Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.855 produits)
- Apoptose(6.375 produits)
- Cycle cellulaire/point de contrôle(4.911 produits)
- Chromatine/Épigénétique(2.633 produits)
- Signalisation du cytosquelette(1.588 produits)
- Altération de l'ADN/réparation de l'ADN(2.868 produits)
- Endocrinologie/Hormones(3.765 produits)
- Enzyme(3.673 produits)
- GPCR/G-Protéine(9.054 produits)
- Immunologie et Inflammation(3.954 produits)
- Virus de la grippe(300 produits)
- Signalisation JAK/STAT(417 produits)
- Signalisation MAPK(1.259 produits)
- Transporteur membranaire/Canal ionique(3.163 produits)
- Métabolisme(10.157 produits)
- Microbiologie/Virologie(7.674 produits)
- Neuroscience(10.550 produits)
- Autres inhibiteurs(35.862 produits)
- Oxydation-Réduction(41 produits)
- Signalisation PI3K/Akt/mTOR(1.438 produits)
- Protéases/Protéasome(1.692 produits)
- Cellules souche et Dérivés(733 produits)
- Tyrosine Kinase/Adaptateurs(1.992 produits)
- Ubiquitination(1.744 produits)
Affichez 16 plus de sous-catégories
66512 produits trouvés pour "Inhibiteurs"
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N-Acetyl-D-mannosamine
CAS :N-Acetyl-D-mannosamine (ManNAc) is a drug potentially for the treatment of hereditary inclusion body myopathy.Formule :C8H15NO6Degré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :221.21Selisistat R-enantiomer
CAS :Selisistat R-enantiomer (EX-527 (R-enantiomer)) is a SIRT1 inhibitor with much less activity than the R-enantiomer of Selisistat (IC50 of SIRT1 > 100 μM).Formule :C13H13ClN2ODegré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :248.71Ref: TM-T15263
1mg101,00€2mg150,00€5mg245,00€1mL*10mM (DMSO)269,00€10mg356,00€25mg597,00€50mg835,00€100mg1.108,00€DMAT
CAS :DMAT (Casein kinase II Inhibitor) is a potent and specific inhibitor of CK2(IC50 value of 130 nM).Formule :C9H7Br4N3Degré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :476.79Desmethylglycitein
CAS :Desmethylglycitein (6,7,4'-Trihydroxyisoflavone) , is a novel inhibitor of PKCα in suppressing solar UV-induced matrix metalloproteinase 1, which hasFormule :C15H10O5Degré de pureté :97.93%Couleur et forme :SolidMasse moléculaire :270.24AZD5153 6-Hydroxy-2-naphthoic acid
CAS :AZD5153 6-Hydroxy-2-naphthoic acid (AZD5153) is a potent triazolopyridazine-based Bromodomain (BRD4) and Extraterminal (BET) inhibitor used in cancer treatmentsFormule :C25H33N7O3·C11H8O3Degré de pureté :97.26% - ≥95%Couleur et forme :SolidMasse moléculaire :667.75Rizatriptan benzoate
CAS :Rizatriptan benzoate (MK-462 Benzoate) selectively binds to and activates serotonin (5-HT) 1B receptors and 5-HT 1D receptors providing relief of migraineFormule :C22H25N5O2Degré de pureté :99% - 99.79%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :391.47Ref: TM-T1512
10mg44,00€1mL*10mM (DMSO)48,00€25mg74,00€50mg119,00€100mg173,00€200mg259,00€500mg437,00€HBT1
CAS :HBT1 is an AMPA receptor potentiator that induces production of brain-derived neurotrophic factor (BDNF) and exhibits little agonistic effect in primary neuronsFormule :C16H17F3N4O2SDegré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :386.39SR3335
