Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.524 produits)
- Apoptose(5.793 produits)
- Cycle cellulaire/point de contrôle(4.452 produits)
- Chromatine/Épigénétique(2.242 produits)
- Signalisation du cytosquelette(1.382 produits)
- Altération de l'ADN/réparation de l'ADN(2.826 produits)
- Endocrinologie/Hormones(3.507 produits)
- Enzyme(3.640 produits)
- GPCR/G-Protéine(8.333 produits)
- Immunologie et Inflammation(3.527 produits)
- Virus de la grippe(296 produits)
- Signalisation JAK/STAT(404 produits)
- Signalisation MAPK(1.203 produits)
- Transporteur membranaire/Canal ionique(2.792 produits)
- Métabolisme(9.449 produits)
- Microbiologie/Virologie(6.981 produits)
- Neuroscience(9.926 produits)
- Autres inhibiteurs(37.921 produits)
- Oxydation-Réduction(41 produits)
- Signalisation PI3K/Akt/mTOR(1.400 produits)
- Protéases/Protéasome(1.597 produits)
- Cellules souche et Dérivés(830 produits)
- Tyrosine Kinase/Adaptateurs(2.015 produits)
- Ubiquitination(1.650 produits)
Affichez 16 plus de sous-catégories
66639 produits trouvés pour "Inhibiteurs"
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KRAS G12C inhibitor 50
CAS :<p>KRAS G12C inhibitor 50 is a KRAS G12C inhibitor (IC50: 46.7 nM).</p>Formule :C31H34N8O2Couleur et forme :SolidMasse moléculaire :550.65QTX125 TFA
<p>QTX125 TFA: Potent, selective HDAC6 inhibitor with antitumor effects.</p>Formule :C25H20F3N3O7Couleur et forme :SolidMasse moléculaire :531.44Leukotriene F-4 sulfone
CAS :<p>Leukotriene F-4 sulfone induces vascular permeability changes.</p>Formule :C28H44N2O10SCouleur et forme :SolidMasse moléculaire :600.72Antitumor agent-48
<p>Antitumor agent-48, a 2,3-dehydrosilybin derivative, exhibits cytotoxicity on MCF-7, NCI-H1299, HepG2, HT29 cells; IC50 ranging 8.06-16.51 µM.</p>Formule :C35H34N2O14Couleur et forme :SolidMasse moléculaire :706.65Isoleucyl tRNA synthetase-IN-2
CAS :<p>Isoleucyl tRNA synthetase-IN-2 is a selective and potent inhibitor (Ki: 114 nM) that targets isoleucyl tRNA synthetase (IleRS).</p>Formule :C22H33N5O8SCouleur et forme :SolidMasse moléculaire :527.59DNA-PK-IN-2
CAS :<p>DNA-PK-IN-2 is an inhibitor of the DNA-PK enzyme complex, useful in cancer research.</p>Formule :C20H23N5O3Couleur et forme :SolidMasse moléculaire :381.43METTL3-IN-2
CAS :<p>METTL3-IN-2, a potent METTL3 inhibitor, exhibits an IC50 value of 6.1 nM, effectively impairing the proliferation of Caov3 cancer cells.</p>Formule :C25H26N8OCouleur et forme :SolidMasse moléculaire :454.53RhlR antagonist 1
<p>RhlR antagonist 1: IC50 of 26 μM, selective for RhlR, inhibits P. aeruginosa biofilm and virulence factors.</p>Formule :C12H10F2OCouleur et forme :SolidMasse moléculaire :208.22R,4R-Sacubitril
CAS :<p>2R,4R-Sacubitril is the impurity of Sacubitril. Sacubitril is used in combination with valsartan for the treatment of patients with heart failure.</p>Formule :C24H29NO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :411.49Trk-IN-8
<p>Trk-IN-8: TRK inhibitor with IC50 of 0.42 nM (TRKA), 0.89 nM (TRKA-G595R), 1.5 nM (TRKC-G623R).</p>Formule :C18H16F2N6O2Couleur et forme :SolidMasse moléculaire :386.36Rostratin B
CAS :<p>Rostratin B, a cytotoxic disulfide, demonstrates in vitro cytotoxicity against human colon carcinoma (HCT-116), exhibiting an IC50 value of 1.9 μg/mL.</p>Formule :C18H20N2O6S2Couleur et forme :SolidMasse moléculaire :424.49Resolvin E2
CAS :<p>RvE2, a bioactive lipid from the SPM family, is made from EPA and reduces inflammatory neutrophil infiltration and helps treat NAFLD and other diseases.</p>Formule :C20H30O4Couleur et forme :SolidMasse moléculaire :334.45HIV-1 inhibitor-40
<p>HIV-1 inhibitor-40 (4ab) is a potent NNRTI (EC50: 1.9 nM), non-toxic in vivo, and a sensitive CYP inhibitor.</p>Formule :C25H18N6O2Couleur et forme :SolidMasse moléculaire :434.45ChemR23-IN-3
<p>ChemR23-IN-3 is a potent thiazole-based ChemR23 inhibitor with an IC 80 value of 12 nM.</p>Formule :C31H33N5O5S2Couleur et forme :SolidMasse moléculaire :619.75UK-432097
CAS :<p>UK 432097 is an adenosine A2A agonist.</p>Formule :C40H47N11O6Couleur et forme :SolidMasse moléculaire :777.87MM-589 TFA
CAS :<p>MM-589 TFA is a potent WD repeat domain 5 (WDR5)inhibitor and mixed lineage leukemia (MLL) protein-protein interaction.</p>Formule :C30H45F3N8O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :686.72Alkannin
CAS :<p>Alkannin: potent, tumor-specific PKM2 inhibitor; non-inhibitory to PKM1/PKL; potential anticancer agent.</p>Formule :C16H16O5Couleur et forme :SolidMasse moléculaire :288.3Fusarisetin A
CAS :<p>Fusarisetin A, a pentacyclic fungal metabolite, is an acinar morphogenesis inhibitor .</p>Formule :C22H31NO5Couleur et forme :SolidMasse moléculaire :389.49P300 bromodomain-IN-1
<p>P300 bromodomain-IN-1 blocks c-Myc, induces G1/G0 arrest, apoptosis. Potent EP300 inhibitor (IC50: 49 nM).</p>Formule :C29H31ClN4O4Couleur et forme :SolidMasse moléculaire :535.03LSD1-IN-22
<p>LSD1-IN-22: potent LSD1 inhibitor, K_i 98 nM, curbs cancer cell growth.</p>Formule :C9H8BrF2NCouleur et forme :SolidMasse moléculaire :248.07CaMKIIα-IN-1
