Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.847 produits)
- Apoptose(6.334 produits)
- Cycle cellulaire/point de contrôle(4.889 produits)
- Chromatine/Épigénétique(2.616 produits)
- Signalisation du cytosquelette(1.579 produits)
- Altération de l'ADN/réparation de l'ADN(2.868 produits)
- Endocrinologie/Hormones(3.753 produits)
- Enzyme(3.673 produits)
- GPCR/G-Protéine(9.027 produits)
- Immunologie et Inflammation(3.938 produits)
- Virus de la grippe(300 produits)
- Signalisation JAK/STAT(415 produits)
- Signalisation MAPK(1.259 produits)
- Transporteur membranaire/Canal ionique(3.160 produits)
- Métabolisme(10.131 produits)
- Microbiologie/Virologie(7.628 produits)
- Neuroscience(10.543 produits)
- Autres inhibiteurs(35.859 produits)
- Oxydation-Réduction(40 produits)
- Signalisation PI3K/Akt/mTOR(1.435 produits)
- Protéases/Protéasome(1.692 produits)
- Cellules souche et Dérivés(732 produits)
- Tyrosine Kinase/Adaptateurs(1.991 produits)
- Ubiquitination(1.727 produits)
Affichez 16 plus de sous-catégories
66512 produits trouvés pour "Inhibiteurs"
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BAY-693
CAS :BAY-693 is a ERK5 negative control agent with IC50 (ERK5) = 6400 nM. Its analog, BAY-885, is a potent and selective ERK5 (MAPK7) inhibitor with IC50 of 40 nMFormule :C26H30F3N7O2Couleur et forme :SolidMasse moléculaire :529.56AL-GDa62
AL-GDa62, a gastric cancer treatment lead, has EC50 of 3.2 μM (MCF10A-WT) and 2 μM (MCF10A-CDH1 -/-).Formule :C24H28FN3OCouleur et forme :SolidMasse moléculaire :393.5MtTMPK-IN-7
MtTMPK-IN-7 inhibits MtbTMPK (IC50: 47 μM), active against M. brevis (MIC: 2.3-4.7 μM), useful for tuberculosis research.Formule :C27H29ClN6O3Couleur et forme :SolidMasse moléculaire :521.01MDL-27788
CAS :MDL-27788 is a tricyclic inhibitor.Formule :C24H26N2O5SCouleur et forme :SolidMasse moléculaire :454.54Pyruvate Carboxylase-IN-2
CAS :Pyruvate Carboxylase-IN-2, erianin analog, inhibits PC with IC50s of 0.065/0.097 μM in lysate/cell assays, targets HCC.Formule :C21H22O8Couleur et forme :SolidMasse moléculaire :402.39L 156903
CAS :L 156903 is a bioactive chemical. It also inhibits the binding of neurotensin to brain tissue.Formule :C35H41N7O5SCouleur et forme :SolidMasse moléculaire :671.81GDC-0339
CAS :GDC-0339: oral Pim kinase inhibitor for multiple myeloma (Kis: Pim1 - 0.03 nM, Pim2 - 0.1 nM, Pim3 - 0.02 nM), well-tolerated.Formule :C20H22F3N7OSCouleur et forme :SolidMasse moléculaire :465.5KRas G12C inhibitor 2
CAS :KRas G12C inhibitor 2 is a compound that inhibits KRas G12C.Formule :C32H37N7O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :567.68OncoFAP
CAS :OncoFAP is an ultra-high affinity fibroblast activating protein (FAP) ligand with potential tumour targeting.Formule :C21H19F2N5O5Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :459.40Antifungal agent 11
Antifungal agent 11 has a good antifungal effect.Formule :C21H19F2N7O3S2Couleur et forme :SolidMasse moléculaire :519.55Valopicitabine
CAS :Valopicitabine is an effective prodrug of the effective anti-HCV drug 2'-C-methylcytidine and can be used as a promising antiviral drug for the study of chronicFormule :C15H24N4O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :356.37VEGFR-2-IN-18
VEGFR-2-IN-18 is a potent VEGFR-2 inhibitor with a 60 nM IC50, promoting cell apoptosis and anticancer effects.Formule :C20H13ClN4O2Couleur et forme :SolidMasse moléculaire :376.8Dopamine D3 receptor ligand-1
Dopamine D 3 receptor ligand is a potent, selective, high-affinity dopamine D3 receptor ligand that is 89 times more selective for D3 (Ki: 8 nM) than D2 (Ki:Formule :C27H29N5OCouleur et forme :SolidMasse moléculaire :439.55GW311616
CAS :GW-311616 is a long duration, orally bioavailable, and selective human neutrophil elastase (HNE) inhibitor (IC50: 22 nM; Ki: 0.31 nM).Formule :C19H31N3O4SCouleur et forme :SolidMasse moléculaire :397.53Galectin-8-IN-1
Galectin-8-IN-1 selectively binds galectin-8N with 48 μM affinity, 15x more than galectin-3.Formule :C16H18N2O6Couleur et forme :SolidMasse moléculaire :334.32Murizatoclax
CAS :AMG 397 is an oral MCL1 inhibitor .Formule :C42H57ClN4O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :765.44Revamilast
CAS :Revamilast, also known as GRC4039, is a phosphodiesterase IV inhibitor for potentially treating of asthma and rheumatoid arthritisFormule :C18H9Cl2F2N3O4Couleur et forme :SolidMasse moléculaire :440.18GSK8814
CAS :GSK8814 is a selective and ATAD2/2B bromodomain chemical probe and inhibitor (binding constant pKd=8.1 and a pKi=8.9 in BROMOscan).Formule :C28H35F2N5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :527.61MDL-43291
CAS :MDL-43291 is a leukotriene receptor antagonist.Formule :C25H42O4SCouleur et forme :SolidMasse moléculaire :438.66Steroid sulfatase/17β-HSD1-IN-3
Steroid sulfatase/17β-HSD1-IN-3 (compound 19) is a dual inhibitor of steroid sulfatase (STS) and 17β-hydroxysteroid dehydrogenase type 1 (17β HSD1).Formule :C19H17ClN2O5SCouleur et forme :SolidMasse moléculaire :420.87EED ligand 1
EED ligand 1: potent PRC2 inhibitor targeting EED subunit.Formule :C19H19FN8OCouleur et forme :SolidMasse moléculaire :394.41PfPKG-IN-1
PfPKG-IN-1, an imidazole-based inhibitor, targets the Plasmodium falciparum cyclic guanosine monophosphate-dependent protein kinase (PfPKG).Formule :C24H22ClN7OSCouleur et forme :SolidMasse moléculaire :492ChemR23-IN-3
