Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.838 produits)
- Apoptose(6.316 produits)
- Cycle cellulaire/point de contrôle(4.881 produits)
- Chromatine/Épigénétique(2.615 produits)
- Signalisation du cytosquelette(1.570 produits)
- Altération de l'ADN/réparation de l'ADN(2.868 produits)
- Endocrinologie/Hormones(3.753 produits)
- Enzyme(3.673 produits)
- GPCR/G-Protéine(9.023 produits)
- Immunologie et Inflammation(3.903 produits)
- Virus de la grippe(300 produits)
- Signalisation JAK/STAT(415 produits)
- Signalisation MAPK(1.258 produits)
- Transporteur membranaire/Canal ionique(3.159 produits)
- Métabolisme(10.130 produits)
- Microbiologie/Virologie(7.618 produits)
- Neuroscience(10.516 produits)
- Autres inhibiteurs(35.844 produits)
- Oxydation-Réduction(40 produits)
- Signalisation PI3K/Akt/mTOR(1.431 produits)
- Protéases/Protéasome(1.688 produits)
- Cellules souche et Dérivés(729 produits)
- Tyrosine Kinase/Adaptateurs(1.983 produits)
- Ubiquitination(1.727 produits)
Affichez 16 plus de sous-catégories
66513 produits trouvés pour "Inhibiteurs"
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PARP1-IN-12
PARP1-IN-12: potent PARP1 inhibitor, IC50 2.99 nM, triggers cell apoptosis, G2/M arrest, induces DSBs in BRCA-deficient cells.Formule :C43H56FN5O5Couleur et forme :SolidMasse moléculaire :741.93BChE-IN-3
BChE-IN-3: Selective, pseudo-irreversible BChE inhibitor (IC50: 56.9 nM); borderline reversible AChE inhibitor.Formule :C26H41N3O2Couleur et forme :SolidMasse moléculaire :427.62FXIa-IN-9
CAS :FXIa-IN-9, a potent FXIa inhibitor (K i : human 0.17 nM, rabbit 0.5 nM), forms hydrogen bonds and has anticoagulant properties.Formule :C23H18Cl2F3N9O2Couleur et forme :SolidMasse moléculaire :580.35PTP1B-IN-16
PTP1B-IN-16: selective benzimidazole inhibitor of PTP1B, Ki: 12.6 μM, potential for type 2 diabetes research.Formule :C26H18ClN3O4SCouleur et forme :SolidMasse moléculaire :503.96Tubulin polymerization-IN-34
"Tubulin-IN-34 inhibits oxazolylisoindole microtubule assembly, selective for VL51 lymphoma."Formule :C31H35N3O6Couleur et forme :SolidMasse moléculaire :545.63CU-2010
CAS :CU-2010 is a synthetic compound that reduces blood loss and aids recovery post-cardiac surgery.Formule :C37H42N6O6SCouleur et forme :SolidMasse moléculaire :698.83RS 12254
CAS :RS 12254 is a dopamine agonist and antihypertensive agent.Formule :C28H40N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :468.63AZD4625
AZD4625 (Compound 21) is a selective, potent, orally active, covalent and mutagenic mutant GTPaseKRASG12C inhibitor.Formule :C24H21ClF2N4O3Couleur et forme :SolidMasse moléculaire :486.9GDC-6036-NH
CAS :GDC-6036-NH is a precursor of compound 17a /b, which is a RAS inhibitor that can be used in cancer research.Formule :C26H30ClF4N7ODegré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :568.01HIV-1 inhibitor-14
HIV-1 inhibitor-14: potent, broad HIV-1 RT inhibitor. IC50=0.14μM. Effective against wild-type and resistant strains, EC50=5.79-28.3nM.Formule :C29H32N6O4SCouleur et forme :SolidMasse moléculaire :560.67PptT-IN-3
PptT-IN-3 (5p), an inhibitor of PptT in Mycobacterium tuberculosis, IC50=3.5μM, is key for TB research.Formule :C16H27N5O3SCouleur et forme :SolidMasse moléculaire :369.48(2S,3R)-LP99
CAS :(2S,3R)-LP99 is a less active enantiomer of LP99.Formule :C26H30ClN3O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :516.05GSK1820795A
CAS :GSK1820795A: Telmisartan analog, selective hGPR132a antagonist, blocks yeast activation by N-acylamides, angiotensin II antagonist, partial PPARγ agonist.Formule :C35H34N8Couleur et forme :SolidMasse moléculaire :566.7MRS-2339
CAS :MRS-2339 is a P2X receptor activator.Formule :C12H15ClN5O6PCouleur et forme :SolidMasse moléculaire :391.70PRMT5-IN-1
CAS :PRMT5-IN-1 is a covalent inhibitor of protein arginine methyltransferase 5 (PRMT5)(IC50 of 11 nM for PRMT5/MEP50).Formule :C19H19ClN4O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :418.83G12Si-1
G12Si-1 selectively binds and inhibits K-Ras(G12S) to block oncogenic signaling and nucleotide exchange.Formule :C29H32ClN5O3Couleur et forme :SolidMasse moléculaire :534.05JAK3-IN-11
CAS :JAK3-IN-11: potent oral JAK3 inhibitor (IC50=1.7 nM), noncytotoxic, >588-fold selectivity, blocks T-cell growth; useful in autoimmune research.Formule :C23H23N5O2Couleur et forme :SolidMasse moléculaire :401.46GSK3368715 3HCl
CAS :GSK3368715, a potent inhibitor of type I protein arginine methyltransferases (PRMT), could inhibit PRMT1, 3, 4, 6 and 8 with Kiapp vaules ranging from 1.5 to 81Formule :C20H41Cl3N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :475.92LTD4 antagonist 1
CAS :LTD4 antagonist 1 is a potent and orally active antagonist of leukotriene D4 (LTD4; Ki: 0.57 nM).Formule :C31H32F3N3O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :615.669-O-Demethyltrigonostemone
CAS :9-O-Demethyltrigonostemone is a natural IDO1 inhibitor, cytotoxic and antiplasmodial agent from the Roots of Strophioblachia fimbricalyx.Formule :C19H20O4Couleur et forme :SolidMasse moléculaire :312.36Bafilomycin C1
