Inhibiteurs
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.834 produits)
- Apoptose(6.315 produits)
- Cycle cellulaire/point de contrôle(4.877 produits)
- Chromatine/Épigénétique(2.613 produits)
- Signalisation du cytosquelette(1.568 produits)
- Altération de l'ADN/réparation de l'ADN(2.871 produits)
- Endocrinologie/Hormones(3.754 produits)
- Enzyme(3.672 produits)
- GPCR/G-Protéine(9.020 produits)
- Immunologie et Inflammation(3.905 produits)
- Virus de la grippe(300 produits)
- Signalisation JAK/STAT(415 produits)
- Signalisation MAPK(1.257 produits)
- Transporteur membranaire/Canal ionique(3.155 produits)
- Métabolisme(10.133 produits)
- Microbiologie/Virologie(7.620 produits)
- Neuroscience(10.473 produits)
- Autres inhibiteurs(35.846 produits)
- Oxydation-Réduction(40 produits)
- Signalisation PI3K/Akt/mTOR(1.429 produits)
- Protéases/Protéasome(1.689 produits)
- Cellules souche et Dérivés(732 produits)
- Tyrosine Kinase/Adaptateurs(1.982 produits)
- Ubiquitination(1.726 produits)
66515 produits trouvés pour "Inhibiteurs"
Dazostinag disodium
CAS :Dazostinag disodium (TAK-676) is a synthetic novel interferon gene (STING) agonist.Cost-effective and quality-assured.Formule :C21H20F2N8Na2O10P2S2Degré de pureté :98.84% - 99.96%Couleur et forme :SolidMasse moléculaire :754.48ELOVL1-IN-2
CAS :ELOVL1-IN-2 weakly inhibits ELOVL1 enzyme (IC50: 21 μM) and shows moderate potency in HEK293 cells (IC50: 6.7 μM).Formule :C18H15FN2ODegré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :294.32ZD 7155 hydrochloride
CAS :ZD 7155 hydrochloride is an angiotensin II receptor type 1 (AT1 receptor) antagonist.Formule :C26H27ClN6ODegré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :474.98Ref: TM-T13390
1mg42,00€5mg88,00€1mL*10mM (DMSO)90,00€10mg135,00€25mg235,00€50mg396,00€100mg635,00€200mg887,00€AKT Kinase Inhibitor
CAS :AKT Kinase Inhibitor is an Akt inhibitor with antitumor activity that selectively inhibits cell proliferation in a dose-dependent manner.Cost-effective and quality-assured.Formule :C16H19N7O3Degré de pureté :97.83% - 99.13%Couleur et forme :SolidMasse moléculaire :357.37Ref: TM-T10276
1mg129,00€5mg313,00€1mL*10mM (DMSO)341,00€10mg537,00€25mg840,00€50mg1.125,00€100mg1.521,00€BAY-3827
CAS :BAY-3827 is an AMPK inhibitor with antiproliferative activity and antitumor activity. BAY-3827 inhibits the phosphorylation of acetyl CoA carboxylase 1.Formule :C27H25FN6ODegré de pureté :99.90%Couleur et forme :SolidMasse moléculaire :468.53Ref: TM-T73350
1mg52,00€5mg113,00€1mL*10mM (DMSO)117,00€10mg177,00€25mg334,00€50mg560,00€100mg792,00€500mg1.575,00€Glycosyltransferase-IN-1
Glycosyltransferase-IN-1 is a glycosyltransferase inhibitor with bacteriostatic activity, inhibiting MSSA, MRSA, Bacillus subtilis, and Enterobacteriaceae.Formule :C19H21N5ODegré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :335.4Treprostinil diethanolamine
CAS :Treprostinil diethanolamine (UT-15C) is a potent agonist of EP2, DP1 and IP, with values of 3.6, 4.4, 32.1, 212, 826, 2505 and 4680 nM for EP2, DP1, IP, EP1,Formule :C27H45NO7Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :495.65HRO761
CAS :HRO761 is a potent Werne r syndrome RecQ DNA deconjugase (WRN) inhibitor that can be used to study cancers such as colon and stomach cancer.Formule :C31H31ClF3N9O5Degré de pureté :98.74% - 99.62%Couleur et forme :SolidMasse moléculaire :702.08Ref: TM-T72107
1mg57,00€5mg118,00€10mg167,00€25mg280,00€50mg475,00€100mg708,00€1mL*10mM (DMSO)778,00€EZM0414
CAS :EZM0414 is a potent, selective, orally bioavailable inhibitor of SETD2 with IC50 of 18 nM in SETD2 biochemical assay and IC50 of 34 nM in a cellular assay.Formule :C22H29FN4O2Degré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :400.49Zelasudil
CAS :Zelasudil (RXC007) is a Rho-related (ROCK) kinase inhibitor for the study of idiopathic pulmonary fibrosis and inflammation.Formule :C22H21F2N7ODegré de pureté :99.15%Couleur et forme :SolidMasse moléculaire :437.445Ref: TM-T69665
1mg92,00€5mg168,00€1mL*10mM (DMSO)170,00€10mg248,00€25mg421,00€50mg587,00€100mg820,00€GLPG0974
CAS :GLPG0974 is an antagonist of FFA2/GPR43 with IC50 of 9 nM.Formule :C25H25ClN2O4SDegré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :484.99KI696
CAS :KI696 is a high-affinity probe that potently inhibits the interaction of Keap1 and NRF2.Formule :C28H30N4O6SDegré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :550.63Ref: TM-T11758L
1mg137,00€5mg281,00€1mL*10mM (DMSO)341,00€10mg423,00€25mg707,00€50mg1.018,00€100mg1.468,00€200mg1.963,00€STK-15
CAS :STK-15 is a candidate for use as a fatty acid binding protein 5 (FABP5) inhibitor.Formule :C34H29NO5Degré de pureté :98.05%Couleur et forme :SolidMasse moléculaire :531.6Vofopitant
CAS :Vofopitant (GR 205171) is a potent NK1 receptor antagonist with anxiolytic and antiemetic activity for the study of post-traumatic stress disorder (PTSD).Formule :C21H23F3N6ODegré de pureté :97.86%Couleur et forme :SolidMasse moléculaire :432.44Cap-dependent endonuclease-IN-1
CAS :Cap-dependent endonuclease-IN-1: potent, oral inhibitor with antiviral properties against influenza.Formule :C27H22F2N2O6SDegré de pureté :99.53% - 99.61%Couleur et forme :SolidMasse moléculaire :540.54Dual FAAH/sEH-IN-1
CAS :Dual FAAH/sEH-IN-1 inhibits both sEH (IC50: 9.6 nM) and FAAH (IC50: 7 nM), offering potent anti-inflammatory effects.
