Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.519 produits)
- Apoptose(5.787 produits)
- Cycle cellulaire/point de contrôle(4.446 produits)
- Chromatine/Épigénétique(2.235 produits)
- Signalisation du cytosquelette(1.381 produits)
- Altération de l'ADN/réparation de l'ADN(2.824 produits)
- Endocrinologie/Hormones(3.500 produits)
- Enzyme(3.639 produits)
- GPCR/G-Protéine(8.317 produits)
- Immunologie et Inflammation(3.516 produits)
- Virus de la grippe(296 produits)
- Signalisation JAK/STAT(404 produits)
- Signalisation MAPK(1.200 produits)
- Transporteur membranaire/Canal ionique(2.787 produits)
- Métabolisme(9.416 produits)
- Microbiologie/Virologie(6.968 produits)
- Neuroscience(9.919 produits)
- Autres inhibiteurs(37.928 produits)
- Oxydation-Réduction(41 produits)
- Signalisation PI3K/Akt/mTOR(1.400 produits)
- Protéases/Protéasome(1.596 produits)
- Cellules souche et Dérivés(831 produits)
- Tyrosine Kinase/Adaptateurs(2.015 produits)
- Ubiquitination(1.649 produits)
Affichez 16 plus de sous-catégories
66626 produits trouvés pour "Inhibiteurs"
Trier par
Degré de pureté (%)
0
100
|
0
|
50
|
90
|
95
|
100
Myxothiazol
CAS :<p>Myxothiazol blocks mitochondrial complex III and triggers SESN2, a gene important for stress response.</p>Formule :C25H33N3O3S2Couleur et forme :SolidMasse moléculaire :487.68Anti-inflammatory agent 6
<p>Anti-inflammatory agent 6 blocks IKKα/β, IκBα, and NF-κB p65 phosphorylation, key to controlling inflammation.</p>Formule :C22H20O12Couleur et forme :SolidMasse moléculaire :476.39Scytonemin
CAS :<p>Scytonemin, a cyanobacterial pigment, inhibits cancer cell growth by decreasing Plk1 activity, especially effective on U266 myeloma cells.</p>Formule :C36H20N2O4Couleur et forme :SolidMasse moléculaire :544.55DNA crosslinker 2 dihydrochloride
CAS :<p>Potent DNA crosslinker 2 binds minor groove, increases Tm by 1.2°C, and inhibits NCI-H460, A2780, MCF-7 cancer cells.</p>Formule :C15H22Cl2N8OCouleur et forme :SolidMasse moléculaire :401.29Carbonic anhydrase inhibitor 10
<p>CA inhibitor 10 targets MCF-7 cells, IC50: 11.9 μM; potent h CA IX inhibitor, Ki: 6.2 nM. Anti-cancer research.</p>Formule :C14H17N5O3SCouleur et forme :SolidMasse moléculaire :335.38CHK1-IN-4
CAS :<p>CHK1-IN-4 is a potent inhibitor of checkpoint kinase 1 (chk1) and potently inhibits chk1 phosphorylation in the tumor cells with anti-tumor activity.</p>Formule :C18H18BrN7O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :444.29Antibacterial agent 69
<p>Antibacterial agent 69 is a novel structural antimicrobial modulator that can be used against lethal multidrug-resistant bacterial infections (MIC: 2.978 μM).</p>Formule :C24H19N3O4SCouleur et forme :SolidMasse moléculaire :445.49LRRK2-IN-4
CAS :<p>LRRK2-IN-4: Potent, selective LRRK2 inhibitor, oral, BBB-penetrating, IC50=2.6 nM, potential for Parkinson's.</p>Formule :C25H29ClF2N6O2Couleur et forme :SolidMasse moléculaire :518.99α-Glucosidase-IN-18
<p>α-Glucosidase-IN-18 (7B) is an orally active inhibitor of α-glucosidase, displaying an IC 50 value of 3.96 μM.</p>Formule :C23H19NO2SCouleur et forme :SolidMasse moléculaire :373.47HIV-1 inhibitor-41
<p>HIV-1 inhibitor-41 (B23): Oral non-nucleoside reverse transcriptase blocker, EC50 of 50 nM (E138K), 20.8 nM (WT), low hERG/CYP impact, non-toxic.</p>Formule :C16H15F2N3OSCouleur et forme :SolidMasse moléculaire :335.37HDAC/HSP90-IN-4
<p>HDAC/HSP90-IN-4 inhibits HDAC (20 IC50=194nM, 26 IC50=360nM) & HSP90α (20 IC50=153nM, 26 IC50=77nM), affects cancer cell survival and invasion.</p>Formule :C20H23N3O6Couleur et forme :SolidMasse moléculaire :401.15869BTK-IN-16
CAS :<p>BTK-IN-16 is a potential inhibitor of wild-type BTK and C481S mutants.BTK-IN-16 can be used to study various autoimmune diseases and cancers caused by BTK.</p>Formule :C15H14N4O2Degré de pureté :99.04%Couleur et forme :SoildMasse moléculaire :282.3WAY-855
CAS :<p>WAY-855 is an EAAT2-preferring, nonsubstrate inhibitor of high-affinity glutamate uptake.</p>Formule :C9H11NO4Couleur et forme :SolidMasse moléculaire :197.19HDAC-IN-9
<p>HDAC-IN-9, a dual tubulin/HDAC inhibitor, impedes A549 cell invasion/migration and shows strong anti-tumor/angiogenic effects.</p>Formule :C33H38N2O4Couleur et forme :SolidMasse moléculaire :526.67BTK-IN-10
CAS :<p>BTK-IN-10 is a potent inhibitor of BTK, acting on wild-type BTK (IC50<5 nM) or mutant BTK (C481S) (IC50<5 nM).</p>Formule :C25H24F2N4O2Couleur et forme :SolidMasse moléculaire :450.48ODN 2088
CAS :<p>ODN 2088 is a potent inhibitor of TLR3, TLR7 and TLR9 that is non-cytotoxic and shows inhibition of the release of IFN-α and IL-6.</p>Couleur et forme :Solidα-Glucosidase-IN-19
<p>Alpha-Glucosidase-IN-19 (Compound 6B) is an orally active alpha-glucosidase inhibitor (IC50: 3.63 μM) with antidiabetic effects.</p>Formule :C31H25NOSCouleur et forme :SolidMasse moléculaire :459.6Antibacterial synergist 1
<p>Compound 20P is a potent antibacterial, inhibits biofilms with IC50 4.5 μM, and reduces pyocyanin at IC50 8.6 μM.</p>Formule :C19H24N2O4Couleur et forme :SolidMasse moléculaire :344.4DX-9065A HCl hydrate
CAS :<p>DX-9065a: Competitive fXa/prothrombinase inhibitor; blocks proinflammatory events; Ki ~10-20 nM.</p>Formule :C26H39ClN4O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :571.06(R)-ONO-2952
<p>(R)-ONO-2952 is the R-enantiomer of ONO-2952. ONO-2952 is selective and oral effective TSPO antagonist, with Kis of 0.330-9.30 nM inhibiting rat and human TSPO.</p>Formule :C22H20ClFN2O2Couleur et forme :SolidMasse moléculaire :398.86Laulimalide
CAS :<p>Microtubule stabilizer; halts cancer cell growth (IC50: 3-30 nM); arrests cells in prometaphase; prevents bipolar spindle formation.</p>Formule :C30H42O7Couleur et forme :SolidMasse moléculaire :514.65Apoptosis inducer 5
<p>Apoptosis Inducer 5, a lignan enantiomer extracted from Crataegus pinnatifida, demonstrates cytotoxic properties through inducing apoptosis and autophagy in</p>Formule :C23H26O7Couleur et forme :SolidMasse moléculaire :414.45RN941