CAS :vacuolar H+-ATPases (V-ATPases) inhibitorFormule :C39H60O12Degré de pureté :98%Couleur et forme :Light Tan SolidMasse moléculaire :720.89Antifungal agent 43
Antifungal agent 43 inhibits biofilms with low toxicity to human cancer cells.Formule :C24H26N4Se2Couleur et forme :SolidMasse moléculaire :528.41Saprisartan potassium
CAS :Saprisartan potassium is an Angiotensin II Type 1 receptor antagonist and antihypertensive agent.Formule :C25H21BrF3KN4O4SCouleur et forme :SolidMasse moléculaire :649.52CB30865
CAS :CB30865 (ZM 242421) is a selective and highly effective nicotinamide phosphoribosyltransferase (Nampt) inhibitor with potential antitumor activity.Formule :C26H22BrN5O2Degré de pureté :99.04%Couleur et forme :SolidMasse moléculaire :516.39ATM-3507 trihydrochloride (1861449-70-8 free base)
ATM-3507 trihydrochloride is a potent tropomyosin inhibitor (IC50s: 3.83-6.84 μM in human melanoma cell lines).Formule :C37H49Cl3FN5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :721.17PF-06372222
CAS :PF-06372222: a small-molecule that modulates GCGR and antagonizes GLP-1R, affecting insulin and glucagon.Formule :C26H28F3N5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :515.53TD-0212 TFA
CAS :TD-0212 TFA is an oral AT1 receptor antagonist & NEP inhibitor with pKi 8.9 & pIC50 9.2.Formule :C30H35F4N3O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :641.67Tubulin inhibitor 13
CAS :Tubulin inhibitor 13 (E27), IC50 16.1 μM, blocks tubulin polymerization, cancer cell migration, and invasion, induces apoptosis.Formule :C25H21N3O4Couleur et forme :SolidMasse moléculaire :427.45Revexepride
CAS :Revexepride, a 5-HT4 agonist, may boost CYP3A4, used for treating GERD.Formule :C21H32ClN3O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :425.95Ladirubicin
CAS :Ladirubicin, as an anthracyclines analog is the leading compound of alkylcyclines.Formule :C29H31NO11SCouleur et forme :SolidMasse moléculaire :601.62NRX-2663
CAS :NRX-2663 boosts β-catenin binding to E3 ligase SCFβ-TrCP (Kd: 54.8 nM, EC50: 22.9 nM).Formule :C20H13F3N2O5Couleur et forme :SolidMasse moléculaire :418.32PF 03709270
CAS :PF 03709270 is an oral prodrug of sulopenem with broad-spectrum antibacterial effects on gram-positive and gram-negative bacteria.Formule :C19H27NO7S3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :477.61MSX-3
CAS :MSX-3 is an antagonist of the A2A adenosine receptor and a prodrug of MSX-2.Formule :C21H23N4Na2O7PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :520.389Moflomycin
CAS :Moflomycin is an anthracycline derivative. It exhibits a higher antileukemic activity compared to other anthracyclines.Formule :C25H25IO10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :612.36Homomoschatoline
CAS :Homomoschatoline is an antibacterial isolated from Artabotrys crassifolius.Formule :C19H15NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :321.33Finafloxacin
CAS :Finafloxacin is a pH-activated fluoroquinolone, most effective at pH 5.0-6.0, targeting bacterial topoisomerases, used for UTIs and H. pylori infections.Formule :C20H19FN4O4Couleur et forme :SolidMasse moléculaire :398.39(S)-3-Hydroxy Midostaurin
CAS :(S)-3-Hydroxy Midostaurin is a potent inhibitor of kinases(IC50 of <400 nM for 13 kinases (VEGFR-2, TRK-A, FLT3, et)).Formule :C35H30N4O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :586.64MNK1/2-IN-6
MNK1/2-IN-6: Strong, selective MNK1/2 inhibitor; IC50s: MNK1 at 2.3 nM, MNK2 at 3.4 nM; triggers dose-dependent apoptosis.Formule :C27H24N6OCouleur et forme :SolidMasse moléculaire :448.52L 156903
CAS :L 156903 is a bioactive chemical. It also inhibits the binding of neurotensin to brain tissue.Formule :C35H41N7O5SCouleur et forme :SolidMasse moléculaire :671.81PDE4B-IN-3
PDE4B-IN-3 is a potent inhibitor of PDE4B (IC50: 0.94 μM) and exhibits anti-inflammatory effects.Formule :C30H35N3O4S2Couleur et forme :SolidMasse moléculaire :565.75Polvitolimod
CAS :Polvitolimod is a TLR7 agonist used to treat infectious disease and cancer.Formule :C13H14FN5O4Couleur et forme :SolidMasse moléculaire :323.28Anticancer agent 143
CAS :Anticancer Agent 143 (Compound 369), a potent dual inhibitor targeting PTPN2 and PTP1B, exhibits IC50 values below 2.5 nM.Formule :C19H15BrF2N3O6PS2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :594.34AChE/GSK-3β-IN-1
CAS :AChE/GSK-3β-IN-1 is a potent dual AChE/GSK-3β inhibitor that crosses the blood-brain barrier and acts on hAChE (IC50: 1.2 nM), hBChE (IC50: 149.8 nM) and hGSK-Formule :C31H35N7O3SCouleur et forme :SolidMasse moléculaire :585.72CDK2-IN-9
CDK2-IN-9: potent CDK2 inhibitor (IC50: 0.63 μM), anti-proliferative, arrests S/G2M cell cycle, induces apoptosis, promising for melanoma study.Formule :C21H16ClN3O4SCouleur et forme :SolidMasse moléculaire :441.89YK5
