Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.519 produits)
- Apoptose(5.786 produits)
- Cycle cellulaire/point de contrôle(4.444 produits)
- Chromatine/Épigénétique(2.235 produits)
- Signalisation du cytosquelette(1.382 produits)
- Altération de l'ADN/réparation de l'ADN(2.823 produits)
- Endocrinologie/Hormones(3.499 produits)
- Enzyme(3.639 produits)
- GPCR/G-Protéine(8.314 produits)
- Immunologie et Inflammation(3.516 produits)
- Virus de la grippe(296 produits)
- Signalisation JAK/STAT(404 produits)
- Signalisation MAPK(1.199 produits)
- Transporteur membranaire/Canal ionique(2.786 produits)
- Métabolisme(9.417 produits)
- Microbiologie/Virologie(6.967 produits)
- Neuroscience(9.920 produits)
- Autres inhibiteurs(37.931 produits)
- Oxydation-Réduction(41 produits)
- Signalisation PI3K/Akt/mTOR(1.399 produits)
- Protéases/Protéasome(1.596 produits)
- Cellules souche et Dérivés(832 produits)
- Tyrosine Kinase/Adaptateurs(2.015 produits)
- Ubiquitination(1.646 produits)
Affichez 16 plus de sous-catégories
66627 produits trouvés pour "Inhibiteurs"
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5-OxoETE
CAS :<p>5-OxoETE, a dehydrogenase-oxidized 5-HETE, raises neutrophil Ca²⁺ (EC50=2nM) & drives eosinophil migration & MAPK pathway.</p>Formule :C20H30O3Degré de pureté :98.59%Couleur et forme :SolidMasse moléculaire :318.45sodium 4-pentynoate
CAS :<p>sodium 4-pentynoate is a alkynylacetate analogue.</p>Formule :C5H5NaO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :120.08Alminoprofen
CAS :<p>Alminoprofen: NSAID; reduces anaphylactic bronchoconstriction at 30 mg/kg intraduodenally.</p>Formule :C13H17NO2Couleur et forme :SolidMasse moléculaire :219.28L-690330
CAS :<p>L-690330 inhibits human/bovine inositol monophosphatase; Ki: 0.19-0.42 μM. 10x potency vs. mouse/rat IMPase.</p>Formule :C8H12O8P2Couleur et forme :SolidMasse moléculaire :298.123-Methylcrotonylglycine
CAS :<p>3-Methylcrotonylglycine is an acyl glycine, a normal amino acid metabolite found in urine.</p>Formule :C7H11NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :157.17Golgicide A-2
CAS :<p>GCA-2 is a potent enantiomer of GCA, selectively and efficiently kills An. stephensi larvae, useful for dengue research.</p>Formule :C17H14F2N2Couleur et forme :SolidMasse moléculaire :284.31Deoxypseudouridine
CAS :<p>Deoxypseudouridine is a nucleotide analog.</p>Formule :C9H12N2O5Couleur et forme :SolidMasse moléculaire :228.2TD-106
CAS :<p>TD-106 is a modulator of cereblon (CRBN), and can be used for targeted protein degradation. BRD4 PROTACs with TD-106 induce BRD4 degradation.</p>Formule :C12H11N5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :273.25HT-2 Toxin
CAS :<p>HT-2 Toxin, a deacetylated metabolite of T-2 toxin, impairs protein synthesis and hinders cell proliferation in plants.</p>Formule :C22H32O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :424.49(S,S)-Valifenalate
CAS :<p>(S,S)-Valifenalate is an acylamino acid fungicide and is used to control a wide range of fungi belonging to the class of Oomycetes.</p>Formule :C19H27ClN2O5Couleur et forme :SolidMasse moléculaire :398.88Phosal 50 PG
CAS :<p>Phosal 50 PG is a co-solvent used as an emulsifier and stabilizer in the pharmaceutical and cosmetic industries.Phosal 50 PG is used as a dietary supplement.</p>Degré de pureté :98%Couleur et forme :SolidAniline-2,4-diphosphonic acid tetraethyl ester;
CAS :<p>Intermediates and building blocks - phosphorous compounds; nucleophile</p>Formule :C14H25NO6P2Couleur et forme :SolidMasse moléculaire :365.3Ceritinib D7
CAS :<p>Ceritinib D7 (LDK378 D7) is a deuterium-labeled Ceritinib. Ceritinib is an ATP-competitive inhibitor of ALK tyrosine kinase.</p>Formule :C28H36ClN5O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :565.184',5'-Dibromofluorescein
CAS :<p>4',5'-Dibromofluorescein (Eosinic acid) is a fluorescent dye that can be used as a ligand for protein characterization by spectroscopic analysis.</p>Formule :C20H10Br2O5Couleur et forme :Orange Solid PowderMasse moléculaire :490.10SIRT-IN-3
CAS :<p>SIRT-IN-3: potent SIRT1 inhibitor (IC50=17μM), 4x selective over SIRT2, 14x over SIRT3 (IC50s: 74μM & 235μM).</p>Formule :C13H12N2OCouleur et forme :SolidMasse moléculaire :212.25N-Octylmaleimide
CAS :<p>N-Octylmaleimide is an alkylmaleimide, which can inhibit rat liver glucose 6-phosphatase.</p>Formule :C12H19NO2Couleur et forme :SolidMasse moléculaire :209.28PDK1-IN-RS2
CAS :<p>PDK1-IN-RS2, a PIFtide mimic, selectively inhibits PDK1, blocking S6K1 activation (Kd: 9 μM).</p>Formule :C15H9ClN2O2S3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :380.89STING agonist-23
CAS :<p>CF502 (STING agonist-23) is a non-nucleotide that activates STING pathway, boosts immune responses, and shows activity against SARS-CoV.</p>Formule :C33H35N13O4Couleur et forme :SolidMasse moléculaire :677.72Cysteinylglycine TFA
CAS :<p>Cysteinylglycine TFA is an endogenous metabolite. It is used in disease diagnosis.</p>Formule :C7H11F3N2O5SCouleur et forme :SolidMasse moléculaire :292.23Muzolimine
CAS :<p>Muzolimine: a long-acting, high-capacity diuretic for kidney failure/hypertension; withdrawn due to serious neurological side effects.</p>Formule :C11H11Cl2N3OCouleur et forme :SolidMasse moléculaire :272.132-Nitrosopyridine
CAS :<p>2-Nitrosopyridine: used in antibiotic synthesis, Click/Diels-Alder reactions, excellent dienophile.</p>Formule :C5H4N2OCouleur et forme :SolidMasse moléculaire :108.1(Rac)-Rotigotine hydrochloride
CAS :<p>(Rac)-Rotigotine hydrochloride is a racemate of Rotigotine. Rotigotine is a full agonist of dopamine receptor, a partial the 5-HT1A receptor agonist.</p>Formule :C19H26ClNOSCouleur et forme :SolidMasse moléculaire :351.93Canagliflozin-d4
CAS :<p>Canagliflozin D4 is a deuterium-labeled Canagliflozin. Canagliflozin is an SGLT2 inhibitor.</p>Formule :C24H25FO5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :448.54GRK2 Inhibitor