ChemR23-IN-3 is a potent thiazole-based ChemR23 inhibitor with an IC 80 value of 12 nM.Formule :C31H33N5O5S2Couleur et forme :SolidMasse moléculaire :619.75Antibacterial agent 99
CAS :Compound 7b (Antibacterial agent 99) is an effective agent with antibacterial, antifungal properties and no haemolytic activity.Formule :C27H27BrN2Couleur et forme :SolidMasse moléculaire :459.42Gemilukast
CAS :Gemilukast (ONO-6950) is a cysteinyl leukotriene 1 and 2 receptor inhibitor that inhibits bronchoconstriction and is used in the treatment of asthma.Formule :C36H37F2NO5Degré de pureté :98.27% - 99.5%Couleur et forme :SolidMasse moléculaire :601.68Ref: TM-T11388
1mg109,00€5mg260,00€1mL*10mM (DMSO)344,00€10mg447,00€25mg865,00€50mg1.341,00€100mg2.385,00€LY367385 hydrochloride
CAS :LY367385 hydrochloride: selective mGluR1a antagonist, IC50 = 8.8 μM, neuroprotective, anticonvulsant, antiepileptic.Formule :C10H12ClNO4Couleur et forme :SolidMasse moléculaire :245.66SC13
CAS :SC13, a novel mitragynine analog, exhibits low-efficacy agonism at Mu opioid receptors and provides antinociception while minimizing adverse effects.Formule :C26H30N2O5Couleur et forme :SolidMasse moléculaire :450.53NDM-1 inhibitor-3
NDM-1 inhibitor-3 is a New Delhi Metallo-β-lactamase-1 (NDM-1) inhibitor (Ki : 4 μM) widely found in nature and is associated with antibiotic resistance.Formule :C16H12O4Degré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :268.26BAY-091
CAS :BAY-091 is a novel potent and highly selective PIP4K2A kinase inhibitor.Formule :C26H21FN4O2Degré de pureté :97.66% - 99.23%Couleur et forme :SoildMasse moléculaire :440.47Ref: TM-T60147
500mgÀ demander1mg78,00€5mg168,00€1mL*10mM (DMSO)178,00€10mg269,00€25mg427,00€50mg610,00€100mg820,00€Teslexivir hydrochloride
CAS :Teslexivir (BTA074) HCl inhibits HPV 6/11 by blocking E1-E2 protein interaction, vital for DNA replication. Used in condyloma research.Formule :C35H37BrClN3O4Couleur et forme :SolidMasse moléculaire :679.04P-gp inhibitor 2
CAS :Potent P-gp inhibitor 2 reverses Doxorubicin resistance in colorectal carcinoma cells with IC50 of 0.22 µM.Formule :C29H26N2O6Couleur et forme :SolidMasse moléculaire :498.53Onalespib lactate
CAS :Onalespib lactate is a second-generation, potent and selective HSP90 Inhibitor with antitumor activity.Formule :C27H37N3O6Couleur et forme :SolidMasse moléculaire :499.6(1R,3S)-THCCA-Asn
(1R,3S)-THCCA-Asn (4j) is a selective inhibitor of thrombin (IC50: 0.07-0.14 μM) with anti-thrombotic effects.Formule :C24H24N4O6Couleur et forme :SolidMasse moléculaire :464.47Antioxidant agent-3
Antioxidant agent-3 shows strong DPPH and ABTS+ radical scavenging (IC50: 26.58, 30.31 μM). Boosts ROS, SOD, GSH; lowers LDH in H2O2-exposed HepG2 cells.Formule :C18H14O8Couleur et forme :SolidMasse moléculaire :358.3Napsagatran hydrate
CAS :Napsagatran hydrate is a novel and specific inhibitor of thrombin.Formule :C26H36N6O7SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :576.66SOS1-IN-6
CAS :SOS1-IN-6 (compound 33-P1) is a potent inhibitor of SOS1, acting on SOS1-G12D (IC50: 14.9 nM) and SOS1-G12V (IC50: 73.3 nM).Formule :C26H28F3N3O2Couleur et forme :SolidMasse moléculaire :471.51Fostriecin (free base)
CAS :Fostriecin inhibits PP2A/PP4 (IC50s = 3.2/3 nM), weakly affects topoisomerase II/PP1 (IC50s = 40/131 μM), doesn't inhibit PP2B, and may modify epigenetics.Formule :C19H27O9PCouleur et forme :SolidMasse moléculaire :430.39LY 245769
CAS :LY 245769 is an inhibitor of leukotriene E4 (LTE4).Formule :C25H33F3N8OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :550.64BMS-066
CAS :BMS-066 is an IKKβ/Tyk2 pseudokinase inhibitor. With IC50s of 9 nM and 72 nM, respectively.Formule :C19H21N7O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :379.42G247
G247 inhibits MsbA by keeping NBDs apart, blocking ATPase activity.Formule :C24H19Cl2FO3Couleur et forme :SolidMasse moléculaire :445.31RORγt modulator 5
CAS :RORγt modulator 5, a potent RORγt modulator, exhibits a dissociation constant (K_i) of <100 nM.Formule :C27H22F5N3O6SCouleur et forme :SolidMasse moléculaire :611.54Nonsteroidal aromatase inhibitor 1
Compound 13h, a nonsteroidal aromatase inhibitor, has a potent IC50 of 0.09 nM against CYP19A1, showing promise for breast cancer research.Formule :C22H16N4O2Couleur et forme :SolidMasse moléculaire :368.39IAB15
CAS :IAB15 is a potent inhibitor of T-type calcium channel that can be used in the research of epilepsy [1].Formule :C15H14F3NO2Couleur et forme :SolidMasse moléculaire :297.27MEK1/2-IN-2
MEK1/2-IN-2 is a potent, ATP-competitive MEK1/2 inhibitor that exhibits equal inhibitory effects on wild-type MEK1/2 and a group of MEK1/2 mutant cells.Formule :C28H22ClFN6OCouleur et forme :SolidMasse moléculaire :512.97rel-MDM2/4-p53-IN-2
Potent dual MDM2/MDM4 inhibitor & p53 activator; IC50: 70.7 nM (MDM2), 81.4 nM (MDM4); regulates cell cycle, triggers apoptosis, anti-cancer.Formule :C25H17Cl3FN3O3Couleur et forme :SolidMasse moléculaire :532.78NF-κB-IN-4
NF-κB-IN-4 (compound 17) is a potent inhibitor of NF-κB pathway which can cross blood brain barrier (BBB).Formule :C18H15FN4OCouleur et forme :SolidMasse moléculaire :322.34GSK699
CAS :GSK699 is a potent, cell penetrant PCAF/GCN5 PROTAC.