CAS :<p>RN941 is a highly potent Bruton's tyrosine kinase (BTK) inhibitor.</p>Formule :C34H34FN7O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :639.68LY2934747
CAS :<p>LY2934747 is a novel, potent, and systemically bioavailable mGlu2/3 receptor agonist, exhibiting both antipsychotic and analgesic properties in vivo.</p>Formule :C10H13NO4Couleur et forme :SolidMasse moléculaire :211.21Lp-PLA2-IN-5
CAS :<p>Lp-PLA2-IN-5 inhibits Lp-PLA2 and PAF-AH, potentially useful in Alzheimer's and atherosclerosis studies.</p>Formule :C23H18F5N3O4Couleur et forme :SolidMasse moléculaire :495.4UAWJ9-36-1
CAS :<p>UAWJ9-36-1: potent broad-spectrum coronavirus Protease inhibitor; IC50 = 51 nM.</p>Formule :C23H29N3O5Couleur et forme :SolidMasse moléculaire :427.49Anti-inflammatory agent 13
<p>Pentacyclic triterpene, Anti-inflammatory 13 inhibits DAMP/PAMP inflammation models.</p>Formule :C30H48O4Couleur et forme :SolidMasse moléculaire :472.7Anticancer agent 14
<p>Anticancer agent 14: a potent breast cancer inhibitor; induces cell death, disrupts mito. membrane potential (IC50: 0.20-0.65 μM).</p>Formule :C29H34N2O3Couleur et forme :SolidMasse moléculaire :458.59NR1H4 activator 1
CAS :<p>NR1H4 activator 1 is a potent and selective agonist of Famesoid X Receptor (FXR).</p>Formule :C34H53NO7SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :619.85GLPG0974
CAS :<p>GLPG0974 is an antagonist of FFA2/GPR43 with IC50 of 9 nM.</p>Formule :C25H25ClN2O4SDegré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :484.99AZD-5672
CAS :<p>AZD-5672 is an antagonist of CCR5 with an IC50 of 0.32 nM.</p>Formule :C32H38F2N2O5S2Degré de pureté :98.1%Couleur et forme :SolidMasse moléculaire :632.78NB-360
CAS :<p>NB-360: potent, brain-penetrant BACE1/2 inhibitor; IC50s: 5-6 nM; high selectivity vs pepsin, cathepsin E/D.</p>Formule :C21H19F4N5O2Degré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :449.4Vofopitant
CAS :<p>Vofopitant (GR 205171) is a potent NK1 receptor antagonist with anxiolytic and antiemetic activity for the study of post-traumatic stress disorder (PTSD).</p>Formule :C21H23F3N6ODegré de pureté :97.86%Couleur et forme :SolidMasse moléculaire :432.44Evixapodlin
CAS :<p>Evixapodlin (PD-1/PD-L1-IN 7) is a human PD-1/PD-L1 protein/protein interaction inhibitor (IC50: 0.213).Evixapodlin has anticancer and antiviral activities.</p>Formule :C34H36Cl2N8O4Degré de pureté :99.07%Couleur et forme :SolidMasse moléculaire :691.61AM103
CAS :<p>AM103 is an effective and selective inhibitor of FLAP (IC50 = 4.2 nM).</p>Formule :C36H38N3NaO4SDegré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :631.76USP5-IN-1
<p>USP5-IN-1, a powerful USP5 deubiquitinase inhibitor, selectively binds with 2.8 μM affinity, blocking USP5's di-ubiquitin cleavage.</p>Formule :C19H20ClN3O5SDegré de pureté :99.76%Couleur et forme :SoildMasse moléculaire :437.9Pocenbrodib
CAS :<p>Pocenbrodib (FT-7051) is a potent inhibitor of the bromodomain of the CBP/p300 family with potential antitumour activity and is palatable for cancer research.</p>Formule :C28H32FN3O6Degré de pureté :98.48% - 99.54%Couleur et forme :SolidMasse moléculaire :525.57D75-4590
CAS :<p>D75-4590, a β-1,6-Glucan synthetase inhibitor, combats fungal infections by targeting cell walls.</p>Formule :C21H27N5Degré de pureté :98.56% - 98.85%Couleur et forme :SolidMasse moléculaire :349.47AZD5462
CAS :<p>AZD5462 is a potent orally available relaxin receptor RXFP1 agonist for the study of heart failure and cancer.</p>Formule :C30H41FN2O6Degré de pureté :98.32% - 99.63%Couleur et forme :SolidMasse moléculaire :544.65Cbl-b-IN-3
CAS :<p>Cbl-b-IN-3 is a potent inhibitor of casitas b lineage lymphoma proto-oncogene-b (Cbl-b) (ic50 < 1 nM).Cost-effective and quality-assured.</p>Formule :C30H34F3N5ODegré de pureté :99%Couleur et forme :SolidMasse moléculaire :537.62Odevixibat
CAS :<p>Odevixibat (A4250) is a selective oral inhibitor for ileal bile acid transport, potentially treating primary biliary cirrhosis.</p>Formule :C37H48N4O8S2Degré de pureté :99.53% - 99.83%Couleur et forme :SolidMasse moléculaire :740.93AKT Kinase Inhibitor
CAS :<p>AKT Kinase Inhibitor is an Akt inhibitor with antitumor activity that selectively inhibits cell proliferation in a dose-dependent manner.Cost-effective and quality-assured.</p>Formule :C16H19N7O3Degré de pureté :97.83% - 99.13%Couleur et forme :SolidMasse moléculaire :357.37(+)-Tetrabenazine
CAS :<p>(+)-Tetrabenazine ((3R,11bR)-Tetrabenazine) is a reversible vesicular monoamine transporter 2 (VMAT-2) inhibitor, inhibits transport by VMAT2 with 10-fold</p>Formule :C19H27NO3Degré de pureté :98.31%Couleur et forme :SolidMasse moléculaire :317.42Milademetan
CAS :<p>Milademetan (DS-3032), an MDM2 inhibitor, exhibits antitumor activity, induces G1 cell cycle arrest and apoptosis, and can be used to study solid tumors.</p>Formule :C30H34Cl2FN5O4Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :618.53BCL6-IN-3
CAS :<p>BCL6-IN-3: potent BCL6 inhibitor, 70 nM GI50 in SU-DHL4, affects cell functions, antitumor.</p>Formule :C24H31ClF2N6O2Degré de pureté :98.17%Couleur et forme :SolidMasse moléculaire :508.99Obicetrapib
CAS :<p>Obicetrapib (AMG-899) is an inhibitor of cholesteryl ester transfer protein.</p>Formule :C32H31F9N4O5Degré de pureté :99.26% - >99.99%Couleur et forme :SolidMasse moléculaire :722.6SB-224289 hydrochloride
CAS :<p>SB-224289 hydrochloride (SB-224289A) is a selective antagonist of 5-HT1B receptor, with anxiolytic effect.</p>Formule :C32H33ClN4O3Degré de pureté :97.82% - 98.99%Couleur et forme :SolidMasse moléculaire :557.08BMS 299897
CAS :<p>BMS 299897, a sulfonamide γ-secretase inhibitor, inhibits Aβ production with an IC50 of 7 nM in HEK293 cells overexpressing APP.</p>Formule :C24H21ClF3NO4SDegré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :511.94LSN3318839
CAS :<p>LSN3318839 is a potent and orally available glucagon-like peptide-1 receptor (GLP-1R) modulator.LSN3318839 enhances GLP-1R G-protein-coupled signaling and can</p>Formule :C26H23Cl2N3O2Degré de pureté :99.21%Couleur et forme :SolidMasse moléculaire :480.39Eravacycline dihydrochloride