CAS :<p>GRK2 Inhibitor is an inhibitor of β-Adrenergic Receptor Kinase 1 (β ARK1).</p>Formule :C12H9NO6Couleur et forme :SolidMasse moléculaire :263.2Loviride
CAS :<p>Loviride, a reverse transcriptase inhibitor with IC50 of 0.3 μM, blocks HIV-1/2 and SIV in MT-4 cells.</p>Formule :C17H16Cl2N2O2Couleur et forme :SolidMasse moléculaire :351.23Metrizoic acid
CAS :<p>Metrizoic acid is an ionic contrast medium. Metrizoic acid displays high osmolality and has a risk of inducing allergic reactions.</p>Formule :C12H11I3N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :627.9402PIH
CAS :<p>PIH inhibits ciliogenesis by destabilizing microtubules and blocking Hh signaling, hindering cilia formation and alpha-tubulin disassembly.</p>Formule :C20H19N5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :361.46Golgicide A-1
CAS :<p>Golgicide A-1 (GCA-1) is a moderately potent cis-diastereomer variant of Golgicide A (GCA) specifically designed to inhibit mosquito reproduction.</p>Formule :C17H14F2N2Couleur et forme :SolidMasse moléculaire :284.313,5-Diphenyl pyridine
CAS :<p>Heterocyclic compounds-pyridine,</p>Formule :C17H13NCouleur et forme :SolidMasse moléculaire :231.29Decyl-TPP bromide
CAS :<p>Decyl-TPP bromide ((1-Decyl)triphenylphosphonium bromide) may be used as an intermediate for chemical synthesis and an inactive control or as a reference to</p>Formule :C28H36BrPDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :483.46Rosmanol
CAS :<p>Rosmanol has antioxidant, anti-inflammatory, CNS effects; induces apoptosis in cancer cells; modulates GABAA receptors.</p>Formule :C20H26O5Degré de pureté :98.82% - 99.79%Couleur et forme :SolidMasse moléculaire :346.424-Hydroxy-6-methylcoumarin
CAS :<p>4-Hydroxy-6-methylcoumarin (4-HMC) is a naturally occurring phenolic compound, a derivative of coumarin, found in a variety of plants, fungi, and bacteria. It has anti-inflammatory and anti-tumor activity.4-HMC is used as a flavoring agent, preservative and antioxidant in the food industry.</p>Formule :C10H8O3Degré de pureté :99.95%Couleur et forme :White PowderMasse moléculaire :176.17Ethyl 4-hydroxyphenylacetate
CAS :<p>Ethyl 4-hydroxyphenylacetate is a selective inhibitor of monoamine oxidase A.</p>Formule :C10H12O3Degré de pureté :99.89%Couleur et forme :Slightly Yellow LiquidMasse moléculaire :180.2Ref: TM-FR12415
Produit arrêtéPamoic acid
CAS :<p>Pamoic acid is the orphan G protein-coupled receptor GPR35 agonist. Pamoic acid activates ERK and beta-arrestin2 and causes antinociceptive activity.</p>Formule :C23H16O6Degré de pureté :99.99%Couleur et forme :Fine Yellow PowderMasse moléculaire :388.37TFLLR-NH2 2TFA(197794-83-5(free base))
<p>TFLLR-NH2 2TFA(197794-83-5(free base)) is an agonist of PAR1 (EC50 :1.9 μM).</p>Formule :C35H55F6N9O10Degré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :875.87Tropinone
CAS :<p>Tropinone used as an intermediate in the synthesis of atropine sulfate, and is a decane alkaloid.</p>Formule :C8H13NODegré de pureté :99.90%Couleur et forme :Beige To Brown Crystalline PowderMasse moléculaire :139.1910Z-Nonadecenoic acid
CAS :<p>10Z-Nonadecenoic acid is a long-chain fatty acid with anti-tumor activity.</p>Formule :C19H36O2Degré de pureté :99.43%Couleur et forme :SolidMasse moléculaire :296.49Isonicotinic acid
CAS :<p>Isonicotinic acid is a metabolite of Isoniazid.Isonicotinic acid is a useful isomer of nicotinic acid. Isoniazid is converted to Isonicotinic acid by hydrazinolysis, with the biotransformation also to be catalyzed by cytochrome P450 enzymes, such as CYP2C.</p>Formule :C6H5NO2Degré de pureté :99.68%Couleur et forme :White To Off-White Crystalline SolidMasse moléculaire :123.114-Hydroxybenzyl cyanide
CAS :<p>4-Hydroxybenzyl cyanide (4-Hydroxyphenylacetonitrile) shows strong antioxidative activity.</p>Formule :C8H7NODegré de pureté :98.13%Couleur et forme :Light Brown SolidMasse moléculaire :133.154-Methoxycoumarine
CAS :<p>4-Methoxycoumarine has antitumour effects.</p>Formule :C10H8O3Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :176.17Sculponeatin O
CAS :<p>Sculponeatin O may have protective effects on the lipid peroxidation-damaged live cells.</p>Formule :C28H40O4Degré de pureté :95.00%Couleur et forme :SolidMasse moléculaire :440.61Lupinine
CAS :<p>Lupinine is an alkaloid capable of counteracting ethanol anesthesia. Lupinine is an AChE and BChE inhibitor and potential CD69 activator found in species of Loranthus, Calia, and Lupinus. It may also inhibit heparin.</p>Formule :C10H19NODegré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :169.26Ref: TM-FR16605
Produit arrêté2-Methyl-5-HT hydrochloride
CAS :<p>2-Methyl-5-HT hydrochloride (2-Methyl-5-hydroxytryptamine) is a potent and selective 5-HT3 receptor agonist with anti-depressive-like effects.</p>Formule :C11H15ClN2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :226.7NLX-204 hydrochloride(2170405-10-2 free base)
<p>NLX-204 hydrochloride is a potent and selective ERK1/2 phosphorylation-preferring serotonin 5 HT1A receptor agonist(pKi = 10.19).</p>Formule :C20H23Cl2F2N3O2Degré de pureté :99.59%Couleur et forme :SolidMasse moléculaire :446.32Coumaran
CAS :<p>Coumaran (2,3-Dihydrobenzofuran) is an acetylcholinesterase (AChE) inhibitor isolated from leaves of L. camara. Coumaran(2,3-Dihydrobenzofuran) can be used as a biopesticide. 2,3-dihydrobenzofuran is a member of the class of 1-benzofurans that is the 2,3-dihydroderivative of benzofuran. It has a role as a metabolite.</p>Formule :C8H8ODegré de pureté :99.61%Couleur et forme :LiquidMasse moléculaire :120.15CTB
CAS :<p>CTB (Cholera Toxin B subunit) is an activator of p300 histone acetyltransferase and induces apoptosis in MCF-7 cells.</p>Formule :C16H13ClF3NO2Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :343.73L-(+)-Abrine