Formule :C45H51BrN8O7Couleur et forme :SolidMasse moléculaire :895.84IDO1-IN-13
IDO1-IN-13 is a potent IDO1 inhibitor (IC50: 61.6 nM, EC50: 30 nM in HeLa) that reduces kyn/trp ratio by 51% in SK-OV-3 tumors.Formule :C20H16BrN5O2SCouleur et forme :SolidMasse moléculaire :470.34BTK-IN-10
CAS :BTK-IN-10 is a potent inhibitor of BTK, acting on wild-type BTK (IC50<5 nM) or mutant BTK (C481S) (IC50<5 nM).Formule :C25H24F2N4O2Couleur et forme :SolidMasse moléculaire :450.48Laulimalide
CAS :Microtubule stabilizer; halts cancer cell growth (IC50: 3-30 nM); arrests cells in prometaphase; prevents bipolar spindle formation.Formule :C30H42O7Couleur et forme :SolidMasse moléculaire :514.65OICR12694
CAS :OICR12694 (JNJ-65234637) is an orally active inhibitor of B cell lymphoma 6 (BCL6) .Formule :C29H28ClF3N8O4Couleur et forme :SolidMasse moléculaire :645.03Cap-dependent endonuclease-IN-6
CAS :Cap-dependent endonuclease-IN-6 (compound 13) is a Cap-dependent endonuclease (CEN) inhibitor that inhibits influenza virus.Formule :C23H21N3O3SCouleur et forme :SolidMasse moléculaire :419.5MetRS-IN-1
CAS :MetRS-IN-1 (Compound 27) is an inhibitor of E. coli methionyl-tRNA synthetase (MetRS) with an IC50 value of 237 nM [1].Formule :C15H13N3O4SCouleur et forme :SolidMasse moléculaire :331.35CEP-7055
CAS :CEP-18770: oral proteasome inhibitor; blocks NF-kappaB; may cause cancer cell apoptosis; less toxic than bortezomib in normal cells.Formule :C32H35N3O4Couleur et forme :SolidMasse moléculaire :525.64γ-Secretase modulator 11 hydrochloride
CAS :γ-Secretase modulator 11 hydrochloride is a potent, orally active γ-secretase modulator (IC50: 0.029 μM).Formule :C28H23ClF2N4O2Couleur et forme :SolidMasse moléculaire :520.96MK-3402
CAS :MK-3402 is a metallo-beta-lactamase inhibitor. MK-3402can be used in the research of bacteria .Formule :C15H19N9O5S2Couleur et forme :SolidMasse moléculaire :469.50QPX7728 bis-acetoxy methyl ester
CAS :QPX7728 bis-acetoxy methyl ester is an inhibitor of boronic acid β-lactamase.Formule :C15H14BFO8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :352.08Dinalbuphine sebacate
CAS :Dinalbuphine sebacate: long-acting nalbuphine prodrug, μ-opioid partial agonist/antagonist, κ-opioid high-efficacy agonist.Formule :C52H68N2O10Couleur et forme :SolidMasse moléculaire :881.1CXCR7 modulator 2
CAS :CXCR7 modulator 2 is a 7-type C-X-C chemokine receptor (CXCR7) modulator with a Ki of 13 nM.Formule :C29H42N6O3Couleur et forme :SolidMasse moléculaire :522.68PARP10/15-IN-2
CAS :PARP10/15-IN-2 (Compound 8h) blocks PARP10/15, has IC50s: 0.15μM/0.37μM, cell-permeable, prevents apoptosis.Formule :C15H11FN2O3Couleur et forme :SolidMasse moléculaire :286.26sEH inhibitor-2
SEH inhibitor-2 is an orally active sEH blocker (IC50=0.9 nM) with predicted 71.2-88.4% absorption, potentially aiding cardiovascular health.Formule :C23H18N4O3Couleur et forme :SolidMasse moléculaire :398.41NNC-11-1585
CAS :NNC-11-1585 is an M(1) and M(2) muscarinic acetylcholine receptor (mAChR) agonist.Formule :C18H19N3OSCouleur et forme :SolidMasse moléculaire :325.43APJ receptor agonist 3
CAS :APJ receptor agonist 3 is a highly effective and orally administerable agonist of the APJ receptor, demonstrating a potent EC50 value of 0.027 nM.Formule :C26H29ClN4O5Couleur et forme :SolidMasse moléculaire :512.98Dyrk1A-IN-2
Dyrk1A-IN-2 is a DYRK1A inhibitor (EC50: 37 nM). dyrk1A-IN-2 exhibits efficient promotion of human β-cell replication, as well as low cytotoxicity.Formule :C27H32N6O4Couleur et forme :SolidMasse moléculaire :504.58AAK1-IN-2 TFA
AAK1-IN-2 TFA (compound (S)-31) is a selective and potent AAK1 inhibitor (IC50: 5.8 nM) that can cross the blood-brain barrier.Formule :C24H22F6N4O4Couleur et forme :SolidMasse moléculaire :544.45Cathepsin C-IN-3
Cathepsin C-IN-3 is a potent inhibitor of histone C (IC50: 61.79 nM) and also inhibits THP-1 cells (IC50: 101.5 nM) and U937 cells (IC50: 86.5 nM).Formule :C28H21F3N6OSCouleur et forme :SolidMasse moléculaire :546.57G-4120
CAS :G-4120 is a biochemical that has been shown to have a dose-dependent complete inhibition of arterial and venous thrombosis.Formule :C26H36N8O11SCouleur et forme :SolidMasse moléculaire :668.68DGY-08-097
CAS :DGY-08-097: potent HCV NS3 degrader, low resistance risk, strong inhibition in cells, DC50 of 50nM at 4h.Formule :C60H76N10O14Couleur et forme :SolidMasse moléculaire :1161.3(Z)-Lanoconazole
(Z)-Lanoconazole, an imidazole antifungal for dermatophytosis and onychomycosis, inhibits fungal ergosterol production.Formule :C14H10ClN3S2Couleur et forme :SolidMasse moléculaire :319.83MB725
CAS :MB725 is a strong and selective inducer of viability reduction in several cancer cell lines containing the oncogenic p53-Y220C mutation.Formule :C18H21IN4O2SCouleur et forme :SolidMasse moléculaire :484.35S1PR1 agonist 2