CAS :<p>Eravacycline dihydrochloride (TP-434-046) is a potent and broad-spectrum antibacterial agent against six E. coli (MICs: 0.125-0.25 mg/L).</p>Formule :C27H33Cl2FN4O8Degré de pureté :94.59% - 95%Couleur et forme :SolidMasse moléculaire :631.48Elacytarabine
CAS :<p>Elacytarabine (M7594 0037), a lipid-conjugated derivative of the nucleoside analog cytarabine, is an antineoplastic drug. It has cytotoxicity in solid tumors.</p>Formule :C27H45N3O6Degré de pureté :97.69%Couleur et forme :SolidMasse moléculaire :507.66DN02
<p>DN02: a potent, selective BRD8(1) bromodomain probe; Ki=32 nM; 30x more affine than BRD8(2).</p>Formule :C22H24FN3O3Degré de pureté :98.22% - 99.74%Couleur et forme :SolidMasse moléculaire :397.44NRX-1532
<p>NRX-1532 is a small molecule β-catenin:β-TrCP interaction enhancer.</p>Formule :C16H11F3N4O2Degré de pureté :98.95% - 99.68%Couleur et forme :SolidMasse moléculaire :348.28HOIPIN-8 sodium
CAS :<p>HOIPIN-8 sodium is a LUBAC inhibitor for the study of inflammatory and immune diseases.</p>Formule :C23H15F2N4NaO3Degré de pureté :97.34%Couleur et forme :SolidMasse moléculaire :456.38Tuvusertib
CAS :<p>Tuvusertib (M1774), an oral ATR inhibitor (Ki<1µM), selectively blocks CHK1 phosphorylation, disrupts DNA repair, and induces tumor cell apoptosis.</p>Formule :C16H12F2N8ODegré de pureté :98.44% - 99.66%Couleur et forme :SolidMasse moléculaire :370.32Zotizalkib
CAS :<p>TPX-0131: potent, selective, CNS-ready, oral ALK inhibitor (WT IC50: 1.4nM, G1202R/L1196M IC50: 0.3nM) with robust antitumor effects.</p>Formule :C21H20F3N5O3Degré de pureté :98.7%Couleur et forme :SolidMasse moléculaire :447.41SJ6986
CAS :<p>SJ6986 is a potent, selective and orally active GSPT1/2 degrader. SJ6986 degrades GSPT1 with a DC 50 of 2.1 nM (D max 99%) [1].</p>Formule :C20H14F3N3O7SDegré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :497.4AZD 3147
CAS :<p>AZD 3147 inhibits mTORC1 (40.7 nM), mTORC2 (5.75 nM), and PI3Kα/β/δ/γ (912/5495/9333/6310 nM IC50s).</p>Formule :C24H31N5O4S2Degré de pureté :99.99%Couleur et forme :SolidMasse moléculaire :517.66BE1218
CAS :<p>BE1218 is a liver X receptor (LXR) inverse agonist active on LXRα and LXRβ with an IC50 of 9 nM and 7 nM, respectively.</p>Formule :C30H30FNO4S2Degré de pureté :99.7%Couleur et forme :SoildMasse moléculaire :551.69KI696
CAS :<p>KI696 is a high-affinity probe that potently inhibits the interaction of Keap1 and NRF2.</p>Formule :C28H30N4O6SDegré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :550.63Picrotoxinin
CAS :<p>Picrotoxinin blocks chloride channels, antagonizes GABAA noncompetitively (IC50: 1.15 μM, α1β2γ2L), and induces convulsions.</p>Formule :C15H16O6Degré de pureté :98.07%Couleur et forme :SolidMasse moléculaire :292.28L-371,257
CAS :<p>L-371,257 is a competitive antagonist of oxytocin receptor with pA2 of 8.4 and Ki of 19 nM. L-371,257 shows a Ki of 3.7 nM for vasopressin receptor 1a.</p>Formule :C28H33N3O6Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :507.58INCB054329
CAS :<p>INCB054329 is a BET inhibitor targeting BRD2/3/4 and BRDT with IC50s ranging from 1-119 nM.</p>Formule :C19H16N4O3Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :348.36ALOX15-IN-2
CAS :<p>ALOX15-IN-2: Potent ALOX15 inhibitor. IC50: 1.55 μM for LA; 2.79 μM for AA. Stops linoleic/arachidonic acid oxidation.</p>Formule :C23H29N3O4SDegré de pureté :98.10%Couleur et forme :SolidMasse moléculaire :443.56Gepotidacin mesylate dihydrate
CAS :<p>Gepotidacin mesylate dihydrate (GSK2140944 mesylate dihydrate) is an antibiotic and an inhibitor of bacterial type II topoisomerase.</p>Formule :C25H36N6O8SDegré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :580.65NDI-034858
CAS :<p>NDI-034858 (TAK-279) is a tyrosine kinase 2 (TYK2) inhibitor (Kd<200 pM) that targets the JH2 structural domain of Tyk2 for the treatment of autoimmune diseases</p>Formule :C23H24N8O3Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :460.49O-Propargyl-Puromycin
CAS :<p>O-Propargyl-Puromycin (OP-puro) is a potent protein synthesis inhibitor, a puromycin acetylene analog.</p>Formule :C24H29N7O5Degré de pureté :97.83% - 99.70%Couleur et forme :SolidMasse moléculaire :495.53EZM0414
CAS :<p>EZM0414 is a potent, selective, orally bioavailable inhibitor of SETD2 with IC50 of 18 nM in SETD2 biochemical assay and IC50 of 34 nM in a cellular assay.</p>Formule :C22H29FN4O2Degré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :400.49IDX184
CAS :<p>IDX184 is a potent, orally active, targeted HCV polymerase inhibitor and nucleoside polymerase.IDX184 effectively inhibits HCV polymerase (IC50=0.31 μM, Ki=52.3</p>Formule :C25H35N6O9PSDegré de pureté :97.15%Couleur et forme :SolidMasse moléculaire :626.62BLU2864
CAS :<p>BLU2864: oral PRKACA inhibitor, IC50=0.3 nM, potential in cancer/poly. kidney disease research.</p>Formule :C24H19F3N4O2Degré de pureté :97.58% - 99.92%Couleur et forme :SoildMasse moléculaire :452.43VX-984
CAS :<p>VX-984 (M9831) is an oral DNA-PK inhibitor, crossing the blood-brain barrier, targeting GBM and NSC-LC.</p>Formule :C23H21D2N7ODegré de pureté :97.65% - 99.98%Couleur et forme :SolidMasse moléculaire :415.49AChE/BChE-IN-10
CAS :<p>AChE/BChE-IN-10 inhibits AChE/BChE (IC50: 0.176/0.47 μM), crosses the blood-brain barrier, and prevents Aβ-aggregation.</p>Formule :C26H30N2O2Degré de pureté :99.55% - 99.88%Couleur et forme :SoildMasse moléculaire :402.53BDZ-g
CAS :<p>BDZ-g: potent, selective AMPA receptor antagonist; useful for researching neurological disorders.</p>Formule :C21H21N5O2SDegré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :407.49USP15-IN-1
CAS :<p>USP15-IN-1 is a potent USP15 inhibitor (IC50 is 3.76 μM).</p>Formule :C22H23N3O3Degré de pureté :99.509% - 99.81%Couleur et forme :SolidMasse moléculaire :377.44FABPs ligand 6
CAS :<p>FABPs ligand 6 (MF6) is an inhibitor of FABP5 and FABP7.</p>Formule :C28H27FN2O3Degré de pureté :97.45%Couleur et forme :SolidMasse moléculaire :458.52Tigemonam
CAS :<p>Tigemonam is a monobactam, a novel orally administered monobactam that protects against gram-negative aerobic bacterial pathogens. Cost-effective and quality-assured.</p>Formule :C12H15N5O9S2Degré de pureté :99.03% - >99.99%Couleur et forme :SolidMasse moléculaire :437.41Glycosyltransferase-IN-1
