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Caspasi

Caspasi

Gli inibitori delle caspasi sono composti che bloccano l'attività delle caspasi, una famiglia di proteasi che sono esecutori centrali dell'apoptosi. Le caspasi clivano substrati specifici all'interno della cellula per innescare il processo apoptotico, portando alla morte cellulare programmata. Gli inibitori delle caspasi sono utilizzati per studiare i meccanismi dell'apoptosi, nonché per prevenire la morte cellulare indesiderata in vari modelli di ricerca. Questi inibitori sono anche esplorati in contesti terapeutici per proteggere le cellule dall'apoptosi in malattie come la neurodegenerazione. Presso CymitQuimica, offriamo una vasta gamma di inibitori delle caspasi di alta qualità per supportare la tua ricerca in apoptosi, morte cellulare e campi correlati.

Trovati 143 prodotti di "Caspasi"

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  • Aspirin

    CAS:
    Aspirin (Acetylsalicylic Acid) is a COX inhibitor. Aspirin has anti-inflammatory, antipyretic and analgesic activities. Cost-effective and quality-assured.
    Formula:C9H8O4
    Purezza:99.78% - 99.91%
    Colore e forma:White Solid Crystalline
    Peso molecolare:180.16
  • Thiabendazole

    CAS:
    <p>Thiabendazole (2-(4-Thiazolyl)benzimidazole) is a benzimidazole derivative with anthelminthic property.</p>
    Formula:C10H7N3S
    Purezza:99.14%
    Colore e forma:Light Yellow Powder
    Peso molecolare:201.25
  • Diclofenac diethylamine

    CAS:
    Diclofenac Diethylamine, a non-selective COX inhibitor, is utilized as a nonsteroidal anti-inflammatory drug (NSAID).
    Formula:C18H22Cl2N2O2
    Purezza:99.81% - 99.87%
    Colore e forma:Solid
    Peso molecolare:369.29
  • Crustecdysone

    CAS:
    <p>Crustecdysone (Hydroxyecdysone) is a steroid hormone that regulates the processes of molting or ecdysis in insects.</p>
    Formula:C27H44O7
    Purezza:99.06% - 99.67%
    Colore e forma:Canary Yellow Fine Powder
    Peso molecolare:480.63
  • Diclofenac

    CAS:
    Diclofenac: a nonsteroidal compound inhibiting COX-1 and COX-2, reducing pro-inflammatory prostaglandins.
    Formula:C14H11Cl2NO2
    Purezza:99.69% - 99.97%
    Colore e forma:Crystals From Ether-Petroleum Ether Solid
    Peso molecolare:296.15
  • Lacidipine

    CAS:
    Lacidipine (SN-305) is a slow-acting, long-duration lipophilic dihydropyridine calcium blocker that prevents reflex tachycardia and lowers blood pressure.
    Formula:C26H33NO6
    Purezza:99.98%
    Colore e forma:White-To-Off-White Crystalline Solid
    Peso molecolare:455.54
  • Ac-FLTD-CMK

    CAS:
    <p>Ac-FLTD-CMK, an abscisicin D derivative, selectively inhibits inflammatory caspases-1, -4, and -11 (IC50: 46.7 nM, 1.49 μM, 329 nM) but not caspase-3.</p>
    Formula:C26H37ClN4O8
    Purezza:95.17%
    Colore e forma:Solid
    Peso molecolare:569.05
  • Ac-YVAD-CMK

    CAS:
    <p>Ac-YVAD-CMK: Irreversible Caspase-1 inhibitor; halts pyroptosis, IL-1β/IL-18; neuroprotective and anti-inflammatory.</p>
    Formula:C24H33ClN4O8
    Purezza:97.08% - 99.909%
    Colore e forma:Solid
    Peso molecolare:540.99
  • Oxidopamine hydrobromide