<p>CaMKIIα-IN-1 (Compound 4d) is an orally active inhibitor of Ca 2+ /calmodulin-dependent protein kinase II α (CaMKIIα) with a Kd of 219 nM for CaMKIIα WT hub.</p>Formule :C14H11ClO4Couleur et forme :SolidMasse moléculaire :278.69ROPA
CAS :<p>ROPA, a potent PKCalpha and PKCgamma activator, promotes tumor growth through PKC-activation.</p>Formule :C28H32O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :464.55CD73-IN-12
<p>CD73-IN-12, a compound from CN114437038A, shows strong anti-tumor activity by effectively inhibiting CD73 enzyme.</p>Formule :C17H14F2N4O2Couleur et forme :SolidMasse moléculaire :344.32LRRK2-IN-4
CAS :<p>LRRK2-IN-4: Potent, selective LRRK2 inhibitor, oral, BBB-penetrating, IC50=2.6 nM, potential for Parkinson's.</p>Formule :C25H29ClF2N6O2Couleur et forme :SolidMasse moléculaire :518.99(S)-Seco-Duocarmycin SA
CAS :<p>(S)-Seco-Duocarmycin SA is a DNA alkylating agent and antibiotic with potent antitumor activity that can be used to synthesize ADC compounds.</p>Formule :C25H24ClN3O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :513.939-cis-β-Carotene
CAS :<p>9-cis-β-Carotene, a precursor of retinal, is cleaved by beta-carotene oxygenase 1 (BCMO1) to produce 9-cis-retinal.</p>Formule :C40H56Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :536.87Belatacept
CAS :<p>Belatacept (BMS 224818), a T-cell costimulation inhibitor, targets CD80/86 for transplant immunosuppression.</p>Couleur et forme :LiquidNI-Pano
<p>NI-Pano (CH-03) is a novel hypoxia-activated KDAC inhibitor capable of O2-dependent release of the compound panobinostat.</p>Formule :C26H28N6O4Couleur et forme :SolidMasse moléculaire :488.54CDK4/6-IN-10
<p>CDK4/6-IN-10: Oral CDK4 (IC50: 22 nM) & CDK6 (IC50: 10 nM) inhibitor with anti-cancer potential for MM research.</p>Couleur et forme :SolidYM-60828 dihydrochloride
CAS :<p>YM-60828 dihydrochloride is a Factor Xa (FXa) inhibitor and anticoagulant used in the treatment of venous thromboembolic disease.</p>Formule :C27H33Cl2N5O5SCouleur et forme :SolidMasse moléculaire :610.55SphK1-IN-1
<p>SphK1-IN-1: SphK1 ATPase inhibitor, IC50=2.48 μM, potential for cancer research.</p>Formule :C22H22N6O2Couleur et forme :SolidMasse moléculaire :402.45S1PR1 agonist 1
CAS :<p>S1PR1 agonist 1 is a potent agonist of S1PR1. S1PR1 agonist 1 has potential in autoimmune diseases.</p>Formule :C29H30N4O4Couleur et forme :SolidMasse moléculaire :498.57Unoprostone
CAS :<p>Unoprostone is a prostaglandin F2α analogs (PGAs), and reduces intraocular pressure and is used topically for glaucoma or ocular hypertension.</p>Formule :C22H38O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :382.53Finafloxacin
CAS :<p>Finafloxacin is a pH-activated fluoroquinolone, most effective at pH 5.0-6.0, targeting bacterial topoisomerases, used for UTIs and H. pylori infections.</p>Formule :C20H19FN4O4Couleur et forme :SolidMasse moléculaire :398.39Mu opioid receptor antagonist 2
<p>Compound 25: potent, selective MOR antagonist, crosses blood-brain barrier (Ki: 0.37 nM, EC50: 0.44 nM), for OUD research.</p>Formule :C25H28N2O4SCouleur et forme :SolidMasse moléculaire :452.57BTK-IN-16
CAS :<p>BTK-IN-16 is a potential inhibitor of wild-type BTK and C481S mutants.BTK-IN-16 can be used to study various autoimmune diseases and cancers caused by BTK.</p>Formule :C15H14N4O2Degré de pureté :99.04%Couleur et forme :SoildMasse moléculaire :282.3SB 204070 hydrochloride
CAS :<p>SB 204070 hydrochloride is an inhibitor of beta-lactamase, it is isolated from Spondias mombin.</p>Formule :C19H27ClN2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :382.88HDAC-IN-35
<p>HDAC-IN-35 (Compound 14) is an effective and selective inhibitor of VEGFR-2 and HDAC, with IC50 values of 13.2 and 0.166 μM for VEGFR-2 and HDAC6, respectively.</p>Formule :C17H13ClF3N3O3Couleur et forme :SolidMasse moléculaire :399.75GSK268
<p>GSK268 is a BET inhibitor.</p>Formule :C26H27N5O3Couleur et forme :SolidMasse moléculaire :457.53Ivaltinostat formic
<p>Ivaltinostat (CG-200745) is an oral panHDAC inhibitor, inducing apoptosis and enhancing cancer drug sensitivity.</p>Formule :C25H35N3O6Couleur et forme :SolidMasse moléculaire :473.56ZBH-1205
CAS :<p>ZBH-1205, a camptothecin derivative, shows strong antitumor effects via apoptosis, outperforming cpt-11 and sn38 in topoisomerase-1 inhibition.</p>Formule :C29H31N3O8Couleur et forme :SolidMasse moléculaire :549.57SSTR5 antagonist 2 hydrochloride
<p>SSTR5 antagonist 2 hydrochloride: potent, oral SSTR5 blocker with potential in type 2 diabetes research.</p>Formule :C32H36ClFN2O5Couleur et forme :SolidMasse moléculaire :583.09OncoFAP
CAS :<p>OncoFAP is an ultra-high affinity fibroblast activating protein (FAP) ligand with potential tumour targeting.</p>Formule :C21H19F2N5O5Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :459.40TLR7/8 antagonist 1
<p>Compound 16c, an imidazoquinoline, is a TLR7/8 agonist; IC50: 3.91 μM (TLR7), 2.19 μM (TLR8); targets TLR-2050 for disease treatment.</p>Formule :C24H27N5O2Couleur et forme :SolidMasse moléculaire :417.5Cdc7-IN-18
CAS :<p>Cdc7-IN-18 (1-2) inhibits CDC7 enzyme (IC50: 1.29 nM) and COLO205 cell proliferation (IC50: 53.62 nM).</p>Formule :C19H21N5OSCouleur et forme :SolidMasse moléculaire :367.47(S)-JDQ-443