CAS :YK5 is an allosteric inhibitor pocket of Hsp70 and represents a previously unknown chemical tool to investigate cellular mechanisms associated with Hsp70.Formule :C18H24N8O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :432.50GLS1 Inhibitor-6
GLS1 Inhibitor-6: IC50=68nM, 220x more selective for GLS2, has anti-tumor and pro-apoptosis effects.Formule :C37H52N6O3SCouleur et forme :SolidMasse moléculaire :660.91Luffolide
CAS :Luffolide, a Luffariella sponge metabolite, shares manoalide's anti-inflammatory traits and fully inhibits PLA2's cleavage of phosphatidylcholine.Formule :C27H40O6Couleur et forme :SolidMasse moléculaire :460.60SSTR4 agonist 4
CAS :SSTR4 agonist 4, potent in pain research, shows promise in rodent pain models, with potential for Alzheimer's due to hippocampus activity.Formule :C19H26N4OCouleur et forme :SolidMasse moléculaire :326.44Sapintoxin D
CAS :Sapintoxin D is a fluorescent phorbol ester and selective activator of protein kinase C.Formule :C30H37NO8Couleur et forme :SolidMasse moléculaire :539.62DSM705 hydrochloride
DSM705 hydrochloride: potent antimalarial, pyrrole-based DHODH inhibitor effective against Plasmodium, non-toxic to mammalian DHODH.Formule :C19H20ClF3N6OCouleur et forme :SolidMasse moléculaire :440.85CB1/2 agonist 1
Potent CB1/2 agonist 1; crosses blood-brain barrier; anti-inflammatory, analgesic; for multiple sclerosis research.Formule :C21H24BrFN2O2Couleur et forme :SolidMasse moléculaire :435.33Mf 268
CAS :Mf 268 is a pseudo-reversible carbamate-type inhibitor which interacts with the catalytic and regulatory anionic site of the enzyme.Formule :C28H46N4O3Couleur et forme :SolidMasse moléculaire :486.69AL-GDa62
AL-GDa62, a gastric cancer treatment lead, has EC50 of 3.2 μM (MCF10A-WT) and 2 μM (MCF10A-CDH1 -/-).Formule :C24H28FN3OCouleur et forme :SolidMasse moléculaire :393.5RORγt modulator 5
CAS :RORγt modulator 5, a potent RORγt modulator, exhibits a dissociation constant (K_i) of <100 nM.Formule :C27H22F5N3O6SCouleur et forme :SolidMasse moléculaire :611.54BI 703704
CAS :BI 703704, a soluble guanylate cyclase (sGC) activator, inhibits the progression of diabetic nephropathy in the ZSF1 rat [1].Formule :C32H37N3O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :559.72NBD-14189
CAS :NBD-14189: Potent HIV-1 entry blocker, binds gp120, IC50: 89 nM, strong antiviral (EC50 <200 nM).Formule :C18H16F4N4O2SCouleur et forme :SolidMasse moléculaire :428.40TAS05567
CAS :TAS05567 is a potent, highly selective, and ATP-competitive Syk inhibitor (IC50: 0.37 nM).Formule :C21H29N9O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :439.51CK2-IN-3
CK2-IN-3: potent, selective CK2 inhibitor; Kd=12 nM, IC50: 1.51 μM (CK2α), 7.64 μM (CK2α'). For cancer research.Formule :C22H26N4O7Couleur et forme :SolidMasse moléculaire :458.46Menin-MLL inhibitor 26
CAS :Menin-MLL inhibitor 26: Active reference, inhibits cell growth, used in leukemia research.Formule :C27H29F3N6O3SCouleur et forme :SolidMasse moléculaire :574.628-Deazafolic acid
CAS :8-Deazafolic acid inhibits folate-dependent bacteria S. faecium & L. casei, and fights lymphoid leukemia L1210 in mice.Formule :C20H20N6O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :440.41FMK-MEA
CAS :FMK-MEA is a potent and selective p90 Ribosomal S6 Kinase (RSK) inhibitor.Formule :C21H26FN5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :399.46CYP2C1/CYP2C19-IN-2
CYP2C1/CYP2C19-IN-2 is a potent inhibitor of CYP2C9/CYP2C19 without liver toxicity or genotoxicity and can be used to study Zika virus (ZIKV) infection.Formule :C27H28N2O6SCouleur et forme :SolidMasse moléculaire :508.59PDHK-IN-5
PDHK-IN-5, potent PDHK2 (0.006 μM IC50) & PDHK4 (0.0329 μM IC50) inhibitor, may be explored for cancer and diabetes treatment.Formule :C30H31N5O2Couleur et forme :SolidMasse moléculaire :493.6Etamicastat
CAS :Etamicastat can be used in the research of cardiovascular diseases.Formule :C14H15F2N3OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :311.35RAD51-IN-5
CAS :RAD51-IN-5 blocks RAD51; may aid mitochondrial disorder research. (WO2021164746A1, cmpd 3)Formule :C26H38N4O5S2Couleur et forme :SolidMasse moléculaire :550.73PM-060184
CAS :PM-060184, a tubulin polymerisation inhibitor, is used potentially for the treatment of solid tumours and breast cancer.Formule :C31H45N3O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :571.7PD-L1-IN-1
PD-L1-IN-1, potent PD-L1 inhibitor with 115 nM IC50, suppresses tumors, boosts immune response, and spares healthy cells.Formule :C21H23N5O2Couleur et forme :SolidMasse moléculaire :377.44BTK-IN-15
BTK-IN-15: Oral BTK inhibitor, IC50 0.7 nM, induces cancer cell apoptosis, selective with anti-tumor effects.Formule :C28H24FN5O2Couleur et forme :SolidMasse moléculaire :481.52BRD50837
CAS :BRD50837 is a potent and selective inhibitor of Sonic Hedgehog (Shh).Formule :C26H32ClN3O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :550.07AK-295
CAS :AK 295, also known as CX 295, is a dipeptide inhibitor of alpha-ketoamide calpain.Formule :C26H40N4O6Couleur et forme :SolidMasse moléculaire :504.62Quorum Sensing-IN-1
