
Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.782 produits)
- Apoptose(6.263 produits)
- Cycle cellulaire/point de contrôle(4.792 produits)
- Chromatine/Épigénétique(2.441 produits)
- Signalisation du cytosquelette(1.528 produits)
- Altération de l'ADN/réparation de l'ADN(2.965 produits)
- Endocrinologie/Hormones(3.707 produits)
- Enzyme(3.667 produits)
- GPCR/G-Protéine(9.009 produits)
- Immunologie et Inflammation(3.875 produits)
- Virus de la grippe(301 produits)
- Signalisation JAK/STAT(414 produits)
- Signalisation MAPK(1.248 produits)
- Transporteur membranaire/Canal ionique(3.033 produits)
- Métabolisme(10.209 produits)
- Microbiologie/Virologie(7.592 produits)
- Neuroscience(10.381 produits)
- Autres inhibiteurs(36.040 produits)
- Oxydation-Réduction(42 produits)
- Signalisation PI3K/Akt/mTOR(1.442 produits)
- Protéases/Protéasome(1.724 produits)
- Cellules souche et Dérivés(826 produits)
- Tyrosine Kinase/Adaptateurs(2.035 produits)
- Ubiquitination(1.717 produits)
Affichez 16 plus de sous-catégories
66683 produits trouvés pour "Inhibiteurs"
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Citalopram hydrobromide
CAS :Citalopram hydrobromide (XU-62-320) , a selective serotonin reuptake inhibitor (SSRI), selectively inhibits the CNS neuronal reuptake of serotonin, therebyFormule :C20H22BrFN2ODegré de pureté :99.81%Couleur et forme :White Crystalline PowderMasse moléculaire :405.304Ascaridole
CAS :Ascaridole (NSC-406266) acts as an anthelmintic compound that repels parasitic helminths (worms) in humans and plants and has weak antimalarial activity.Formule :C10H16O2Degré de pureté :99.82% - 99.93%Couleur et forme :SolidMasse moléculaire :168.23Sabatolimab
CAS :Sabatolimab (MBG453) is a humanized IgG4 antibody that inhibits TIM-3 to modulate immunity and shows promise as an immunosuppressant.Degré de pureté :> 95% - > 95%Couleur et forme :LiquidMasse moléculaire :145 kDa (average)BJJF078
CAS :BJJF078, an aminopiperidine, inhibits human/mouse TG2 (IC50: 41/54 nM) and TG1 (IC50: 0.16 μM), may be used in MS studies.Formule :C27H29N3O6SDegré de pureté :99.56%Couleur et forme :SoildMasse moléculaire :523.6Lin28-let-7a antagonist 1
CAS :Lin28-let-7a antagonist 1, with an IC50 of 4.03 μM for Lin28A-let-7a-1 interaction,and shows a clear antagonistic effect against the Lin28-let-7a interaction.Formule :C31H29N5O7Degré de pureté :99.44%Couleur et forme :SolidMasse moléculaire :583.59Ref: TM-T11851
1mg92,00€5mg216,00€10mg329,00€25mg593,00€50mg893,00€100mg1.311,00€1mL*10mM (DMSO)281,00€L-Cycloserine
CAS :L-Cycloserine irreversibly inhibits E. coli GABA aminotransferase, raising GABA levels, an inhibitory neurotransmitter.Formule :C3H6N2O2Degré de pureté :99.75% - 99.99%Couleur et forme :Crystals White PowderMasse moléculaire :102.09(R)-AZD 9639
CAS :(R)-AZD 9639 is the R-isomer of AZD 9639, a novel respiratory syncytial virus (RSV) fusion inhibitor with antiviral activity.Formule :C21H15ClN4O2Degré de pureté :99.48% - 99.64%Couleur et forme :SoildMasse moléculaire :390.823-Hydroxykynurenamine Dihydrochloride