<p>Glycosyltransferase-IN-1 is a glycosyltransferase inhibitor with bacteriostatic activity, inhibiting MSSA, MRSA, Bacillus subtilis, and Enterobacteriaceae.</p>Formule :C19H21N5ODegré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :335.4SYM2206
CAS :<p>SYM2206 is a low affinity non-competitive AMPA receptor antagonist with an IC50 value of 1.6 μM.SYM2206 exhibits anticancer activity by blocking Nav1.6-mediated</p>Formule :C20H22N4O3Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :366.41BQ-788
CAS :<p>BQ-788 is an ETB receptor antagonist with potential hypertensive activity that inhibits exogenous ET-1-induced elevation of coronary perfusion pressure.</p>Formule :C34H51N5O7Degré de pureté :98.81%Couleur et forme :SolidMasse moléculaire :641.8Cort108297
CAS :<p>Cort108297: selective GR modulator/antagonist, high GR affinity (Ki: 0.45nM), no other steroid receptor affinity.</p>Formule :C26H25F4N3O3SDegré de pureté :98.36% - 99.94%Couleur et forme :SolidMasse moléculaire :535.55KU-60019
CAS :<p>KU-60019 is a specific inhibitor of ATM kinase (IC50: 6.3 nM).</p>Formule :C30H33N3O5SDegré de pureté :98.05% - 98.50%Couleur et forme :SolidMasse moléculaire :547.67Moiramide B
CAS :<p>Moiramide B is an acetyl coenzyme A carboxylase inhibitor with antimicrobial activity, strongly inhibiting Gram-positive bacteria.</p>Formule :C25H31N3O5Degré de pureté :98.53% - 99.90%Couleur et forme :SolidMasse moléculaire :453.53SY-5609
CAS :<p>SY-5609 (CDK7-IN-3) is a selective non-covalent CDK7 inhibitor, with weak inhibitory activity against CDK2, CDK9 and CDK12.Cost-effective and quality-assured.</p>Formule :C23H26F3N6OPDegré de pureté :99.34% - >99.99%Couleur et forme :SolidMasse moléculaire :490.46GSK3368715 dihydrochloride
CAS :<p>GSK3368715 dihydrochloride (EPZ019997 dihydrochloride) is a PRMTs inhibitor , with anticancer activity, for the study of advanced solid tumors.</p>Formule :C20H40Cl2N4O2Degré de pureté :99.66% - 99.66%Couleur et forme :SolidMasse moléculaire :439.46BMS-986141
CAS :<p>BMS-986141(UDM-003183) is a selective and potent protease-activated receptor-4 (PAR-4) antagonist with oral activity and an IC50 value of 0.4 nM.BMS-98614</p>Formule :C27H23N5O5S2Degré de pureté :98.43% - 99.26%Couleur et forme :SolidMasse moléculaire :561.63BODIPY FL prazosin
CAS :<p>BODIPY FL prazosin is an α1-adrenergic antagonist that inhibits α1a-AR and α1b-AR.</p>Formule :C28H32BF2N7O3Degré de pureté :97.27%Couleur et forme :SolidMasse moléculaire :563.41NRX-103095
CAS :<p>NRX-103095 increases β-catenin binding to SCFβ-TrCP E3 ligase; EC50 is 163 nM for pSer33/Ser37 affinity boost.</p>Formule :C22H16Cl2F3N3O3SDegré de pureté :99.58% - 99.95%Couleur et forme :SolidMasse moléculaire :530.35Cap-dependent endonuclease-IN-1
CAS :<p>Cap-dependent endonuclease-IN-1: potent, oral inhibitor with antiviral properties against influenza.</p>Formule :C27H22F2N2O6SDegré de pureté :98.88% - 99.09%Couleur et forme :SolidMasse moléculaire :540.54AChE-IN-26
CAS :<p>AChE-IN-26 (compound 4a) is an AChE (acetylcholinesterase) inhibitor (IC50: 0.42 μM).</p>Formule :C21H21BrN2O3Degré de pureté :99.24% - 99.85%Couleur et forme :SoildMasse moléculaire :429.31Lometrexol
CAS :<p>Lometrexol (LY 264618) is an antifolate that inhibits GARFT, blocks purine synthesis, induces apoptosis, and has anticancer properties.</p>Formule :C21H25N5O6Degré de pureté :97.76% - 99.56%Couleur et forme :SolidMasse moléculaire :443.45NRX-103094
CAS :<p>NRX-103094 boosts β-catenin binding to SCFβ-TrCP ligase with EC50 62 nM and Kd 0.6 nM.</p>Formule :C20H11Cl2F3N2O4SDegré de pureté :99.13%Couleur et forme :SolidMasse moléculaire :503.28PF-07258669
CAS :<p>PF-07258669 is a selective melanocortin 4 receptor (MC4) antagonist used in the study of cachexia and loss of appetite.</p>Formule :C25H27FN6O2Degré de pureté :99.9%Couleur et forme :SolidMasse moléculaire :462.52BMS453
CAS :<p>BMS453 (BMS-189453), a synthetic retinoid, is a potent and selective agonist of RARβ and a potent testicular toxin.</p>Formule :C27H24O2Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :380.48Aldometanib
CAS :<p>Aldometanib (LXY-05-029) is an oral aldolase inhibitor that maintains metabolic balance by blocking FBP and activating lysosomal AMPK.</p>Formule :C27H43Cl2IN2Degré de pureté :99.32% - 99.55%Couleur et forme :SolidMasse moléculaire :593.46SDZ 220-040
CAS :<p>SDZ 220-040 是一种选择性哺乳动物 NMDA 受体拮抗剂，可诱导根系生长的部分无重力模式 。</p>Formule :C16H16Cl2NO6PDegré de pureté :98.13%Couleur et forme :SolidMasse moléculaire :420.18AZ12601011
CAS :<p>AZ12601011 is a TGFBR1 kinase inhibitor that inhibits the growth of breast tumors.</p>Formule :C19H15N5Degré de pureté :98.81%Couleur et forme :SolidMasse moléculaire :313.36Umibecestat
CAS :<p>Umibecestat inhibits human and mouse BACE-1 (IC50: 11 nM & 10 nM), potentially for Alzheimer's research.</p>Formule :C19H15ClF7N5O2Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :513.8Enbezotinib
CAS :<p>Enbezotinib is an inhibitor of RET autophosphorylation and can be used in cancer research.</p>Formule :C21H21FN6O3Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :424.43Vecabrutinib
CAS :<p>Vecabrutinib (SNS-062) is a potent and noncovalent BTK and ITK inhibitor (Kd: 0.3 nM and 2.2 nM, respectively). Vecabrutinib displays an IC50 of 24 nM for ITK.</p>Formule :C22H24ClF4N7O2Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :529.92STK-15
CAS :<p>STK-15 is a candidate for use as a fatty acid binding protein 5 (FABP5) inhibitor.</p>Formule :C34H29NO5Degré de pureté :98.05%Couleur et forme :SolidMasse moléculaire :531.6Aleglitazar
CAS :<p>Aleglitazar (R1439) (R1439) is a potent dual PPARα/γ agonist, with IC50s of 38 nM and 19 nM for human PPARa and PPARγ, respectively.</p>Formule :C24H23NO5SDegré de pureté :99.03%Couleur et forme :SolidMasse moléculaire :437.51LY2979165
CAS :<p>LY2979165 (mGlu2 agonist) is an orthosteric agonist of mGluR2 and can be used in studies about serving as an anti-depressant.</p>Formule :C13H22N6O6SDegré de pureté :98.41%Couleur et forme :SolidMasse moléculaire :390.42ELOVL1-IN-2