CAS :<p>L-(+)-Abrine (L-N-Methyltryptophan) is a toxic protein found in the jequirity seed.,can be used as a biomarker for abrin exposure.</p>Formule :C12H14N2O2Degré de pureté :98.71% - ≥95%Couleur et forme :White PowderMasse moléculaire :218.25Elamipretide 2TFA
CAS :<p>Elamipretide 2TFA (RX-31 2TFA) is a novel mitochondrion-targeted antioxidant.</p>Formule :C36H51F6N9O9Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :867.84AM-2232
CAS :<p>AM-2232 (UNII-40KCH8YIKP) is a potent and unselective agonist of the cannabinoid receptors.</p>Formule :C24H20N2ODegré de pureté :99.37%Couleur et forme :SolidMasse moléculaire :352.43Dimethylamine hydrochloride
CAS :<p>Dimethylamine hydrochloride, found in urine, comes from food compound TMAO and NO synthesis inhibitor ADMA, processed by DDAH enzyme.</p>Formule :C2H8ClNDegré de pureté :98% - 99.89%Couleur et forme :White Solid CrystallineMasse moléculaire :81.54MTP 131 acetate
CAS :<p>MTP 131 (acetate) is a small mitochondrially-targeted tetrapeptide.</p>Formule :C34H53N9O7Degré de pureté :99.9%Couleur et forme :SolidMasse moléculaire :699.84Ref: TM-T35689
Produit arrêté7-Methoxy-1-tetralone
CAS :<p>7-Methoxy-1-tetralone may have insecticidal activity.</p>Formule :C11H12O2Degré de pureté :99.93%Couleur et forme :White CrystalMasse moléculaire :176.21Elamipretide
CAS :<p>Elamipretide (SS-31, MTP-131, Bendavia) is a mitochondria-focused peptide that curbs toxic ROS and stabilizes cardiolipin.</p>Formule :C32H49N9O5Degré de pureté :98.53% - 99.85%Couleur et forme :SolidMasse moléculaire :639.79Ref: TM-TP1095
Produit arrêtéDanoprevir sodium
CAS :<p>Danoprevir sodium is an NS3/4A protease inhibitor used in the treatment of Hepatitis C</p>Formule :C35H45FN5NaO9SCouleur et forme :SolidMasse moléculaire :753.82Elamipretide Triacetate
CAS :<p>Elamipretide TriTFA, a tetrapeptide, targets mitochondria, associates with cardiolipin, studied for treating Leber's Optic Neuropathy.</p>Formule :C38H61N9O11Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :819.94Ref: TM-T8644
Produit arrêtép-Toluic Acid
CAS :<p>p-Toluic Acid (4-Methylbenzoic acid) belongs to the class of organic compounds known as benzoic acids. 4-Methylbenzoic acid has been primarily detected in saliva. Within the cell, 4-methylbenzoic acid is primarily located in the cytoplasm.</p>Formule :C8H8O2Degré de pureté :99.44%Couleur et forme :Physical Description White Powder Sublimes (Ntp 1992)Masse moléculaire :136.15SR17018
CAS :<p>SR17018 is an mu-opioid-receptor (MOR) agonist, binding with GTPγS, with an EC50 of 97 nM.</p>Formule :C19H18Cl3N3ODegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :410.72Cebranopadol
CAS :<p>Cebranopadol (GRT6005) is an analgesic NOP and opioid receptor agonist with Kis of 0.9 nM, 0.7 nM, 2.6 nM, 18 nM for human NOP, μ-opioid (MOP), κ-opioid (KOP)</p>Formule :C24H27FN2ODegré de pureté :98.32% - 99.78%Couleur et forme :SolidMasse moléculaire :378.48Compound T69202(SC)
CAS :<p>NBQX (FG9202), an AMPA/kainate receptor blocker, counters glutamate toxicity; water-soluble as disodium salt, has anticonvulsant properties.</p>Formule :C12H6N4Na2O6SCouleur et forme :SolidMasse moléculaire :380.2415SR-4370
CAS :<p>SR-4370 is an HDAC inhibitor. SR- 4370 exhibited IC50 values of 0.5 μM, 0.1 μM and 0.06 μM towards HDAC1, HDAC2 and HDAC3, resp.</p>Formule :C17H18F2N2ODegré de pureté :99.50%Couleur et forme :SolidMasse moléculaire :304.33Oxindole
CAS :<p>Oxindole (Indolin-2-one) is an aromatic heterocyclic building block. 2-indolinone derivatives have become lead compounds in the research of kinase inhibitors.Oxindole structure has been used in receptor tyrosine kinases (RTKs) inhibitors such as SU4984 and intedanib, the RTK family represents an important therapeutic target for anti-cancer drug development.</p>Formule :C8H7NODegré de pureté :99.34%Couleur et forme :Off-White Crystalline PowderMasse moléculaire :133.15Desidustat
CAS :<p>Desidustat is an inhibitor of HIF hydroxylase.</p>Formule :C16H16N2O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :332.31Ref: TM-T5176
Produit arrêtéIGFBP-1 Protein, Rat, Recombinant
<p>IGF-binding proteins prolong the half-life of the IGFs and have been shown to either inhibit or stimulate the growth promoting effects of the IGFs on cell culture. They alter the interaction of IGFs with their cell surface receptors. Promotes cell migration. IGFBP-1 Protein, Rat, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 26.9 kDa and the accession number is P21743.</p>Masse moléculaire :26.9 kDa (predicted)COR-001
CAS :<p>Ziltivekimab (COR-001) is a human IL-6 antibody, lowers CRP, and may treat inflammation and heart issues in CKD.</p>Degré de pureté :95%Couleur et forme :Odour LiquidARGX-112
CAS :<p>Temtokibart is a humanized IgG1 λ2 antibody that specifically targets IL22RA1, and is expressed by cells that are deficient in the glutamine synthetase gene.</p>Couleur et forme :Odour LiquidOkadaic acid
CAS :<p>Okadaic acid, a polyether marine toxin, is a highly potent and selective protein phosphatase (PP) inhibitor.</p>Formule :C44H68O13Degré de pureté :98%Couleur et forme :White Crystals Or PowderMasse moléculaire :805Fotemustine
CAS :<p>Fotemustine: antineoplastic, chloroethylates DNA, blocks synthesis, causes cell arrest/apoptosis, lipophilic, crosses blood-brain barrier.</p>Formule :C9H19ClN3O5PCouleur et forme :SolidMasse moléculaire :315.69Benzovindiflupyr
CAS :<p>Benzovindiflupyr: a fungicide that inhibits SDH (IC50=5.2nM), halts S. sclerotiorum growth (EC50=0.011μg/ml), and protects crops like eggplants.</p>Formule :C18H15Cl2F2N3OCouleur et forme :SolidMasse moléculaire :398.23BET-IN-15
CAS :<p>BET-IN-15 (compound 1) is a potent, orally active inhibitor of BET, demonstrating inhibitory IC50 values of 0.64 nM for BRD4-BD1 and 0.25 nM for BRD4-BD2.</p>Formule :C21H18F2N4O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :444.45PAD4-IN-2