CAS :<p>(S)-JDQ-443, an isomer of JDQ-443, is a selective, potent oral KRAS G12C inhibitor with antitumor properties.</p>Formule :C29H28ClN7OCouleur et forme :SolidMasse moléculaire :526.03PF 03709270
CAS :<p>PF 03709270 is an oral prodrug of sulopenem with broad-spectrum antibacterial effects on gram-positive and gram-negative bacteria.</p>Formule :C19H27NO7S3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :477.61JAK1/TYK2-IN-3
<p>JAK1/TYK2-IN-3, orally active, selectively inhibits TYK2 (IC50: 6 nM), JAK1 (37 nM), JAK2 (140 nM), JAK3 (362 nM), and has anti-inflammatory effects.</p>Couleur et forme :SolidAnticancer agent 35
<p>Compound 10, a sulfonylurea, inhibits A549, A431, PACA2 cells with IC50s: 18.1, 4.0, 18.9 μg/mL.</p>Formule :C15H13N3O3S3Couleur et forme :SolidMasse moléculaire :379.48FCE-27262
CAS :<p>FCE-27262 is a prostaglandin H2/thromboxane A2 receptor antagonist.</p>Formule :C23H31N3O3Couleur et forme :SolidMasse moléculaire :397.51TAS05567
CAS :<p>TAS05567 is a potent, highly selective, and ATP-competitive Syk inhibitor (IC50: 0.37 nM).</p>Formule :C21H29N9O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :439.51Mibefradil dihydrochloride hydrate
CAS :<p>Mibefradil dihydrochloride hydrate is a long-acting antihypertensive blocking high-voltage L calcium channels.</p>Formule :C29H42Cl2FN3O4Couleur et forme :SolidMasse moléculaire :586.57BMS-986339
CAS :<p>BMS-986339: oral, potent FXR agonist; binds to His298/ASN287; for PBC, PSC, NASH, anti-fibrosis research.</p>Formule :C35H41F4N3O4Couleur et forme :SolidMasse moléculaire :643.71Alentemol hydrobromide
CAS :<p>Alentemol hydrobromide is a Dopamine agonist.</p>Formule :C19H26BrNODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :364.32ATM Inhibitor-1
CAS :<p>ATM Inhibitor-1 is a highly potent, selective and orally active ATM inhibito (IC50: 0.7 nM) anti-tumor activity.</p>Formule :C27H36N6O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :492.61Org-6906
CAS :<p>DCB-3503, a tylophorine analog, may treat cancer and suppress immunity by blocking protein synthesis and modulating HSC70's ATPase activity.</p>Formule :C13H16ClNDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :221.73Encephalitic alphavirus-IN-1
<p>Alphavirus-IN-1 blocks VEEV (EC50: 0.24 μM) & EEEV (EC50: 0.16 μM), non-toxic, stable in mice plasma.</p>Formule :C27H25FN6O2Couleur et forme :SolidMasse moléculaire :484.52MurB-IN-1
<p>MurB-IN-1 (compound 44) inhibits key bacterial enzyme MurB with 3.57 μM affinity, offering treatment potential against P. aeruginosa.</p>Formule :C12H7Cl2F3N2O2Couleur et forme :SolidMasse moléculaire :339.1GSK-3036656 free base
CAS :<p>GSK656 (GSK3036656) inhibits Mtb LeuRS with IC50 of 0.20 μM, promising for tuberculosis treatment.</p>Formule :C10H13BClNO4Couleur et forme :SolidMasse moléculaire :257.48AXKO-0046
<p>AXKO-0046 is an indole derivative and small-molecule LDHB selective inhibitor.</p>Formule :C25H33N3Couleur et forme :SolidMasse moléculaire :375.55UCN-01
CAS :<p>inhibitor of Akt, protein kinase C, PDK1 and cyclin-dependent kinases</p>Formule :C28H26N4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :482.53EGFR/HER2-IN-5
<p>EGFR/HER2-IN-5: Irreversible, oral dual EGFR inhibitor, IC50 0.6 nM, targets L858R/T790M mutations, anti-tumor in vivo for lung cancer study.</p>Couleur et forme :SolidJH295 hydrate
<p>JH295 hydrate: potent, irreversible Nek2 inhibitor (IC50 = 770 nM), selective, doesn't target Cdk1, Aurora B or Plk1.</p>Formule :C18H18N4O3Couleur et forme :SolidMasse moléculaire :338.36CBP/p300-IN-18
<p>CBP/p300-IN-18 (compound 8) is a potent inhibitor of EP300/CBP HAT, acting on HAT EP300 (IC50: 0.056 μM) and LK2 H3K27 (IC50: 0.46 μM).</p>Formule :C25H27FN4O3Couleur et forme :SolidMasse moléculaire :450.51Tubulin polymerization-IN-34
<p>"Tubulin-IN-34 inhibits oxazolylisoindole microtubule assembly, selective for VL51 lymphoma."</p>Formule :C31H35N3O6Couleur et forme :SolidMasse moléculaire :545.63LasR-IN-3
<p>LasR-IN-3 inhibits LasR in Pseudomonas, disrupting its dimer, causing loss of function.</p>Formule :C22H19N3O2Couleur et forme :SolidMasse moléculaire :357.41Arterolane
CAS :<p>Arterolane is an antimalarial compound. For against P. falciparum Ro73 and W2, the IC50s are both 1.1 nM.</p>Formule :C22H36N2O4Couleur et forme :SolidMasse moléculaire :392.53RORγt Inverse agonist 2
CAS :<p>RORγt Inverse agonist 2 is a selective, orally active inverse agonist of RORγt(EC50 of 119 nM).</p>Formule :C27H25F8NO5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :627.54HIV-1 inhibitor-44
<p>HIV-1 inhibitor-44 (compound 11l) is an HIV-1 reverse transcriptase inhibitor that exhibits activity against wild-type HIV-1 strains (EC50: 0.209 μM).</p>Formule :C23H26N2O4SCouleur et forme :SolidMasse moléculaire :426.53Kri 1314
CAS :<p>Kri 1314 is a cyclohexyl-norstatine-containing dipeptide renin inhibitor which has potential for the treatment of hypertension.</p>Formule :C38H51N5O7Couleur et forme :SolidMasse moléculaire :689.84trans-RdRP-IN-5
<p>Trans-RdRP-IN-5 is a potent inhibitor of the influenza virus RNA-dependent RNA polymerase (RdRP), with applications in influenza virus research.</p>Formule :C23H21N3O5Couleur et forme :SolidMasse moléculaire :419.43GYKI-53784