CAS :S1PR1 agonist 2 is potent for autoimmune research (from WO2021175225A1).Formule :C25H25N5O4Couleur et forme :SolidMasse moléculaire :459.50A 76889
CAS :A 76889 is an inhibitor of HIV-1 protease.Formule :C44H58N8O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :794.98AFM-30a hydrochloride
AFM-30a hydrochloride: selective PAD2 inhibitor, EC50 9.5 μM; blocks H3 guanylation, EC50 0.4 μM; used for cancer and autoimmune research.Formule :C24H28ClFN6O3Couleur et forme :SolidMasse moléculaire :502.97Lunacalcipol
CAS :Lunacalcipol is used for the treatment of Secondary Hyperparathyroidism.Formule :C28H42O4SCouleur et forme :SolidMasse moléculaire :474.7(25S)-δ7-Dafachronic acid
CAS :(25S)-delta7-Dafachronic acid, an orphan nuclear receptor DAF-12 ligand, inhibits the dauer-promoting activity of DAF-12.Formule :C27H42O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :414.62NMDA receptor antagonist-3
NMDA antagonist-3: recovery rate 40% at 100 μM, low toxicity in SH-SY5Y, human stem cells.Formule :C13H19N3O6Couleur et forme :SolidMasse moléculaire :313.31D1R antagonist 1
CAS :Compound 12a (D1R antagonist 1) is a D1R antagonist that participates in both G-protein-coupled and β-arrestin-mediated signaling pathways [1].Formule :C22H26BrNO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :448.35COX-2/PI3K-IN-1
COX-2/PI3K-IN-1 (compound 5d) is a potent inhibitor of PI3K (IC50: 1.14 nM). COX-2/PI3K-IN-1 is a selective inhibitor of COX-2 (Ki: 3.24 nM).Formule :C19H14ClN5S2Couleur et forme :SolidMasse moléculaire :411.93rel-SB-612111 hydrochloride
CAS :NOP receptor antagonistFormule :C24H30Cl3NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :454.86HIF-2α-IN-7
CAS :HIF-2α-IN-7 is a hypoxia inducible factor 2α (HIF-2α) inhibitor.Formule :C18H9F6NO2Couleur et forme :SolidMasse moléculaire :385.26MC4355
MC4355 is a dual inhibitor of EZH2 and histone deacetylase (HDAC).Formule :C30H36N4O5Couleur et forme :SolidMasse moléculaire :532.63AChE/BChE-IN-3 hydrochloride
AChE/BChE-IN-3 (BMC-1) HCl is a dual inhibitor with IC50s: eqBChE 0.383 μM, elAChE 6.08 μM.Formule :C15H25ClN2O3Couleur et forme :SolidMasse moléculaire :316.82Mu opioid receptor antagonist 2
Compound 25: potent, selective MOR antagonist, crosses blood-brain barrier (Ki: 0.37 nM, EC50: 0.44 nM), for OUD research.Formule :C25H28N2O4SCouleur et forme :SolidMasse moléculaire :452.57Flurdihydroergotamine
CAS :Flurdihydroergotamine, a serotonin 5HT1 receptor agonist, is used as an antimigraine drug.Formule :C34H36F3N5O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :651.68BMS-986339
CAS :BMS-986339: oral, potent FXR agonist; binds to His298/ASN287; for PBC, PSC, NASH, anti-fibrosis research.Formule :C35H41F4N3O4Couleur et forme :SolidMasse moléculaire :643.71PI4KIIIbeta-IN-11
CAS :PI4KIIIbeta-IN-11 is a PI4KIIIβ inhibitor (mean pIC50=9.1) that can be used to study diseases caused by RNA viruses and Plasmodium falciparum.Formule :C33H39N7O3Couleur et forme :SolidMasse moléculaire :581.71METTL3-IN-2
CAS :METTL3-IN-2, a potent METTL3 inhibitor, exhibits an IC50 value of 6.1 nM, effectively impairing the proliferation of Caov3 cancer cells.Formule :C25H26N8OCouleur et forme :SolidMasse moléculaire :454.53BRD4 D1-IN-1
BRD4 D1-IN-1 selectively inhibits BRD4 D1 (IC50 <0.092 μM, Kd 18 nM) with >500-fold specificity versus D2.Formule :C32H37F3N6OCouleur et forme :SolidMasse moléculaire :578.67CI-1029
CAS :CI-1029: HIV protease inhibitor, combats mutant strains, high efficacy, good bioavailability in animals.Formule :C28H37NO4SCouleur et forme :SolidMasse moléculaire :483.66Anticancer agent 12
Anticancer agent 12 shows cytotoxic activity in malignant cells with no hepatotoxicity.Formule :C16H17BrN4O2SCouleur et forme :SolidMasse moléculaire :409.3Cilengitide hydrochloride
CAS :Cilengitide hydrochloride is a salt that may combat cancer by blocking specific integrins, disrupting cell interactions and angiogenesis.Formule :C27H41ClN8O7Couleur et forme :SolidMasse moléculaire :625.12TD-0212
CAS :TD-0212: Oral dual antagonist for AT1 (pKi 8.9) & NEP inhibitor (pIC50 9.2).Formule :C28H34FN3O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :527.65YW3-56
CAS :YW3-56 is a potent peptidylarginine deiminase (PAD) inhibitor, with an IC50 of 1-5 μM for PAD4.Formule :C27H32ClN5O2Couleur et forme :SolidMasse moléculaire :494.03Antitumor agent-78
Antitumor agent-78 blocks GPx-4, raises COX2, triggers apoptosis, halts EMT, and stifles cancer cell growth and migration.Couleur et forme :SoildIMR687
CAS :IMR687: a PDE9 inhibitor that could improve memory in Alzheimer's by slowing cGMP hydrolysis.Formule :C21H26N6O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :394.47KRAS G12D inhibitor 3