CAS :<p>PAD4-IN-2 (compound 5i) is a PAD4 inhibitor with an IC50 value of 1.94 μM, shown to suppress tumor growth in mice through specific inhibition of the PAD4-H3cit-</p>Formule :C20H23BClN7O6Couleur et forme :SolidMasse moléculaire :503.7Aminobutane bisphosphonate
CAS :<p>Aminobutane bisphosphonate curbs bone loss; may manage hypercalcemia in cancer.</p>Formule :C4H13NO6P2Couleur et forme :SolidMasse moléculaire :233.1PPARγ-IN-2
CAS :<p>"PPARγ-IN-2 (Compound 5a), a PPARγ inhibitor, exhibits an EC50 of 0.106 μM in inhibiting TG accumulation in 3T3-L1 preadipocytes.</p>Formule :C19H21N5ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :335.4Fostedil
CAS :<p>Fostedil enhances heart function, maintains blood flow during partial/total coronary occlusions, and lowers aortic pressure.</p>Formule :C18H20NO3PSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :361.4PKUMDL-LTQ-301
CAS :<p>PKUMDL-LTQ-301 is a potent inhibitor of HipA toxin. PKUMDL-LTQ-301 also inhibits E. coli persistence.</p>Formule :C30H28N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :480.55CGP 44532
CAS :<p>CGP 44532 a GABAB receptor agonist.</p>Formule :C4H12NO3PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :153.12Pazinaclone
CAS :<p>Pazinaclone is a non-benzodiazepine (GABAA) partial agonist with sedative and anxiolytic activity.</p>Formule :C25H23ClN4O4Degré de pureté :97.79% - 99.07%Couleur et forme :SolidMasse moléculaire :478.93Lp-PLA2-IN-15
CAS :<p>Lp-PLA2-IN-15 (example 2) is an inhibitor of lipoprotein-associated phospholipase A2 (Lp-PLA2) with potential application in Alzheimer's disease research [1].</p>Formule :C22H17F5N4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :480.39SR14150
CAS :<p>SR14150 is a partial agonist of high-affinity NOP receptor.</p>Formule :C21H30N2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :326.48Neurokinin antagonist 1
CAS :<p>Neurokinin antagonist 1 is a potent is a neuropeptide antagonist that can be used to study neurological disorders.</p>Formule :C38H40N4O3Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :600.75IDX-375
CAS :<p>IDX-375, a HCV NS5B polymerase inhibitor, is used potentially for the treatment of HCV infection.</p>Formule :C29H50N5O7PSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :643.78MEN11467
CAS :<p>MEN11467 is a novel, orally available, potent and selective peptidomimetic tachykinin NK 1 receptor antagonist for the study of acute colon cancer.</p>Formule :C38H40N4O3Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :600.75Phenazolam
CAS :<p>Phenazolam is an analytical reference standard categorized as a benzodiazepine. [1] This product is intended for research and forensic applications.</p>Formule :C17H12BrClN4Couleur et forme :SolidMasse moléculaire :387.66AKOS-22
CAS :<p>AKOS-22: potent VDAC1 inhibitor, Kd=15.4 μM; prevents mitochondrial dysfunction and apoptosis.</p>Formule :C22H21ClF3N3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :467.87UBP1112
CAS :<p>group III mGlu receptor antagonist</p>Formule :C10H14NO5PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :259.2Fosfonet sodium
CAS :<p>Fosfonet sodium is a sodium salt of phosphonoacetic acid, effective against herpesviruses by inhibiting viral DNA polymerase.</p>Formule :C2H4NaO5PCouleur et forme :SolidMasse moléculaire :162.01Gacyclidine
CAS :<p>Gacyclidine (OTO311), an NMDA receptor blocker, treats tinnitus and injuries in the brain and spinal cord.</p>Formule :C16H25NSDegré de pureté :99.85% - 99.92%Couleur et forme :SolidMasse moléculaire :263.44D(-)-Octopamine CSA salt
CAS :<p>D(-)-Octopamine CSA salt is an agonist of octopamine receptors.</p>Formule :C18H27NO6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :385.48HBV-IN-34
CAS :<p>HBV-IN-34 (compound 17i) is a potent inhibitor of HBsAg production, demonstrating remarkable in vitro anti-HBV efficacy with EC50 values of 0.018 μM for HBV DNA</p>Formule :C21H19F2N7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :407.42Questiomycin A derivatives 18 TFA
<p>Questiomycin A derivative 18 TFA exhibits antibacterial, anticancer properties and inhibits GRP78.</p>Formule :C16H12F3N3O5Degré de pureté :98.45%Couleur et forme :SoildMasse moléculaire :383.07Mavodelpar free base
CAS :<p>Mavodelpar free acid (REN001 free acid) is an selective agonist of PPARδ.</p>Formule :C31H30FNO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :515.57CH-100
CAS :<p>CH-100 is a Chinese herbal medicine previously used in the treatment of human hepatitis C.</p>Formule :C14H22ClNO3Couleur et forme :SolidMasse moléculaire :287.78(E)-Crotylbarbital
CAS :<p>(E)-Crotylbarbital, a Crotylbarbital isomer, is a sedative with hypnotic, anticonvulsant properties, aiding sleep and mental stability.</p>Formule :C10H14N2O3Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :210.23PL265
CAS :<p>PL265 is a long-acting dual ENKephalinase inhibitor (DENKi) with analgesic potential.</p>Formule :C27H35N2O9PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :562.55FM-24 HCl
CAS :<p>FM-24 HCl is a long acting beta-adrenergic receptor antagonist.</p>Formule :C19H30ClNO2Couleur et forme :SolidMasse moléculaire :339.9Radafaxine hydrochloride
CAS :<p>Radafaxine hydrochloride is an inhibitor of DAT and NET transporters, and nAChR family modulator.</p>Formule :C13H19Cl2NO2Degré de pureté :98%Masse moléculaire :292.2Glutaminyl Cyclase Inhibitor 4
CAS :<p>Glutaminyl Cyclase Inhibitor 4 is a potent, selective glutaminyl cyclase (QC) inhibitor (IC50: 6.1 nM). It is a potent anti-Alzheimer’s agent.</p>Formule :C22H33N5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :415.53SB251023
CAS :<p>SB251023 is an agonist of β3-adrenoceptor.</p>Formule :C28H34NO6PCouleur et forme :SolidMasse moléculaire :511.55YM 298198 Hydrochloride