CAS :SR3335 (ML 176) is a selective inverse agonist of RORα, competitively inhibiting the binding of 25-hydroxycholesterol to the ligand binding domain (Ki: 220 nM).Formule :C13H9F6NO3S2Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :405.34Ref: TM-T5160
1mg34,00€5mg74,00€1mL*10mM (DMSO)82,00€10mg119,00€25mg233,00€50mg371,00€100mg595,00€200mg833,00€2-Amino-4-hydroxypyrrolo[2,3- d]pyrimidi
CAS :2-Amino-4-hydroxypyrrolo[2,3-d]pyrimidine serves as an intermediate.Formule :C6H6N4ODegré de pureté :99.21% - 99.42%Couleur et forme :SolidMasse moléculaire :150.14LANOSTEROL
CAS :Lanosterol (3β-Hydroxy-8,24-lanostadiene) is a tetracyclic triterpenoid which is the compound from which all steroids are derived.Formule :C30H50ODegré de pureté :97.99% - 99.67%Couleur et forme :SolidMasse moléculaire :426.72JAK-IN-5 hydrochloride
CAS :JAK-IN-5 hydrochloride is a JAK inhibitor [1].Formule :C27H32ClFN6OCouleur et forme :SolidMasse moléculaire :511.03Folcisteine
CAS :Folcisteine (3-Acetylthiazolidine-4-carboxylic acid) is a kind of plant growth regulator.Formule :C6H9NO3SDegré de pureté :97.39%Couleur et forme :White Crystalline PowderMasse moléculaire :175.206Sumaresinolic Acid
CAS :Sumaresinolic Acid, a natural lignan in flaxseed, sesame, wheat bran, may reduce inflammation, improve lipids, and offer antioxidant benefits.Formule :C30H48O4Degré de pureté :98.17%Couleur et forme :SolidMasse moléculaire :472.7Ref: TM-T8772
1mg84,00€5mg168,00€1mL*10mM (DMSO)198,00€10mg245,00€25mg404,00€50mg567,00€100mg767,00€200mg1.018,00€2,6,6-Trimethyl-2,4-cycloheptadien-1-one
CAS :2,6,6-Trimethyl-2,4-cycloheptadien-1-one: a terpene in plants like parsley; key in essential oils, with medicinal benefits.Formule :C10H14ODegré de pureté :97.95%Couleur et forme :SolidMasse moléculaire :150.224,7-DIHYDROXYCOUMARIN
CAS :4,7-Dihydroxycoumarin: Natural enzyme inhibitor in parsley, chamomile; binds DNA, impacts genes, cell cycle, and can trigger tumor cell apoptosis.Formule :C9H6O4Degré de pureté :99.16% - 99.2%Couleur et forme :SolidMasse moléculaire :178.14TAS6417
CAS :Zipalertinib (TAS6417, CLN-081) is a novel, highly potent, orally active covalent EGFR tyrosine kinase inhibitor.Cost-effective and quality-assured.Formule :C23H20N6ODegré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :396.44Ref: TM-T16996
1mg93,00€2mg117,00€5mg178,00€1mL*10mM (DMSO)203,00€10mg295,00€25mg595,00€50mg795,00€100mg1.071,00€200mg1.468,00€Duvelisib hydrate
CAS :Duvelisib (IPI-145, INK-1197) is an oral PI3K delta/gamma inhibitor with potential anti-cancer and immunomodulatory effects.Formule :C22H19ClN6O2Couleur et forme :SolidMasse moléculaire :434.884Tetrahydrocoptisine
CAS :Tetrahydrocoptisine (Stylopine) quells inflammation, protects against ALI, guards the gut, and blocks key pro-inflammatory pathways.Formule :C19H17NO4Degré de pureté :99.76% - ≥95%Couleur et forme :SolidMasse moléculaire :323.34STING agonist-1