Quorum Sensing-IN-1 is a small-molecule inhibitor of quorum sensing.Formule :C13H10N2O2S2Couleur et forme :SolidMasse moléculaire :290.36RET-IN-10
CAS :RET-IN-10: Potent RET inhibitor, may treat congenital megacolon and tumors (Patent WO2021135938A1, compound 18).Formule :C29H28N8OSCouleur et forme :SolidMasse moléculaire :536.65Porphobilinogen
CAS :Porphobilinogen act as a phytotoxin, a metabotoxin, and a neurotoxin.Formule :C10H14N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :226.23Chitin synthase inhibitor 8
Chitin synthase inhibitor 8 is a chitin synthase (CHS) inhibitor with broad-spectrum antifungal effects that can be used in studies related to fungal infectionsFormule :C23H23N3O5Couleur et forme :SolidMasse moléculaire :421.45BPN-15606 besylate
BPN-15606 besylate is a potent oral γ-secretase regulator reducing Aβ42 and Aβ40 with good pharmacokinetics. IC50: 7 nM (Aβ42), 17 nM (Aβ40).Formule :C29H29FN6O4SCouleur et forme :SolidMasse moléculaire :576.64RORγt/DHODH-IN-3
RORγt/DHODH-IN-3 (compound (S)-14d) is a potent, orally active dual inhibitor of RORγt (IC50: 0.098 μM) and DHODH (IC50: 0.432 μM).RORγt/DHODH-IN-1 hasFormule :C24H26ClF6N3O3SCouleur et forme :SolidMasse moléculaire :585.99JTE 151A
CAS :JTE-151 is a novel RORγ inverse agonist.Formule :C26H30ClN3O5Couleur et forme :SolidMasse moléculaire :499.99Streptothricin F
CAS :Streptothricin F is a biochemical.Formule :C19H34N8O8Couleur et forme :SolidMasse moléculaire :502.52(+)-Sparteine sulfate pentahydrate
(+)-sparteine (sulfate pentahydrate) is a ganglion blocker that competitively blocks nicotinic acetylcholine receptors in neurons.Formule :C15H38N2O9SCouleur et forme :SolidMasse moléculaire :422.54ERK1/2 inhibitor 6
CAS :ERK1/2 inhibitor 6 - potent cancer/inflammation treatment from WO2021063335A1.Formule :C27H29ClFN7O5Couleur et forme :SolidMasse moléculaire :586.01GDC-0927 Racemate
CAS :GDC-0927 Racemate is a degrader of estrogen receptor, is used in the research of ER-related diseases, potently inhibits ER-α activity, with an IC50 of 0.2 nM.Formule :C28H28FNO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :461.52Abarelix acetate
CAS :Abarelix acetate: synthetic GnRHR antagonist, spikes histamine, lowers LH and testosterone temporarily, used in advanced prostate cancer.Formule :C72H95ClN14O14·xC2H4O2Couleur et forme :SolidMasse moléculaire :1476.14COX-2-IN-10
COX-2-IN-10 is a potent COX-2 inhibitor, reducing IL-6, TNF-α, IL-1β, PGE2 (IC50=2.54 μM), and iNOS expression.Formule :C31H32FN5O2SCouleur et forme :SolidMasse moléculaire :557.68T01-1
CAS :T01-1, a derivative of camptothecin, is an anticancer agent demonstrating significant anti-proliferative activity.Formule :C26H29N3O6SCouleur et forme :SolidMasse moléculaire :511.59Dihydrokainic acid
CAS :EAAT2(GLT1)-selective non-transportable inhibitor of L-glutamate and L-aspartate uptakeFormule :C10H17NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :215.25(Rac)-BI 703704
CAS :(Rac)-BI 703704 is a potent activator of soluble guanylyl cyclase (sGC).Formule :C32H37N3O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :559.72FGFR-IN-6
CAS :FGFR-IN-6 (Compound 5) is an FGFR inhibitor.Formule :C23H22N6O3Couleur et forme :SolidMasse moléculaire :430.46Vps34-IN-3
Vps34-IN-3 is a potent, selective, and orally bioavailable inhibitor of VPS34 kinase .Formule :C14H20N4O2Couleur et forme :SolidMasse moléculaire :276.33Daeatal
CAS :Dynorphin A ethylamide (1-9), the opioid activities were examined in the bioassays.Formule :C56H93N19O10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1192.46PF-06751979
CAS :PF-06751979 is an inhibitor of β-site amyloid precursor protein cleaving enzyme 1 (BACE1) (IC50 of 7.3 nM in BACE1 binding assay).Formule :C18H19F2N5O3S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :455.5Quinagolide Free Base
CAS :Quinagolide Free Base is a non-ergot dopamine D(2)-agonist.Formule :C20H33N3O3SCouleur et forme :SolidMasse moléculaire :395.56RO5461111
CAS :RO5461111: Oral Cathepsin S inhibitor, IC50 of 0.4 nM (human) & 0.5 nM (mouse), reduces T/B cell activation, treats lung inflammation & lupus nephritis.Formule :C27H24F6N4O4SCouleur et forme :SolidMasse moléculaire :614.56DNA-PK-IN-8
CAS :DNA-PK-IN-8: Potent, selective oral DNA-PK inhibitor, IC50 = 0.8 nM, boosts anti-cancer effects with Doxorubicin.Formule :C19H22N8O2Couleur et forme :SolidMasse moléculaire :394.43(-)-Cevimeline hydrochloride hemihydrate
(-)-Cevimeline HCl hemihydrate, a muscarinic agonist, treats Sjogren's xerostomia. Quick absorption, species-dependent metabolism.Formule :C10H19ClNO1·5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :244.78FAK inhibitor 6
CAS :Compound 26F: potent enzyme inhibitor (IC50=28.2nM), low cytotoxicity (IC50=3.32μM), induces dose-dependent apoptosis in MDA-MB-231, blocks G0/G1 phase.Formule :C25H24FN5O2SCouleur et forme :SolidMasse moléculaire :477.55ABL-001-Amide-PEG3-acid