CAS :<p>GYKI-53784 (LY 303070) is an effective selective AMPA receptor antagonist.</p>Formule :C19H20N4O3Couleur et forme :SolidMasse moléculaire :352.39U 80215
CAS :<p>U 80215 is an enzyme-competitive inhibitor.</p>Formule :C42H60N8O6SCouleur et forme :SolidMasse moléculaire :805.04NMDAR/HDAC-IN-1
<p>Compound 9d is a dual NMDAR and HDAC inhibitor with high NMDAR affinity (Ki=0.59 μM) and inhibits HDAC1-3,6,8; crosses the blood-brain barrier.</p>Formule :C22H28N2O3Couleur et forme :SolidMasse moléculaire :368.47AZ-PFKFB3-67 quarterhydrate
<p>AZ-PFKFB3-67 quarterhydrate inhibits PFKFB3 (IC50: 11 nM), PFKFB2 (159 nM), and PFKFB1 (1130 nM).</p>Formule :C26H27N5O4Couleur et forme :SolidMasse moléculaire :460.01Terpendole E
CAS :<p>Terpendole E is an atypical L5 site inhibitor.</p>Formule :C28H39NO3Couleur et forme :SolidMasse moléculaire :437.61Acetoxycycloheximide
CAS :<p>Acetoxycycloheximide triggers TNF receptor 1, prompts apoptosis, and cytochrome c release by activating c-Jun N-terminal kinase.</p>Formule :C17H25NO6Couleur et forme :SolidMasse moléculaire :339.38Anti-inflammatory agent 10
<p>Tilomisole-derived benzimidazole-thiazole, orally active, favors COX-2 inhibition over COX-1.</p>Formule :C17H13BrN4O3S2Couleur et forme :SolidMasse moléculaire :465.34CS-0777
CAS :<p>CS-0777 is a potent, selective, and orally active S1P1 agonist (sphingosine 1-phosphate receptor modulator).</p>Formule :C21H31N2O5PCouleur et forme :SolidMasse moléculaire :422.45Dehatrine
CAS :<p>Dehatrine: alkaloid from Beilschmiedia madang, inhibits Plasmodium falciparum K1 growth.</p>Formule :C37H38N2O6Couleur et forme :SolidMasse moléculaire :606.71PARP10/15-IN-3
<p>Compound 8a, a dual PARP10 & PARP15 inhibitor, has IC50s: PARP10 at 0.14μM & PARP15 at 0.40μM; it's cell-permeable & anti-apoptotic.</p>Formule :C12H12N2O3Couleur et forme :SolidMasse moléculaire :232.24MRGPRX1 agonist 3
<p>Compound 1f, a potent MRGPRX1 agonist, has an EC50 of 0.22 μM, useful for neuropathic pain studies.</p>Formule :C14H11FN2OSCouleur et forme :SolidMasse moléculaire :274.31MK-8876
CAS :<p>MK-8876 is an Inhibitor of HCV NS5B Site D.</p>Formule :C32H24F2N4O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :614.62Calcipotriol Impurity C
CAS :<p>Calcipotriol Impurity C is the impurity of Calcipotriol. Calcipotriol is a VDR-like receptors ligand.</p>Formule :C27H40O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :412.614D-473
CAS :<p>D-473 is a novel orally active triple reuptake inhibitor targeting dopamine, serotonin and norepinephrine transporters.</p>Formule :C26H27F2NO3Couleur et forme :SolidMasse moléculaire :439.49PD-149163
CAS :<p>PD-149163: brain-penetrating, selective NTR1 agonist; shows pro-cognitive, anti-psychotic, anxiolytic effects.</p>Formule :C42H71N9O6Couleur et forme :SolidMasse moléculaire :798.07Homomoschatoline
CAS :<p>Homomoschatoline is an antibacterial isolated from Artabotrys crassifolius.</p>Formule :C19H15NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :321.33AChE-IN-10
<p>AChE-IN-10 (24r) inhibits AChE (IC50=2.4 nM), reducing amyloid buildup, tau phosphorylation, and promotes neuron health.</p>Formule :C23H27F2NO4SCouleur et forme :SolidMasse moléculaire :451.53Antitubercular agent-22
<p>Antitubercular agent-22 combats Candida albicans (MIC: 2.34 μg/ml) and M. tuberculosis (MIC: 2 μg/ml).</p>Formule :C24H28FN5O8Couleur et forme :SolidMasse moléculaire :533.51Mibefradil
CAS :<p>Mibefradil is a calcium channel blocker with moderate selectivity for T-type Ca2+ channels (IC50s: 2.7 μM and 18.6 μM for T-type and L-type currents).</p>Formule :C29H38FN3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :495.63EGFR/HER2-IN-4
<p>EGFR/HER2-IN-4: oral, irreversible dual EGFR inhibitor (IC50: 0.6 nM), targets L858R/T790M mutations, potent anti-lung cancer effects in vivo.</p>Couleur et forme :SolidMTL-CEBPA
<p>MTL-CEPBA is a small activating RNA that targets C/EBPα upregulation and exhibits anti-inflammatory and anti-cancer effects.</p>Couleur et forme :SolidMenin-MLL inhibitor 4
CAS :<p>Menin-MLL inhibitor 4 has antitumor activity.Menin-MLL inhibitor 4 is an inhibitor of Menin- MLL (mixed-lineage leukemia protein) interaction .</p>Formule :C32H38FN7O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :587.69ONO-5334
CAS :<p>ONO-5334: selective cathepsin K inhibitor, potential for osteoporosis study; Ki: 0.10 nM (human), 0.049 nM (rabbit), 0.85 nM (rat).</p>Formule :C21H34N4O4SDegré de pureté :98.22% - 99.60%Couleur et forme :SolidMasse moléculaire :438.58FTI 276 TFA
CAS :<p>FTI 276 TFA targets plasmodium falciparum & humans, inhibits PFT with IC50s: 0.9 nM (parasite) & 0.5 nM (human).</p>Formule :C23H28F3N3O5S2Couleur et forme :SolidMasse moléculaire :547.61EGFR-IN-48
<p>EGFR-IN-48: potent EGFR inhibitor, oral, IC50: 0.193-66.7 nM, blocks EGFR mutants & BaF3/PC-9 cell proliferation.</p>Couleur et forme :SolidJAK2/FLT3-IN-1 TFA
<p>JAK2/FLT3-IN-1 (TFA), an oral JAK2/FLT3 inhibitor, shows anticancer properties; IC50: JAK2 (0.7 nM), FLT3 (4 nM), JAK1 (26 nM), JAK3 (39 nM).</p>Formule :C27H35F4N7O3Couleur et forme :SolidMasse moléculaire :581.61Olanzapine/Samidorphan