<p>3-Hydroxykynurenamine HCl (3-OH-Kynurenamine HCl) is an immunomodulatory biogenic amine that induces and promotes cell death.</p>Formule :C9H14Cl2N2O2Degré de pureté :99.53% - 99.69%Couleur et forme :SolidMasse moléculaire :252.04Antiarol
CAS :Antiarol (3,4,5-trimethoxyphenol) is a member of aromatic phenols and exhibits moderate DPPH free radical scavenging activity.Formule :C9H12O4Degré de pureté :99.61%Couleur et forme :Slightly Brown PowderMasse moléculaire :184.19Articaine hydrochloride
CAS :Articaine hydrochloride (Hoe-045) is a thiophene-containing local anesthetic pharmacologically similar to MEPIVACAINE.Formule :C13H21ClN2O3SDegré de pureté :99.76%Couleur et forme :White Crystalline PowderMasse moléculaire :320.84CEP-28122 mesylate salt (1022958-60-6 free base)
CEP-28122 mesylate salt (1022958-60-6 free base) is a highly selective orally active ALK inhibitor (IC50: 1.9 nM in an enzyme-based TRF assay).Formule :C29H39ClN6O6SDegré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :635.17JNJ-39758979
CAS :JNJ-39758979: selective H4 receptor antagonist, Kis 12.5/5.3/25 nM (human/mouse/monkey), blocks histamine cAMP inhibition (pA2 7.9).Formule :C11H19N5Degré de pureté :98.33% - 99.62%Couleur et forme :SolidMasse moléculaire :221.3Ref: TM-T11723L
1mg48,00€5mg97,00€10mg156,00€25mg255,00€50mg369,00€100mg543,00€200mg738,00€1mL*10mM (DMSO)105,00€Methyl-Hesperidin
CAS :<p>Methyl Hesperidin, a flavanone glycoside (flavonoid) (C28H34O15), is abundant in citrus fruits. Its aglycone form is called hesperetin.</p>Formule :C29H36O15Degré de pureté :98.51% - 99.01%Couleur et forme :Light Yellow Crystalline Powder Slightly Bitter TasteMasse moléculaire :624.5871Vildagliptin
CAS :Vildagliptin (LAF237), an oral DPP-4 inhibitor with hypoglycemic effects, is metabolized and excreted in urine.Formule :C17H25N3O2Degré de pureté :97.81% - >99.99%Couleur et forme :White Crystalline PowderMasse moléculaire :303.40Etofibrate
CAS :Etofibrate is a combination of clofibrate and niacin, used to treat hyperlipemia.Formule :C18H18ClNO5Degré de pureté :98.74%Couleur et forme :White To Off-White SolidMasse moléculaire :363.79Sulfacetamide sodium monohydrate
CAS :Sulfacetamide sodium monohydrate is a sulfonamide antibiotic. It has been investigated for the treatment of rosacea and pityriasis versicolor.Formule :C8H9N2NaO3S·H2ODegré de pureté :99.92%Couleur et forme :White Crystalline PowderMasse moléculaire :254.2BAY-2402234
CAS :BAY-2402234: a selective DHODH inhibitor targeting myeloid cancers with low-nanomolar potency.Formule :C21H18ClF5N4O4Degré de pureté :98.9%Couleur et forme :SolidMasse moléculaire :520.84Ref: TM-T14501
1mg173,00€2mg246,00€5mg368,00€10mg567,00€25mg905,00€50mg1.225,00€100mg1.644,00€1mL*10mM (DMSO)424,00€Chlorpropamide
CAS :<p>Chlorpropamide (Diabinese) is a sulfonylurea hypoglycemic agent used in the treatment of non-insulin-dependent diabetes mellitus not responding to dietary</p>Formule :C10H13ClN2O3SDegré de pureté :98.90%Couleur et forme :Crystals From Dil Ethanol Physical Description White Crystalline Powder With A Slight Odor (Ntp 1992)Masse moléculaire :276.74Hypoxanthine