CAS :<p>ELOVL1-IN-2 weakly inhibits ELOVL1 enzyme (IC50: 21 μM) and shows moderate potency in HEK293 cells (IC50: 6.7 μM).</p>Formule :C18H15FN2ODegré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :294.32JNJ-6204
CAS :<p>JNJ-6204 is a deuterated compound that efficiently inhibits CSNK1D and CSNK1E.</p>Formule :C19H11D6FN6ODegré de pureté :97.42% - 99.87%Couleur et forme :SolidMasse moléculaire :370.41NRX-252114
CAS :<p>NRX-252114 promotes mutant β-catenin degradation, binding it to E3 ligase SCFβ-TrCP (EC50: 6.5 nM; Kd: 0.4 nM).</p>Formule :C22H12Cl2F3N3O2SDegré de pureté :99.70%Couleur et forme :SolidMasse moléculaire :510.32Suzetrigine
CAS :<p>Suzetrigine (VX-548) is an oral NaV1.8 inhibitor with analgesic properties for acute pain research.</p>Formule :C21H20F5N3O4Degré de pureté :98.08% - 99.27%Couleur et forme :SolidMasse moléculaire :473.39ZD 7155 hydrochloride
CAS :<p>ZD 7155 hydrochloride is an angiotensin II receptor type 1 (AT1 receptor) antagonist.</p>Formule :C26H27ClN6ODegré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :474.98WAY-213613 hydrochloride
CAS :<p>WAY-213613 hydrochloride: potent, selective GLT-1/EAAT2 inhibitor (IC50 85 nM); weaker for EAAT1/3; inactive at glutamate receptors; research tool for CNS.</p>Formule :C16H13BrF2N2O4Degré de pureté :99.14% - 99.37%Couleur et forme :SoildMasse moléculaire :415.19LLY-283
CAS :<p>LLY-283, PRMT5 inhibitor, IC50 22 nM, Kd 6 nM, oral, selective, with antitumor effects.</p>Formule :C17H18N4O4Degré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :342.35DRF-1042
CAS :<p>DRF-1042 is a camptothecin analog with anticancer and insecticidal activity and is used to study solid tumors such as prostate and colon cancer.</p>Formule :C22H20N2O6Degré de pureté :98.34%Couleur et forme :SolidMasse moléculaire :408.4SB-423562
CAS :<p>SB-423562 is a calcium-sensing receptor (CaSR) antagonist and can be used in studies about osteoporosis.</p>Formule :C26H32N2O4Degré de pureté :99.22%Couleur et forme :SolidMasse moléculaire :436.54CP-642931
CAS :<p>CP-642931 (Sorbitol dehydrogenase-IN-1) is a sorbitol dehydrogenase inhibitor used in the study of diabetes mellitus and cardiovascular disease.</p>Formule :C17H25N7ODegré de pureté :99.67% - >99.99%Couleur et forme :SolidMasse moléculaire :343.43Dual FAAH/sEH-IN-1
CAS :<p>Dual FAAH/sEH-IN-1 inhibits both sEH (IC50: 9.6 nM) and FAAH (IC50: 7 nM), offering potent anti-inflammatory effects.</p>Formule :C25H22ClN3O3S2Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :512.04Simmitecan hydrochloride
CAS :<p>Simmitecan hydrochloride is a camptothecin derivative, a topoisomerase I inhibitor with anticancer activity, which can be used to study is solid tumors.</p>Formule :C34H39ClN4O6Degré de pureté :98.20% - 98.93%Couleur et forme :SolidMasse moléculaire :635.15MAO-B-IN-17
CAS :<p>MAO-B-IN-17 is a selective and potent monoamine oxidase B (MAO-B) inhibitor (IC50: 5.08 μM) for the study of central nervous system disorders like Parkinson's.</p>Formule :C17H17F2NO2Degré de pureté :99.41%Couleur et forme :SoildMasse moléculaire :305.32DRB18
CAS :<p>DRB18 inhibits GLUT proteins, altering glucose metabolism and inducing cancer cell death by G1/S arrest and oxidative stress.</p>Formule :C22H23ClN2O2Degré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :382.88Dersimelagon
CAS :<p>Dersimelagon (MT-7117) is an orally active, selective melanocortin 1 receptor (MC1R) agonist.Cost-effective and quality-assured.</p>Formule :C36H45F4N3O5Degré de pureté :97.35% - 98.23%Couleur et forme :SolidMasse moléculaire :675.75Etamicastat hydrochloride
CAS :<p>Etamicastat hydrochloride (BIA 5-453 hydrochloride) is a peripherally selective dopamine beta-hydroxylase inhibitor that reduces hypertension.</p>Formule :C14H16ClF2N3OSDegré de pureté :98.54%Couleur et forme :SolidMasse moléculaire :347.81Dazostinag disodium
CAS :<p>Dazostinag disodium (TAK-676) is a synthetic novel interferon gene (STING) agonist.Cost-effective and quality-assured.</p>Formule :C21H20F2N8Na2O10P2S2Degré de pureté :98.84% - 99.96%Couleur et forme :SolidMasse moléculaire :754.48MIV-247
CAS :<p>MIV-247 is a cathepsin S inhibitor that attenuates mechanically abnormal pain in preclinical neuropathic pain models and can be used to study myocardial injury.</p>Formule :C17H24F3N3O4Degré de pureté :99.27%Couleur et forme :SolidMasse moléculaire :391.39Treprostinil diethanolamine
CAS :<p>Treprostinil diethanolamine (UT-15C) is a potent agonist of EP2, DP1 and IP, with values of 3.6, 4.4, 32.1, 212, 826, 2505 and 4680 nM for EP2, DP1, IP, EP1,</p>Formule :C27H45NO7Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :495.65Darizmetinib
CAS :<p>Darizmetinib (HRX215) is an MKK4 inhibitor.</p>Formule :C21H17F2N5O3SDegré de pureté :98.03% - 99.57%Couleur et forme :SolidMasse moléculaire :457.45Vofopitant dihydrochloride
CAS :<p>Vofopitant dihydrochloride (GR 205171A) is a tachykinin NK1 receptor antagonist and a potential compound for the treatment of pathologic vomiting.</p>Formule :C21H25Cl2F3N6ODegré de pureté :98.99%Couleur et forme :SolidMasse moléculaire :505.36HRO761
CAS :<p>HRO761 is a potent Werne r syndrome RecQ DNA deconjugase (WRN) inhibitor that can be used to study cancers such as colon and stomach cancer.</p>Formule :C31H31ClF3N9O5Degré de pureté :98.74% - 99.62%Couleur et forme :SolidMasse moléculaire :702.08PREP inhibitor-1
CAS :<p>PREP inhibitor-1 is a prolyl oligopeptidase (PREP) inhibitor for the study of Alzheimer's disease.</p>Formule :C22H28N4O2Degré de pureté :98.78%Couleur et forme :SoildMasse moléculaire :380.48JTK-109
CAS :<p>JTK-109 is an inhibitor of hepatitis C virus NS5B RNA-dependent RNA polymerase inhibitor and inhibits G1b and G3a subgenomic replicons and recombinant enzymes.</p>Formule :C37H33ClFN3O4Degré de pureté :98.48% - 99.68%Couleur et forme :SolidMasse moléculaire :638.13CCF0058981