CAS :<p>Olanzapine/Samidorphan, a tablet blending olanzapine and samidorphan, targets schizophrenia and bipolar I, curbing weight gain.</p>Formule :C38H46N6O4SCouleur et forme :SolidMasse moléculaire :682.88Cilobamine (free base)
CAS :<p>Cilobamine: a stimulant antidepressant, inhibits norepinephrine-dopamine reuptake, based on dichloroisoprenaline structure.</p>Formule :C17H23Cl2NOCouleur et forme :SolidMasse moléculaire :328.28HIV-1 inhibitor-52
CAS :<p>HIV-1 inhibitor-52: potent, broad-spectrum with EC50s 1.6-6.4 nM against various HIV-1 strains.</p>Formule :C46H72FNO5SCouleur et forme :SolidMasse moléculaire :770.13rel-SB-612111 hydrochloride
CAS :<p>NOP receptor antagonist</p>Formule :C24H30Cl3NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :454.86hCA XII/II/IX-IN-1
<p>hCA XII/II/IX-IN-1 inhibits hCA I/II/IX/XII (IC50: 2.6, 0.004, 0.005, 0.001 μM) with anticancer properties.</p>Formule :C25H34N4O7SCouleur et forme :SolidMasse moléculaire :534.63Antibiotic MA 144M2
CAS :<p>Antibiotic MA 144M2, an anthracycline glycoside, targets gram-positive bacteria and tumors, derived from Streptomyces and aclacinomycin A conversion.</p>Formule :C42H55NO16Couleur et forme :SolidMasse moléculaire :829.88PI3Kα-IN-8
<p>PI3Kα-IN-8 is a selective inhibitor of PI3Kα (IC50: 0.012 μM).</p>Formule :C26H27BrN4O2Couleur et forme :SolidMasse moléculaire :507.42Pol I-IN-1
<p>Pol I-IN-1 is a powerful inhibitor of RNA polymerase I (Pol I), specifically targeting the large catalytic subunit RPA194, demonstrating an inhibition</p>Formule :C23H22N4O2Couleur et forme :SolidMasse moléculaire :386.45eIF4A3-IN-6
CAS :<p>eIF4A3-IN-6 is a potent eIF4A inhibitor, potentially used for treating eIF4A-related diseases like cancer. (US20170145026A1)</p>Formule :C26H25N3O5Couleur et forme :SolidMasse moléculaire :459.49GNE-203
CAS :<p>GNE-203 is a Met inhibitor.</p>Formule :C30H29Cl2F3N8O3Couleur et forme :SolidMasse moléculaire :677.50p38 MAPK-IN-3
<p>Compound 2c is a potent p38α MAPK inhibitor with antitumor effects, enhancing apoptosis and ROS.</p>Formule :C22H17BrO2Couleur et forme :SolidMasse moléculaire :393.27Cicaprost
CAS :<p>Cicaprost (ZK 96480) is an IP agonist with artery relaxing effects; EC50 is 5.8 nM.</p>Formule :C22H30O5Couleur et forme :SolidMasse moléculaire :374.47PNU-140457
CAS :<p>PNU-140457 is a bio-active chemical.</p>Formule :C14H14FN5O3Couleur et forme :SolidMasse moléculaire :319.29N'-(2-Fluorophenyl)pyrazine-2-carbohydrazide
<p>N'-(2-Fluorophenyl)pyrazine-2-carbohydrazide is a Ole1p desaturase inhibitor as well as antifungal agent [1].</p>Formule :C11H9FN4OCouleur et forme :SolidMasse moléculaire :232.21CXCR2 antagonist 7
<p>CXCR2 antagonist 7 is a powerful blocker with IC50s: 0.044 μM for binding, 0.66 μM for calcium mobilization.</p>Formule :C14H14F2N6OSCouleur et forme :SolidMasse moléculaire :352.36MDL-100240
CAS :<p>MDL-100240 inhibits ACE/neprilysin, effective against hypertension-induced heart/vascular changes.</p>Formule :C26H28N2O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :480.58FGFR4-IN-6
<p>FGFR4-IN-6: covalent, reversible FGFR4 blocker, 5.4 nM IC50, good oral bioavailability, reduces Hep3B2.1-7 tumors in mice, low toxicity.</p>Formule :C31H33N7O4Couleur et forme :SolidMasse moléculaire :567.64HbF inducer-1
<p>HbF inducer-1 is a fetal hemoglobin inducer which is orally bioavailable.</p>Formule :C18H19N3O3Couleur et forme :SolidMasse moléculaire :325.36MtTMPK-IN-8
<p>MtTMPK-IN-8 inhibits MtbTMPK, has low cytotoxicity, shows 0.78-9.4 μM activity against Mycobacterium, useful for tuberculosis research.</p>Formule :C24H24N6O7Couleur et forme :SolidMasse moléculaire :508.48CI 992
CAS :<p>CI 992 is a novel potent inhibitor of primate renin.</p>Formule :C33H52N6O7S2Couleur et forme :SolidMasse moléculaire :708.93Vindeburnol
CAS :<p>Vindeburnol is a cerebral vasodilator vincamine analog that bears neuroprotective properties.</p>Formule :C17H20N2OCouleur et forme :SolidMasse moléculaire :268.35Nurr1 agonist 1
<p>Nurr1 agonist 1 is an inverse agonist tool for the neuroprotective transcription factor Nurr1 which is an appealing target to treat neurodegenerative diseases.</p>Formule :C16H14N2O2Couleur et forme :SolidMasse moléculaire :266.29Gamendazole
CAS :<p>Gamendazole is a novel drug candidate for male contraception. It has been shown to reduce fertility in male rats without affecting testosterone levels.</p>Formule :C18H11Cl2F3N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :415.19NS2B/NS3-IN-4
CAS :<p>Compound 34e inhibits DENV2/ZIKV proteases; IC50: 0.69 µM (DENV2), 1.04 µM (ZIKV).</p>Formule :C15H11NO4Couleur et forme :SolidMasse moléculaire :269.25GSK 366
CAS :GSK 366 is a potent kynurenine-3-monooxygenase (KMO) inhibitor (IC50s: 0.7 nM and 2.3 nM for P. fluorescens-KMO and human KMO).Formule :C17H16ClN3O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :361.78LL-Z 1640-4
CAS :A signal-specific JNK/p38 pathway and TAK 1 inhibitorFormule :C19H24O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :364.39PD-1/PD-L1-IN-13
<p>PD-1/PD-L1-IN-13 is a potent immune checkpoint PD-1/PD-L1 inhibitor with an IC50 value of 10.2 nM for PD-1/PD- L1 interaction.PD-1/PD-L1-IN-13 promotes CD8+ T-</p>Formule :C36H34ClF2N3O9Couleur et forme :SolidMasse moléculaire :726.12Utrophin modulator 1