Formule :C25H22ClN3O3S2Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :512.04NRX-252114
CAS :NRX-252114 promotes mutant β-catenin degradation, binding it to E3 ligase SCFβ-TrCP (EC50: 6.5 nM; Kd: 0.4 nM).Formule :C22H12Cl2F3N3O2SDegré de pureté :99.70%Couleur et forme :SolidMasse moléculaire :510.32Moiramide B
CAS :Moiramide B is an acetyl coenzyme A carboxylase inhibitor with antimicrobial activity, strongly inhibiting Gram-positive bacteria.Formule :C25H31N3O5Degré de pureté :98.53% - 99.90%Couleur et forme :SolidMasse moléculaire :453.53BQ-788
CAS :BQ-788 is an ETB receptor antagonist with potential hypertensive activity that inhibits exogenous ET-1-induced elevation of coronary perfusion pressure.Formule :C34H51N5O7Degré de pureté :98.81%Couleur et forme :SolidMasse moléculaire :641.8Ref: TM-T10595
1mg130,00€2mg178,00€5mg313,00€1mL*10mM (DMSO)341,00€10mg447,00€25mg713,00€50mg964,00€100mg1.305,00€500mg2.592,00€Elacytarabine
CAS :Elacytarabine (M7594 0037), a lipid-conjugated derivative of the nucleoside analog cytarabine, is an antineoplastic drug. It has cytotoxicity in solid tumors.Formule :C27H45N3O6Degré de pureté :97.69%Couleur et forme :SolidMasse moléculaire :507.66NDI-034858
CAS :NDI-034858 (TAK-279) is a tyrosine kinase 2 (TYK2) inhibitor (Kd<200 pM) that targets the JH2 structural domain of Tyk2 for the treatment of autoimmune diseasesFormule :C23H24N8O3Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :460.49Vecabrutinib
CAS :Vecabrutinib (SNS-062) is a potent and noncovalent BTK and ITK inhibitor (Kd: 0.3 nM and 2.2 nM, respectively). Vecabrutinib displays an IC50 of 24 nM for ITK.Formule :C22H24ClF4N7O2Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :529.92Ref: TM-T17220
1mg82,00€5mg177,00€1mL*10mM (DMSO)207,00€10mg289,00€25mg470,00€50mg623,00€100mg874,00€DRB18
CAS :DRB18 inhibits GLUT proteins, altering glucose metabolism and inducing cancer cell death by G1/S arrest and oxidative stress.Formule :C22H23ClN2O2Degré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :382.88Ref: TM-T22317
1mg89,00€5mg215,00€1mL*10mM (DMSO)236,00€10mg340,00€25mg687,00€50mg1.108,00€100mg1.485,00€500mg2.962,00€DN02
DN02: a potent, selective BRD8(1) bromodomain probe; Ki=32 nM; 30x more affine than BRD8(2).Formule :C22H24FN3O3Degré de pureté :98.22% - 99.74%Couleur et forme :SolidMasse moléculaire :397.44Tuvusertib
CAS :Tuvusertib (M1774), an oral ATR inhibitor (Ki<1µM), selectively blocks CHK1 phosphorylation, disrupts DNA repair, and induces tumor cell apoptosis.Formule :C16H12F2N8ODegré de pureté :98.44% - 99.66%Couleur et forme :SolidMasse moléculaire :370.32Ref: TM-T10406
1mg58,00€5mg124,00€1mL*10mM (DMSO)142,00€10mg187,00€25mg363,00€50mg505,00€100mg717,00€Enbezotinib
CAS :Enbezotinib is an inhibitor of RET autophosphorylation and can be used in cancer research.Formule :C21H21FN6O3Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :424.43Ref: TM-T62285
1mg77,00€5mg166,00€1mL*10mM (DMSO)182,00€10mg253,00€25mg414,00€50mg567,00€100mg745,00€SYM2206
CAS :SYM2206 is a low affinity non-competitive AMPA receptor antagonist with an IC50 value of 1.6 μM.SYM2206 exhibits anticancer activity by blocking Nav1.6-mediatedFormule :C20H22N4O3Degré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :366.41Milademetan
CAS :Milademetan (DS-3032), an MDM2 inhibitor, exhibits antitumor activity, induces G1 cell cycle arrest and apoptosis, and can be used to study solid tumors.Formule :C30H34Cl2FN5O4Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :618.53Ref: TM-T12040
1mg93,00€5mg167,00€1mL*10mM (DMSO)221,00€10mg260,00€25mg492,00€50mg802,00€100mg1.378,00€BE1218
CAS :BE1218 is a liver X receptor (LXR) inverse agonist active on LXRα and LXRβ with an IC50 of 9 nM and 7 nM, respectively.
Formule :C30H30FNO4S2Degré de pureté :99.7%Couleur et forme :SoildMasse moléculaire :551.69Zotizalkib
CAS :TPX-0131: potent, selective, CNS-ready, oral ALK inhibitor (WT IC50: 1.4nM, G1202R/L1196M IC50: 0.3nM) with robust antitumor effects.Formule :C21H20F3N5O3Degré de pureté :98.7%Couleur et forme :SolidMasse moléculaire :447.41Ref: TM-T9414
1mg114,00€5mg268,00€1mL*10mM (DMSO)303,00€10mg439,00€25mg879,00€50mg1.395,00€100mg1.873,00€BCL6-IN-3
CAS :BCL6-IN-3: potent BCL6 inhibitor, 70 nM GI50 in SU-DHL4, affects cell functions, antitumor.Formule :C24H31ClF2N6O2Degré de pureté :98.17%Couleur et forme :SolidMasse moléculaire :508.99Ref: TM-T10487
500mgÀ demander1mg109,00€5mg241,00€10mg355,00€1mL*10mM (DMSO)370,00€25mg532,00€50mg745,00€100mg1.018,00€BDZ-g
CAS :BDZ-g: potent, selective AMPA receptor antagonist; useful for researching neurological disorders.Formule :C21H21N5O2SDegré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :407.49BODIPY FL prazosin
CAS :BODIPY FL prazosin is an α1-adrenergic antagonist that inhibits α1a-AR and α1b-AR.
Formule :C28H32BF2N7O3Degré de pureté :97.27%Couleur et forme :SolidMasse moléculaire :563.41Aldometanib
CAS :Aldometanib (LXY-05-029) is an oral aldolase inhibitor that maintains metabolic balance by blocking FBP and activating lysosomal AMPK.Formule :C27H43Cl2IN2Degré de pureté :99.32% - 99.55%Couleur et forme :SolidMasse moléculaire :593.46JNJ-6204
CAS :JNJ-6204 is a deuterated compound that efficiently inhibits CSNK1D and CSNK1E.Formule :C19H11D6FN6ODegré de pureté :97.42% - 99.87%Couleur et forme :SolidMasse moléculaire :370.41Tigemonam
CAS :Tigemonam is a monobactam, a novel orally administered monobactam that protects against gram-negative aerobic bacterial pathogens. Cost-effective and quality-assured.Formule :C12H15N5O9S2Degré de pureté :97.71% - >99.99%Couleur et forme :SolidMasse moléculaire :437.41CP-642931
CAS :CP-642931 (Sorbitol dehydrogenase-IN-1) is a sorbitol dehydrogenase inhibitor used in the study of diabetes mellitus and cardiovascular disease.Formule :C17H25N7ODegré de pureté :99.67% - >99.99%Couleur et forme :SolidMasse moléculaire :343.43CCF0058981
CAS :CCF0058981: noncovalent inhibitor for SARS-CoV-2 & -1 proteases; IC50s: 68 nM (SC2) & 19 nM (SC1). Potential COVID-19 research use.