CAS :<p>YM 298198 HCl: non-competitive mGlu1 antagonist, Ki=19 nM. Inactive on mGlu2-7, stronger than CPCCOEt.</p>Formule :C18H22N4OSCouleur et forme :SolidMasse moléculaire :342.46Trimetoquinol HCl hydrate
CAS :<p>Trimetoquinol hydrochloride possesses differential and selective beta-adrenergic properties.</p>Formule :C19H26ClNO6Couleur et forme :SolidMasse moléculaire :399.87FGFR1 inhibitor-10
CAS :<p>FGFR1 inhibitor-10 (Compound 4i), with an IC50 of 28 nM, effectively inhibits FGFR1 phosphorylation.</p>Formule :C26H30F3N7O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :561.62JAK2-IN-9
CAS :<p>Compound A8, known as JAK2-IN-9, is a selective JAK2 inhibitor with an IC50 of 5 nM.</p>Formule :C20H24N6O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :412.51PS372424 HCl
CAS :<p>PS372424 activates CXCR3, triggers ERK phosphorylation, and inhibits CXCL11's effect on CD45+ cell migration in humanized mice.</p>Formule :C33H45ClN6O4Couleur et forme :SolidMasse moléculaire :625.21MitoE10
CAS :<p>MitoE10 is an effective mitochondrial targeting antioxidant.</p>Formule :C42H55O5PSCouleur et forme :SolidMasse moléculaire :702.92Anti-NASH agent 1
CAS :<p>Anti-NASH Agent 1 (Compound 3d), derived from Elafibranor, serves as a strong PPAR-α/δ agonist aimed at treating nonalcoholic steatohepatitis (NASH).</p>Formule :C26H33NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :423.54DPX-3778
CAS :<p>DPX-3778, a triethanolamine salt, boosts tobacco callus growth 4-5x at 0.124-2.48 μM and slows aging with IAA and kinetin.</p>Formule :C16H23ClN4O6Couleur et forme :SolidMasse moléculaire :402.83Dioxifedrine
CAS :<p>Dioxifedrine is a beta-2 -adrenergic agonist with bronchodilator activity.</p>Formule :C10H15NO3Couleur et forme :SolidMasse moléculaire :197.23Oxitropium Bromide
CAS :<p>Oxitropium bromide, a mAChR blocker, treats asthma and COPD as an anticholinergic bronchodilator.</p>Formule :C19H26BrNO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :412.32(S)-Coriolic acid
CAS :<p>(S)-Coriolic acid, a 15-LOX metabolite and signaling molecule, modulates cell growth, tumor adhesion, receptor expression, and can cause mitochondrial damage.</p>Formule :C18H32O3Degré de pureté :97.67% - 98.04%Couleur et forme :SolidMasse moléculaire :296.44Cebranopadol ((1α,4α)stereoisomer)
CAS :<p>Cebranopadol ((1α,4α)stereoisomer) is a stereoisomer of cebranopadol which is a potent ORL-1 agonist.</p>Formule :C24H27FN2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :378.48EGFR-IN-82
CAS :<p>EGFR-IN-82 (Compound 8a) is a potent, orally active inhibitor of EGFR, exhibiting IC50 values of 0.09 nM for EGFR L858R/T790M/C797S and 0.06 nM for EGFR Del19/</p>Formule :C32H41BrN9O2PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :694.6ALPK1-IN-2
CAS :<p>ALPK1-IN-2 is a potent inhibitor of ALPK1 (α-kinase 1) (IC50: 95 nM). ALPK1-IN-2 inhibits NF-κB (IC50: 1.31 μM).</p>Formule :C20H18F2N4O2SCouleur et forme :SolidMasse moléculaire :416.44Saxitoxinol
CAS :<p>Saxitoxinol is an analog of saxitoxin, a known voltage-gated sodium channel blocker.</p>Formule :C10H17N7O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :283.29BChE-IN-17
CAS :<p>BChE-IN-17 (compound 6n) is a potent, selective inhibitor of butyrylcholinesterase (BChE), demonstrating inhibitory half-maximal inhibitory concentrations (</p>Formule :C23H23BrN2O4S2Couleur et forme :SolidMasse moléculaire :535.47Culmerciclib
CAS :<p>Culmerciclib is a cell cycle protein-dependent kinase (CDK) inhibitor that exhibits antitumour effects.</p>Formule :C24H27FN8Couleur et forme :SolidMasse moléculaire :446.52Ceronapril
CAS :<p>Ceronapril (SQ 29852) is an orally active and potent angiotensin-converting enzyme (ACE) inhibitor (IC50 : 36 nM) for the study of dementia and hypertension.</p>Formule :C21H33N2O6PDegré de pureté :97.94%Couleur et forme :SolidMasse moléculaire :440.47Lp-PLA2-IN-16
CAS :<p>Lp-PLA2-IN-16 (Example 1) is an inhibitor of lipoprotein-associated phospholipase A2 (Lp-PLA2) with potential applications in Alzheimer's disease research [1].</p>Formule :C22H17F5N4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :480.39Bromadoline maleate
CAS :<p>Bromadoline is an opioid analgesic selective for the μ-opioid receptor.</p>Formule :C19H25BrN2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :441.322Lp-PLA2-IN-12
CAS :<p>Lp-PLA2-IN-12 (compound 19), an Lp-PLA2 inhibitor, is utilized in researching neurodegenerative diseases including Alzheimer's disease (AD), glaucoma, age-</p>Formule :C24H23F2N5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :467.47KP372-1
CAS :<p>KP372-1, an Akt inhibitor, blocks PI3K signaling, arrests cell growth, and triggers apoptosis in head/neck squamous cell carcinoma.</p>Formule :C20H8N12O2Couleur et forme :SolidMasse moléculaire :448.36CXCR4-IN-1
CAS :<p>CXCR4-IN-1 (Example C5), with an IC50 of 20 nM, is a potent inhibitor of CXCR4, applicable for the research of various conditions such as cancer, HIV, diabetic</p>Formule :C23H32N6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :392.54Erythrityl Tetranitrate
CAS :<p>Erythrityl Tetranitrate, a vasodilator similar to nitroglycerin, was first in "sustained release" tablets; may cause "nitro headache."</p>Formule :C4H6N4O12Couleur et forme :SolidMasse moléculaire :302.11GR 218,231
CAS :<p>GR 218,231 is a selective antagonist of D3 dopamine receptor.</p>Formule :C24H33NO3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :415.59DprE1-IN-8
CAS :<p>DprE1-IN-8 is a potent inhibitor of DprE1, exhibiting an IC50 of less than 0.75 μM.</p>Formule :C19H12F3N5O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :463.39HPK1-IN-18
CAS :<p>HPK1-IN-18: Potent, specific inhibitor of HPK1, a MAP4K enzyme, for cancer research and treatment.</p>Formule :C24H24N4Couleur et forme :LiquidMasse moléculaire :368.47anti-TNBC agent-2