<p>UM1 upregulates utrophin, has EC50 of 0.11 μM, useful in DMD research.</p>Formule :C22H18N6OCouleur et forme :SolidMasse moléculaire :382.42Tilpisertib fosmecarbil
CAS :<p>Tilpisertib fosmecarbil is a potent inhibitor of serine/threonine kinases with anti-inflammatory properties.</p>Formule :C35H36ClN8O7PCouleur et forme :SolidMasse moléculaire :747.14Antifungal agent 11
<p>Antifungal agent 11 has a good antifungal effect.</p>Formule :C21H19F2N7O3S2Couleur et forme :SolidMasse moléculaire :519.55LY 541850
CAS :<p>LY541850 is a selective orthosteric mGlu2 agonist and mGlu3 antagonist with IC50 values of 0.161 μM and 0.038 μM, respectively.LY 541850 is claimed from human</p>Formule :C9H13NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :199.2PF-06795071
CAS :<p>PF-06795071 is an effective and selective covalent inhibitor of MAGL (IC50: 3 nM).</p>Formule :C18H17F4N3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :399.34Isoleucyl tRNA synthetase-IN-1
CAS :<p>Isoleucyl tRNA synthetase-IN-1 is a selective and potent inhibitor (Ki: 88 nM) that targets isoleucyl tRNA synthetase (IleRS).</p>Formule :C23H35N5O7SCouleur et forme :SolidMasse moléculaire :525.62DAD dichloride
<p>DAD dichloride is a 3rd-gen photoelectric switch, blocks K+ channels, and helps in visual function research.</p>Formule :C26H42Cl2N6OCouleur et forme :SolidMasse moléculaire :525.56MCTR2
CAS :<p>MCTR2, synthesized from DHA in macrophages, aids in tissue repair and reduces inflammation by promoting eicosanoid PGD2 and PGF2α decrease.</p>Formule :C27H40N2O6SCouleur et forme :SolidMasse moléculaire :520.68CM-414
CAS :<p>CM-414: HDAC/PDE5 inhibitor, targeting Alzheimer’s, IC50s: PDE5 (60 nM), HDAC1/2/3/6. Reduces Aβ, pTau in mice, boosts cognition.</p>Formule :C23H29N5O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :439.51Factor B-IN-4
CAS :<p>Factor B-IN-4 is a potent inhibitor (IC50: 1 μM) of complement factor B. Factor B-IN-4 can be used to study inflammatory and immune-related diseases.</p>Formule :C27H32N2O4Couleur et forme :SolidMasse moléculaire :448.55GABAA receptor agonist 1
<p>Compound 3e, a potent GABAA agonist, targets GABA sites and has potential anti-depressive effects in mice.</p>Formule :C20H30O3Couleur et forme :SolidMasse moléculaire :318.45GLS1 Inhibitor-5
<p>GLS1 Inhibitor-5 (24y): Selective, oral glutaminase 1 inhibitor; IC50 68 nM; induces apoptosis; anti-tumor.</p>Couleur et forme :SolidNorbinaltorphimine dihydrochloride
CAS :<p>Norbinaltorphimine dihydrochloride is a selective and potent κ opioid receptor antagonist that induces itch-associated responses in mice.</p>Formule :C40H45Cl2N3O6Degré de pureté :98.17% - 99.88%Couleur et forme :SolidMasse moléculaire :734.71Peridinin
CAS :<p>Peridinin is an exceptionally potent and membrane-embedded inhibitor of bilayer lipid peroxidation.</p>Formule :C39H50O7Couleur et forme :SolidMasse moléculaire :630.81L 668411
CAS :<p>L 668411, the 2,3-ditritiated methyl ester of L 659699, inhibits HMG-CoA synthase.</p>Formule :C19H30O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :338.44NLRP3-IN-7
<p>NLRP3-IN-7 (Compound 36) is a selective inhibitor of the NLRP3 inflammasome and is able to assemble the NLRP3 inflammasome.</p>Formule :C18H15ClN2O4S3Couleur et forme :SolidMasse moléculaire :454.97RK-582
CAS :<p>RK-582: oral spiroindolinone tankyrase inhibitor, halts colon cancer growth in COLO-320DM mouse model.</p>Formule :C27H35FN6O3Couleur et forme :SolidMasse moléculaire :510.6PD 134922
CAS :<p>PD 134922 is a HIV-1 protease inhibitors. Inactivation of the protease prevents infectious virion formation.</p>Formule :C37H61N5O7SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :719.97GSK3368715
CAS :<p>GSK3368715 is an orally active, reversible, and S-adenosyl-L-methionine (SAM) uncompetitive type I protein arginine methyltransferases (PRMTs) inhibitor (IC50s</p>Formule :C20H38N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :366.54K203
<p>K203 is a potent tabun-inhibited AChE reactivator and is an important antidote to organophosphorus poisoning.</p>Formule :C16H18Br2N4O2Couleur et forme :SolidMasse moléculaire :458.15GSK1820795A
CAS :<p>GSK1820795A: Telmisartan analog, selective hGPR132a antagonist, blocks yeast activation by N-acylamides, angiotensin II antagonist, partial PPARγ agonist.</p>Formule :C35H34N8Couleur et forme :SolidMasse moléculaire :566.7Anticancer agent 143
CAS :<p>Anticancer Agent 143 (Compound 369), a potent dual inhibitor targeting PTPN2 and PTP1B, exhibits IC50 values below 2.5 nM.</p>Formule :C19H15BrF2N3O6PS2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :594.34AChE-IN-24
<p>AChE-IN-24: Strong AChE blocker, crosses blood-brain barrier, IC50=0.053 μM, useful for AD research.</p>Formule :C22H30N2O4S2Couleur et forme :SolidMasse moléculaire :450.61SARS-CoV-2 nsp14-IN-1
<p>SARS-CoV-2 nsp14-IN-1 inhibits Nsp14 Mtase with an IC50 of 0.061 μM, affecting multiple substrates.</p>Formule :C20H20N6O5SCouleur et forme :SolidMasse moléculaire :456.48PCTR1
CAS :<p>PCTR1, derived from DHA, hastens inflammation resolution and boosts macrophage function, reducing PGE2, PGD2, and TXB2 in mice.</p>Formule :C32H47N3O9SCouleur et forme :SolidMasse moléculaire :649.8WS-898