ABL-001-Amide-PEG3-acid, an analogue to ABL-001, primarily serves as a labeled chemical or fluorescent probe.Formule :C29H33ClF2N6O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :683.06Anti-ToCV agent 1
Anti-ToCV agent 1 can be used as a potential anti-ToCV drug.Formule :C22H19FN2O5SCouleur et forme :SolidMasse moléculaire :442.46Diguanosine 5′-triphosphate lithium
Diguanosine 5′-triphosphate (Gp3G) lithium is a dinucleoside triphosphate and a virus-specific oligonucleotide.Diguanosine 5′-triphosphate lithium is requiredFormule :C20H27N10O18P3·xLiCouleur et forme :SolidPefcalcitol
CAS :Pefcalcitol is a novel antipsoriatic prodrug candidate containing a 16-en-22-oxa-vitamin D3 structure.Formule :C26H34F5NO4Couleur et forme :SolidMasse moléculaire :519.54Protease-Activated Receptor-1 antagonist 3
PAR-1 antagonist 3: potent (IC50: 7 nM), binds hERG K+ channels (IC50: 9 μM).Formule :C30H34N4O3Couleur et forme :SolidMasse moléculaire :498.62Elongation factor P-IN-1
EFP-IN-1: potent β-lysine derivative, inhibits EFP, slows E. coli growth.Formule :C14H31N3O2Couleur et forme :SolidMasse moléculaire :273.41CHK1-IN-4
CAS :CHK1-IN-4 is a potent inhibitor of checkpoint kinase 1 (chk1) and potently inhibits chk1 phosphorylation in the tumor cells with anti-tumor activity.Formule :C18H18BrN7O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :444.29HIF-1/2α-IN-1
HIF-1/2α-IN-1, an orally active compound, functions as an inhibitor of HIF-2α.Formule :C17H16N6O4Couleur et forme :SolidMasse moléculaire :368.35Edotecarin
CAS :Edotecarin is a potent topoisomerase I inhibitor. It can decrease single-strand DNA cleavage (IC50: 50 nM).Formule :C29H28N4O11Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :608.55Keap1-Nrf2-IN-1 TFA
Keap1-Nrf2-IN-1 TFA (compound35) is a potent inhibitor (IC50: 43 nM) protecting against acetaminophen liver damage.Formule :C26H25F3N2O9SCouleur et forme :SolidMasse moléculaire :598.54BRD-7880
CAS :BRD-7880 is a potent and highly specific inhibitor of aurora kinases B and C.Formule :C32H38N4O7Couleur et forme :SolidMasse moléculaire :590.67KDM1/CDK1-IN-1
KDM1/CDK1-IN-1 inhibits KDM1 (IC50: 0.096 μM) & CDK1 (IC50: 0.078 μM), blocks HOP-92 G2/M phase, induces apoptosis, toxic to cancer cells.Formule :C22H17N5O3SCouleur et forme :SolidMasse moléculaire :431.47PD 113271
CAS :PD 113,271 is an analog of the fermentation products fostriecin with antitumor activity in vitro and in vivo.Formule :C19H27O10PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :446.39VU0463271 quarterhydrate
VU0463271 quarterhydrate is a potent KCC2 antagonist, with an IC 50 of 61 nM [1].Formule :C19H20N4O2S2Couleur et forme :SolidMasse moléculaire :387P-gp inhibitor 2
CAS :Potent P-gp inhibitor 2 reverses Doxorubicin resistance in colorectal carcinoma cells with IC50 of 0.22 µM.Formule :C29H26N2O6Couleur et forme :SolidMasse moléculaire :498.53PSB 36
CAS :A1 adenosine receptor antagonistFormule :C21H30N4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :386.49LY210073
CAS :LY210073 is an antagonist of the Leukotriene B4 (LTB4) receptor (IC50: 6.2 nM).Formule :C30H28O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :516.54Sdz 210-096
CAS :Sdz 210-096: a 14 beta-benzyl morphinan, mu/kappa opiate receptor antagonist, stimulates LH secretion in rats.Formule :C27H31NO2Couleur et forme :SolidMasse moléculaire :401.54NusB-IN-1
NusB-IN-1 (22r) is an oral bacterial rRNA inhibitor, effective against MRSA and VRSA.Formule :C21H16N2O3Couleur et forme :SolidMasse moléculaire :344.36A2A receptor antagonist 2
A2A receptor antagonist 2 is a highly selective and potent antagonist of the adenosine A2Areceptor (IC50: 8.3 nM).Formule :C25H28FN7O3Couleur et forme :SolidMasse moléculaire :493.53Diacylglycerol acyltransferase inhibitor-1
CAS :Diacylglycerol Acyltransferase Inhibitor-1, a diacylglycerol acyltransferase (DGAT1) inhibitor, effectively suppresses the activity of DGAT1.Formule :C21H23N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :377.44VEGFR-2-IN-14
VEGFR-2-IN-14 (Compound 5) is a potent inhibitor of VEGFR-2, which inhibits the growth of HepG2 cells in the Pre-G1 phase and induces apoptosis.Formule :C24H23N3O3SCouleur et forme :SolidMasse moléculaire :433.52Cyclic-di-GMP sodium
c-di-GMP sodium: STING activator, regulates bacteria biofilm, motility, virulence.Formule :C20H24N10NaO14P2Couleur et forme :SolidMasse moléculaire :713.08464NI-Pano
NI-Pano (CH-03) is a novel hypoxia-activated KDAC inhibitor capable of O2-dependent release of the compound panobinostat.Formule :C26H28N6O4Couleur et forme :SolidMasse moléculaire :488.54Bilanafos
CAS :Bilanafos is an agent of Anti-Bacterial.Formule :C11H22N3O6PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :323.28Lapaquistat
CAS :Lapaquistat: active TAK-475 metabolite; reduces cholesterol synthesis and statin myotoxicity.Formule :C31H39ClN2O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :603.1TRK-IN-19
TRK-IN-19 (I-10) inhibits TRKA (1.1 nM IC50) & TRKAG595R (5.3 nM), promising for cancer research.Formule :C22H26FN5O2Couleur et forme :SolidMasse moléculaire :411.47MK-7128