CAS :KRAS G12D Inhibitor 3, a compound targeting the KRAS G12D mutation, demonstrates potent antitumor efficacy with an inhibitory concentration (IC50) of less thanFormule :C34H31ClF3N5O2Couleur et forme :SolidMasse moléculaire :634.09SARS-CoV-2-IN-24
SARS-CoV-2-IN-24 blocks PLpro, altering its shape and stopping virus replication—useful for SARS-CoV-2 research.Formule :C27H30N4O5Couleur et forme :SolidMasse moléculaire :490.55HBV-IN-19 TFA
CAS :HBV-IN19 TFA suppresses HBsAg, hampers HBV infection, and aids in HBV research.Formule :C26H31F3N2O8Couleur et forme :SolidMasse moléculaire :556.53hA3AR agonist 1
hA3AR agonist 1 is a potent human A 3 adenosine receptor (hA 3 AR) agonist (Ki = 2.40 nM) .Formule :C10H14N6OSCouleur et forme :SolidMasse moléculaire :266.32FTI-2148
CAS :FTI-2148 blocks RAS-related FT-1 & GGT-1; IC50: 1.4 nM & 1.7 μM.Formule :C24H28N4O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :452.57Serlopitant
CAS :Serlopitant is a selective antagonist of Neurokinin-1 (NK-1) receptor.Formule :C29H28F7NO2Couleur et forme :SolidMasse moléculaire :555.53GSK864
CAS :GSK864 is an inhibitor of isocitrate dehydrogenase 1 (IDH1) mutant. GSK864 inhibits IDH1 mutants R132C, R132H, and R132G (IC50: 8.8, 15.2, and 16.6 nM).Formule :C30H31FN6O4Degré de pureté :97.07%Couleur et forme :SolidMasse moléculaire :558.6Antitumor agent-54
Compound C11 inhibits 14-3-3η protein (KD: 35 μM), targets liver cancer cells, blocks G1-S phase, and induces apoptosis.Formule :C29H32N2O3Couleur et forme :SolidMasse moléculaire :456.58TX2-121-1
CAS :TX2-121-1 targets HER3 for proteasome-mediated degradation to inhibit HER3-dependent signalling and growth.Formule :C42H52N8O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :716.91BRD0418
CAS :BRD0418 acts as an upregulator of TRIB1 expression by leading to reprogramming of hepatic lipoprotein metabolism from adipogenesis to clearance it.Formule :C29H32N2O5Degré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :488.57Nrf2/HO-1 activator 2
Compound 13m, a difluoro derivative, activates Nrf2/HO-1, showing neuroprotective and antioxidant effects, useful in PD research.Formule :C20H16F2O5Couleur et forme :SolidMasse moléculaire :374.33SLC4101431
SLC4101431 is a potent SphK2 inhibitor with Ki value of 90 nM.Formule :C29H28ClN7OSCouleur et forme :SolidMasse moléculaire :558.1Novokinin
CAS :Angiotensin AT2 receptor agonistFormule :C39H61N11O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :795.97ATP synthase inhibitor 2
CAS :ATP synthase inhibitor 2 blocks P. aeruginosa ATP synthase; IC50=10 μg/mL, fully inhibits at 128 μg/mL.Formule :C21H22N2O3SCouleur et forme :SolidMasse moléculaire :382.48PTP1B-IN-19
PTP1B-IN-19, a benzimidazole, selectively inhibits protein tyrosine phosphatase 1B with a Ki of 23.3 μM, potential for type 2 diabetes research.Formule :C26H19N3O4SCouleur et forme :SolidMasse moléculaire :469.51AMXI-5001 hydrochloride
AMXI-5001 hydrochloride, an oral inhibitor of PARP1/2 and microtubules, shows greater potency and selective anti-cancer effects.Formule :C25H21ClFN5O3Couleur et forme :SolidMasse moléculaire :493.92CDK1-IN-5
CDK1-IN-5 is a selective inhibitor for CDK1 (IC50: 42.19 nM), CDK2, CDK5, halting cancer cell growth.Formule :C27H26ClN5OSCouleur et forme :SolidMasse moléculaire :504.05NB-533
CAS :NB-533 is a macrocyclic peptidic BACE-1 inhibitor.Formule :C33H55N3O4Couleur et forme :SolidMasse moléculaire :557.81Antiangiogenic agent 3
Antiangiogenic agent 3 blocks HUVEC cell migration, chemotaxis, and lowers Src, cdc42, MAPK gene expression.Formule :C19H20O7Couleur et forme :SolidMasse moléculaire :360.36Heme Oxygenase-1-IN-2
Heme Oxygenase-1-IN-2 is a novel inhibitor of heme oxygenase-1 (HO-1), displaying potent antiproliferative activity in vitro, with an IC50 value of 0.95 μM.Formule :C19H18ClN3OCouleur et forme :SolidMasse moléculaire :339.82CYP1B1-IN-2
CYP1B1-IN-2 (compound 9j) is a highly potent and selective inhibitor of CYP1B1, a cytochrome P450 enzyme. It exhibits an IC50 value of 0.52 nM [1].Formule :C20H11F3O2Couleur et forme :SolidMasse moléculaire :340.3KP 10614
CAS :KP 10614 is a new prostacyclin analog that inhibits platelet-polymorphonuclear leukocyte interaction.Formule :C23H32O4Couleur et forme :SolidMasse moléculaire :372.50P-gp modulator 3
P-gp modulator 3 (Compound 37) is a potent, competitive, metabotropic P-glycoprotein (P-gp) modulator.Formule :C31H37N3O5Couleur et forme :SolidMasse moléculaire :531.64Ganoderic acid R
CAS :Ganoderic acid R: potent anticancer, induces apoptosis, cytotoxic to MDR and sensitive tumor cells.Formule :C34H50O6Couleur et forme :SolidMasse moléculaire :554.76HDAC2-IN-1