Formule :C24H19ClN6ODegré de pureté :98.94%Couleur et forme :SoildMasse moléculaire :442.9Ref: TM-T60095
500mgÀ demander1mg46,00€2mg60,00€5mg92,00€10mg160,00€25mg324,00€50mg449,00€100mg562,00€SB-224289 hydrochloride
CAS :SB-224289 hydrochloride (SB-224289A) is a selective antagonist of 5-HT1B receptor, with anxiolytic effect.Formule :C32H33ClN4O3Degré de pureté :98.99% - 99.96%Couleur et forme :SolidMasse moléculaire :557.08ALOX15-IN-2
CAS :ALOX15-IN-2: Potent ALOX15 inhibitor. IC50: 1.55 μM for LA; 2.79 μM for AA. Stops linoleic/arachidonic acid oxidation.Formule :C23H29N3O4SDegré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :443.56Ref: TM-T62606
1mg46,00€5mg90,00€1mL*10mM (DMSO)100,00€10mg160,00€25mg313,00€50mg537,00€100mg767,00€500mg1.558,00€AChE-IN-26
CAS :AChE-IN-26 (compound 4a) is an AChE (acetylcholinesterase) inhibitor (IC50: 0.42 μM).
Formule :C21H21BrN2O3Degré de pureté :99.24% - 99.85%Couleur et forme :SoildMasse moléculaire :429.31NRX-103095
CAS :NRX-103095 increases β-catenin binding to SCFβ-TrCP E3 ligase; EC50 is 163 nM for pSer33/Ser37 affinity boost.Formule :C22H16Cl2F3N3O3SDegré de pureté :99.85% - 99.95%Couleur et forme :SolidMasse moléculaire :530.35Ref: TM-T63730
1mg142,00€5mg344,00€1mL*10mM (DMSO)404,00€10mg557,00€25mg1.108,00€50mg1.783,00€100mg2.673,00€BAY-8400
BAY-8400 is an orally active, potent and selective DNA-dependent protein kinase ( DNA-PK ) inhibitor ( IC 50 =81 nM) which shows synergistic efficacy inFormule :C21H17F2N5ODegré de pureté :99.53%Couleur et forme :SolidMasse moléculaire :393.39Ref: TM-T9498
1mg80,00€5mg147,00€1mL*10mM (DMSO)161,00€10mg215,00€25mg439,00€50mg750,00€100mg1.009,00€XMD-17-51 Trifluoroacetate
CAS :XMD-17-51 Trifluoroacetate is a pyrimido-diazepinone compound that regulates protein kinases.Formule :C23H25F3N8O3Degré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :518.49Rineterkib
CAS :Rineterkib (ERK-IN-1) is an inhibitor of RAF and ERK1/2 activating mutations in the MAPK pathway.Formule :C26H27BrF3N5O2Degré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :578.42Ref: TM-T11224
1mg87,00€5mg170,00€1mL*10mM (DMSO)224,00€10mg318,00€25mg538,00€50mg765,00€100mg1.035,00€Gemcitabine elaidate hydrochloride
CAS :CP-4126, a lipophilic pro-drug of Gemcitabine, converts to active form by esterases, allowing oral administration with dose-dependent effects.
Formule :C27H44ClF2N3O5Degré de pureté :98.50% - 99.6%Couleur et forme :SolidMasse moléculaire :564.11CK2 inhibitor 2
CAS :CK2 Inhibitor 2, characterized as a potent, selective, and orally active inhibitor of CK2, demonstrates an impressive IC50 value of 0.66 nM.Formule :C21H17ClN4O2Degré de pureté :99.02%Couleur et forme :SolidMasse moléculaire :392.84Ref: TM-T35557
1mg62,00€5mg138,00€1mL*10mM (DMSO)152,00€10mg215,00€25mg425,00€50mg637,00€100mg853,00€200mg1.153,00€10-Methoxycamptothecin
CAS :10-Methoxycamptothecin is a natural bioactive derivative of camptothecin (CPT) isolated from Camptotheca acuminata and possesses high anti-cancer properties.Formule :C21H18N2O5Degré de pureté :98.36%Couleur et forme :SolidMasse moléculaire :378.38TGFβRI-IN-3
CAS :TGFβRI-IN-3 inhibits TGFβR1 with an IC 50 of 0.79 nM with 2000-fold selectivity against MAP4K4.Formule :C28H23N3O2SDegré de pureté :99.85%Couleur et forme :SoildMasse moléculaire :465.57Ref: TM-T9523
1mg84,00€5mg177,00€1mL*10mM (DMSO)177,00€10mg281,00€25mg552,00€50mg859,00€100mg1.234,00€500mg2.457,00€(E/Z)-GSK5182
CAS :GSK5182 is a racemic mix of (E/Z) isomers, a selective ERRγ inverse agonist (IC50: 79 nM), and induces ROS in liver cancer.Formule :C27H31NO3Degré de pureté :97.58%Couleur et forme :SolidMasse moléculaire :417.54Ref: TM-T7709
1mg77,00€5mg167,00€1mL*10mM (DMSO)177,00€10mg260,00€25mg477,00€50mg707,00€100mg1.063,00€LY3143921 hydrate
CAS :LY3143921 ((S)-Example 2) hydrate is an orally active CDC7 kinase inhibitor with broad in vitro anticancer activity [1].Formule :C16H14FN5O2Degré de pureté :98.43%Couleur et forme :SolidMasse moléculaire :327.31ARN19702
CAS :ARN19702: orally active, brain-penetrant, selective NAAA inhibitor, IC50 230 nM, broad analgesic profile.Formule :C21H22FN3O3S2Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :447.55Ref: TM-T9528
1mg52,00€5mg113,00€1mL*10mM (DMSO)124,00€10mg177,00€25mg350,00€50mg560,00€100mg880,00€200mg1.189,00€500mg1.765,00€Sinefungin
CAS :Sinefungin (Adenosyl-Ornithine) is an effective inhibitor of virion mRNA(guanine-7-)-methyltransferase, mRNA(nucleoside-2'-)-methyltransferase, and viralFormule :C15H23N7O5Degré de pureté :98% - 98.12%Couleur et forme :SolidMasse moléculaire :381.39BRD0639
CAS :BRD0639 is a first-in-class PRMT5-substrate interaction inhibitor for PBM-dependent PRMT5 activity studies.Formule :C21H22ClN5O4SDegré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :475.95SR 11302
CAS :SR 11302 is an inhibitor of activator protein-1 (AP-1).Formule :C26H32O2Degré de pureté :98.65%Couleur et forme :SolidMasse moléculaire :376.53Ref: TM-T23384
1mg93,00€5mg137,00€1mL*10mM (DMSO)150,00€10mg205,00€25mg356,00€50mg587,00€100mg888,00€JAK2-IN-7
CAS :JAK2-IN-7 selectively inhibits JAK2 (IC50: 3 nM), shows 14-fold selectivity over JAK1/3, FLT3, induces G0/G1 arrest, apoptosis, and has antitumor effects.Formule :C26H33N7ODegré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :459.59Ref: TM-T35900
1mg138,00€5mg334,00€1mL*10mM (DMSO)339,00€10mg597,00€25mg1.234,00€50mg1.648,00€100mg2.232,00€PD 151746
CAS :PD151746: calpain inhibitor, Ki μ-calpain=0.26μM, Ki m-calpain=5.33μM; reduces oxLDL cytotoxicity.Formule :C11H8FNO2SDegré de pureté :98.63% - ≥95%Couleur et forme :SolidMasse moléculaire :237.25Rolapitant hydrochloride
CAS :Rolapitant HCl is a potent NK1 antagonist, non-CYP3A4 interactive, with anti-emetic effects and a Ki of 0.66 nM.Formule :C25H27ClF6N2O2Degré de pureté :98.35% - 99.79%Couleur et forme :SolidMasse moléculaire :536.94Ref: TM-T3724
1mg153,00€5mg365,00€1mL*10mM (DMSO)439,00€10mg520,00€25mg780,00€50mg1.054,00€100mg1.425,00€200mg1.882,00€Durlobactam sodium salt
CAS :Durlobactam sodium salt (ETX2514) have an IC50 values of 4, 14 and 190 nM against class A KPC-2, class C AmpC and class D OXA-24.Cost-effective and quality-assured.Formule :C8H10N3NaO6SDegré de pureté :97.01% - 99.03%Couleur et forme :SolidMasse moléculaire :299.23FGI-106 tetrahydrochloride
CAS :FGI-106 tetrahydrochloride demonstrates potent inhibitory activity across a broad spectrum of viruses, including those causing hemorrhagic fevers such as EbolaFormule :C28H42Cl4N6Degré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :604.48Ref: TM-T11281L
1mg82,00€5mg161,00€1mL*10mM (DMSO)207,00€10mg245,00€25mg406,00€50mg572,00€100mg772,00€200mg1.035,00€INCB086550
CAS :INCB086550 (PD-1/PD-L1-IN-8) (example 24) is a PD-1/PD-L1 inhibitor, with an IC50 <= 10 nM.Formule :C41H39N7O4Degré de pureté :98.49%Couleur et forme :SolidMasse moléculaire :693.79Sebetralstat
CAS :Sebetralstat (KVD900) is an inhibitor of plasma kallikrein and can be used in studies about metabolic diseases.