CAS :MK-7128 is a CB1 receptor inverse agonist.Formule :C29H25ClF2N4O2Couleur et forme :SolidMasse moléculaire :534.98SSR 146977
CAS :NK3 receptor antagonistFormule :C35H42Cl2N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :621.64Belotecan
CAS :Belotecan (CKD-602) inhibits DNA topoisomerase I, blocks cell cycle, induces apoptosis, and is a camptothecin-derived anticancer agent.Formule :C25H27N3O4Couleur et forme :SolidMasse moléculaire :433.5AG-7404
CAS :AG-7404: strong protease inhibitor, fights poliovirus, EC50 0.080-0.674 μM, effective on V-073-resistant strains.Formule :C26H29N5O7Couleur et forme :SolidMasse moléculaire :523.54(-)-Adenophorine
CAS :(-)-Adenophorine is a moderate alpha-l-fucosidase inhibitor.Formule :C8H17NO4Couleur et forme :SolidMasse moléculaire :191.22Basroparib
CAS :Basroparib is an inhibitor of ribose polymerase (PARP) and has shown antitumour effects.Formule :C18H21F2N7O3Couleur et forme :SolidMasse moléculaire :421.4Macropa-NCS
CAS :Macropa-NCS is a macropa bifunctional analog with antitumor activity and can be used to study prostate cancer.Formule :C27H35N5O8SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :589.66rel-SB-612111 hydrochloride
CAS :NOP receptor antagonistFormule :C24H30Cl3NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :454.86PRMT5-IN-3
CAS :PRMT5-IN-3 is a PRMT5 inhibitor.PRMT5-IN-3 is a combined DNA damaging agent that is synthetically lethal to tumor cells.Formule :C22H23F3N4O3Couleur et forme :SolidMasse moléculaire :448.44Leualacin
CAS :Leualacin is a novel calcium blocker from Hapsidospora irregularis.Formule :C31H47N3O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :573.72Holothurinogenin
CAS :Holothurinogenin, as a lanosterol derivative, has toxic to nerve tissue.Formule :C30H46O4Couleur et forme :SolidMasse moléculaire :470.68Merigolix
CAS :Merigolix is a potent gonadotrophin releasing hormone (GnRH) antagonist .Formule :C36H35F7N4O6Couleur et forme :SolidMasse moléculaire :752.68LLS30
CAS :LLS30 inhibits Gal-1, reduces its binding affinity, and may help treat advanced prostate cancer.Formule :C34H33Cl4N5O3Couleur et forme :SolidMasse moléculaire :701.47PRN694
CAS :PRN694 is a potent, irreversible ITK/RLK inhibitor with IC50s: 0.3/1.4 nM; offers lasting effector cell suppression.Formule :C28H35F2N5O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :543.67BET-IN-8
BET-IN-8 (Compound 27) is a potent inhibitor of BET (Ki: 0.83 μM, Kd: 0.571 μM), which ameliorates LPS-induced sepsis in vivo.BET-IN-8 has shown potential inFormule :C22H21N3O4SCouleur et forme :SolidMasse moléculaire :423.48HIF-1α-IN-4
HIF-1α-IN-4 is an inhibitor of HIF-1α with IC50 of 24 nM in HEK293T cells which has potential antitumor effects.Formule :C16H12N2O3Couleur et forme :SolidMasse moléculaire :280.28Heparastatin
CAS :Heparastatin is an inhibitor of heparanase.Formule :C8H11F3N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :272.18Atorvastatin 3-Deoxyhept-2E-Enoic Acid
CAS :Atorvastatin 3-Deoxyhept-2E-Enoic Acid, an impurity in Atorvastatin, lowers blood lipids as an HMG-CoA reductase inhibitor.Formule :C33H33FN2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :540.62Ornoprostil
CAS :Ornoprostil, a prostaglandin E1 analogue, acts as a mucosal protectant.Formule :C23H38O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :410.54HDAC6-IN-9
CAS :HDAC6-IN-9 is a γ-secretase modulator that can significantly reduce the level of Aβ42 in mouse brain and can be used to study neurological diseases.Formule :C19H16N2O3Degré de pureté :98.84%Couleur et forme :SolidMasse moléculaire :320.345-HT7R antagonist 1
5-HT7R antagonist 1 is a G protein-biased antagonist with Ki of 6.5 nM for 5-HT 7R.Formule :C14H18Cl2N4Couleur et forme :SolidMasse moléculaire :313.23HIF-2α-IN-7
CAS :HIF-2α-IN-7 is a hypoxia inducible factor 2α (HIF-2α) inhibitor.Formule :C18H9F6NO2Couleur et forme :SolidMasse moléculaire :385.26DRX-065
CAS :DRX-065, a deuterated R-enantiomer of pioglitazone, treats NASH without PPARγ weight gain issues.Formule :C19H20N2O3SCouleur et forme :SolidMasse moléculaire :357.45PARP-1/HDAC-IN-1
CAS :PARP-1/HDAC-IN-1 is a PARP-1 and HDAC6 inhibitor with anticancer, antimigratory, and antiangiogenic activities and is used in tumor research.Formule :C22H18N4O4Degré de pureté :95.94%Couleur et forme :SolidMasse moléculaire :402.4LY 292728
CAS :LY 292728 is a highly potent antagonist of leukotriene B4 receptor.Formule :C34H29FO9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :600.59(S)-5-hydroxy-6-methoxy Duloxetine maleate
(S)-5-hydroxy-6-methoxy Duloxetine, an active metabolite of the (S)-duloxetine, functions as a serotonin (5-HT) and norepinephrine reuptake inhibitor.Formule :C19H21NO3S·C4H4O4Couleur et forme :SolidMasse moléculaire :459.51HBV-IN-20
HBV-IN-20 is a potent, orally active HBV inhibitor (EC50: 0.46 μM). HBV-IN-20 is a classical type II CpAM (core protein assembly regulator).Couleur et forme :SolidMDL-28050