<p>WS-898 boosts paclitaxel efficacy in resistant cells by inhibiting ABCB1; IC50: SW620/Ad300 - 5.0 nM, KB-C2 - 3.67 nM, HEK293/ABCB1 - 3.68 nM.</p>Formule :C33H25N7OSCouleur et forme :SolidMasse moléculaire :567.66P-gp modulator 1
CAS :<p>P-gp modulator 1 is a high affinity and orally available P-glycoprotein (Pgp) modulator</p>Formule :C41H72N2O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :689.02PPO-IN-1
<p>PPO-IN-1 is a potent inhibitor of protoporphyrinogen IX oxidase (PPO) (Ki: 2.5 nM).</p>Formule :C18H10F3N3O4SCouleur et forme :SolidMasse moléculaire :421.35GRPR antagonist-1
<p>GRPR antagonist-1 targets GRPR, kills specific cancer cells (e.g., PC3, Pan02, HGC-27), and promotes apoptosis by modulating Bcl-2 and Bax.</p>Formule :C29H33F3N4O4Couleur et forme :SolidMasse moléculaire :558.59MLKL-IN-6
<p>MLKL-IN-6 (compound P28) is a mixed lineage kinase inhibitor that specifically targets the Mixed Lineage Kinase domain-like (MLKL) protein.</p>Formule :C20H18N4O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :394.388-iso Prostaglandin F3α
CAS :<p>8-iso PGF3α is an isoprostane produced from the free-radical peroxidation of EPA.</p>Formule :C20H32O5Couleur et forme :SolidMasse moléculaire :352.47Tandutinib (MLN518) HCl
Tandutinib antagonizes FLT3, PDGFR, and c-Kit with an IC50 of ~200 nM.Formule :C31H43ClN6O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :599.16Elongation factor P-IN-2
<p>Elongation factor P-IN-2, a β-lysine derivative, is a potent EFP inhibitor reducing E. coli growth.</p>Formule :C16H35N3O2Couleur et forme :SolidMasse moléculaire :301.47RORγt inhibitor 2
CAS :<p>RORγt Inhibitor 2, a potent inhibitor of RORγt, exhibits an IC50 of 9.2 nM and is utilized in the study of cancer, inflammation, or autoimmune diseases that are</p>Formule :C31H33F5N2O7SCouleur et forme :SolidMasse moléculaire :672.66di-Val-L-dC
CAS :<p>Di-Val-L-dC, a reverse transcriptase inhibitor, is used potentially for treatment of HBV infection.</p>Formule :C19H31N5O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :425.48LY593093
CAS :<p>LY593093 is a selective partial orthosteric agonist of M1 muscarinic acetylcholine receptor.</p>Formule :C32H30FN3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :507.6Galectin-3-IN-2
<p>Galectin-3-IN-2 inhibits galactose lectin-3 (Gal-3) with an 8.3 μM IC50, impacting cancer-related metabolism.</p>Formule :C24H30FN3O10SCouleur et forme :SolidMasse moléculaire :571.57THR-β agonist 5
CAS :<p>THR-β agonist 5 (compound 54) is a potent THR-β agonist, with an EC 50 of <50 nM [1].</p>Formule :C22H23N5O2Couleur et forme :SolidMasse moléculaire :389.45QPX7728 methoxy acetoxy methy ester
CAS :<p>QPX7728 methoxy acetoxy methy ester is an inhibitor of boronic acid β-lactamase.</p>Formule :C14H14BFO7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :324.07PD-1/PD-L1-IN-30
CAS :<p>PD-1/PD-L1-IN-30: Cancer research inhibitor with 0.018 μM IC50.</p>Formule :C29H28F3NO5Couleur et forme :SolidMasse moléculaire :527.53DS34942424
<p>DS34942424 is an orally potent analgesic which did not exhibit mu opioid receptor agonist activity.</p>Formule :C15H17FN2OCouleur et forme :SolidMasse moléculaire :260.31KRAS G12C inhibitor 33
CAS :<p>KRAS G12C inhibitor 33 is a KRAS G12C inhibitor that can be used to study cancer.</p>Formule :C30H33N7O3Couleur et forme :SolidMasse moléculaire :539.63Intoplicine
CAS :<p>Intoplicine is an inhibitor of DNA topoisomerase I and II.</p>Formule :C21H24N4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :348.44Carbonic anhydrase inhibitor 8
<p>R-13, a carbonic anhydrase inhibitor, has Ki of 60.7 nM (hCA I), 320.7 nM (hCA II), and 2298 nM (hCA IV).</p>Formule :C20H25N3O4SCouleur et forme :SolidMasse moléculaire :403.5(R)-NVS-ZP7-4
CAS :<p>(R)-NVS-ZP7-4, an R-isomer, inhibits ZIP7 to study ER zinc impact & Notch pathway.</p>Formule :C28H28FN5OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :501.62CXCR4 antagonist 3
<p>CXCR4 antagonist 3, aka compound 12a, has 11 nM IC50, shares TIQ15 traits, and is promising in HIV research.</p>Formule :C22H31N5Couleur et forme :SolidMasse moléculaire :365.52EGFR-IN-47
<p>EGFR-IN-47: strong oral EGFRL858R/T790M/C797S blocker, induces cell death; promising for NSCLC research. IC50: 0.01 μM.</p>Formule :C29H35N7Couleur et forme :SolidMasse moléculaire :481.64(rel)-AR234960
CAS :(rel)-AR234960 is an active relative configuration of AR234960. AR234960 is a non-peptide agonist of MAS.Formule :C27H30FN5O5SCouleur et forme :SolidMasse moléculaire :555.63D-Cl-amidine hydrochloride
<p>D-Cl-amidine hydrochloride is a potent and highly selective inhibitor of PAD1. It exhibits excellent tolerance and does not induce significant toxicity [1].</p>Formule :C14H20Cl2N4O2Couleur et forme :SolidMasse moléculaire :347.24Antibacterial agent 112
<p>Compound 112: Powerful antibacterial, MIC 1250 μM against B. subtilis, E. coli, E. faecalis, S. typhimurium, S. aureus; also an HIV-1 antibody.</p>Formule :C35H23N5O5Couleur et forme :SolidMasse moléculaire :593.59Anticancer agent 78