Formule :C26H26FN5O4Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :491.51LSZ-102
CAS :LSZ-102 is an effective and selective degrader of estrogen receptor (IC50 = 0.2 nM) and can be used in studies about ERα positive breast cancer.Formule :C25H17F3O4SDegré de pureté :98.56%Couleur et forme :SolidMasse moléculaire :470.46FX-11
CAS :FX-11: potent LDHA inhibitor (Ki 8 μM), activates PKM2, reduces ATP, induces oxidative stress/ROS, cell death, shows antitumor effects.Formule :C22H22O4Degré de pureté :98.95% - 98.95%Couleur et forme :SolidMasse moléculaire :350.41Clorophene
CAS :Clorophene (Clorofene) is an antimicrobial agent and can be used in personal care products.Formule :C13H11ClODegré de pureté :99.87%Couleur et forme :White To Light Tan Or Pink Flakes Phenolic Odor (Ntp 1992)Masse moléculaire :218.68TEM1/CD248 Protein, Mouse, Recombinant (His)
TEM1/CD248 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with C-His tag. The predicted molecular weight is 73.6 kDa and the accession number is Q91V98.
Couleur et forme :SolidMasse moléculaire :73.6 kDa (predicted). Due to glycosylation, the protein migrates to 75-140 kDa based on Tris-Bis PAGE result.GAS6 Protein, Human, Recombinant (His)
GAS6 (Growth arrest-specific protein 6) is also known as AXL receptor tyrosine kinase ligand, AXLLG, is a multimodular protein that is up-regulated by a wide variety of cell types in response to growth arrest. Gas6 binds and induces signaling through the receptor tyrosine kinases Axl, Dtk, and Mer whose signaling is implicated in cell growth and survival, cell adhesion and cell migration. GAS6/AXL signaling plays a role in various processes such as endothelial cell survival during acidification by preventing apoptosis, optimal cytokine signaling during human natural killer cell development, hepatic regeneration, gonadotropin-releasing hormone neuron survival and migration, platelet activation, or regulation of thrombotic responses. GAS6 Protein, Human, Recombinant (His) is expressed in HEK293 cells.
Degré de pureté :＞99.90%Couleur et forme :SoildMasse moléculaire :72.7 KDa (Predicted), 80-90 KDa (Reducing conditions)TCblR Protein, Human, Recombinant (His)
TCblR Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with C-6xHis tag. The predicted molecular weight is 32-58 KDa and the accession number is Q9NPF0.
Couleur et forme :SolidMasse moléculaire :32-58 KDa (reducing condition)4-Ethoxycoumarin
CAS :4-Ethoxycoumarin has antimicrobial activity.
Formule :C11H10O3Degré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :190.23-Acetylcoumarin
CAS :3-Acetylcoumarin as a practical ligand for copper-catalyzed CN coupling reactions at room temperature. It has neuroprotective and acaricidal properties.
Formule :C11H8O3Degré de pureté :99.41%Couleur et forme :Yellow Crystalline PowderMasse moléculaire :188.182'-Hydroxy-4'-methylacetophenone
CAS :2'-Hydroxy-4'-methylacetophenone, a phenolic compound isolated from Angelicae koreana roots possesses acaricidal property. 2'-Hydroxy-4'-methylacetophenone has acaricidal activity, it could be used in the preparation of 4'-methyl-2'-[(p-tolylsulfonyl) oxy] acetophenone.
Formule :C9H10O2Degré de pureté :99.88%Couleur et forme :Black LiquidMasse moléculaire :150.17Relacorilant
CAS :Relacorilant is an oral glucocorticoid receptor antagonist with Ki of 7.2 nM, potential for treating Cushing's syndrome.
Formule :C27H22F4N6O3SDegré de pureté :98.53% - 99%Couleur et forme :SolidMasse moléculaire :586.56Ref: TM-T16727
Produit arrêtéPRGL493
CAS :PRGL493 blocks ACSL4, halts PC3/MDA-MB-231 cancer cell spread, and inhibits MA-10 tumor progesterone. Effective in mouse PC3 tumor model at 0.25 mg/kg.Formule :C25H21N7O2Degré de pureté :98.80% - 99.11%Couleur et forme :SolidMasse moléculaire :451.483-Methoxyphenylacetic acid
CAS :3-Methoxyphenylacetic acid belongs to the class of organic compounds known as anisoles. 3-Methoxyphenylacetic acid is slightly soluble (in water) and a weakly acidic compound (based on its pKa).3-Methoxyphenylacetic acid (m-Methoxyphenylacetic acid), a m-hydroxyphenylacetic acid (m-OHPAA) derivative, is a phytotoxin in Rhizoctonia solani. 3-Methoxyphenylacetic acid is used to develop a toxin-mediated bioassay for resistance to rhizoctonia root rot
Formule :C9H10O3Degré de pureté :98.61%Couleur et forme :White SolidMasse moléculaire :166.17α-Terpineol
CAS :Terpineol possesses antifungal activity against Trichophyton mentagrophytes, it also exhibits strong antimicrobial activity against periodontopathic and cariogenic bacteria. α-Terpineol (Terpineol) shows anticonvulsant, and anti-inflammatory activities, it inhibits the gene expression of the IL-6 receptor.
Formule :C10H18ODegré de pureté :97.55%Couleur et forme :Colorless LiquidMasse moléculaire :154.25Anisylacetone
CAS :Anisylacetone (Anisylacetone) is an effective lure for the male melon fly.