CAS :<p>Hypoxanthine, a purine derivative, is a metabolite in nucleic acid synthesis and oxidizes to uric acid via xanthine.</p>Formule :C5H4N4ODegré de pureté :98.39% - 99.86%Couleur et forme :SolidMasse moléculaire :136.11CYM50308
CAS :CYM50308 is a high affinity agonist of sphingosine-1-phosphate receptor 4 (S1P4-R) (EC50: 56 nM).Formule :C20H21F2N3O2SDegré de pureté :99.43% - 99.77%Couleur et forme :SolidMasse moléculaire :405.46Ref: TM-T15032
1mg62,00€5mg140,00€10mg202,00€25mg324,00€50mg455,00€100mg597,00€200mg842,00€500mg1.225,00€Ascorbyl palmitate
CAS :<p>Ascorbyl palmitate (L-Ascorbic acid 6-hexadecanoate), an ester formed from ascorbic acid and palmitic acid, produces a fat-soluble form of vitamin C.</p>Formule :C22H38O7Degré de pureté :99.52%Couleur et forme :White Or Yellowish White Powder White Or Yellowish-White Powder With A Citrus-Like OdourMasse moléculaire :414.53MRTX0902
CAS :MRTX0902 is an effective and high selective inhibitor of SOS1 with an IC50 of 46 nM and a Ki of 2 nM.Formule :C22H24N6ODegré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :388.47Phthalic acid mono-2-ethylhexyl ester
CAS :Phthalic acid mono-2-ethylhexyl ester (Phthalic Acid Monooctyl Ester is a major bioactive metabolite of DEHP, which inhibits the 17, 20 lyase activity of CYP17.Formule :C16H22O4Degré de pureté :98.01%Couleur et forme :Physical Description Clear Colorless To Cloudy White Viscous Liquid (Ntp 1992)Masse moléculaire :278.34Ethoxyquin
CAS :<p>Ethoxyquin (Santoflex) is an antioxidant used in animal feeds.</p>Formule :C14H19NODegré de pureté :97.15% - 98.73%Couleur et forme :Yellow Liquid Mercaptan-Like Odor (Ntp 1992)Masse moléculaire :217.31Ximoprofen
CAS :Ximoprofen is a novel anti-inflammatory compound for the study of spondylitis.Formule :C15H19NO3Degré de pureté :98.06% - 98.13%Couleur et forme :SolidMasse moléculaire :261.32Orelabrutinib
CAS :<p>Orelabrutinib (ICP-022) is an orally active and irreversible inhibitor of Bruton's tyrosine kinase (BTK).</p>Formule :C26H25N3O3Degré de pureté :97.77% - 99.54%Couleur et forme :SolidMasse moléculaire :427.49Clevidipine
CAS :Clevidipine (Clevidipine butyrate) is a dihydropyridine L-type calcium channel blocker that is selective for vascular smooth muscle and is indicated for bloodFormule :C21H23Cl2NO6Degré de pureté :99.40%Couleur et forme :PowderMasse moléculaire :456.32Lysipressin acetate(50-57-7(fb_acetate))
CAS :<p>Lysipressin acetate (50-57-7), triggers rabbit bladder contraction & activates adenylate cyclase, is an antidiuretic in pigs & marsupials.</p>Formule :C48H69N13O14S2Degré de pureté :98.08%Couleur et forme :SolidMasse moléculaire :1116.28G150
CAS :G150 suppresses DSDNA-induced interferon; IC50: 10.2 nM. It's a potent, selective H-CGAS inhibitor.Formule :C18H16Cl2N4O2Degré de pureté :97.75%Couleur et forme :SolidMasse moléculaire :391.25Ref: TM-T11344
