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Trombina

Trombina

Gli inibitori della trombina sono composti che bloccano la trombina, un enzima coinvolto nel processo di coagulazione del sangue che ha anche un ruolo nella promozione dell'angiogenesi. La trombina può stimolare la formazione di nuovi vasi sanguigni nei tumori, favorendone la crescita e la metastasi. Inibendo la trombina, questi composti possono ridurre l'angiogenesi e la progressione tumorale. Gli inibitori della trombina sono importanti sia nella ricerca sul cancro che nello studio delle malattie vascolari. Presso CymitQuimica, offriamo una selezione di inibitori della trombina di alta qualità per supportare la tua ricerca in emostasi, oncologia e angiogenesi.

Trovati 52 prodotti di "Trombina"

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  • Anti-Coagulation Factor II Antibody (8M286)


    Anti-Coagulation Factor II Antibody (8M286) is a Rabbit antibody targeting Coagulation Factor II. Anti-Coagulation Factor II Antibody (8M286) can be used in ELISA.
    Colore e forma:Odour Liquid
  • Dabigatran ethyl ester

    CAS:
    Dabigatran ethyl ester (Dabigatran (ethyl ester)) is an emerging oral anticoagulant and it also is a direct inhibitor of thrombin activity.
    Formula:C27H29N7O3
    Purezza:99.98%
    Colore e forma:Solid
    Peso molecolare:499.56
  • Coagulation Factor II Protein, Mouse, Recombinant (His)


    Coagulation Factor II Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag.
    Colore e forma:Lyophilized Powder
    Peso molecolare:69.3 kDa (predicted); 85 kDa (reducing conditions)
  • Dabigatran

    CAS:
    <p>Dabigatran (BIBR 953ZW), a thrombin inhibitor, prevents thrombus formation, reducing stroke and embolism risk in nonvalvular atrial fibrillation patients.</p>
    Formula:C25H25N7O3
    Purezza:97.44% - 98.7%
    Colore e forma:Tan Solid
    Peso molecolare:471.51
  • Argatroban Monohydrate

    CAS:
    Argatroban Monohydrate is a specific thrombin inhibitor, which is a non-heparin anticoagulant, prevents the formation of thrombi.
    Formula:C23H38N6O6S
    Purezza:99.51%
    Colore e forma:Solid
    Peso molecolare:526.65
  • TRAP-6

    CAS:
    <p>TRAP-6 (Thrombin Receptor Activator Peptide 6)(2TFA) is an agonist of protease-activated receptor 1 (PAR1).</p>
    Formula:C34H56N10O9
    Purezza:>99.99%
    Colore e forma:Solid
    Peso molecolare:748.87
  • Edoxaban Tosylate Monohydrate

    CAS:
    <p>Edoxaban(DU-176) is an oral factor Xa (FXa) inhibitor in clinical development for stroke prevention.</p>
    Formula:C31H40ClN7O8S2
    Purezza:99.86% - 99.91%
    Colore e forma:Solid
    Peso molecolare:738.27
  • Dabigatran Etexilate Mesylate

    CAS:
    Dabigatran Etexilate Mesylate (BIBR 1048MS) is the orally active prodrug of dabigatran. Dabigatran is a reversible and selective, direct thrombin inhibitor.
    Formula:C34H41N7O5·CH4O3S
    Purezza:99.91%
    Colore e forma:Solid
    Peso molecolare:723.84
  • Bivalirudin

    CAS:
    <p>Bivalirudin (BG-8967) is a reversible inhibitor of α- and ζ-thrombin (Kis = 2.56 and 1.84 nM, respectively), enzymes that exhibit high fibrinogen-clotting</p>
    Formula:C98H138N24O33
    Purezza:98.8% - >99.99%
    Colore e forma:White To Off-White Powder
    Peso molecolare:2180.29
  • H-D-Phe-Pip-Arg-pNA dihydrochloride

    CAS:
    <p>H-D-Phe-Pip-Arg-pNA dihydrochloride (S-2238) is a sensitive and accurate thrombin detection substrate for measuring antithrombin-heparin cofactor (AT-III).</p>
    Formula:C27H38Cl2N8O5
    Purezza:99.47%
    Colore e forma:Solid
    Peso molecolare:625.55
  • AEBSF hydrochloride

    CAS:
    AEBSF hydrochloride (Pefabloc SC) is an irreversible inhibitor of serine proteases, such as chymotrypsin, kallikrein, thrombin, plasmin, and trypsin.
    Formula:C8H11ClFNO2S
    Purezza:98% - 99.81%
    Colore e forma:White Powder
    Peso molecolare:239.69
  • Cycloolivil

    CAS:
    <p>Cycloolivil (Isoolivil) is a natural polyphenolic compound with a significant radical scavenging activity present in olive trees.</p>
    Formula:C20H24O7
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:376.4
  • NQ301

    CAS:
    NQ301, an antithrombotic agent, inhibits collagen-challenged rabbit platelet aggregation (IC50: 10 mg/mL).
    Formula:C18H12ClNO3
    Purezza:99.74% - 99.76%
    Colore e forma:Solid
    Peso molecolare:325.75
  • Ximelagatran

    CAS:
    Ximelagatran, oral direct thrombin inhibitor, transforms to active melagatran in body.
    Formula:C24H35N5O5
    Purezza:95.48% - 99.60%
    Colore e forma:Solid
    Peso molecolare:473.57
  • MNS

    CAS:
    MNS is a tyrosine kinases inhibitor, inhibits Syk, Src, p97 with IC50 of 2.5 μM, 29.3 μM and 1.7 μM, respectively.
    Formula:C9H7NO4
    Purezza:98.53%
    Colore e forma:Yellow Powder
    Peso molecolare:193.16
  • Enoxaparin sodium

    CAS:
    Enoxaparin, a low-weight heparin approved by FDA for STEMI, enhances antithrombin and prevents clotting by inhibiting factors XIa, IXa, Xa, IIa.
    Formula:C42H59N3Na4O35S2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:1322
  • Lusutrombopag

    CAS:
    Lusutrombopag (Mulpleta) is an orally bioavailable, small molecule thrombopoietin (TPO) receptor agonist for chronic liver disease (CLD) patients with
    Formula:C29H32Cl2N2O5S
    Purezza:99.96%
    Colore e forma:Solid
    Peso molecolare:591.55
  • Avatrombopag

    CAS:
    <p>Avatrombopag (YM477) is a new oral thrombopoietin (TPO) receptor agonist, activating TPO receptor and increasing megakaryocytic proliferation/differentiation</p>
    Formula:C29H34Cl2N6O3S2
    Purezza:99.01% - 99.63%
    Colore e forma:Solid
    Peso molecolare:649.65
  • Argatroban

    CAS:
    Argatroban (MCI-9038), a specific thrombin inhibitor, which is a non-heparin anticoagulant, prevents the formation of thrombi.
    Formula:C23H36N6O5S
    Purezza:99.77% - >99.99%
    Colore e forma:White To Off-White Crystalline Solid
    Peso molecolare:508.63
  • Atopaxar

    CAS:
    <p>Atopaxar (E5555), a reversible PAR-1 thrombin receptor antagonist, interferes with platelet signaling.</p>
    Formula:C29H38FN3O5
    Purezza:97.07% - 98.07%
    Colore e forma:Solid
    Peso molecolare:527.63