CAS :STING agonist-1 (G10) is a human-specific STING agonist,elicits antiviral activity against emerging Alphaviruses.Formule :C21H16ClFN2O3SDegré de pureté :99.07%Couleur et forme :SolidMasse moléculaire :430.88Trifluoperazine
CAS :Trifluoperazine (trifluoroperazine) is a Dopamine D2 receptor inhibitor(IC50 : 1.2 nM), and Treatment of schizophrenia.Formule :C21H24F3N3SDegré de pureté :98.3% - 99.46%Couleur et forme :White To Yellowish Crystalline PowderMasse moléculaire :407.5JNJ-39758979 2HCl
CAS :JNJ-39758979 2HCl is an antagonist of histamine receptor H4.Formule :C11H21Cl2N5Couleur et forme :SolidMasse moléculaire :294.22Galgravin
CAS :Galgravin combats inflammation, safeguards neurons, promotes neurite growth, and resists Abeta25-35 and MPP+ toxicity.Formule :C22H28O5Degré de pureté :99.75% - 99.88%Couleur et forme :SolidMasse moléculaire :372.45Ref: TM-TN1038
1mg195,00€5mg487,00€1mL*10mM (DMSO)495,00€10mg702,00€25mg1.063,00€50mg1.459,00€100mg1.963,00€Rhamnetin
CAS :Rhamnetin (beta-Rhamnocitrin), a quercetin derivative found in Coriandrum sativum, has antioxidant and anti-inflammatory activities.Formule :C16H12O7Degré de pureté :99.61% - 99.905%Couleur et forme :SolidMasse moléculaire :316.26Ref: TM-TN1419
1mg60,00€5mg130,00€1mL*10mM (DMSO)137,00€10mg200,00€25mg338,00€50mg497,00€100mg708,00€BEBT-908
CAS :BEBT-908 (PI3Kα inhibitor 1) is a selective PI3Kα inhibitor (IC50 <0.1 μM). BEBT-908 also inhibits HDAC (0.1 μM≤IC50≤1 μM).Formule :C23H25N9O3SDegré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :507.57Ref: TM-T16529
1mg94,00€5mg222,00€1mL*10mM (DMSO)249,00€10mg334,00€25mg562,00€50mg802,00€100mg1.063,00€200mg1.459,00€[Ala107]-MBP (104-118) acetate
[Ala107]-MBP (104-118) acetate ([Ala107]-MBP ) is synthetic peptide analog of bovine myelin basic protein (MBP).Formule :C59H108N20O21Degré de pureté :99.23%Couleur et forme :SolidMasse moléculaire :1553.72Reversine
CAS :Reversine, a small synthetic purine analogue (2, 6-disubstituted purine), is a potent inhibitior of Aurora A/B/C(IC50s=150-500 nM).Formule :C21H27N7ODegré de pureté :98% - 99.45%Couleur et forme :SolidMasse moléculaire :393.49Ref: TM-T1825
1mg35,00€2mg50,00€5mg66,00€1mL*10mM (DMSO)66,00€10mg84,00€25mg156,00€50mg212,00€100mg371,00€Pseudoprotodioscin
CAS :1. Pseudoprotodioscin has moderate cytotoxicity.Formule :C51H82O21Degré de pureté :99.19% - ≥95%Couleur et forme :SolidMasse moléculaire :1031.18Ref: TM-T5S0246
2mg39,00€5mg62,00€10mg94,00€1mL*10mM (DMSO)99,00€25mg137,00€50mg193,00€100mg286,00€200mg423,00€Episyringaresinol 4'-O-β-D-glncopyranoside
CAS :Episyringaresinol 4'-O-β-D-glncopyranoside ((-)-Syringaresinol 4-O-β-D-glucopyranosi) inhibits proliferation through G(1) arrest and induction of apoptosis.Formule :C28H36O13Degré de pureté :98.74% - 99.89%Couleur et forme :SolidMasse moléculaire :580.58Fmoc-Val-Cit-PAB-MMAE
CAS :Fmoc-Val-Cit-PAB-MMAE: ADC linker plus MMAE, a tubulin inhibitor drug-linker for ADCs.Formule :C73H104N10O14Degré de pureté :98.2%Couleur et forme :SolidMasse moléculaire :1345.67AZD3264
CAS :AZD3264 is a new type IKK2 inhibitor.Formule :C21H23N5O4SDegré de pureté :98.98% - 99.17%Couleur et forme :SolidMasse moléculaire :441.5Ref: TM-T6771