Formule :C11H14O2Degré de pureté :99.74%Couleur et forme :LiquidMasse moléculaire :178.23EGFR-IN-7
CAS :EGFR-IN-7 (TQB3804) is a selective and potent EGFR kinase inhibitor.
Formule :C32H41BrN9O2PDegré de pureté :95.32% - 99.64%Couleur et forme :SolidMasse moléculaire :694.6(-)-Isopulegol
CAS :Isopulegol has antioxidant, and neuroactive properties. It also has gastroprotective effects induced by isopulegol appear to be mediated, at least in part, by endogenous prostaglandins, K+ATP channel opening and antioxidant proprieties related to GSH increased.
Formule :C10H18ODegré de pureté :99.89%Couleur et forme :LiquidMasse moléculaire :154.25m-PEG12-Mal
m-PEG12-Mal is a PEG-based PROTAC linker that can be used in the synthesis of PROTACs[1].
Formule :C32H58N2O15Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :710.81Trk-IN-6
CAS :Trk-IN-6 shows excellent in vitro potency on a panel of TRK mutants ( IC 50 = 0.2-0.7 nM).
Formule :C21H21F3N6O2Couleur et forme :SolidMasse moléculaire :446.43TLQP-21 TFA
TLQP-21 TFA （TLQP-21 Trifluoroacetate） 是一种 VGF 衍生肽，可通过结合后折叠机制激活C3aR1 受体。
Degré de pureté :98%Lupinine hydrochloride
CAS :Lupinine hydrochloride is a bioactive chemical.
Formule :C10H20ClNOMasse moléculaire :205.73OVA Peptide 323-339
OVA Peptide (323-339) is an Ovalbumin epitope crucial for hypersensitivity in BALB/c mice.
Formule :C74H120N26O25Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1773.91A031
CAS :A031: PROTAC AR degrader, IC50 < 0.25 μM, inhibits prostate cancer growth in zebrafish.
Formule :C50H61ClN10O7SCouleur et forme :SolidMasse moléculaire :981.6Melarsonyl dipotassium
CAS :Melarsonyl dipotassium, also known as melarsonic acid dipotassium, is a potent anthelmintic agent with the ability to effectively inhibit parasites.
Formule :C13H13AsK2N6O4S2Couleur et forme :SolidMasse moléculaire :534.52PROTAC BTK Degrader-3
CAS :PROTAC BTK Degrader-3 is a potent degrader of Bruton's tyrosine kinase (BTK), exhibiting a DC50 (median degradation concentration) of 10.9 nM in Mino cells.
Formule :C41H40N10O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :752.82MRS2802
CAS :MRS2802 is a P2Y14 receptor agonist, its EC50 value for P2Y14 receptor is 63 nM.Formule :C10H14F2N2O11P2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :438.169HX103
CAS :HX103: Fluorogenic EGFR-TKI probe; inhibits various EGFR mutations; predicts NSCLC treatment response. IC50: 1.3-977 nM.
Formule :C26H25ClFN7O5SCouleur et forme :SolidMasse moléculaire :602.04gp91ds-tat
gp91ds-tat is a useful organic compound for research related to life sciences and the catalog number is T35393.
Degré de pureté :98%Couleur et forme :SolidCarbamic acid, N-(O,O-dimethylphosphorothioyl)-N-methyl-, m-isopropylphenyl ester
CAS :Carbamic acid, N-(O,O-dimethylphosphorothioyl)-N-methyl-, m-isopropylphenyl ester is a bioactive chemical.Formule :C13H20NO4PSCouleur et forme :SolidMasse moléculaire :317.34Compound N060-0121
Compound N060-0121 is a useful organic compound for research related to life sciences and the catalog number is T131219.
Couleur et forme :SolidCap-dependent endonuclease-IN-22
CAS :Cap-dependent endonuclease-IN-22 is a powerful inhibitor of cap-dependent endonuclease (CEN) [1].
Formule :C37H37ClF2N6O7S2Couleur et forme :SolidMasse moléculaire :815.31HDAC3/6-IN-2
CAS :HDAC3/6-IN-2 inhibits HDAC6/3 with IC50s 0.368/0.635 μM; promotes cancer cell apoptosis and histone acetylation.
Formule :C49H67N5O6Couleur et forme :SolidMasse moléculaire :822.09NE97220
CAS :NE97220 is a bioactive chemical.Formule :C7H12N2O6P2Couleur et forme :SolidMasse moléculaire :282.13Zelavespib hydrochloride
Zelavespib (PU-H71) hydrochloride is a potent inhibitor of Hsp90, exhibiting an IC50 value of 51 nM in MDA-MB-468 cells.Degré de pureté :98%Couleur et forme :Odour SolidContezolid acefosamil
CAS :Contezolid acefosamil (MRX-4), oral prodrug of Contezolid (MRX-I), treats multidrug-resistant Gram-positive bacteria, including MRSA.
Formule :C20H18F3N4O8PCouleur et forme :SolidMasse moléculaire :530.353Cgp 11130
CAS :Cgp 11130 is a bio-active chemical.Formule :C10H12FNO2Couleur et forme :SolidMasse moléculaire :197.21LH1306
CAS :LH1306 inhibits PD-1/PD-L1 interaction, IC50: 25 nM (HTRF assay); boosts Jurkat cell activation, EC50: 334-4,214 nM.
Formule :C38H48N6O6Couleur et forme :SolidMasse moléculaire :684.838AI 3-25755
CAS :AI 3-25755 is a biochemical.Formule :C11H15ClNO4PSCouleur et forme :SolidMasse moléculaire :323.733-Hydroxyephedrine
CAS :3-Hydroxyephedrine is a bioactive chemical.Formule :C10H15NO2Couleur et forme :SolidMasse moléculaire :181.23CAY10735
CAS :CAY10735: Anticancer agent; inhibits growth/migration in various cancer cells; reduces tumor in mouse models. IC50=0.674-11.56μM.
Formule :C44H60FN3O4Couleur et forme :SolidMasse moléculaire :713.979MCAAD-3
CAS :MCAAD-3, a near-infrared Aβ imaging probe, exhibits blood-brain barrier permeability and strong affinity for Aβ polymers (Ki >106 nM).
Formule :C17H18N2O2Couleur et forme :SolidMasse moléculaire :282.34Aflatoxin M1
CAS :Aflatoxin M1, a toxic metabolite of Aflatoxin B1, is produced by Aspergillus fungi, with a toxicity order: B1 > M1 > G1 > B2 > M2 > G2.
Formule :C17H12O7Couleur et forme :SolidMasse moléculaire :328.2762-AEMP TFA
CAS :2-AEMP TFA is a potent and rapidly acting antagonist of GABA(A)-ρ1 receptors. 2-AEMP is an analog of GABA.Formule :C3H10NO3PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :139.091Kbz probe 1
CAS :Kbz probe 1, an adaptable probe utilized for examining histone benzoylation and interactions within living cells, showcases extensive versatility.
Formule :C13H17ClF2N2O3Couleur et forme :SolidMasse moléculaire :322.73(±)5-HETE
CAS :(±)5-HETE is one of the six monohydroxy fatty acids produced by the non-enzymatic oxidation of arachidonic acid.