<p>Anticancer agent 78: anti-aromatase (IC50=0.9 μM), cytotoxic, potential in breast cancer research.</p>Formule :C19H14BrNO4Couleur et forme :SolidMasse moléculaire :400.22Agarospirol
CAS :<p>Agarospirol has partial anti-inflammatory activity.</p>Formule :C15H26ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :222.37VEGFR-2-IN-17
<p>VEGFR-2-IN-17 (15a) is a potent VEGFR-2 inhibitor with an IC50 of 67.25 nM, showing significant antitumor effects.</p>Formule :C21H14ClN3O2Couleur et forme :SolidMasse moléculaire :375.81iMDK quarterhydrate
<p>iMDK quarterhydrate, PI3K inhibitor, blocks MDK growth; suppresses NSCLC safely with MEK inhibitor.</p>Formule :C21H15FN2O3SCouleur et forme :SolidMasse moléculaire :380.91CYP2C9/CYP2C19-IN-1
<p>CYP2C9/CYP2C19-IN-1 is a potent inhibitor of CYP2C9/CYP2C19 without liver toxicity or genotoxicity and can be used to study Zika virus (ZIKV) infection.</p>Formule :C27H28N2O6SCouleur et forme :SolidMasse moléculaire :508.59MAP855
CAS :<p>MAP855: potent, selective, oral MEK1/2 inhibitor; IC50=3 nM, pERKEC50=5 nM; effective on wild-type/mutant MEK1/2.</p>Formule :C28H23ClF2N6O3Couleur et forme :SolidMasse moléculaire :564.97UB 165
CAS :<p>Subtype-selective nicotinic agonist</p>Formule :C13H15ClN2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :234.72Cav 3.2 inhibitor 3
<p>Cav 3.2 inhibitor 3 is a potent inhibitor of the Cav3.2 T-type Ca2+channel (IC50: 0.1534 μM) and has a low binding affinity for D2 receptors.</p>Formule :C32H37N3O2Couleur et forme :SolidMasse moléculaire :495.66RmlA-IN-2
<p>RmlA-IN-2: Strong RmlA blocker, hinders l-rhamnose synthesis & alters bacterial wall permeability (IC50: 0.303 μM).</p>Formule :C22H26BrN5O4SCouleur et forme :SolidMasse moléculaire :536.44RdRP-IN-5
CAS :<p>RdRP-IN-5 (compound 20), a potent inhibitor of the influenza virus RNA-dependent RNA polymerase (RdRP), has potential application in influenza research [1].</p>Formule :C23H21N3O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :419.43Calphostin D
CAS :<p>Calphostins, PKC inhibitors from Cladosporium cladosporioides, include A, B, C, D, I; C is most potent.</p>Formule :C30H30O10Couleur et forme :SolidMasse moléculaire :550.55WQ3810
CAS :<p>WQ3810 is an orally active fluoroquinolone, has potent antibacterial activities.</p>Formule :C22H22F3N5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :461.4412(S)-HEPE
CAS :<p>12(S)-HEPE, made from EPA by 12-LO, is an anti-inflammatory ω-3 derivative affecting leukotriene formation.</p>Formule :C20H30O3Couleur et forme :SolidMasse moléculaire :318.45Antitumor agent-43
<p>Antitumor agent-43 (Compound 4B) is a potent antitumor agent that induces cell cycle arrest at G2/M phase.</p>Formule :C16H8N2O3Couleur et forme :SolidMasse moléculaire :276.25Casein Kinase II Inhibitor IV Hydrochloride
CAS :<p>Casein Kinase II Inhibitor IV HCl promotes keratinocyte differentiation, potential for skin disorder therapy.</p>Formule :C24H24ClN5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :465.93RWJ-445167
CAS :<p>RWJ-445167 is a thrombin and factor Xa dual inhibitor(Ki of 4.0 nM and 230 nM, respectively), with potent antithrombotic activity.</p>Formule :C18H24N6O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :436.49IL-17 modulator 1 disodium
CAS :<p>Potent, orally active IL-17 Modulator 1 (disodium) from patent WO 2020127685, used in psoriasis and arthritis research.</p>Formule :C28H37N6NaO6PCouleur et forme :SolidMasse moléculaire :607.604ZK-Thiazolidinone
CAS :<p>ZK-Thiazolidinone (TAL), ATP-competitive PLK1 inhibitor, disrupts cell division processes in vitro and in vivo, targeting human/mouse tumors.</p>Formule :C23H26F3N5O2SCouleur et forme :SolidMasse moléculaire :493.55CD73-IN-2
<p>CD73-IN-2 is a potent inhibitor of CD73 (IC50: 0.09 nM).</p>Formule :C17H25ClN5O7PCouleur et forme :SolidMasse moléculaire :477.84Teoprolol
CAS :<p>Teoprolol is a blocker of β-adrenergic receptor.</p>Formule :C23H30N6O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :454.52(RS)-AMPA
CAS :<p>(RS)-AMPA ((±)-AMPA) is a glutamate analog. (RS)-AMPA is an agonist of effective and selective excitatory neurotransmitter L-glutamic acid.</p>Formule :C7H10N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :186.17VU6028418
<p>VU6028418 is a highly selective, potent, orally active M4mAChR antagonist that acts on hM4 (IC50: 4.1 nM).</p>Couleur et forme :LiquidYKL-1-116
CAS :<p>YKL-1-116 is an effective, selective, and covalent CDK7 inhibitor.</p>Formule :C34H38N8O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :606.72Fosmanogepix
CAS :<p>Fosmanogepix (APX001) is a broad-spectrum oral antifungal that targets Gwt1 enzyme, transforming into active APX001A in the body.</p>Formule :C22H21N4O6PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :468.40J-104871
CAS :<p>J-104871 (UNII-6137X5QNJF) is an FTase inhibitor that inhibits tumor growth in nude mice transplanted with activated H-ras-transformed NIH3T3 cells.</p>Formule :C38H32N2O12Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :708.67Cacospongionolide B
CAS :<p>Cacospongionolide B from Fasciospongia cavernosa inhibits secretory phospholipase A2, curbing inflammation.</p>Formule :C25H36O4Couleur et forme :SolidMasse moléculaire :400.55