1mg126,00€5mg261,00€10mg376,00€25mg645,00€50mg842,00€100mg1.093,00€1mL*10mM (DMSO)285,00€Ciprofloxacin
CAS :Ciprofloxacin (Bay-09867) mainly targets bacterial DNA Gyrase (IC50=0.22-0.31 µM) and topoisomerase IV (IC50=0.3-1.9 µM). antibiotic. High-Quality, Low-Cost!Formule :C17H18FN3O3Degré de pureté :98.77% - 99.91%Couleur et forme :White PowderMasse moléculaire :331.34Telotristat ethyl
CAS :Telotristat ethyl (LX1606) is a orally-delivered inhibitor of tryptophan hydroxylase that reduces serotonin production.Formule :C27H26ClF3N6O3Degré de pureté :98% - 99.89%Couleur et forme :White SolidMasse moléculaire :574.98Oxiracetam
CAS :<p>Oxiracetam (ISF2522), a cyclic derivative of gamma-aminobutyric acid (GABA), is utilized for the treatment of cognitive impairments.</p>Formule :C6H10N2O3Degré de pureté :99.67%Couleur et forme :White Crystalline PowderMasse moléculaire :158.16Org-26576
CAS :Org-26576 is a positive allosteric modulator of the AMPA receptor.Formule :C11H12N2O2Degré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :204.23Ref: TM-T16402
5mg47,00€10mg70,00€25mg104,00€50mg150,00€100mg256,00€200mg379,00€1mL*10mM (DMSO)50,00€K-604 dihydrochloride
CAS :K-604 dihydrochloride is a potent and selective acyl-CoA:cholesterol acyltransferase 1 inhibitor with an IC50 of 0.45±0.06 μM.Formule :C23H32Cl2N6OS3Degré de pureté :99.10% - 99.74%Couleur et forme :SolidMasse moléculaire :575.64Ref: TM-T11733
1mg56,00€2mg81,00€5mg119,00€10mg187,00€25mg378,00€50mg560,00€100mg800,00€1mL*10mM (DMSO)166,00€SU056
CAS :<p>SU056 is a YB-1 inhibitor that induces cell-cycle arrest, apoptosis, and inhibits ovarian cancer cell migration.</p>Formule :C20H16FNO5Degré de pureté :99.89%Couleur et forme :SoildMasse moléculaire :369.34RIPK1-IN-7
CAS :RIPK1-IN-7: Strong, selective RIPK1 inhibitor (Kd=4 nM, IC50=11 nM) with great antimetastasis effects in B16 melanoma.Formule :C25H22F3N5O2Degré de pureté :98.02% - 98.18%Couleur et forme :SolidMasse moléculaire :481.47Ref: TM-T12731
1mg92,00€5mg216,00€10mg329,00€25mg512,00€50mg707,00€100mg944,00€1mL*10mM (DMSO)233,00€Cilnidipine
CAS :Cilnidipine (FRC-8653)(FRC8653) is a dual L- and N-type calcium channel blocker and displays antihypertensive, sympatholytic and neuroprotective activity.Formule :C27H28N2O7Degré de pureté :99.83% - 99.96%Couleur et forme :Yellow Crystalline SolidMasse moléculaire :492.52Lovastatin
CAS :Lovastatin (MK-803) is an HMG-CoA reductase inhibitor. Lovastatin lowers cholesterol and is used as a lipid-lowering agent. Cost-effective and quality-assured.Formule :C24H36O5Degré de pureté :99.66% - 99.92%Couleur et forme :The Substance Is A White-Yellowish To Yellow Powder Solid PowderMasse moléculaire :404.54Ipriflavone
CAS :Ipriflavone (Osteofix) (Osteofix) is a feed additive and a catabolic agent. It is used to inhibit bone resorption.Formule :C18H16O3Degré de pureté :99.6% - 99.82%Couleur et forme :White Crystalline PowderMasse moléculaire :280.32BNC105
CAS :BNC105 is a tubulin polymerization inhibitor. It has potent antiproliferative and tumor vascular disrupting properties.Formule :C20H20O7Degré de pureté :96.57%Couleur et forme :SolidMasse moléculaire :372.37Ref: TM-T14694