Formule :C20H32O3Couleur et forme :SolidMasse moléculaire :320.47Pyrromethene 597
CAS :Pyrromethene 597, a BODIPY laser dye, exhibits a wide tuning range of lasing wavelengths along with high photostability, and can serve as a thermal probe [1] [2Formule :C22H33BF2N2Couleur et forme :SolidMasse moléculaire :374.32Naphthol AS-BR
CAS :C.I. 37575 is a dye.Formule :C36H28N2O6Couleur et forme :SolidMasse moléculaire :584.62Antibacterial agent 83
CAS :Compound 17h is a potent antibacterial against VRE and MRSA, reduces MRSA biofilms, and is stable in liver microsomes.
Formule :C11H5Cl2N3O2Couleur et forme :SolidMasse moléculaire :282.08Thalidomide-PEG2-C2-NH2 TFA
CAS :Thalidomide-O-amido-PEG3-C2-NH2 TFA, a cereblon ligand-PEG linker for PROTAC, is synthesized.
Formule :C21H25F3N4O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :518.44Yhhu 3792
Activates Notch pathway, boosts NSC self-renewal and neurogenesis, enhances mice memory.
Couleur et forme :SolidRhizocticin A
CAS :Rhizocticin A is a potential inhibitor of threonine synthase.Formule :C11H22N5O6PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :351.3N2S2-CBMBC
CAS :N2S2-CBMBC, a bromo-benzyl ether, binds to 99mTc for PD-L1 tumor imaging, offering a real-time alternative to immunohistochemistry.
Formule :C34H33BrClN3O3S2Couleur et forme :SolidMasse moléculaire :711.131-(2,3-Dichlorphenyl)-piperazine
CAS :1-(2,3-Dichlorphenyl)-piperazine (DCPP) is a potent DHCR7 inhibitor. DHCR7 is the last enzyme in cholesterol biosynthesis.Formule :C10H12Cl2N2Degré de pureté :98%Couleur et forme :Brown OilMasse moléculaire :231.12Xibornol
CAS :Xibornol (Nanbacine) 具有广谱的抗菌和抗病毒活性，可用于研究革兰氏阳性菌感染和人呼吸道合胞病毒与人冠状病毒229E感染。Formule :C18H26OCouleur et forme :SolidMasse moléculaire :258.41-Oleoyl Lysophosphatidic Acid
CAS :1-Oleoyl Lysophosphatidic Acid (1-Oleoyl LPA) is a biologically active phospholipid that can be used to study cancer and atherosclerosis.
Formule :C21H41O7PCouleur et forme :SolidMasse moléculaire :436.52Mitoquinone-cyclodextrin
CAS :Mitoquinone-cyclodextrin is a mitochondria-targeted, 1:1 mix of Mitoquinone mesylate and cyclodextrin, aiming to combat oxidative damage.
Formule :C80H117O42PSCouleur et forme :SolidMasse moléculaire :1813.81PROTAC BRD4 Degrader-6
CAS :Compound 32a: PROTAC BRD4 Degrader-6, IC50 = 2.7 nM, degrades BRD4, halts BxPC3 pancreatic cancer cell growth, induces apoptosis for research.
Formule :C43H40F2N10O10SCouleur et forme :SolidMasse moléculaire :926.9Spiratisanin A
CAS :Spiratisanin A is a natural product from Spiraea japonica.
Formule :C29H40O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :436.63LCMV gp33-41 (TFA) (151705-84-9 free base)
LCMV gp33-41 (TFA) is an 11-aa peptide, MHC class I H-2Db-bound, presented to CTLs.Formule :C50H74N11F3015SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1158.24PROTAC VEGFR-2 degrader-2
CAS :PROTAC VEGFR-2 degrader-2 has minimal VEGFR-2 inhibition (IC50 > 1μM) and low anti-proliferative effect on EA.hy926 cells (IC50 > 100μM).
Formule :C50H56FN9O6SCouleur et forme :SolidMasse moléculaire :930.1Patent Blue V
CAS :Patent Blue V (Acid blue 1), a biological dye, serves as an intraocular stain in retinectomy—surgical removal of the inner limiting membrane (ILM).Formule :C27H31N2NaO6S2Couleur et forme :SolidMasse moléculaire :566.67Azido-PEG12-t-butyl ester
CAS :Azido-PEG12-t-butyl ester, a soluble PEG with azide/reactive t-butyl, forms triazoles via Click Chemistry; deprotectable in acid.
Formule :C31H62N3O14Couleur et forme :SolidMasse moléculaire :700.84AT-1002 TFA
AT-1002 TFA, a 6-mer synthetic peptide, functions as a tight junction regulator and absorption enhancer.
Formule :C34H54F3N9O9SCouleur et forme :SolidMasse moléculaire :821.91N-Deacetyllapaconitine
N-Deacetyllapaconitine is a useful organic compound for research related to life sciences and the catalog number is T131546.
Formule :C30H42N2O7Couleur et forme :SolidMasse moléculaire :542.6733'-O-Angeloylhamaudol
3'-O-Angeloylhamaudol is a useful organic compound for research related to life sciences and the catalog number is T124112.
Formule :C20H22O6Couleur et forme :SolidMasse moléculaire :358.39HJM-561
CAS :HJM-561 is a potent and selective EGFR PROTAC with oral bioavailability, capable of overcoming osimertinib-resistant EGFR triple mutations and demonstrating
Formule :C45H51ClN9O5PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :864.37Stibosamine
CAS :Stibosamine is a bioactive chemical.Formule :C10H19N2O3SbCouleur et forme :SolidMasse moléculaire :337.033Neuraminic acid
CAS :Neuraminic acid: acidic amino sugar, 9 carbon chain, from pyruvic acid + D-mannosamine, in active mucoproteins.Formule :C9H17NO8Couleur et forme :SolidMasse moléculaire :267.23PEG2-bis(phosphonic acid)
CAS :PEG2-bis(phosphonic acid) is a PEG Linker.Formule :C6H16O8P2Couleur et forme :SolidMasse moléculaire :278.13Propiram fumarate HCl
CAS :Propiram fumarate HClis an orally available Opioid receptors agonist with analgesic activity for the study of musculoskeletal pain.
Formule :C16H25N3O·xClHDegré de pureté :99.25%Couleur et forme :SoildPROTAC MDM2 Degrader-4
CAS :PROTAC MDM2 Degrader-4 targets MDM2 for degradation with E3 ligase via a linked inhibitor.
Formule :C70H74Cl4N8O14Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1393.19Pomalidomide-amido-PEG3-C2-NH2
CAS :Cereblon Ligand-Linker 22: A pomalidomide-based E3 ligase conjugate with a PEG3 linker for PROTACs.
Formule :C22H28N4O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :476.48Ephedrine levulinate
CAS :Ephedrine levulinate: alkaloid, stimulates alpha/beta-adrenergic receptors, boosts norepinephrine release.
Formule :C15H21NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :263.337Diacetoxyscirpenol
CAS :Diacetoxyscirpenol: a fungal mycotoxin causing blood disorders in humans/animals.