CAS :<p>CCF0058981: noncovalent inhibitor for SARS-CoV-2 & -1 proteases; IC50s: 68 nM (SC2) & 19 nM (SC1). Potential COVID-19 research use.</p>Formule :C24H19ClN6ODegré de pureté :98.94%Couleur et forme :SoildMasse moléculaire :442.9Emprumapimod
CAS :<p>Emprumapimod, an oral p38α MAPK inhibitor, targets RPMI-8226 cells, curbs LPS-induced IL-6; IC50: 100 pM; for cardiomyopathy, acute pain.</p>Formule :C24H29F2N5O3Degré de pureté :99.21% - >99.99%Couleur et forme :SolidMasse moléculaire :473.52Rupintrivir
CAS :<p>Rupintrivirvr (AG7088) is a mimetic peptide inhibitor of rhinovirus (HRV) 3C cysteine protease with antiviral activity for the study of viral infections.</p>Formule :C31H39FN4O7Degré de pureté :97.72% - 99.35%Couleur et forme :SolidMasse moléculaire :598.66BAY-3827
CAS :<p>BAY-3827 is an AMPK inhibitor with antiproliferative activity and antitumor activity. BAY-3827 inhibits the phosphorylation of acetyl CoA carboxylase 1.</p>Formule :C27H25FN6ODegré de pureté :99.90%Couleur et forme :SolidMasse moléculaire :468.53Zelasudil
CAS :<p>Zelasudil (RXC007) is a Rho-related (ROCK) kinase inhibitor for the study of idiopathic pulmonary fibrosis and inflammation.</p>Formule :C22H21F2N7ODegré de pureté :99.15%Couleur et forme :SolidMasse moléculaire :437.445Iclepertin
CAS :<p>Iclepertin (BI-425809) is a GlyT1 inhibitor.Iclepertin is used for the treatment of Alzheimer;s disease and other CNS disorders.</p>Formule :C20H18F6N2O5SDegré de pureté :98.89% - 98.93%Couleur et forme :SolidMasse moléculaire :512.42Sinefungin
CAS :<p>Sinefungin (Adenosyl-Ornithine) is an effective inhibitor of virion mRNA(guanine-7-)-methyltransferase, mRNA(nucleoside-2'-)-methyltransferase, and viral</p>Formule :C15H23N7O5Degré de pureté :98.12%Couleur et forme :SolidMasse moléculaire :381.39JAK2-IN-7
CAS :<p>JAK2-IN-7 selectively inhibits JAK2 (IC50: 3 nM), shows 14-fold selectivity over JAK1/3, FLT3, induces G0/G1 arrest, apoptosis, and has antitumor effects.</p>Formule :C26H33N7ODegré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :459.59CK2 inhibitor 2
CAS :<p>CK2 Inhibitor 2, characterized as a potent, selective, and orally active inhibitor of CK2, demonstrates an impressive IC50 value of 0.66 nM.</p>Formule :C21H17ClN4O2Degré de pureté :99.02%Couleur et forme :SolidMasse moléculaire :392.84ARN19702
CAS :<p>ARN19702: orally active, brain-penetrant, selective NAAA inhibitor, IC50 230 nM, broad analgesic profile.</p>Formule :C21H22FN3O3S2Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :447.55Rolapitant hydrochloride
CAS :<p>Rolapitant HCl is a potent NK1 antagonist, non-CYP3A4 interactive, with anti-emetic effects and a Ki of 0.66 nM.</p>Formule :C25H27ClF6N2O2Degré de pureté :98.35% - 99.79%Couleur et forme :SolidMasse moléculaire :536.94LY3143921 hydrate
CAS :<p>LY3143921 ((S)-Example 2) hydrate is an orally active CDC7 kinase inhibitor with broad in vitro anticancer activity [1].</p>Formule :C16H14FN5O2Degré de pureté :98.43%Couleur et forme :SolidMasse moléculaire :327.3110-Methoxycamptothecin
CAS :<p>10-Methoxycamptothecin is a natural bioactive derivative of camptothecin (CPT) isolated from Camptotheca acuminata and possesses high anti-cancer properties.</p>Formule :C21H18N2O5Degré de pureté :98.36%Couleur et forme :SolidMasse moléculaire :378.38XMD-17-51 Trifluoroacetate
CAS :<p>XMD-17-51 Trifluoroacetate is a pyrimido-diazepinone compound that regulates protein kinases.</p>Formule :C23H25F3N8O3Degré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :518.49TGFβRI-IN-3
CAS :<p>TGFβRI-IN-3 inhibits TGFβR1 with an IC 50 of 0.79 nM with 2000-fold selectivity against MAP4K4.</p>Formule :C28H23N3O2SDegré de pureté :99.85%Couleur et forme :SoildMasse moléculaire :465.57SR 11302
CAS :<p>SR 11302 is an inhibitor of activator protein-1 (AP-1).</p>Formule :C26H32O2Degré de pureté :98.65%Couleur et forme :SolidMasse moléculaire :376.53BAY-8400
<p>BAY-8400 is an orally active, potent and selective DNA-dependent protein kinase ( DNA-PK ) inhibitor ( IC 50 =81 nM) which shows synergistic efficacy in</p>Formule :C21H17F2N5ODegré de pureté :99.53%Couleur et forme :SolidMasse moléculaire :393.39(E/Z)-GSK5182
CAS :<p>GSK5182 is a racemic mix of (E/Z) isomers, a selective ERRγ inverse agonist (IC50: 79 nM), and induces ROS in liver cancer.</p>Formule :C27H31NO3Degré de pureté :97.58%Couleur et forme :SolidMasse moléculaire :417.54BRD0639
CAS :<p>BRD0639 is a first-in-class PRMT5-substrate interaction inhibitor for PBM-dependent PRMT5 activity studies.</p>Formule :C21H22ClN5O4SDegré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :475.95Gemcitabine elaidate hydrochloride
CAS :<p>CP-4126, a lipophilic pro-drug of Gemcitabine, converts to active form by esterases, allowing oral administration with dose-dependent effects.</p>Formule :C27H44ClF2N3O5Degré de pureté :98.50% - 99.6%Couleur et forme :SolidMasse moléculaire :564.11FGI-106 tetrahydrochloride
CAS :<p>FGI-106 tetrahydrochloride demonstrates potent inhibitory activity across a broad spectrum of viruses, including those causing hemorrhagic fevers such as Ebola</p>Formule :C28H42Cl4N6Degré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :604.48Rineterkib
CAS :<p>Rineterkib (ERK-IN-1) is an inhibitor of RAF and ERK1/2 activating mutations in the MAPK pathway.</p>Formule :C26H27BrF3N5O2Degré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :578.42Durlobactam sodium salt
CAS :<p>Durlobactam sodium salt (ETX2514) have an IC50 values of 4, 14 and 190 nM against class A KPC-2, class C AmpC and class D OXA-24.Cost-effective and quality-assured.</p>Formule :C8H10N3NaO6SDegré de pureté :97.01% - 99.03%Couleur et forme :SolidMasse moléculaire :299.23PD 151746
CAS :<p>PD151746: calpain inhibitor, Ki μ-calpain=0.26μM, Ki m-calpain=5.33μM; reduces oxLDL cytotoxicity.</p>Formule :C11H8FNO2SDegré de pureté :98.63% - ≥95%Couleur et forme :SolidMasse moléculaire :237.25Sebetralstat
CAS :<p>Sebetralstat (KVD900) is an inhibitor of plasma kallikrein and can be used in studies about metabolic diseases.</p>Formule :C26H26FN5O4Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :491.51LSZ-102