CAS :<p>Anti-TNBC agent-2 (3j), a purine derivative, acts as an anti-triple negative breast cancer (TNBC) therapeutic.</p>Formule :C28H37ClFN7ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :542.09ALPK1-IN-1
CAS :<p>ALPK1-IN-1 (A001) strongly inhibits ALPK1, key for innate immunity & NF-κB signaling via TIFA/TRAF.</p>Formule :C25H32N6O2SCouleur et forme :SolidMasse moléculaire :480.63CK176
CAS :<p>CK176 is an HIV-1 inhibitor, 11x more effective than I-XW-053 in human PBMCs.</p>Formule :C21H12IN3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :465.24AMPK activator C2
CAS :<p>AMPK activator C2 is an AMPK allosteric activator.</p>Formule :C7H6NO6PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :231.1Albuterol stearate
CAS :<p>Albuterol stearate, a salt form of Albuterol, is a selective beta2 agonist for treating asthma and COPD, with 29x preference for beta2 over beta1.</p>Formule :C31H57NO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :523.799PSB-6426
CAS :<p>PSB-6426 is the first potent and selective human nucleoside triphosphate diphosphohydrolase-2 inhibitor.</p>Formule :C22H29N4O10PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :540.46H 35-25
CAS :<p>H 35-25 is a beta 2-antagonist.</p>Formule :C13H21NOCouleur et forme :SolidMasse moléculaire :207.31anti-TNBC agent-3
CAS :<p>Anti-TNBC agent-3 (compound 3g) is a compound that induces apoptosis and possesses anti-cancer cell proliferation properties.</p>Formule :C29H39F2N7OCouleur et forme :SolidMasse moléculaire :539.66AEF0117
CAS :<p>AEF0117 is a signaling inhibitor of CB1-SSi that inhibits cannabinoid self-administration and can be used to study cannabis withdrawal.</p>Formule :C29H40O3Degré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :436.63Ref: TM-T79909
Produit arrêtéXilmenolone
CAS :<p>Xilmenolone acts as a positive allosteric modulator of the GABA_A receptor [1].</p>Formule :C26H37N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :423.59Azilsartan mepixetil potassium
CAS :<p>Azilsartan medoxomil potassium (QR-01019K), an angiotensin II receptor antagonist, exhibits a potent and sustained antihypertensive effect, along with a more</p>Formule :C36H33KN6O8Couleur et forme :SolidMasse moléculaire :716.78Antibacterial agent 157
CAS :<p>Compound B12 (Antibacterial agent 157) is a fungicidal agent that can impact protein synthesis in Botrytis cinerea.</p>Formule :C26H23BrF4N2O3Couleur et forme :SolidMasse moléculaire :567.37Bumetanide sodium
CAS :<p>Bumetanide sodium, a potent diuretic, blocks NKCC1 (IC50: 0.68 μM) and NKCC2 (IC50: 4.0 μM).</p>Formule :C17H19N2NaO5SCouleur et forme :SolidMasse moléculaire :386.4CGP 56999A
CAS :<p>CGP 56999A is a GABA(B) receptor antagonist; it boosts BDNF and reduces dopamine loss in rat striatum.</p>Formule :C19H30NO5PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :383.42And1-IN-1
CAS :<p>And1-IN-1, also known as compound III, is a potent inhibitor of And1 [1].</p>Formule :C15H11BCl2O2Couleur et forme :SolidMasse moléculaire :304.96VISTA-IN-2
CAS :<p>VISTA-IN-2 (Compound 1) is a V-domain Ig suppressor of T-cell activation (VISTA) inhibitor that promotes the degradation of VISTA in cells via autophagy,</p>Formule :C23H23N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :357.45BCR-ABL-IN-8
CAS :<p>BCR-ABL-IN-8 (compound 26f) is a BCR-ABL inhibitor featuring a trimethoxy group [1].</p>Formule :C30H33N7O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :571.63Davelizomib
CAS :<p>Davelizomib is a proteasome inhibitor that exhibits antineoplastic activity [1].</p>Formule :C21H26BF2N3O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :481.25TrkB-IN-1
CAS :<p>TrkB-IN-1 is a potent, orally active agonist of the TrkB receptor, with favorable pharmacokinetic (PK) properties.</p>Formule :C19H16N2O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :368.34Antitumor photosensitizer-1
CAS :<p>Antitumor Photosensitizer-1 (Compound 8) is a potent photosensitizer with remarkable photodynamic anti-tumor properties and minimal skin photo-toxicity,</p>Formule :C42H51N5O6Couleur et forme :SolidMasse moléculaire :721.88LT-540-717
CAS :<p>LT-540-717 (compound 32), a potent FLT3 inhibitor (IC50=0.62 nM), exhibits antiproliferative activity and effectively inhibits various acquired FLT3 mutations,</p>Formule :C24H24N8O2Couleur et forme :SolidMasse moléculaire :456.5JAK1-IN-11
CAS :<p>JAK1-IN-11 (compound 11) serves as a potent inhibitor of Janus kinases, exhibiting nanomolar inhibitory concentrations with IC50 values of 0.02 nM (JAK1) and 0.</p>Formule :C26H36N6O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :528.67Insecticidal agent 6
CAS :<p>Compound Im (Insecticidal agent 6) is a potent inhibitor of insect ryanodine receptors (RyRs), exhibiting an EC50 of 0.6308 µM against S.</p>Formule :C19H14BrCl2N5O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :527.16RIOK2-IN-2
CAS :<p>RIOK2-IN-2 (8) functions as an inhibitor of RIOK2, exhibiting IC50 values of 3.02 μM in MKN-1 cells and 5.34 μM in MOLT4 cells [1].</p>Formule :C27H23F3N6O2Couleur et forme :SolidMasse moléculaire :520.51LFS-1107
CAS :<p>LFS-1107, a reversible CRM1 inhibitor (Kd: 12.5 pM), selectively targets and eliminates ENKTL cells, offering potential for cancer research applications [1].</p>Formule :C12H11N5OS2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :305.38BET-IN-14
CAS :<p>BET-IN-14 is a pan BET inhibitor with an IC50 of 5.35 nM, demonstrating oral activity and anticancer properties [1].</p>Formule :C30H37N7O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :527.66Estrogen receptor modulator 8
CAS :<p>Estrogen Receptor Modulator 8 (compound 4) is an orally active inhibitor targeting Estrogen Receptor/ERR α with potent efficacy (IC50 = 0.437 nM in MCF-7 cells</p>Formule :C25H24F4N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :460.46Antibacterial agent 160