1mg49,00€2mg66,00€5mg98,00€1mL*10mM (DMSO)108,00€10mg152,00€25mg295,00€50mg475,00€100mg762,00€500mg1.521,00€Protirelin Acetate(24305-27-9 free base)
CAS :Protirelin Acetate(24305-27-9 free base) (Thyroliberin Acetate) is a tripeptide that stimulates the release of thyrotropin and prolactin.Formule :C18H26N6O6Degré de pureté :98.78%Couleur et forme :SolidMasse moléculaire :422.44Ref: TM-T6956L
5mg52,00€10mg64,00€1mL*10mM (DMSO)78,00€25mg118,00€50mg178,00€100mg320,00€200mg464,00€Cytidine 5'-diphosphate disodium
CAS :Cytidine 5'-diphosphate disodium (CDP sodium salt) produces CTP to support DNA and RNA biosynthesis and ribonucleotide reductase to produce dCMP.Formule :C9H13N3Na2O11P2Degré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :447.14Guanabenz hydrochloride
CAS :Guanabenz hydrochloride (NE56490) is an orally active α2-adrenoceptor agonist with hypotensive effects.Formule :C8H9Cl3N4Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :267.54BTS
CAS :BTS (N-Tosylbenzylamine) is a potent inhibitor of Ca2+-stimulated myosin S1 ATPase (IC50 : 5 μM) .Formule :C14H15NO2SDegré de pureté :99.45%Couleur et forme :White Crystalline SolidMasse moléculaire :261.34JH-X-119-01
CAS :JH-X-119-01 is a highly potent and selective covalent inhibitor of IRAK-1.Formule :C25H20N6O3Degré de pureté :98.42%Couleur et forme :SolidMasse moléculaire :452.46Ref: TM-T9203
1mg63,00€2mg92,00€5mg137,00€1mL*10mM (DMSO)150,00€10mg200,00€25mg356,00€50mg532,00€100mg740,00€PD-161570
CAS :PD-161570 is a potent and ATP-competitive human FGF-1 receptor inhibitor with an IC50 of 39.9 nM and a Ki of 42 nM.Formule :C26H35Cl2N7ODegré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :532.51Ref: TM-T23127
1mg34,00€5mg96,00€1mL*10mM (DMSO)118,00€10mg141,00€25mg289,00€50mg465,00€100mg662,00€200mg888,00€Doxazosin HCl
CAS :Doxazosin HCl, a salt, blocks alpha(1)-adrenoceptors, reducing catecholamine-induced vasoconstriction for vasodilation.Formule :C23H26ClN5O5Couleur et forme :SolidMasse moléculaire :487.94β-Estradiol 17-hemisuccinate
CAS :beta-Estradiol 17-hemisuccinate selectively stains estrogen receptor (ER)-rich cells.Formule :C22H28O5Degré de pureté :99.62%Couleur et forme :SolidMasse moléculaire :372.45Ref: TM-T9604
1mg52,00€5mg108,00€1mL*10mM (DMSO)112,00€10mg160,00€25mg248,00€50mg351,00€100mg477,00€200mg622,00€Vildagliptin dihydrate
CAS :Vildagliptin dihydrate: potent, selective DPP-IV inhibitor with 3.5 nM IC50, high oral bioavailability, effective against hyperglycemia.Formule :C17H29N3O4Couleur et forme :SolidMasse moléculaire :339.436Dacomitinib
CAS :Dacomitinib (PF299) is an oral selective inhibitor of EGFR, ERBB2, ERBB4 with IC50s: 6, 45.7, 73.7 nM.Formule :C24H25ClFN5O2Degré de pureté :99.4% - 99.72%Couleur et forme :SolidMasse moléculaire :469.94Ref: TM-T2483
1mg35,00€2mg50,00€5mg74,00€1mL*10mM (DMSO)74,00€10mg120,00€25mg170,00€50mg215,00€100mg334,00€200mg421,00€500mg692,00€(E)-KPT330
CAS :(E)-RN (KPT 330) is a CRM1-selective inhibitor of nuclear export. (E)-RN inhibits protein trafficking from the nucleus and induces cell cycle arrest.