CAS :MDL-28050 is a synthetic analog of hirudin 55-65 C-terminal fragment and a peptide inhibitor.Formule :C61H88N10O23Couleur et forme :SolidMasse moléculaire :1329.4Methysergide maleate
CAS :Methysergide prevents migraines/cluster headaches; treats serotonin syndrome, carcinoid-induced diarrhea; risk of fibrosis limits use.Formule :C25H31N3O6Degré de pureté :98%Couleur et forme :White To Off-WhiteMasse moléculaire :469.54SR 33805 oxalate
CAS :Ca2+ channel antagonistFormule :C34H42N2O9SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :654.77USP7-IN-6
CAS :USP7-IN-6 is a potent inhibitor of ubiquitin-specific protease 7 (USP7, IC50: 6.8 nM).Formule :C41H43N7O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :729.89SCH 563705
CAS :SCH 563705 is a CXCR2 and CXCR1 antagonist used in the study of acute respiratory syndrome, chronic obstructive pulmonary disease, and inflammation.Formule :C23H27N3O5Degré de pureté :98.03%Couleur et forme :SolidMasse moléculaire :425.48SCO-792
SCO-792: potent, reversible oral enteropeptidase inhibitor, with slow in vitro dissociation and in vivo protein digestion blocking.Formule :C22H22N4O8·xH2OCouleur et forme :SolidCHF-6366
CAS :CHF-6366: M3 antagonist & β2 agonist (pKi 10.4/11.4), mild Ca channel blocker, used in COPD study.Formule :C42H48N6O8Couleur et forme :SolidMasse moléculaire :764.87GSK065
CAS :GSK065 is a potent inhibitor of kynurenine-3-monooxygenase (KMO).Formule :C17H15ClN2O4Couleur et forme :SolidMasse moléculaire :346.77SB 258741 hydrochloride
SB 258741 hydrochloride is a potent antagonist of the 5-HT 7 receptor, designed specifically for studying schizophrenia [1].Formule :C19H31ClN2O2SCouleur et forme :SolidMasse moléculaire :386.98PD 134922
CAS :PD 134922 is a HIV-1 protease inhibitors. Inactivation of the protease prevents infectious virion formation.Formule :C37H61N5O7SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :719.9712(S)-HETE
CAS :Enpatoran hydrochloride (M5049 hydrochloride) is a TLR7/8 inhibitor with antiviral activity that is used in the study of autoimmune diseases.
Formule :C20H32O3Couleur et forme :SolidMasse moléculaire :320.47PF-06815345 hydrochloride
CAS :PF-06815345 HCl is an oral, potent PCSK9 inhibitor, IC50 13.4 μM, lowers PCSK9 in mice.Formule :C27H30Cl2FN9O4Couleur et forme :SolidMasse moléculaire :634.49AChE-IN-10
AChE-IN-10 (24r) inhibits AChE (IC50=2.4 nM), reducing amyloid buildup, tau phosphorylation, and promotes neuron health.Formule :C23H27F2NO4SCouleur et forme :SolidMasse moléculaire :451.53KUSC-5037
KUSC-5037 inhibits HIF-1 (IC50 = 1.2 μM) and mitochondrial complex V/FoF1ATP synthase.Formule :C18H17F3N6O2Couleur et forme :SolidMasse moléculaire :406.13651L-Sepiapterin
CAS :L-Sepiapterin aids in making BH4, a coenzyme essential for eNOS, enhancing artery function and angiogenesis, while suppressing ovarian cancer cell growth.Formule :C9H11N5O3Couleur et forme :SolidMasse moléculaire :237.22Antioxidant agent-8
Antioxidant agent-8, an oral Aβ 1-42 inhibitor, reduces fibril aggregation & promotes disaggregation; it's neuroprotective & BBB permeable.Formule :C13H12O5Couleur et forme :SolidMasse moléculaire :248.23SB-612111
CAS :SB-612111: potent ORL-1 antagonist, Ki=0.33 nM; μ-, κ-, δ-receptor Ki=57.6, 160.5, 2109 nM; blocks nociceptin's pain effect.Formule :C24H29Cl2NOCouleur et forme :SolidMasse moléculaire :418.40K027
K027 is a potent organophosphate (OP) inhibitor of acetylcholinesterase (AChE) reactivation. k027 can be used to study Alzheimer's disease.Formule :C15H18Br2N4O2Couleur et forme :SolidMasse moléculaire :446.14iNOs-IN-1
iNOs-IN-1 (YPW) is a strong iNOS inhibitor with dose-dependent anti-inflammatory properties, reducing IL-6, iNOS, and NO levels.Formule :C25H30N4O5Couleur et forme :SolidMasse moléculaire :466.53MRTX849 ethoxypropanoic acid
CAS :MRTX849 is a KRAS G12C ligand and PROTAC linker for creating potent LC-2, degrading KRAS G12C with DC50 of 0.25-0.76 μM.Formule :C37H43ClFN7O5Couleur et forme :SolidMasse moléculaire :720.24TrxR-IN-2
TrxR-IN-2 is a potential thioredoxin reductase (TrxR) inhibitor. TrxR-IN-2 has research value in the chemotherapy of drug-resistant hepatocellular carcinoma.Formule :C22H22N4O4Couleur et forme :SolidMasse moléculaire :406.43YM 202074
CAS :metabotropic glutamate receptor type 1 (mGlu1) antagonistFormule :C56H72N8O16S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1177.34LY 215890
CAS :LY 215890 is a compound that exhibits potent Gram-negative and Gram-positive antibacterial activity.Formule :C13H12ClN5O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :385.78BACE1-IN-2
CAS :BACE1-IN-2 is a BACE1 inhibitor (IC50: 22 nM).Formule :C19H15F4N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :421.35Sekdel sequence
CAS :Sekdel sequence, as a signal, leads to retention of at least two proteins in the endoplasmic reticulum of animal cells.Formule :C29H49N7O14Couleur et forme :SolidMasse moléculaire :719.74L-threo-Sphingosine C-18