Formule :C19H26O7Degré de pureté :98%Couleur et forme :Solid SolidMasse moléculaire :366.41Araliadiol
CAS :Araliadiol is a polyacetylenic compound isolated from the leaves of Aralia cordata Thunb. Araliadiol inhibits MCF-7 cell growth (IC50: 6.41 μg/mL).Formule :C15H20O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :232.32(3,4-Dihydroxy-5-methoxybenzoyl)taraxerol
CAS :(3,4-Dihydroxy-5-methoxybenzoyl)taraxerol is a natural products from plants
Formule :C38H56O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :592.85STING agonist-9
CAS :STING agonist-9 (Compound 45): potent, EC50 1.2 nM h-STING, 32.82 μM m-STING; antitumor [1].
Formule :C39H47N13O6SCouleur et forme :SolidMasse moléculaire :825.94Phenol, m-(2-(methylamino)ethyl)-, hydrochloride
CAS :Phenol, m-(2-(methylamino)ethyl)-, hydrochloride is a biaoctive chemical.Formule :C9H14ClNOCouleur et forme :SolidMasse moléculaire :187.67Apratoxin A
CAS :Apratoxin A is a potent cytotoxin isolated from the marine cyanobacterium Lyngbya majuscula Harvey ex Gomont.Formule :C45H69N5O8SCouleur et forme :SolidMasse moléculaire :840.13Mouse IgG3 κ, Isotype Control
Mouse IgG3 kappa Isotype Control is a monoclonal antibody serving as an isotype control specifically for mouse IgG3κ antibodies.
Couleur et forme :Odour Liquid(5R)-Platyphyllone
CAS :(5R)-Platyphyllone has a wide range of applications in life science related research.
Formule :C19H22O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :314.381MitoPY1
CAS :a fluorescent probe for imaging hydrogen peroxide (H2O2) in mitochondria of living cellsFormule :C52H53BN2O5PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :827.77H-L-Photo-lysine hydrochloride
H-L-Photo-lysine HCl is a diazirine lysine for site-specific protein incorporation and in vivo cross-linking.Formule :C11H21ClN4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :308.76BD-9136
BD-9136, a highly selective BRD4 degrader, demonstrates the capability to inhibit tumor growth without inducing adverse effects in mice, showing potential forFormule :C44H44N10O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :824.95SIAIS117
CAS :SIAIS117: A Brigatinib-VHL-1 ALK PROTAC; degrades ALK G1202R, inhibits SR/H2228 cells, may fight small cell lung cancer.
Formule :C57H76ClN10O7PSCouleur et forme :SolidMasse moléculaire :1111.77Questiomycin A derivatives 12
Questiomycin A derivatives 12 is a Questiomycin A derivative.
Formule :C16H14N2O3Degré de pureté :99.79%Couleur et forme :SoildMasse moléculaire :282.29Antiviral agent 8
CAS :Antiviral agent 8, surpassing lead compounds crocin-1 and crocin-2, has been identified as a potent and promising candidate with enhanced antiviral activities.
Formule :C36H38F2O4Couleur et forme :SolidMasse moléculaire :572.693FGFR-IN-1
CAS :FGFR-IN-1 targets FGFR1-3 with IC50 <100 nM. (US20130338134A1, ex 219)
Formule :C26H24F2N4O6SCouleur et forme :SolidMasse moléculaire :558.55Phototherapeutic agent-1
CAS :Phototherapeutic agent-1: a light-activated, ROS-generating cancer cell killer with aggregation-induced emission.
Formule :C39H33F6N2O2PS3Couleur et forme :SolidMasse moléculaire :802.85Elamipretide acetate
Elamipretide acetate (MTP 131), a small tetrapeptide, targets mitochondria to reduce toxic species and stabilize cardiolipin.
Formule :C34H53N9O7Degré de pureté :99.76%Couleur et forme :SoildMasse moléculaire :699.84RB-OPD
CAS :RB-OPD, aka NO-red, is a fluorescent NO sensor with OPD & rhodamine, excitation at 550 nm & emission at 590 nm, highly sensitive & selective.Formule :C34H36N4O2Couleur et forme :SolidMasse moléculaire :532.688SHP2 protein degrader-1
CAS :SHP2 degrader-1: highly efficient, induces SHP2 degradation & cell apoptosis, shows promise in SHP2-related disease research.
Formule :C42H51Cl2N11O8Couleur et forme :SolidMasse moléculaire :908.84Compound TCFN97859
CAS :Compound TCFN97859 is a useful organic compound for research related to life sciences. The catalog number is T131721 and the CAS number is 103476-99-9.Formule :C19H24O9Couleur et forme :SoildMasse moléculaire :396.392MCA17-1
CAS :MCA17-1 exhibits superior bioactivity compared to the positive control, obeticholic acid (OCA), in the treatment of liver fibrosis.
Formule :C14H15NO5Couleur et forme :SolidMasse moléculaire :277.276BPH-629
CAS :BPH-629 is a bioactive chemical.Formule :C20H18O8P2Couleur et forme :SolidMasse moléculaire :448.3Gd-NMC-3
CAS :Gd-NMC-3, a bimodal imaging probe, exhibits high resolution and sensitivity for tumor imaging with favorable biocompatibility, demonstrating significant
Formule :C77H114Gd2N14O24S2Couleur et forme :SolidMasse moléculaire :1998.44PROTAC ER Degrader-10
CAS :Potent PROTAC ER Degrader-10 for cancer research; from patent WO2021133886, example 36.
Formule :C44H45N5O6Couleur et forme :SolidMasse moléculaire :739.86Dabigatran Acyl-β-D-Glucuronide
CAS :Dabigatran acyl-β-D-glucuronide is a major active metabolite of the thrombin inhibitor dabigatran .Formule :C31H33N7O9Couleur et forme :SolidMasse moléculaire :647.6455-Hydroxydopamine hydrochloride
CAS :5-Hydroxydopamine, a natural amine in urine, targets Luxaphone receptor (IC50: 22 µM); may have antimicrobial & anticancer properties.Formule :C8H12ClNO3Degré de pureté :99.56%Couleur et forme :Off-White To Beige To Grey-Brown PowderMasse moléculaire :205.64Yimitasvir
CAS :Yimitasvir, an oral NS5A inhibitor, treats chronic hepatitis C. Used for research.
Formule :C49H58N8O6Couleur et forme :SolidMasse moléculaire :855.03PROTAC MDM2 Degrader-2
CAS :PROTAC MDM2 Degrader-2: A potent MDM2-targeting compound with PROTAC tech for E3 ligase-mediated degradation.
Formule :C70H76Cl4N10O12Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1391.22Lichenase
CAS :Lichenase, an enzyme, breaks down β-glucans in grains into GOS, aiding polysaccharide degradation in cell walls.Couleur et forme :SolidCAY10736
CAS :CAY10736: Anticancer agent, blocks cell growth & migration in various cancers, effective in mouse models.
Formule :C41H59N3O3SCouleur et forme :SoildMasse moléculaire :673.99PLK1-IN-6
PLK1-IN-6: potent, selective PLK1 inhibitor, IC50 = 0.45 nM, hinders cancer cell growth.
Formule :C28H37N9O3Couleur et forme :SolidMasse moléculaire :547.65LY 280748
CAS :LY 280748 is a bio-active chemical.Formule :C23H29N4NaO2Couleur et forme :SolidMasse moléculaire :416.492',3'-cGAMP-C2-SH
CAS :2', 3'-cGAMP-C2-SH is a ADC cytotoxin.