    CAS:
    <p>Oxidopamine hydrobromide (6-OHDA hydrobromide) is a neurotransmitter dopamine antagonist.</p>
    Formula:C8H12BrNO3
    Purezza:98.22% - 99.88%
    Colore e forma:Beige To Brown Fine Crystalline Powder
    Peso molecolare:250.09
  • Q-VD-OPH

    CAS:
    <p>Q-VD-OPh is an irreversible caspase inhibitor with an IC50 value of 48 nM against caspase-7 and between 25 and 400 nM against caspase-1, 3, 8, 9, 10, 12.</p>
    Formula:C26H25F2N3O6
    Purezza:97.8% - 98.95%
    Colore e forma:Solid
    Peso molecolare:513.5
  • Diclofenac sodium

    CAS:
    <p>Diclofenac sodium (GP 45840) is a non-steroidal anti-inflammatory agent (NSAID) with antipyretic and analgesic actions.</p>
    Formula:C14H10Cl2NNaO2
    Purezza:98.21% - 99.73%
    Colore e forma:White Or Off-White Powder
    Peso molecolare:318.13
  • Fenbufen

    CAS:
    <p>Fenbufen (Lederfen) is a non-steroidal anti-inflammatory drug used primarily to treat inflammation in osteoarthritis, ankylosing spondylitis, and tendinitis.</p>
    Formula:C16H14O3
    Purezza:98.35% - 98.46%
    Colore e forma:White Solid
    Peso molecolare:254.28
  • Dehydrocorydaline chloride

    CAS:
    <p>Dehydrocorydaline chloride (13-Methylpalmatine chloride) is an alkaloid with anti-inflammatory and anti-cancer activity. Can improve the activation of p38 MAPK.</p>
    Formula:C22H24ClNO4
    Purezza:99.53%
    Colore e forma:Solid
    Peso molecolare:401.88
  • ML-9

    CAS:
    <p>ML-9 suppresses MLCK, PKA, and PKC activity with Ki values of 4, 32, and 54 μM, respectively.</p>
    Formula:C15H18Cl2N2O2S
    Purezza:99.69%
    Colore e forma:Crystalline Solid
    Peso molecolare:361.29
  • Terfenadine

    CAS:
    Terfenadine, metabolized to fexofenadine by CYP3A4, is a non-sedative antihistamine targeting H1 receptors.
    Formula:C32H41NO2
    Purezza:98.76% - 99.75%
    Colore e forma:Solid
    Peso molecolare:471.67
  • Oxidopamine hydrochloride

    CAS:
    Oxidopamine hydrochloride (6-Hydroxydopamine hydrochloride) is an neurotransmitter dopamine antagonist.
    Formula:C8H12ClNO3
    Purezza:98.34% - 99.85%
    Colore e forma:Physical Description Beige Solid (Ntp 1992)
    Peso molecolare:205.64
  • Ac-Trp-Glu-His-Asp-Aldehyde

    CAS:
    <p>Ac-Trp-Glu-His-Asp-Aldehyde is a powerful and selective inhibitor of caspase-1, demonstrating a K_i value of 56 pM [1] [2].</p>
    Formula:C28H33N7O9
    Colore e forma:Solid
    Peso molecolare:611.6
  • TNF-α-IN-11


    <p>TNF-α-IN-11 (Compound 10) is a TNF-α inhibitor exhibiting a dissociation constant (K D) of 12.06 μM.</p>
    Formula:C24H26N2O5
    Colore e forma:Solid
    Peso molecolare:422.47
  • IRF1-IN-2

    CAS:
    <p>IRF1-IN-2 is a small molecule IRF1 inhibitor that suppresses pyroptosis, protecting against radiation-induced skin damage.</p>
    Formula:C18H20N2O4S
    Purezza:99.85%
    Colore e forma:Solid
    Peso molecolare:360.43
  • TD1092


    TD1092, a pan-IAP degrader, activates caspase 3/7, induces apoptosis in cancer cells, inhibits NF-κB, and is used in cancer research.
    Formula:C55H70N8O9
    Colore e forma:Solid
    Peso molecolare:987.19