CAS :<p>LSZ-102 is an effective and selective degrader of estrogen receptor (IC50 = 0.2 nM) and can be used in studies about ERα positive breast cancer.</p>Formule :C25H17F3O4SDegré de pureté :98.56%Couleur et forme :SolidMasse moléculaire :470.46FX-11
CAS :<p>FX-11: potent LDHA inhibitor (Ki 8 μM), activates PKM2, reduces ATP, induces oxidative stress/ROS, cell death, shows antitumor effects.</p>Formule :C22H22O4Degré de pureté :98.95%Couleur et forme :SolidMasse moléculaire :350.41INCB086550
CAS :<p>INCB086550 (PD-1/PD-L1-IN-8) (example 24) is a PD-1/PD-L1 inhibitor, with an IC50 <= 10 nM.</p>Formule :C41H39N7O4Degré de pureté :98.49%Couleur et forme :SolidMasse moléculaire :693.79Clorophene
CAS :<p>Clorophene (Clorofene) is an antimicrobial agent and can be used in personal care products.</p>Formule :C13H11ClODegré de pureté :99.87%Couleur et forme :White To Light Tan Or Pink Flakes Phenolic Odor (Ntp 1992)Masse moléculaire :218.68Metrizoic acid
CAS :<p>Metrizoic acid is an ionic contrast medium. Metrizoic acid displays high osmolality and has a risk of inducing allergic reactions.</p>Formule :C12H11I3N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :627.9402Deoxypseudouridine
CAS :<p>Deoxypseudouridine is a nucleotide analog.</p>Formule :C9H12N2O5Couleur et forme :SolidMasse moléculaire :228.23-Methylcrotonylglycine
CAS :<p>3-Methylcrotonylglycine is an acyl glycine, a normal amino acid metabolite found in urine.</p>Formule :C7H11NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :157.17GAS6 Protein, Human, Recombinant (His)
<p>GAS6 (Growth arrest-specific protein 6) is also known as AXL receptor tyrosine kinase ligand, AXLLG, is a multimodular protein that is up-regulated by a wide variety of cell types in response to growth arrest. Gas6 binds and induces signaling through the receptor tyrosine kinases Axl, Dtk, and Mer whose signaling is implicated in cell growth and survival, cell adhesion and cell migration. GAS6/AXL signaling plays a role in various processes such as endothelial cell survival during acidification by preventing apoptosis, optimal cytokine signaling during human natural killer cell development, hepatic regeneration, gonadotropin-releasing hormone neuron survival and migration, platelet activation, or regulation of thrombotic responses. GAS6 Protein, Human, Recombinant (His) is expressed in HEK293 cells.</p>Degré de pureté :＞99.90%Couleur et forme :SoildMasse moléculaire :72.7 KDa (Predicted), 80-90 KDa (Reducing conditions)(S,S)-Valifenalate
CAS :<p>(S,S)-Valifenalate is an acylamino acid fungicide and is used to control a wide range of fungi belonging to the class of Oomycetes.</p>Formule :C19H27ClN2O5Couleur et forme :SolidMasse moléculaire :398.88TCblR Protein, Human, Recombinant (His)
<p>TCblR Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with C-6xHis tag. The predicted molecular weight is 32-58 KDa and the accession number is Q9NPF0.</p>Couleur et forme :SolidMasse moléculaire :32-58 KDa (reducing condition)sodium 4-pentynoate
CAS :<p>sodium 4-pentynoate is a alkynylacetate analogue.</p>Formule :C5H5NaO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :120.08TEM1/CD248 Protein, Mouse, Recombinant (His)
<p>TEM1/CD248 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with C-His tag. The predicted molecular weight is 73.6 kDa and the accession number is Q91V98.</p>Couleur et forme :SolidMasse moléculaire :73.6 kDa (predicted). Due to glycosylation, the protein migrates to 75-140 kDa based on Tris-Bis PAGE result.4',5'-Dibromofluorescein
CAS :<p>4',5'-Dibromofluorescein (Eosinic acid) is a fluorescent dye that can be used as a ligand for protein characterization by spectroscopic analysis.</p>Formule :C20H10Br2O5Couleur et forme :Orange Solid PowderMasse moléculaire :490.10(S)-Rasagiline
CAS :<p>(S)-Rasagiline is rasagiline S-isomer, and is an agent of anti-Parkinson.</p>Formule :C12H13NCouleur et forme :SolidMasse moléculaire :171.243-Hydroxyhippuric acid
CAS :<p>3-Hydroxyhippuric acid is an acyl glycine, which are normally minor metabolites of fatty acids.</p>Formule :C9H9NO4Couleur et forme :SolidMasse moléculaire :195.17TD-106
CAS :<p>TD-106 is a modulator of cereblon (CRBN), and can be used for targeted protein degradation. BRD4 PROTACs with TD-106 induce BRD4 degradation.</p>Formule :C12H11N5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :273.25(Rac)-Rotigotine hydrochloride
CAS :<p>(Rac)-Rotigotine hydrochloride is a racemate of Rotigotine. Rotigotine is a full agonist of dopamine receptor, a partial the 5-HT1A receptor agonist.</p>Formule :C19H26ClNOSCouleur et forme :SolidMasse moléculaire :351.933-Acetylcoumarin
CAS :<p>3-Acetylcoumarin as a practical ligand for copper-catalyzed CN coupling reactions at room temperature. It has neuroprotective and acaricidal properties.</p>Formule :C11H8O3Degré de pureté :99.41%Couleur et forme :Yellow Crystalline PowderMasse moléculaire :188.18(-)-Isopulegol
CAS :<p>Isopulegol has antioxidant, and neuroactive properties. It also has gastroprotective effects induced by isopulegol appear to be mediated, at least in part, by endogenous prostaglandins, K+ATP channel opening and antioxidant proprieties related to GSH increased.</p>Formule :C10H18ODegré de pureté :99.89%Couleur et forme :LiquidMasse moléculaire :154.25α-Terpineol
CAS :<p>Terpineol possesses antifungal activity against Trichophyton mentagrophytes, it also exhibits strong antimicrobial activity against periodontopathic and cariogenic bacteria. α-Terpineol (Terpineol) shows anticonvulsant, and anti-inflammatory activities, it inhibits the gene expression of the IL-6 receptor.</p>Formule :C10H18ODegré de pureté :97.55%Couleur et forme :Colorless LiquidMasse moléculaire :154.25Anisylacetone
CAS :<p>Anisylacetone (Anisylacetone) is an effective lure for the male melon fly.</p>Formule :C11H14O2Degré de pureté :99.74%Couleur et forme :LiquidMasse moléculaire :178.234-Ethoxycoumarin
CAS :<p>4-Ethoxycoumarin has antimicrobial activity.</p>Formule :C11H10O3Degré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :190.2PRGL493
