclin analog, binds to human IP & EP1 receptors with high affinity; inhibits platelet aggregation effectively.</p>Formule :C22H32O4Couleur et forme :SolidMasse moléculaire :360.49Cap-dependent endonuclease-IN-14
CAS :<p>Cap-dependent endonuclease-IN-14 hinders CEN and could treat influenza virus infections. (Patent CN113620948A, compound 1-c).</p>Formule :C30H23FN2O6SCouleur et forme :SolidMasse moléculaire :558.58nAChR antagonist 1
CAS :<p>Compound B15, a potent α7 nAChR antagonist, IC50 = 3.3 μM, promising for research on schizophrenia, Alzheimer's, and inflammation.</p>Formule :C19H22N4O2Couleur et forme :SolidMasse moléculaire :338.4Nurr1 agonist 1
<p>Nurr1 agonist 1 is an inverse agonist tool for the neuroprotective transcription factor Nurr1 which is an appealing target to treat neurodegenerative diseases.</p>Formule :C16H14N2O2Couleur et forme :SolidMasse moléculaire :266.29ONO-9780307
CAS :<p>ONO-9780307 is a specific antagonist of LPA1 (lysophosphatidic acid receptor 1) (IC50: 2.7 nM).</p>Formule :C30H35NO7Couleur et forme :SolidMasse moléculaire :521.6Carbonic anhydrase inhibitor 4
<p>CA inhibitor 4, photoprobe; targets hCA I-XIV; Ki: 640-1166 nM.</p>Formule :C21H18N2O4SCouleur et forme :SolidMasse moléculaire :394.44[D-Leu-4]-OB3
CAS :[D-Leu-4]-OB3 suppresses the expression of genes associated with inflammation, proliferation, and metastasis, as well as the expression of PD-L1.Formule :C29H50N8O12SCouleur et forme :SolidMasse moléculaire :734.82MK-8318
CAS :<p>MK-8318 is an effective and selective antagonist of the CRTh2 receptor (Ki: 5.0 nM).</p>Formule :C27H26F4N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :534.5LRRK2-IN-6
<p>LRRK2-IN-6 is an oral, selective LRRK2 inhibitor crossing the blood-brain barrier, targeting GS (IC50: 4.6μM) and WT LRRK2 (IC50: 49μM).</p>Formule :C23H24F2N4O2SCouleur et forme :SolidMasse moléculaire :458.52Elocalcitol
CAS :<p>Elocalcitol is a calcitriol analog for inhibition of prostate cell growth.</p>Formule :C29H43FO2Couleur et forme :SolidMasse moléculaire :442.65Topo I-IN-1
<p>Topo I-IN-1 (14d) is a powerful Topo I inhibitor with antitumor effects and DNA intercalation, inducing apoptosis.</p>Formule :C20H14BrN3O2Couleur et forme :SolidMasse moléculaire :408.25CV 5975
CAS :<p>CV 5975 is a nonsulfhydryl ACE inhibitor that was investigated for use in hypertension and heart failure.</p>Formule :C22H31N3O5SCouleur et forme :SolidMasse moléculaire :449.56RK-582
CAS :<p>RK-582: oral spiroindolinone tankyrase inhibitor, halts colon cancer growth in COLO-320DM mouse model.</p>Formule :C27H35FN6O3Couleur et forme :SolidMasse moléculaire :510.6HIV-1 inhibitor-52
CAS :<p>HIV-1 inhibitor-52: potent, broad-spectrum with EC50s 1.6-6.4 nM against various HIV-1 strains.</p>Formule :C46H72FNO5SCouleur et forme :SolidMasse moléculaire :770.13Taprostene
CAS :<p>Taprostene (CG-4203), a stable Prostacyclin analogue, protects endothelium and myocardium post-ischemia in cats, with minimal hemodynamic impact.</p>Formule :C24H30O5Couleur et forme :SolidMasse moléculaire :398.49Gabaculine HCl