1mg84,00€5mg160,00€10mg226,00€25mg371,00€50mg520,00€100mg702,00€200mg944,00€1mL*10mM (DMSO)170,00€AZD5423
CAS :AZD5423: Inhaled, potent GR modulator, non-steroidal, curbs allergy asthma symptoms.Formule :C25H21F4N3O3Degré de pureté :98.76%Couleur et forme :SolidMasse moléculaire :487.45TINK-IN-1
CAS :TINK-IN-1 is a selective and potent TNIK inhibitor (IC50: 8 nM).TINK-IN-1 inhibits colorectal cancer cell viability and can be used to study mental retardation.Formule :C24H24N4O3Degré de pureté :99.4%Couleur et forme :SoildMasse moléculaire :416.47Ref: TM-T77660
1mg42,00€2mg52,00€5mg87,00€10mg127,00€25mg250,00€50mg373,00€100mg547,00€500mg1.159,00€Doxepin hydrochloride
CAS :Doxepin hydrochloride, a dibenzoxepin tricyclic, blocks monoamine reuptake and has anticholinergic and antihistaminic effects. Mechanism partly unknown.Formule :C19H22ClNODegré de pureté :99.65% - 99.91%Couleur et forme :White To Off-White PowderMasse moléculaire :315.84Centanafadine hydrochloride
CAS :Centanafadine HCl is a NE/DA reuptake inhibitor, also affects serotonin (IC50: NE 6 nM, DA 38 nM, serotonin 83 nM).Formule :C15H16ClNDegré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :245.75Ref: TM-T10758L
1mg59,00€5mg126,00€10mg202,00€25mg406,00€50mg653,00€100mg1.026,00€200mg1.378,00€500mg2.052,00€1mL*10mM (DMSO)140,00€Baloxavir
CAS :<p>Baloxavir (S-033447) is a first-in-class cap-dependent endonuclease inhibitor of the influenza virus polymerase PA subunit.</p>Formule :C24H19F2N3O4SDegré de pureté :99.26% - 99.87%Couleur et forme :SolidMasse moléculaire :483.494-Amino-5-Chloro-2-Methoxybenzoic Acid
CAS :4-Amino-5-Chloro-2-Methoxybenzoic Acid (Metoclopramide EP Impurity C) is a Metoclopramide metabolite.Formule :C8H8ClNO3Degré de pureté :99.78%Couleur et forme :White To Slightly Beige PowderMasse moléculaire :201.61BLU-945
CAS :<p>BLU-945 is a reversible, potent, highly selective, and orally available epidermal growth factor receptor tyrosine kinase inhibitor (TKIs).Cost-effective and quality-assured.</p>Formule :C28H37FN6O3SDegré de pureté :99.11% - 99.16%Couleur et forme :SolidMasse moléculaire :556.7CP-28888
CAS :CP-28888 (CP 28888-27) is an interferon inducer, a lipoamine with antitumor activity.Formule :C40H76N2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :585.05Amphotericin B
CAS :Amphotericin B (NSC-527017) is a polyene antifungal agent with broad-spectrum activity against many fungal species.Formule :C47H73NO17Degré de pureté :99.75% - ≥98%Couleur et forme :Deep Yellow Prisms Or Needles From N N-Dimethylformamide Physical Description Bright Yellow Powder (Ntp 1992)Masse moléculaire :924.08Ethambutol dihydrochloride
CAS :Ethambutol dihydrochloride (CL40881) is a bacteriostatic antimycobacterial agent, which obstructs the formation of cell wall by inhibiting arabinosylFormule :C10H26Cl2N2O2Degré de pureté :98% - 99.95%Couleur et forme :Crystals White PowderMasse moléculaire :277.24