CAS :<p>Antibacterial Agent 160 is a potent antibacterial agent that rapidly eradicates bacteria and inhibits the formation of bacterial biofilms.</p>Formule :C29H27ClFN3O6Couleur et forme :SolidMasse moléculaire :567.99Bi-Mc-VC-PAB-MMAE
CAS :<p>Bi-Mc-VC-PAB-MMAE is an agent-linker conjugate for antibody-drug conjugates (ADCs), featuring the linker (Fmoc-Val-Cit-PAB) and the potent tubulin inhibitor (</p>Formule :C71H104N12O18Couleur et forme :SolidMasse moléculaire :1413.66DDO-2213
CAS :<p>DDO-2213 is a potent, orally active inhibitor of the WDR5-MLL1 interaction, demonstrating an IC50 of 29 nM and a Kd of 72.9 nM against WDR5.</p>Formule :C24H27ClFN7OCouleur et forme :SolidMasse moléculaire :483.97JAK1-IN-10
CAS :<p>JAK1-IN-10 (compound 9), a cyano-substituted cyclic hydrazine derivative, functions as a potent and selective inhibitor of JAK1 [1].</p>Formule :C15H17N7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :295.34MDL-811
CAS :<p>MDL-811, an allosteric activator of SIRT6, markedly enhances the deacetylation of histone H3 at lysine residues 9, 18, and 56 (H3K9Ac, H3K18Ac, and H3K56Ac),</p>Formule :C25H25BrCl2FN3O5S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :681.42IDO1-IN-22
CAS :<p>IDO1-IN-22 (Compound 3) is an inhibitor of IDO1, demonstrating potent activity with biochemical hIDO1 IC50 of 67.4 nM and HeLa hIDO1 IC50 of 17.6 nM.</p>Formule :C12H12BrFN6O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :387.16Syk-IN-8
CAS :<p>Syk-IN-8 (compound 19q) functions as a Syk inhibitor with demonstrated antiproliferative effects on a variety of hematological tumor cells.</p>Formule :C23H26N10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :442.52EST73502
CAS :<p>EST73502 is a compound that functions as a dual agonist for the μ-opioid receptor (MOR) and an antagonist for the σ1 receptor (σ1R). It is selective, orally active, and possesses the ability to penetrate the blood-brain barrier (BBB). The compound exhibits a Ki value of 64 nM for the MOR and 118 nM for the σ1R. Additionally, EST73502 demonstrates antinociceptive activity [1].</p>Formule :C19H26F2N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :352.426CIAC001
CAS :<p>CIAC001, a pyruvate kinase PKM2 inhibitor, exhibits anti-neuroinflammatory properties.</p>Formule :C20H25N3O2Couleur et forme :SolidMasse moléculaire :339.43BTK-IN-25
CAS :<p>BTK-IN-25 (compound 71) is a potent BTK inhibitor, demonstrating an IC50 of 0.77 nM against BTK(C481S) and achieving an IC50 of 1 nM in DOHH2 cells [1].</p>Formule :C28H27F2N3O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :523.53PI3Kδ-IN-13
CAS :<p>PI3Kδ-IN-13 (compound 89), with an IC50 value of 2.6 nM, is an inhibitor of PI3Kδ, applicable for researching diseases involving cell proliferation, including</p>Formule :C27H39N7O4S2Couleur et forme :SolidMasse moléculaire :589.77Mal-cyclohexane-Gly-Gly-Phe-Gly-Exatecan
CAS :<p>Mal-cyclohexane-Gly-Gly-Phe-Gly-Exatecan is a linker molecule employed in the synthesis of antibody-drug conjugates (ADCs), demonstrating potent antitumor</p>Formule :C55H60FN9O13Couleur et forme :SolidMasse moléculaire :1074.12JAK-IN-34
CAS :<p>JAK-IN-34 (compound 11n) is a potent inhibitor of Janus kinases (JAKs), demonstrating IC50 values of 0.40 nM for JAK1, 0.83 nM for JAK2, 2.10 nM for JAK3,</p>Formule :C27H26N6ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :450.53Sakura 6
CAS :<p>Sakura 6, a synthetic serotonin transporter (SERT)-binding peptide, enhances the interaction between SERT and neuronal nitric oxide synthase.</p>Formule :C31H45N5O7Couleur et forme :SolidMasse moléculaire :599.73S1P1 agonist 6
CAS :<p>Compound I (S1P1 agonist 6) is an S1P1 agonist that mitigates autoimmune activity by inhibiting lymphocyte trafficking and has potential as an immunosuppressive</p>Formule :C25H26F3NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :445.47LM2I
CAS :<p>LM2I, a derivative of Spinosyn A (SPA), serves both as an argininosuccinate synthase (ASS1) enzyme activator and a tumor inhibitor through direct interaction</p>Formule :C47H77N3O11Couleur et forme :SolidMasse moléculaire :860.13PF-05236216 hydrochloride
CAS :<p>PF-05236216 hydrochloride: Brain-penetrant, potent CK1δ/ε inhibitor affecting mouse circadian rhythms.</p>Formule :C18H15FN4OCouleur et forme :SolidMasse moléculaire :322.34Antitumor agent-104
CAS :<p>Antitumor Agent-104 (Compound 9) serves as an antineoplastic by impeding DNA repair mechanisms in tumor cells, primarily through the inhibition of PARP1 enzyme</p>Formule :C31H33FN6O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :556.63URAT1&XO inhibitor 1
CAS :<p>URAT1&XO Inhibitor 1 (compound 29) serves as a dual inhibitor with IC50 values of approximately 10 μM for URAT1 and 1.01 μM for Xanthine Oxidase.</p>Formule :C20H13N5O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :403.41ALPK1-IN-3
CAS :<p>ALPK1-IN-3,serves as an ALPK1 inhibitor that dampens proinflammatory gene expression in the kidney and enhances survival in animal models of sepsis-induced</p>Formule :C20H16F2N4OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :398.43Tibremciclib
CAS :<p>Tibremciclib is a cyclin-dependent kinase 4 (CDK4) inhibitor that exhibits antineoplastic properties [1].</p>Formule :C28H32F2N8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :518.6FOXM1-IN-2
CAS :<p>FOXM1-IN-2, a FOXM1 inhibitor, exhibits antineoplastic activity [1].</p>Formule :C48H47F4N7O12SCouleur et forme :SolidMasse moléculaire :1021.99ROCK2-IN-6
CAS :<p>ROCK2-IN-6 (Comp A) is a selective inhibitor of ROCK2, applicable in the study and treatment of ROCK-mediated, autoimmune, and inflammatory diseases [1].</p>Formule :C26H21F2N7ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :485.49BBDDL2059
CAS :<p>BBDDL2059 is a selective covalent inhibitor targeting EZH2, exhibiting an IC50 of 1.5 nM against the EZH2-Y641F mutant.</p>Formule :C27H36N4O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :512.66Canlitinib