CAS :<p>Gabaculine, an irreversible GABA-T inhibitor (Ki: 2.9 μM), impacts plastid development and affects DPOR/GluTR levels.</p>Formule :C7H10ClNO2Couleur et forme :SolidMasse moléculaire :175.61Carmegliptin dihydrochloride
CAS :<p>Carmegliptin dihydrochloride (RG-1579, RO4876904) is a salt of Camegliptin, a DPP-4 inhibitor for type 2 diabetes.</p>Formule :C20H30Cl2FN3O3Couleur et forme :SolidMasse moléculaire :450.38Tofacitinib Prodrug-1
<p>Tofacitinib Prodrug-1: an oral prodrug reducing Tofacitinib's side effects, treats ulcerative colitis in mice effectively with low toxicity.</p>Formule :C36H39ClN10O7Couleur et forme :SolidMasse moléculaire :759.21Antitumor agent-43
<p>Antitumor agent-43 (Compound 4B) is a potent antitumor agent that induces cell cycle arrest at G2/M phase.</p>Formule :C16H8N2O3Couleur et forme :SolidMasse moléculaire :276.25Carboxylesterase-IN-3
CAS :<p>Carboxylesterase-IN-3 is a potent inhibitor of Carboxylesterase Notum (IC50 ≤ 10 nM).Carboxylesterase-IN-3 has the potential to study cancer diseases.</p>Formule :C11H6Cl2N4OSDegré de pureté :97.49% - 98.47%Couleur et forme :SolidMasse moléculaire :313.16FGFR4-IN-6
<p>FGFR4-IN-6: covalent, reversible FGFR4 blocker, 5.4 nM IC50, good oral bioavailability, reduces Hep3B2.1-7 tumors in mice, low toxicity.</p>Formule :C31H33N7O4Couleur et forme :SolidMasse moléculaire :567.64CI 992
CAS :<p>CI 992 is a novel potent inhibitor of primate renin.</p>Formule :C33H52N6O7S2Couleur et forme :SolidMasse moléculaire :708.93BRL-42715
CAS :<p>BRL-42715 is an effective inhibitor of bacterial beta-lactamases.</p>Formule :C10H7N4NaO3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :286.24Cathepsin C-IN-5
CAS :<p>Cathepsin C-IN-5 (SF38) is a potent, oral Cathepsin C blocker with an IC50 of 59.9 nM; less active against Cat L/S/B/K; has anti-inflammatory effects.</p>Formule :C21H17ClN6OSCouleur et forme :SolidMasse moléculaire :436.92CVS-1578
CAS :<p>CVS-1578 is a potent serine protease inhibitor, targeting the S2S3 thrombin and FXa subsites.</p>Formule :C20H30N6O5SCouleur et forme :SolidMasse moléculaire :466.55MAP3K14-IN-173
CAS :<p>MAP3K14-IN-173 is a potent MAP3K14 kinase inhibitor.</p>Formule :C29H31N7O2Couleur et forme :SolidMasse moléculaire :509.60EZH2-IN-12
<p>EZH2-IN-12 (Compound 5) is a potent inhibitor of EZH2, which has potential for studies of CNS malignancies.</p>Formule :C23H23Cl2N3O3Couleur et forme :SolidMasse moléculaire :460.35Tarloxotinib bromide
CAS :Tarloxotinib bromide (TH-4000) is an irreversible inhibitor of EGFR/HER2.Formule :C24H24Br2ClN9O3Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :681.77BILA 1906 BS
CAS :BILA 1906 BS is an inhibitor of substrate analog protease.Formule :C41H52N6O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :724.95Oxeclosporin
CAS :<p>Oxeclosporin is a hydroxyethyl derivative of serine(8)-cyclosporine; inhibits proliferation and functions of lymphocytes.</p>Formule :C64H115N11O14Couleur et forme :SolidMasse moléculaire :1262.66Fusarochromanone
CAS :<p>Fusarochromanone (FC-101) is a mycotoxin produced by Fusarium oxysporum with potent antiangiogenic, anticancer and antimalarial activities.</p>Formule :C15H20N2O4Degré de pureté :95.31% - 96%Couleur et forme :SolidMasse moléculaire :292.33(R)-Atuveciclib