Formule :C17H11F6N7ODegré de pureté :98.69% - 99.49%Couleur et forme :SolidMasse moléculaire :443.31Nicotinuric acid
CAS :Nicotinuric acid: a minor acyl glycine metabolite of fatty acids, synthesized by glycine N-acyltransferase.Formule :C8H8N2O3Degré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :180.16Isovaleric acid
CAS :Isovaleric acid (Delphinic acid) is a naturally occurring aroma compound found in Bartlett pear brandies, vanilla beans, rape-honey, and banana.Formule :C5H10O2Degré de pureté :97.89%Couleur et forme :Colourless Clear LiquidMasse moléculaire :102.13R-268712
CAS :R-268712 is a potent ALK5 inhibitor with a 2.5 nM IC50, also targeting TGF-β type I receptor orally.Formule :C20H18FN5ODegré de pureté :99.61%Couleur et forme :SolidMasse moléculaire :363.39Ref: TM-T16708
1mg44,00€1mL*10mM (DMSO)92,00€5mg93,00€10mg130,00€25mg250,00€50mg378,00€100mg537,00€200mg762,00€CD73-IN-3
CAS :CD73-IN-3 (LY-3475070) is a potent CD73 inhibitor with a 28 nM IC50, being tested in advanced cancer alone or with pembrolizumab.Formule :C15H18N4O2Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :286.33Ref: TM-T8875
1mg60,00€5mg138,00€1mL*10mM (DMSO)152,00€10mg215,00€25mg359,00€50mg510,00€100mg692,00€200mg888,00€N,N'-Dimethylthiourea
CAS :N,N'-Dimethylthiourea (DMTU) scavenges hydroxyl radicals, blocks their production by neutrophils, and prevents gastric lesions in rats.Formule :C3H8N2SDegré de pureté :≥98%Couleur et forme :Off-White Crystalline PowderMasse moléculaire :104.17Handle region peptide, rat acetate
Handle region peptide, rat acetate is a prorenin receptor antagonist, suppresses the progression of diabetic nephropathy and has anti-inflammatory in the eye.Formule :C56H105N15O14SDegré de pureté :99.01%Couleur et forme :SolidMasse moléculaire :1244.614-Methylesculetin
CAS :4-Methylesculetin (Methylesculetin) is one of the coumarin derivatives with great anti-oxidant and anti-inflammatory activities.Formule :C10H8O4Degré de pureté :97.96%Couleur et forme :Yellow Needle CrystalMasse moléculaire :192.179-hydroxy-4-androstene-3,17-dione
CAS :9-Hydroxy-4-androstene-3,17-dione: a steroid with anti-tumor properties against breast, prostate, and lung cancers.Formule :C19H26O3Degré de pureté :99.65% - 99.77%Couleur et forme :White To Beige Solid PowderMasse moléculaire :302.41GLP-1(7-36), amide
CAS :GLP-1 secretion by human enteroendocrine NCI-H716 cells is augmented in a dose-dependent manner by the addition of CPE.Cost-effective and quality-assured.Formule :C149H226N40O45Degré de pureté :99.85%Couleur et forme :White PowderMasse moléculaire :3297.63
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