CAS :L-threo-Sphingosine C-18 is a protein kinase C inhibitor.Formule :C18H37NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :299.49Alentemol hydrobromide
CAS :Alentemol hydrobromide is a Dopamine agonist.Formule :C19H26BrNODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :364.32RORγt Inverse agonist 2
CAS :RORγt Inverse agonist 2 is a selective, orally active inverse agonist of RORγt(EC50 of 119 nM).Formule :C27H25F8NO5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :627.54L-2'-Fd4C
CAS :L-2'-Fd4C is an L-nucleoside analogue with both anti-human immunodeficiency virus (HIV) and anti-hepatitis B virus (HBV) activity [1].Formule :C9H10FN3O3Couleur et forme :SolidMasse moléculaire :227.19PSMA-1007
CAS :PSMA-1007 is a novel Glu-Ureido-type prostate-specific membrane antigen (PSMA) inhibitor.Formule :C49H55FN8O16Couleur et forme :SolidMasse moléculaire :1030.01DG013A
CAS :DG013A inhibits ERAP1 & ERAP2 (IC50: 33 nM & 11 nM) to research autoimmune diseases & cancer.Formule :C27H37N4O4PCouleur et forme :SolidMasse moléculaire :512.58HSP90-IN-10
HSP90-IN-10 is a potent HSP90 inhibitor, targeting HCC1954 cells (IC50: 6 μM) and inducing apoptosis, sparing normal cells.Formule :C30H26FN3O6Couleur et forme :SolidMasse moléculaire :543.54MK-8876
CAS :MK-8876 is an Inhibitor of HCV NS5B Site D.Formule :C32H24F2N4O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :614.62Metoquizine
CAS :Metoquizine is an anticholinergic compound. It is a muscarinic acetylcholine receptor antagonist that has been used to treat ulcers.Formule :C22H27N5ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :377.48HDAC10-IN-2
HDAC10-IN-2, a selective HDAC10 inhibitor (IC50=20nM), modulates autophagy in FLT3-ITD+ acute myeloid leukemia.Formule :C19H22N2O2Couleur et forme :SolidMasse moléculaire :310.39Beloxepin
CAS :Beloxepin is an oral dual selective inhibitor of serotonin and norepinephrine uptake.Formule :C19H21NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :295.38TRPC4/5-IN-1
TRPC4/5-IN-1, a TRPC5/4 inhibitor with IC50s 0.54 μM/2.06 μM, targets skin inflammation and proteinuric kidney diseases.Formule :C21H21N3OCouleur et forme :SolidMasse moléculaire :331.41α-Amylase-IN-1
CAS :α-Amylase-IN-1 is an α-Amylase inhibitor (IC50: 0.5509 μM).Formule :C18H18N2O3Degré de pureté :99.92%Couleur et forme :SoildMasse moléculaire :310.356-trans-12-epi-Leukotriene B4
CAS :6-trans-12-epi-Leukotriene B4, a metabolite of arachidonic acid, serves as a potent anti-inflammatory agent.Formule :C20H32O4Couleur et forme :SolidMasse moléculaire :336.47hAChE/Aβ1-42-IN-1
CAS :Compound 16 (hAChE/Aβ1-42-IN-1) is a potent inhibitor targeting both hAChE and Aβ1-42 aggregation, demonstrating considerable safety in hepG2 cell lines andFormule :C20H24N6OCouleur et forme :SolidMasse moléculaire :364.44Aplysin
CAS :Aplysin suppresses breast cancer cells and protects liver cells by blocking PI3K/AKT/FOXO3a and preventing oxidative damage.Formule :C15H19BrOCouleur et forme :SolidMasse moléculaire :295.21Antibacterial agent 79
Antibacterial agent 79 is an antibacterial agent.Formule :C18H27N3O2S3Couleur et forme :SolidMasse moléculaire :413.62QPX7728 methoxy acetoxy methy ester
CAS :QPX7728 methoxy acetoxy methy ester is an inhibitor of boronic acid β-lactamase.Formule :C14H14BFO7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :324.07Isoleucyl tRNA synthetase-IN-2
CAS :Isoleucyl tRNA synthetase-IN-2 is a selective and potent inhibitor (Ki: 114 nM) that targets isoleucyl tRNA synthetase (IleRS).Formule :C22H33N5O8SCouleur et forme :SolidMasse moléculaire :527.59PDE4-IN-6
PDE4-IN-6: Potent PDE4 inhibitor, IC50 - 0.125μM (B), 0.43μM (D), anti-inflammatory, for arthritis research.Formule :C25H20FNO5SCouleur et forme :SolidMasse moléculaire :465.49Napsagatran hydrate
CAS :Napsagatran hydrate is a novel and specific inhibitor of thrombin.Formule :C26H36N6O7SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :576.66Tonapofylline
CAS :Tonapofylline, orally active, selectively blocks A1 adenosine receptor (Ki: 7.4 nM), used in heart failure research.Formule :C22H32N4O4Degré de pureté :98.57%Couleur et forme :SolidMasse moléculaire :416.515(S),6(R)-DiHETE
CAS :5(S),6(R)-DiHETE is a dihydroxy fatty acid from LTA4 hydrolysis and weak LTD4 agonist with ED50 of 1.3 μM for guinea pig ileum contraction.Formule :C20H32O4Couleur et forme :SolidMasse moléculaire :336.47HDAC8-IN-2
HDAC8-IN-2 (5o) inhibits both smHDAC8 and hHDAC8 with IC50s of 0.27 μM, 0.32 μM, kills schistosome larvae, and lowers egg laying.Formule :C21H16N2O5Couleur et forme :SolidMasse moléculaire :376.36ADU-S100 disodium salt
CAS :ADU-S100 (MIW815) disodium salt is an activator of stimulator of interferon genes (STING).Formule :C20H22N10Na2O10P2S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :734.51STING agonist-7
STING agonist-7 is an agonist of non-nucleotide STING that binds selectively to mouse STING but not human STING [1].Formule :C17H12N4O4Couleur et forme :SolidMasse moléculaire :336.3