CAS :<p>Atuveciclib (BAY-1143572) is a potent and highly selective, oral PTEFb / CDK9 inhibitor that inhibits CDK9 / CycT1 with an IC 50 of 13 nM [1].</p>Formule :C18H18FN5O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :387.43Flutimide
CAS :<p>Flutimide: Endonuclease inhibitor, IC50 = 3μM, for research on acute respiratory diseases like influenza.</p>Formule :C12H18N2O3Couleur et forme :SolidMasse moléculaire :238.28CL656
CAS :<p>CL656 is a stimulator of interferon genes (STING) activator.</p>Formule :C20H21F2N9O9P2S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :695.51Minnelide
CAS :<p>Minnelide is a prodrug of triptolide,and shows potent antitumor activity in a number of tumor types.</p>Formule :C21H25Na2O10PDegré de pureté :98.49% - 99.59%Couleur et forme :SolidMasse moléculaire :514.37VU6005806
CAS :<p>VU6005806 is a potent M4 PAM with EC50s: 94 nM (human), 28 nM (rat), 87 nM (dog), 68 nM (cyno); studied for neuropsychiatric disorders.</p>Formule :C17H16F3N7O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :439.41AMG-25
CAS :<p>AMG-25 (c-Kit-IN-5-1) is a c-Kit inhibitor that inhibits c-Kit, KDR, p38, Lck, and Src, and can be used for the study of mast cell-associated fibrotic diseases.</p>Formule :C23H17N5O2Degré de pureté :98.16%Couleur et forme :SolidMasse moléculaire :395.41α-Glucosidase-IN-17
CAS :<p>α-Glucosidase-IN-17 (Compound 12B) is a potent and orally active inhibitor of α-glucosidase, demonstrating antidiabetic activity with an inhibitory</p>Formule :C30H27NO2SCouleur et forme :SolidMasse moléculaire :465.61BM635 hydrochloride
<p>BM635 hydrochloride, an MmpL3 inhibitor, strongly blocks Divergent bacteriophage H37Rv (MIC50: 0.08 μM), with doubled in vivo potency.</p>Formule :C25H30ClFN2OCouleur et forme :SolidMasse moléculaire :428.97MM-589
CAS :<p>MM-589 is a potent WD repeat domain 5 (WDR5) inhibitor and mixed lineage leukemia (MLL) protein-protein interaction.</p>Formule :C28H44N8O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :572.70O-GlcNAcase-IN-1
<p>O-GlcNAcase-IN-1 is a potent and novel inhibitor of O-GlcNAcase(OGA) with an IC 50 value of 46 nM.</p>Formule :C15H22N6Couleur et forme :SolidMasse moléculaire :286.38Sekdel sequence
CAS :<p>Sekdel sequence, as a signal, leads to retention of at least two proteins in the endoplasmic reticulum of animal cells.</p>Formule :C29H49N7O14Couleur et forme :SolidMasse moléculaire :719.74Antifungal agent 43
<p>Antifungal agent 43 inhibits biofilms with low toxicity to human cancer cells.</p>Formule :C24H26N4Se2Couleur et forme :SolidMasse moléculaire :528.41Adafosbuvir
CAS :<p>Adafosbuvir has antiviral activity.</p>Formule :C22H29FN3O10PCouleur et forme :SolidMasse moléculaire :545.457NDT-30805
<p>NDT-30805, a triazolopyridine, blocks IL-1β in PBMC (IC50: 0.013μM) & NLRP3 inflammasome, for inflammation research.</p>Formule :C23H22N6SCouleur et forme :SolidMasse moléculaire :414.53BAY 38-7271
CAS :<p>BAY 38-7271: potent neuroprotective, selective CB1/CB2 agonist, Ki of 1.85 nM (CB1) & 5.96 nM (CB2).</p>Formule :C20H21F3O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :430.44β-N-Acetyl-D-hexosaminidase-IN-1