CAS :<p>PRGL493 blocks ACSL4, halts PC3/MDA-MB-231 cancer cell spread, and inhibits MA-10 tumor progesterone. Effective in mouse PC3 tumor model at 0.25 mg/kg.</p>Formule :C25H21N7O2Degré de pureté :98.80% - 99.11%Couleur et forme :SolidMasse moléculaire :451.48Relacorilant
CAS :<p>Relacorilant is an oral glucocorticoid receptor antagonist with Ki of 7.2 nM, potential for treating Cushing's syndrome.</p>Formule :C27H22F4N6O3SDegré de pureté :98.53% - 99%Couleur et forme :SolidMasse moléculaire :586.563-Methoxyphenylacetic acid
CAS :<p>3-Methoxyphenylacetic acid belongs to the class of organic compounds known as anisoles. 3-Methoxyphenylacetic acid is slightly soluble (in water) and a weakly acidic compound (based on its pKa).3-Methoxyphenylacetic acid (m-Methoxyphenylacetic acid), a m-hydroxyphenylacetic acid (m-OHPAA) derivative, is a phytotoxin in Rhizoctonia solani. 3-Methoxyphenylacetic acid is used to develop a toxin-mediated bioassay for resistance to rhizoctonia root rot</p>Formule :C9H10O3Degré de pureté :98.61%Couleur et forme :White SolidMasse moléculaire :166.172'-Hydroxy-4'-methylacetophenone
CAS :<p>2'-Hydroxy-4'-methylacetophenone, a phenolic compound isolated from Angelicae koreana roots possesses acaricidal property. 2'-Hydroxy-4'-methylacetophenone has acaricidal activity, it could be used in the preparation of 4'-methyl-2'-[(p-tolylsulfonyl) oxy] acetophenone.</p>Formule :C9H10O2Degré de pureté :99.88%Couleur et forme :Black LiquidMasse moléculaire :150.17EGFR-IN-7
CAS :<p>EGFR-IN-7 (TQB3804) is a selective and potent EGFR kinase inhibitor.</p>Formule :C32H41BrN9O2PDegré de pureté :95.32% - 99.64%Couleur et forme :SolidMasse moléculaire :694.6PD-1/PD-L1-IN 5 TFA
CAS :<p>PD-1/PD-L1-IN 5 is an inhibitor of PD-1/PD-L1 protein/protein interaction (IC50 of ≤100 nM).</p>Formule :C22H18N4O3S·xC2HF3O2Degré de pureté :98%Couleur et forme :SolidAntitubercular agent-10
CAS :<p>Antitubercular agent-10 shows potent antitubercular activity with a MIC value of 30 nM.</p>Formule :C19H15N5O6S2Couleur et forme :SolidMasse moléculaire :473.48Patecibart
CAS :<p>Patecibart is a humanized immunoglobulin G4-kappa monoclonal antibody that functions as an antagonist to the endothelin receptor A (EDNRA).</p>Degré de pureté :98%Couleur et forme :LiquidNE97220
CAS :<p>NE97220 is a bioactive chemical.</p>Formule :C7H12N2O6P2Couleur et forme :SolidMasse moléculaire :282.13Sodium pyrene-1,3,6,8-tetrasulfonate
CAS :<p>Sodium pyrene-1,3,6,8-tetrasulfonate is a useful organic compound for research related to life sciences.</p>Formule :C16H11NaO12S4Couleur et forme :SolidMasse moléculaire :546.482',3'-cGAMP-C2-SH
CAS :<p>2', 3'-cGAMP-C2-SH is a ADC cytotoxin.</p>Formule :C22H28N10O12P2SCouleur et forme :SolidMasse moléculaire :718.53STING agonist-22
CAS :<p>STING agonist-22 (CF501) boosts vaccines by activating STING, inducing IFN-I and cytokines, aiding in SARS-CoV-2 research.</p>Formule :C40H48N14O6Couleur et forme :SolidMasse moléculaire :820.9AI3-10714
CAS :<p>AI3-10714 is a biochemical.</p>Formule :C14H6F17NO2SCouleur et forme :SolidMasse moléculaire :575.24Patent Blue V
CAS :<p>Patent Blue V (Acid blue 1), a biological dye, serves as an intraocular stain in retinectomy—surgical removal of the inner limiting membrane (ILM).</p>Formule :C27H31N2NaO6S2Couleur et forme :SolidMasse moléculaire :566.67LY 280748
CAS :<p>LY 280748 is a bio-active chemical.</p>Formule :C23H29N4NaO2Couleur et forme :SolidMasse moléculaire :416.49Mitoquinone
CAS :<p>Mitoquinone is a TPP-based, mitochondrially targeted antioxidant .</p>Formule :C37H44O4PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :583.72Phenol, m-(2-(methylamino)ethyl)-, hydrochloride
CAS :<p>Phenol, m-(2-(methylamino)ethyl)-, hydrochloride is a biaoctive chemical.</p>Formule :C9H14ClNOCouleur et forme :SolidMasse moléculaire :187.67Phototherapeutic agent-1
CAS :<p>Phototherapeutic agent-1: a light-activated, ROS-generating cancer cell killer with aggregation-induced emission.</p>Formule :C39H33F6N2O2PS3Couleur et forme :SolidMasse moléculaire :802.85Leishman's stain
CAS :<p>Leishman's stain is a vital dye for staining peripheral blood and bone marrow smears, which appear pale bluish-grey to deep blue when viewed under an oil-</p>Couleur et forme :SolidBD-9136
<p>BD-9136, a highly selective BRD4 degrader, demonstrates the capability to inhibit tumor growth without inducing adverse effects in mice, showing potential for</p>Formule :C44H44N10O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :824.95ABT-491 free base
CAS :<p>ABT-491 free base is a bio-active chemical. Detailed information has not been published.</p>Formule :C28H22FN5O2Couleur et forme :SolidMasse moléculaire :479.51Sinoporphyrin sodium
CAS :<p>Sinoporphyrin sodium hinders cell growth, induces early apoptosis, disrupts F-actin, impairs movement, and may treat cancer; it's a photosensitizer.</p>Formule :C68H70N8Na4O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1235.314Melarsonyl dipotassium
CAS :<p>Melarsonyl dipotassium, also known as melarsonic acid dipotassium, is a potent anthelmintic agent with the ability to effectively inhibit parasites.</p>Formule :C13H13AsK2N6O4S2Couleur et forme :SolidMasse moléculaire :534.52Pyrromethene 597
CAS :<p>Pyrromethene 597, a BODIPY laser dye, exhibits a wide tuning range of lasing wavelengths along with high photostability, and can serve as a thermal probe [1] [2</p>Formule :C22H33BF2N2Couleur et forme :SolidMasse moléculaire :374.32Antibacterial agent 30
CAS :<p>Antibacterial agent 30 exhibits remarkable in vitro activity against Xoo, as evidenced by its EC50 value of 1.9 μg/mL.</p>Formule :C24H24F3NO5Couleur et forme :SolidMasse moléculaire :463.45Antibacterial agent 28
CAS :<p>Antibacterial agent 28 targets MRSA with 0.5-2 μg/mL MIC, showing high potential.</p>Formule :C40H64Br2N4O4Couleur et forme :SolidMasse moléculaire :824.77Methyl Green zinc chloride
CAS :<p>Methyl Green zinc chloride: fluorescent DNA dye for cell/gel staining, viability tests; absorbance at 633/677 nm. Store in dark.</p>Formule :C27H35N3·Br·xCl2Zn·ClCouleur et forme :SolidMasse moléculaire :653.23