HDAC2-IN-1 is an oral HDAC2 inhibitor (IC50: 0.5 μM), crosses the blood-brain barrier, and inhibits HDAC1 and HDAC8.Formule :C22H23ClN4OSCouleur et forme :SolidMasse moléculaire :426.96Kendomycin
CAS :Kendomycin is a proteasome inhibitor and endothelin receptor antagonist. It induces apoptosis in lymphoma.Formule :C29H42O6Couleur et forme :SolidMasse moléculaire :486.64BRD4 Inhibitor-17
BRD4 Inhibitor-17: Potent with 0.33 μM IC50; modulates gene expression, may counter arsenic toxicity.Formule :C16H16FN3O3SCouleur et forme :SolidMasse moléculaire :349.38ABT-072
CAS :ABT-072 is a nonnucleoside NS5B polymerase inhibitor and a candidate drug evaluated for treatment of hepatitis C virus.Formule :C24H27N3O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :469.55Epothilone E
CAS :Epothilone E, a derivative of epothilone, functions by inhibiting microtubule protein activity, thereby halting cell division and exhibiting anti-tumorFormule :C26H39NO7SCouleur et forme :SolidMasse moléculaire :509.66SphK2-IN-1
CAS :SphK2-IN-1 is an SphK2 inhibitor with an IC50 value of 0.359 μM. SphK2-IN-1 can be used to study cancer, inflammation, neurological and cardiovascular diseases.Formule :C23H22ClF3N8OCouleur et forme :SolidMasse moléculaire :518.92FAK-IN-6
FAK-IN-6: Potent FAK inhibitor (IC50=1.415 nM), anti-cancer, for pancreatic studies.Formule :C25H31ClN5O6PSCouleur et forme :SolidMasse moléculaire :596.04Antitrypanosomal agent 5
Antitrypanosal agent 5 is a selective anti-trypanosomal agent that acts on T. brucei (IC50: 1 nM) and HEK293 cells (IC50: 483.3 μM).Formule :C30H30N6O4SCouleur et forme :SolidMasse moléculaire :570.66TP-030-2
CAS :TP-030-2 is a RIPK1 inhibitor (human K i =0.43 nM ; mouse IC 50 =100 nM) .Formule :C23H21BrN4O3Couleur et forme :SolidMasse moléculaire :481.342,3-dinor-11β-Prostaglandin F2α
CAS :2,3-dinor-11β-Prostaglandin F2α (2,3-dinor-11β-PGF2α) was recovered from the urine of both normal monkeys and humans when infused with radiolabeled PGD2, whereFormule :C18H30O5Couleur et forme :SolidMasse moléculaire :326.43CDK4/6-IN-13
CAS :Compounds 10B and 10C: potent cdk4/6 inhibitors with low nM activity, great antiproliferative effects, excellent metabolism, and good pharmacokinetics.Formule :C25H29N7OCouleur et forme :SolidMasse moléculaire :443.54ZIKV-IN-5
ZIKV-IN-5 is an acid-stable, low cytotoxic anti-ZIKV agent with an EC50 value of 0.71 μM. ZIKV-IN-5 showed effective inhibition of ZIKV NS5 MTase activity.Formule :C36H45NO4SiCouleur et forme :SolidMasse moléculaire :583.83AKN-028 acetate
AKN-028 acetate: an oral TK inhibitor for AML research, targets FLT3 with IC50 of 6 nM, inhibits autophosphorylation, and induces apoptosis.Formule :C19H18N6O2Couleur et forme :SolidMasse moléculaire :362.39DH376
CAS :DH376 inhibits DAGLα in a time and dose dependent manner in mouse brain. DH376 shows picomolar activity.Formule :C31H28F2N4O3Couleur et forme :SolidMasse moléculaire :542.58PF-06273340
CAS :PF-06273340 是一种口服具有活力的、具有选择性的外周限制性Trk 泛抑制剂。Formule :C23H22ClN7O3Degré de pureté :98% - 98.00%Couleur et forme :SolidMasse moléculaire :479.92Bilanafos
CAS :Bilanafos is an agent of Anti-Bacterial.Formule :C11H22N3O6PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :323.28ZBH-1205
CAS :ZBH-1205, a camptothecin derivative, shows strong antitumor effects via apoptosis, outperforming cpt-11 and sn38 in topoisomerase-1 inhibition.Formule :C29H31N3O8Couleur et forme :SolidMasse moléculaire :549.57OXS007417
OXS007417 induces AML cell differentiation at 48 nM EC50 and shows potent in vivo antitumor effects.Formule :C20H14F3N3OCouleur et forme :SolidMasse moléculaire :369.34HER2-IN-11
HER2-IN-11 is a psoralen derivative that induces apoptosis. HER2-IN-11 shows light-activated cytotoxicity and also exhibits anti-breast cancer activity [1].Formule :C17H11NO6Couleur et forme :SolidMasse moléculaire :325.27NLRP3-IN-4
NLRP3-IN-4 is an effective, oral NLRP3 inflammasome inhibitor with potent anti-inflammatory effects on colitis.Formule :C22H22N2O5Couleur et forme :SolidMasse moléculaire :394.42Enpp-1-IN-11
Enpp-1-IN-11 inhibits ENPP1 with a 45 nM Ki, is plasma stable, and has low clearance in human/mouse livers, potentially aiding cancer research.Formule :C15H15N5O3SCouleur et forme :SolidMasse moléculaire :345.38ND-654
CAS :ND-654 is an acetyl CoA carboxylase inhibitor.Formule :C29H33N3O8SCouleur et forme :SolidMasse moléculaire :583.65GPR81 agonist 2
CAS :GPR81 agonist 2 is a potent agonist targeting the GPR81 receptor, demonstrating EC50 values of 0.023 µM for hGPR81 and 0.123 µM for hGPR109A, respectively.Formule :C26H27ClN6O5S2Couleur et forme :SolidMasse moléculaire :603.11Carboxylesterase-IN-3
CAS :Carboxylesterase-IN-3 is a potent inhibitor of Carboxylesterase Notum (IC50 ≤ 10 nM).Carboxylesterase-IN-3 has the potential to study cancer diseases.