<p>β-N-Acetyl-D-hexosaminidase-IN-1 is a newly discovered chemical compound that acts as an inhibitor for β-N-acetyl-D-hexosaminidase.</p>Formule :C18H13F2NO2SCouleur et forme :SolidMasse moléculaire :345.36LY503430
CAS :<p>LY503430: Oral AMPA enhancer with nootropic, neuroprotective properties, mitigates 6-OHDA/MPTP brain damage.</p>Formule :C20H25FN2O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :392.49Anticancer agent 142
CAS :<p>Compound 142 (also known as Compound 235) is a PTPN inhibitor with potential applications in cancer research [1].</p>Formule :C13H14BrF2N2O7PS2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :523.26FMK-MEA
CAS :<p>FMK-MEA is a potent and selective p90 Ribosomal S6 Kinase (RSK) inhibitor.</p>Formule :C21H26FN5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :399.46AR-13324 M1 metabolite
CAS :<p>AR-13324 M1 metabolite is a hydrolysis metabolite of AR-13324 mesylate.</p>Formule :C19H19N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :321.37ZK118182 isopropyl ester
CAS :<p>ZK118182 isopropyl ester is a PG analog with potent DP-agonist activity (EC50 = 16.5 nM) and high affinity for the DP receptor (Ki = 74 nM).</p>Formule :C23H37ClO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :428.99XIAP/cIAP1 antagonist-1
<p>Potent oral XIAP/cIAP1 inhibitor with EC50s: XIAP 5.1 nM, cIAP1 0.32 nM; curbs tumor growth in vivo.</p>Couleur et forme :SolidCCG258208
CAS :<p>GRKs-IN-1 has remarkable potency against and selectivity for G protein-coupled receptor kinase 2 GRK2 (IC50: 130 nM) and GRK5 (IC50: 7.1 μM).</p>Formule :C24H25FN4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :452.48AChE-IN-10
<p>AChE-IN-10 (24r) inhibits AChE (IC50=2.4 nM), reducing amyloid buildup, tau phosphorylation, and promotes neuron health.</p>Formule :C23H27F2NO4SCouleur et forme :SolidMasse moléculaire :451.53Tasidotin hydrochloride
CAS :<p>Tasidotin hydrochloride, a dolastatin 15 analog, inhibits microtubule assembly and dynamics.</p>Formule :C32H59ClN6O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :643.30ZD6021
CAS :<p>ZD6021 is an antagonist of neurokinin 1 receptor.</p>Formule :C35H35Cl2N3O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :632.64Bcl-2-IN-8
<p>Bcl-2-IN-8: potent, hinders cell growth/migration, induces apoptosis, promising in triple-negative breast cancer research.</p>Formule :C36H44O6Couleur et forme :SolidMasse moléculaire :572.73Cbl-b-IN-2
CAS :<p>Cbl-b-IN-2 is an oral E3 enzyme inhibitor for immune-modulated diseases and cancer research.</p>Formule :C29H30F5N5O2Couleur et forme :SolidMasse moléculaire :575.57Rostratin B
CAS :<p>Rostratin B, a cytotoxic disulfide, demonstrates in vitro cytotoxicity against human colon carcinoma (HCT-116), exhibiting an IC50 value of 1.9 μg/mL.</p>Formule :C18H20N2O6S2Couleur et forme :SolidMasse moléculaire :424.49HIV-1 inhibitor-44
<p>HIV-1 inhibitor-44 (compound 11l) is an HIV-1 reverse transcriptase inhibitor that exhibits activity against wild-type HIV-1 strains (EC50: 0.209 μM).</p>Formule :C23H26N2O4SCouleur et forme :SolidMasse moléculaire :426.53
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