Formule :C22H28N10O12P2SCouleur et forme :SolidMasse moléculaire :718.53Thalidomide-C2-amido-C2-COOH
CAS :Thalidomide-C2-amido-C2-COOH is a compound that includes a CRBN ligand for the E3 ubiquitin ligase, as well as a linker.
Formule :C19H20N4O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :416.38Fungicide5
CAS :Fungicide5 is a fungicide candidate targeting succinate dehydrogenase ( K i = 0.095 μM).
Formule :C20H13F8N3O2Couleur et forme :SolidMasse moléculaire :479.33CRTh2 antagonist 3
CAS :CRTh2 antagonist 3, a potent molecule, activates PDK1 (EC50=2μM, Kd=8.4μM) and may cause cardiovascular inflammation.Formule :C19H20N2O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :356.44Zanamivir-Cholesterol Conjugate
CAS :Zanamivir-cholesterol conjugate is an extended-duration neuraminidase inhibitor highly effective against drug-resistant influenza strains.
Formule :C61H104N8O15Couleur et forme :SolidMasse moléculaire :1189.544Podoblastin A (D-mannitol)
Podoblastin A (D-mannitol) is a useful organic compound for research related to life sciences and the catalog number is TSP-41077145.
Formule :C20H34O4Masse moléculaire :338.49BPH-830
CAS :BPH-830 is a bioactive chemical.Formule :C17H20NO5PCouleur et forme :SolidMasse moléculaire :349.32ER degrader 2
CAS :ER degrader 2: Potent estrogen receptor disruptor; key for cancer research.
Formule :C34H42F3N5O3Couleur et forme :SolidMasse moléculaire :625.72A 53868A
CAS :A 53868A is an antibiotic, it is isolated from Streptomyces luridus.Formule :C11H22N3O5PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :307.287m-PEG11-Tos
m-PEG11-Tos is a PEG-based PROTAC linker that can be used in the synthesis of PROTACs[1].
Formule :C28H50O13SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :626.75Mitoquinone
CAS :Mitoquinone is a TPP-based, mitochondrially targeted antioxidant .
Formule :C37H44O4PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :583.72Anticancer agent 11
CAS :Anticancer agent 11 suppresses angiogenesis and induces DNA cross-links for broad-spectrum efficacy.
Formule :C20H21N3O2Couleur et forme :SolidMasse moléculaire :335.40PROTAC PARP/EGFR ligand 1
CAS :PROTAC PARP/EGFR ligand 1 enables dual PARP EGFR degrader synthesis via PROTAC.
Formule :C53H56ClF2N9O8Couleur et forme :SolidMasse moléculaire :1020.52PROTAC BRD4 Degrader-16
CAS :PROTAC BRD4 Degrader-16 is a potent degrader of BRD4, exhibiting IC50 values of 34.58 nM for BRD4 (BD1) and 40.23 nM for BRD4 (BD2).
Formule :C46H41N7O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :819.86(D)-PPA 1
CAS :PD-1/PD-L1 binder, Kd 0.51 μM; blocks interaction in flow cytometry at 1 mg/mL; inhibits tumors, extends mouse survival.
Formule :C70H98N20O21Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1555.67PROTAC MDM2 Degrader-3
CAS :PROTAC MDM2 Degrader-3 uses PROTAC tech to efficiently break down MDM2 with a potent inhibitor and E3 ligase ligand.
Formule :C72H78Cl4N8O15Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1437.25Carbostyril 124
CAS :Carbostyril 124 is a useful organic compound for research related to life sciences. The catalog number is T65062 and the CAS number is 19840-99-4.Formule :C10H10N2OCouleur et forme :SolidMasse moléculaire :174.203Coumberone
CAS :Coumberone, a fluorogenic probe, is reduced by AKR1C family to fluorescent coumberol; vital for AKR1C research.Formule :C22H19NO3Couleur et forme :SolidMasse moléculaire :345.398AS-604850
AS-604850: PI3Kγ inhibitor, ATP-competitive, IC50=2.5μM, 30x> PI3Kδ/β, 18x> PI3Kα.
Formule :C11H5F2NO4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :285.227-(Diethylamino)-4-methyl-2H-chromen-2-one
CAS :7-(Diethylamino)-4-methyl-2H-chromen-2-one is a useful organic compound for research related to life sciences.Formule :C14H17NO2Couleur et forme :SolidMasse moléculaire :231.30Antibacterial agent 30
CAS :Antibacterial agent 30 exhibits remarkable in vitro activity against Xoo, as evidenced by its EC50 value of 1.9 μg/mL.
Formule :C24H24F3NO5Couleur et forme :SolidMasse moléculaire :463.45m-PEG1-acid
CAS :M-PEG1-acid, a soluble PEG derivative, has a terminal carboxylic acid for forming amide bonds with primary amines using activators like EDC, DCC.
Formule :C4H8O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :104.10Cytochrome P450 2C9
CAS :Cytochrome P450 2C9 metabolizes acidic drugs, including NSAIDs, anticoagulants, and diuretics.Formule :C37H40FeN5O7SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :754.666-[2-[4-(Ethylsulfonyl)phenyl]-1-methylethenyl]-1,2,3,4-tetrahydro-1,1,4,4-tetramethylnaphthalene
CAS :Degré de pureté :98%Phenarsone sulfoxylate
CAS :Phenarsone sulfoxylate is a biochemical.Formule :C7H8AsNNa2O6SCouleur et forme :SolidMasse moléculaire :355.11Pulcherriminic acid
CAS :Pulcherriminic acid, a cyclic dipeptide, chelates Fe3+, forms pulcherrimin, and has antimicrobial properties used in food, agriculture, and medicine.Formule :C12H20N2O4Couleur et forme :SolidMasse moléculaire :256.30Mca-Ala-Pro-Lys(Dnp)-OH
CAS :Mca-Ala-Pro-Lys(Dnp)-OH, a specific quenched fluorogenic substrate for ACE2, enables the detection of ACE2 activity in various tissues including urinary, heart
Formule :C32H36N6O12Couleur et forme :SolidMasse moléculaire :696.67L-Histidinyl-D-penicillaminatocobalt(III)
CAS :L-Histidinyl-D-penicillaminatocobalt(III) can provide a model for the binding of D-penicillamine to metal ions.Formule :C11H15CoN4O5SCouleur et forme :SolidMasse moléculaire :374.26TAK-448
CAS :TAK-448 (MVT-602), a potent KISS1R agonist, IC50: 460 pM, EC50: 632 pM, trialed for Prostate Cancer and Hypogonadism.Formule :C58H80N16O14Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1225.36Praluzatamab ravtansine
CAS :Sirtratumab vedotin (ASG15-ME) is an antibody-drug conjugate (ADC) that links a SLITRK6-specific human gamma 2 antibody (Igγ2) to the microtubule disruption agent monomethyl auristatin E (MMAE) through a protease-cleavable linker [1].
Degré de pureté :99.40%Couleur et forme :SoildHA-CD44 interaction inhibitor 1
Antitumor agent-109 (compound 6) is a dual-function inhibitor that targets hyaluronic acid and CD44, which are involved in tumor progression and invasion.
Couleur et forme :Odour Solid