CAS :<p>Canlitinib, a tyrosine kinase inhibitor, holds potential for cancer research.</p>Formule :C33H31F2N3O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :619.61ATR-IN-24
CAS :<p>ATR-IN-24 (Compound 1) is an ATR inhibitor with demonstrated anticancer activity [1].</p>Formule :C23H26N6O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :418.49Lerzeparib
CAS :<p>Lerzeparib is a PARP (ADP-ribose polymerase) inhibitor that exhibits antineoplastic activity [1].</p>Formule :C21H20FN3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :365.4diMal-O-CH2COOH
CAS :<p>DiMal-O-CH2COOH is a cleavable linker utilized in antibody-drug conjugates (ADCs).</p>Formule :C13H12N2O7Couleur et forme :SolidMasse moléculaire :308.24FAP-IN-2
CAS :<p>FAP-IN-2 is a 99mTc-labeled, isonitrile-containing derivative of a fibroblast activation protein (FAPI) inhibitor suitable for tumor imaging [1].</p>Formule :C24H28F2N6O3Couleur et forme :SolidMasse moléculaire :486.51Immune cell migration-IN-1
CAS :<p>Immune cell migration-IN-1 (compound 2) serves as a potent inhibitor of immune cell migration, with potential research applications for mitigating conditions</p>Formule :C30H25ClN4O6SCouleur et forme :SolidMasse moléculaire :605.06Py-MAA-Val-Cit-PAB-MMAE
CAS :<p>Py-MAA-Val-Cit-PAB-MMAE (AAJ8D6-PY-Val-Cit-MMAE) serves as an ADC linker for Zapadcine-3a, a broad-spectrum anti-TRAILR2 ADC with antineoplastic properties.</p>Formule :C72H111N13O16SCouleur et forme :SolidMasse moléculaire :1446.79SARS-CoV-2-IN-68
CAS :<p>SARS-CoV-2-IN-68 (compound 6C) is a covalent inhibitor of both SARS-CoV-2 PLpro and Mpro, exhibiting potent antiviral properties by targeting the Zn-finger</p>Formule :C14H12N2OSeDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :303.22JDB175
CAS :<p>JDB175, a selective BTK inhibitor with oral bioavailability, demonstrates excellent penetration through the blood-brain barrier.</p>Formule :C26H21F3N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :478.47STAT3-IN-18
CAS :<p>STAT3-IN-18 (compound SPP), a platinum (IV) complex featuring an axial ligand from sandalwood, suppresses the JAK2-STAT3 pathway in breast cancer (BC) cells and</p>Formule :C18H24Cl2N2O6PtDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :630.38DPP
CAS :<p>DPP, a Platinum(IV) complex with a pterostilbene-derived axial ligand, inhibits the JAK2-STAT3 pathway in breast cancer (BC) cells, demonstrating</p>Formule :C36H40Cl2N2O10PtDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :926.7YK-029A
CAS :<p>YK-029A, an orally active EGFR mutant inhibitor, targets both EGFR T790M and EGFRex20ins mutations.</p>Formule :C27H32N8O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :500.6JAK-IN-27
CAS :<p>JAK-IN-27, also known as compound 1, is an orally active, potent inhibitor of the JAKS family kinases, displaying inhibitory concentrations (IC50s) of 3.0 nM</p>Formule :C20H21F2N7ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :413.42L 689037
CAS :<p>L 689037 is an inhibitor of leukotriene biosynthesis.</p>Formule :C36H37ClN2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :597.14VMAT2-IN-2 tosylate
CAS :<p>VMAT2-IN-2 tosylate is a potent inhibitor of VMAT2 and is applicable in the research of tardive dyskinesia [1].</p>Formule :C27H36F3NO6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :559.64IDO/Tubulin-IN-2
CAS :<p>IDO/Tubulin-IN-2 inhibits TDO/tubulin, effective on U87, HepG2, A549, HCT-116, LO2 cancer cells; IC50 values 0.036-1.04 μM, boosts antitumor action.</p>Formule :C48H40N6O10Couleur et forme :SolidMasse moléculaire :860.87(αR)-Cyclopropaneacetamide-Exatecan
CAS :<p>(αR)-Cyclopropaneacetamide-Exatecan (compound 2-A), an Exenotecan derivative, serves as a cytotoxic agent that effectively inhibits the proliferation of U87MG</p>Formule :C29H28FN3O6Couleur et forme :SolidMasse moléculaire :533.55Yhhu6669
CAS :<p>Yhhu6669 is an anti-HBV agent that suppresses viral DNA and replication by promoting DNA-free capsid assembly, effectively reducing HBV DNA and HBcAg levels in</p>Formule :C29H28ClFN6O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :563.02HPK1-IN-38
CAS :<p>HPK1-IN-38 (compound 15) is an inhibitor of MAP4K1/HPK1, suitable for research into disorders related to HPK1 [1].</p>Formule :C29H29N5O3Couleur et forme :SolidMasse moléculaire :495.57MOR agonist-1
CAS :<p>MOR Agonist-1 is a μ-opioid receptor (MOR) agonist noted for its potent analgesic properties and is utilized in research concerning pain and associated</p>Formule :C22H26ClFN2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :404.91MDVN1003
CAS :<p>MDVN1003 inhibits BTK & PI3Kδ in B cells, blocking NHL growth; it kills lymphoma cells, not erythroblasts.</p>Formule :C22H20FN7ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :417.44APG-2449
CAS :<p>APG-2449 is an orally active inhibitor targeting ALK, ROS1, and FAK, demonstrating antitumor efficacy in mouse models of non-small cell lung cancer (NSCLC) [1].</p>Formule :C33H42ClN5O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :640.24URAT1 inhibitor 5
CAS :<p>URAT1 Inhibitor 5 (compound 16) serves as a powerful inhibitor of URAT1 and is utilized in hyperuricemia research [1].</p>Formule :C18H14BrN3O2SCouleur et forme :SolidMasse moléculaire :416.29HBV-IN-38
CAS :<p>HBV-IN-38 (Example 193), an HBV DNA inhibitor with an EC50 value of ≤100 nM, serves as a research tool for investigating viral infections [1].</p>Formule :C18H16F3N5O4S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :487.48Tauro-Obeticholic Acid sodium
CAS :<p>Tauro-obeticholic acid, a farnesoid X receptor (FXR) agonist and semisynthetic derivative of chenodeoxycholic acid, is an active metabolite of obeticholic acid.</p>Formule :C28H48NO6S·NaCouleur et forme :SolidMasse moléculaire :549.74