Formule :C11H6Cl2N4OSDegré de pureté :97.49% - 98.47%Couleur et forme :SolidMasse moléculaire :313.16Antibacterial agent 75
Antibacterial agent 75 re-sensitizes VRSA to vancomycin.Formule :C22H28N6OCouleur et forme :SolidMasse moléculaire :392.5Cryptopleurine
CAS :Cryptopleurine is an inhibitor of gene products associated with cell proliferation, survival, invasion and angiogenesis. It acts by targeting the NF-κB pathway.Formule :C24H27NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :377.48L162389
CAS :L162389 is an angiotensin II receptor antagonist with a balanced affinity for AT1 and AT2 receptor and stimulates the conversion of phosphatidylinositol.Formule :C31H38N4O4SDegré de pureté :99.11% - 99.57%Couleur et forme :SolidMasse moléculaire :562.72α-Glucosidase-IN-12
α-Glucosidase-IN-12 is a potent inhibitor of α-glucosidase (IC50: 10.20 μM).Formule :C25H30N4O4S2Couleur et forme :SolidMasse moléculaire :514.66RIPK1-IN-14
CAS :RIPK1-IN-14 inhibits RIPK1 with 92 nM IC50 and reduces necrotic apoptosis in U937 cells.Couleur et forme :SoildMRL-494
MRL-494, a small-molecule BamA inhibitor, resists efflux and outer membrane permeability, with antibacterial properties.Formule :C26H35FN16O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :622.66LIT-001 free base
CAS :LIT-001, a nonpeptide OT-R agonist, enhances mouse autism-like behavior, with EC50=55 nM and Ki=226 nM.Formule :C28H33N7O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :531.67LH secretion antagonist 1
CAS :LH secretion antagonist 1 is an antagonist of luteinizing hormone secretion with analgesic activity.Formule :C18H24ClNO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :321.84Chitin synthase inhibitor 6
Compound 9b inhibits CHS with an IC50 of 0.21 mM; it's a broad-spectrum antifungal, effective against resistant strains.Formule :C24H25N3O6Couleur et forme :SolidMasse moléculaire :451.47ERRγ agonist-1
ERRγ agonist-1 can be used in neuropsychological disorders research.Formule :C17H21N5OCouleur et forme :SolidMasse moléculaire :311.38T-3861174
CAS :T-3861174 is a prolyl tRNA synthetase (PRS) inhibitor, exhibiting significant in vitro anti-tumor activity with GCN2-ATF4 pathway activation.Formule :C26H25FN6O2Couleur et forme :SolidMasse moléculaire :472.51β-Glucuronidase-IN-2
β-Glucuronidase-IN-2 is a potent inhibitor of E.Formule :C21H17Cl3O7Couleur et forme :SolidMasse moléculaire :487.71BRD7539
CAS :BRD7539B: PfDHODH inhibitor, IC50 0.033μM; selective vs HsDHODH, IC50 >50μM.Formule :C23H22FN3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :391.44PDE-I2
CAS :PDE-I2 is a parasite schizogony inhibitor.Formule :C25H23N5O8Couleur et forme :SolidMasse moléculaire :521.48Fosmanogepix
CAS :Fosmanogepix (APX001) is a broad-spectrum oral antifungal that targets Gwt1 enzyme, transforming into active APX001A in the body.Formule :C22H21N4O6PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :468.40Antitubercular agent-29
Compound 6xa inhibits drug-resistant tuberculosis with MICs 0.03 μg/mL for DS-Mtb and 0.03-0.06 for DR-Mtb, SI>40 for Vero cells.Formule :C20H12ClN3O5Couleur et forme :SolidMasse moléculaire :409.78Anti-Trypanosoma cruzi agent-1
Anti-Trypanosoma cruzi agent-1 (Compd E5) has a potent anti-Toxoplasma effect.Formule :C23H29N3O5Couleur et forme :SolidMasse moléculaire :427.49(R)-Atuveciclib
CAS :Atuveciclib (BAY-1143572) is a potent and highly selective, oral PTEFb / CDK9 inhibitor that inhibits CDK9 / CycT1 with an IC 50 of 13 nM [1].Formule :C18H18FN5O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :387.43LY3020371 hydrochloride
CAS :LY3020371 HCl: potent mGlu2/3 antagonist, antidepressant-like; Ki: 5.3/2.5 nM, IC50: 16.2 nM for cAMP inhibition.Formule :C15H16ClF2NO5SCouleur et forme :SolidMasse moléculaire :395.81NF-κB-IN-6
NF-κB-IN-6 (Compound 3d) is an anti-inflammatory agent that works by reducing the protein expression of iNOS and COX-2 by suppressing the NF-κB signalingFormule :C14H20N2O3Couleur et forme :SolidMasse moléculaire :264.32AM-6494
CAS :AM-6494 is a potent and orally active BACE1 inhibitor (IC50: 0.4 nM) with in vivo selectivity over BACE2 (IC50: 18.6 nM).Formule :C22H21F2N5O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :473.5AS1940477
CAS :AS1940477 selectively inhibits p38 MAPK α/β, blocks proinflammatory cytokines in cells, and has anti-inflammatory effects in rats.Formule :C24H22FN5O2Couleur et forme :SolidMasse moléculaire :431.46TGFβ1-IN-1
CAS :TGFβ1-IN-1 is a TGF-β1 inhibitor that inhibits the production of TGF-β1-induced fibrosis markers (α-SMA and fibronectin) and can be used in cancer research.Formule :C22H24N2O3Degré de pureté :99.89% - 99.89%Couleur et forme :SolidMasse moléculaire :364.438Ref: TM-T61389
1mg50,00€5mg105,00€1mL*10mM (DMSO)117,00€10mg170,00€25mg340,00€50mg557,00€100mg893,00€200mg1.198,00€Tuberculosis inhibitor 5
Compound 11i: potent, non-toxic anti-tuberculosis biphenyl analogue.Formule :C25H18N2O2SCouleur et forme :SolidMasse moléculaire :410.49U75302
CAS :U75302 is an antagonist of thymosin beta-4 (TB4) receptor with a Ki value of 159 nM on guinea pig lung membranes.Formule :C22H35NO3Degré de pureté :98%Couleur et forme :Light Yellow OilMasse moléculaire :361.52ZK168281
CAS :ZK168281 is a 1α,25(OH)2D3 analog, VDR antagonist with 0.1 nM Kd, and blocks receptor CoA interaction.Formule :C32H46O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :510.70Cav 3.2 inhibitor 1
Cav 3.2 inhibitor 1 targets T-type calcium channels, weakly binds D2 receptors, and aids physical and visceral pain research.Formule :C32H39N3OCouleur et forme :SolidMasse moléculaire :481.67Calphostin A
CAS :Calphostins, from Cladosporium fungus, inhibit PKC; calphostin C is most potent, used as a biochemical tool.Formule :C44H38O12Couleur et forme :SolidMasse moléculaire :758.77CHK1-IN-4
CAS :CHK1-IN-4 is a potent inhibitor of checkpoint kinase 1 (chk1) and potently inhibits chk1 phosphorylation in the tumor cells with anti-tumor activity.Formule :C18H18BrN7O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :444.29Equisetin
CAS :Equisetin: a QSI from Fusarium equiseti, curbs P. aeruginosa virulence, fights Gram-positive bacteria & HIV-1 integrase; not antibacterial to Gram-negative.Formule :C22H31NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :373.49ATX inhibitor 12
Oral ATX inhibitor 12 (IC50: 1.72 nM) at 60 mg/kg prevents lung damage in C57Bl/6J mice.Formule :C30H34FN5O2Couleur et forme :SolidMasse moléculaire :515.62BMS 310705
CAS :BMS 310705, an Epothilone B analog, targets ovarian/renal/bladder/lung cancer, inducing apoptosis via mitochondria.Formule :C27H42N2O6SCouleur et forme :SolidMasse moléculaire :522.70ORP-101
CAS :ORP-101: large, stable molecule with partial μ agonist, full κ antagonist properties.Formule :C60H84N2O8Couleur et forme :SolidMasse moléculaire :961.32FGFR1 inhibitor-6
FGFR1 inhibitor-6, IC50: 16.31 nM, blocks cell cycle at pro-G1/G2/M and induces apoptosis.Formule :C27H19N5O4S2Couleur et forme :SolidMasse moléculaire :541.6Detajmium
CAS :Detajmium is an anti-arrhythmia compound. It is an Na(+)-channel-blocking drug with an extremely long recovery from use-dependent sodium channel block.Formule :C27H42N3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :456.64CDK7/12-IN-1
CAS :CDK7/12-IN-1 is a selective CDK7 (IC50: 3 nM) and CDK12 (IC50: 277 nM) inhibitor, effective against tumor growth.Formule :C25H34N8OCouleur et forme :SolidMasse moléculaire :462.59FTO-IN-5
CAS :FTO-IN-5 is a potent, selective inhibitor targeting the fat mass obesity-associated protein (FTO).Formule :C23H18Cl2N6O6Couleur et forme :SolidMasse moléculaire :545.33AChE/BACE1/GSK3β-IN-1
AChE/BACE1/GSK3β-IN-1 is an orally active, blood-brain barrier-transparent, moderately bioavailable triple inhibitor of AChE/BACE1/GSK3β.Formule :C26H27FN2O4Couleur et forme :SolidMasse moléculaire :450.5Cilazapril HCl
CAS :Cilazapril, also known as Ro 31 2848, is a potent ACE inhibitor used for hypertension.Formule :C22H32ClN3O5Couleur et forme :SolidMasse moléculaire :453.96Antifungal agent 27
Antifungal agent 27 shows moderate action against MRSA, weak against C. albicans, with MICs of 8 μg/mL and 32 μg/mL, respectively.Formule :C18H23N5OSCouleur et forme :SolidMasse moléculaire :357.47Tubulin polymerization-IN-33
Tubulin-IN-33, an oxazoloisoindole, hinders microtubule assembly; effective against NCI cancer cells.Formule :C27H28N2O6Couleur et forme :SolidMasse moléculaire :476.52MK-8970
MK-8970 is an acetal carbonate prodrug of raltegravir with enhanced colonic absorption.Formule :C25H29FN6O8Couleur et forme :SolidMasse moléculaire :560.54Danavorexton
CAS :Danavorexton is an orexin receptor agonist.Formule :C21H32N2O5SCouleur et forme :SolidMasse moléculaire :424.55CP-199330
CAS :CP-199330: non-toxic alternative to Zafirlukast & Pranlukast, blocks cysteyl LT1 receptors.Formule :C28H24ClF3N2O6SCouleur et forme :SolidMasse moléculaire :609.01Macropa-NCS
CAS :Macropa-NCS is a macropa bifunctional analog with antitumor activity and can be used to study prostate cancer.Formule :C27H35N5O8SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :589.66A1-Phytoprostane-I
CAS :A1-Phytoprostane-I: cyclopentenone from α-linolenic acid in plants, induces gene expression & increases phytoalexin synthesis.Formule :C18H28O4Couleur et forme :SolidMasse moléculaire :308.41Aquayamycin
CAS :Aquayamycin is an anthraquinone derivative and inhibitor of the enzyme tyrosine hydroxylase..Formule :C25H26O10Couleur et forme :SolidMasse moléculaire :486.4722-HDHA
CAS :22-HDHA is an oxidation product of docosahexaenoic acid .Formule :C22H32O3Couleur et forme :SolidMasse moléculaire :344.49LRRK2-IN-3
CAS :LRRK2-IN-3: potent, selective oral LRRK2 blocker, BBB-penetrant, IC50 of 0.6 nM in hPBMCs, for Parkinson's research.Formule :C25H29ClF2N6O2Couleur et forme :SolidMasse moléculaire :518.99LXR antagonist 2
LXR antagonist 2 inhibits adipogenesis, downregulates LXR genes, and reduces lipids in hyperlipidemic mice (LXRβ IC50: 0.36μM, LXRα IC50: 2.25μM).
Formule :C34H40N2O5SCouleur et forme :SolidMasse moléculaire :588.76GAT564
GAT564, an allosteric CB1R modulator, shows EC50s of 87 nM (cAMP) & 320 nM (β-arrestin2) and lowers IOP effectively in glaucoma mice.Formule :C20H16N2O2SCouleur et forme :SolidMasse moléculaire :348.42Aβ42-IN-1
CAS :Aβ42-IN-1, compound 1v, is a novel, potent and orally active γ-secretase modulator (GSM).Formule :C29H27ClN4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :499Cap-dependent endonuclease-IN-7
CAS :Cap-dependent endonuclease-IN-7, a potent CEN inhibitor, blocks viral mRNA synthesis and virus spread, with research use for influenza A, B, C.Formule :C36H28FN3O7SCouleur et forme :SolidMasse moléculaire :665.69LRH-1 modulator-1
CAS :LRH-1 modulator-1: potent agonist, boosts IL-10, reduces IL-1b/TNFa, anti-inflammatory in gut.Formule :C28H36N2O2SCouleur et forme :SolidMasse moléculaire :464.66Omaciclovir
CAS :Omaciclovir (ABT-091) is a herpesvirus herpesvirus replication inhibitor with antiviral activity that is used in the study of herpesvirus infections.Formule :C10H15N5O3Degré de pureté :99.46% - 99.46%Couleur et forme :SolidMasse moléculaire :253.26EICAR
CAS :EICAR: IMP dehydrogenase inhibitor with anticancer and antiviral properties, failed in leukemia trials, active against various viruses but not SARS.Formule :C11H13N3O5Couleur et forme :SolidMasse moléculaire :267.24Antibiotic LL Z1640-2
CAS :Antibiotic LL Z1640-2 is an inhibitor against the TAK1 activity.Formule :C19H22O7Couleur et forme :SolidMasse moléculaire :362.38
