
Cromatina/Epigenetica
Gli inibitori della cromatina/epigenetica sono composti che modulano la struttura e la funzione della cromatina o interferiscono con le modificazioni epigenetiche, come la metilazione del DNA e la modifica degli istoni. Questi inibitori sono strumenti essenziali per studiare la regolazione dell'espressione genica e il ruolo dell'epigenetica in malattie come il cancro, i disturbi neurologici e le anomalie dello sviluppo. Mirando ai processi epigenetici, questi inibitori possono alterare i modelli di espressione genica e offrire nuove opportunità terapeutiche. Presso CymitQuimica, offriamo un'ampia selezione di inibitori della cromatina/epigenetica di alta qualità per supportare le tue ricerche in biologia molecolare, genetica ed epigenetica.
Sottocategorie di "Cromatina/Epigenetica"
Trovati 2573 prodotti di "Cromatina/Epigenetica"
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3-TYP
CAS:3-TYP (3-(1H-1,2,3-triazol-4-yl) pyridine) is a selective SIRT3 inhibitor.Formula:C7H6N4Purezza:99.16% - >99.99%Colore e forma:SolidPeso molecolare:146.15Ref: TM-T4108
2mg39,00€5mg52,00€10mg93,00€25mg166,00€50mg248,00€100mg393,00€200mg560,00€1mL*10mM (DMSO)52,00€A-196
CAS:A-196 is a potent and selective inhibitor of SUV420 h1 and SUV420 h2 with IC50 values of 0.025 and 0.144 μM, respectively; more than 100-fold selective overFormula:C18H16Cl2N4Purezza:99.92%Colore e forma:SolidPeso molecolare:359.253,6-Dihydroxyflavone
CAS:3,6-Dihydroxyflavone suppresses the epithelial-mesenchymal transition in breast cancer cells by inhibiting the Notch signaling pathway.Formula:C15H10O4Purezza:99.92%Colore e forma:SolidPeso molecolare:254.24Methyl L-histidinate dihydrochloride
CAS:The inhibitory effect of Methyl L-histidinate dihydrochloride (L-Histidine methyl ester dihydrochloride) on histidine decarboxylase in Sprague-Dawley ratFormula:C7H13Cl2N3O2Purezza:99.74%Colore e forma:White To Off-White PowderPeso molecolare:242.1SNS-314
CAS:SNS-314 inhibits Aurora kinases A and B, blocking cell division in AK-overexpressing tumors.Formula:C18H15ClN6OS2Purezza:98%Colore e forma:SolidPeso molecolare:430.93PFI-2 hydrochloride
CAS:PFI-2 hydrochloride ((R)-PFI-2 hydrochloride) is a potent, highly selective, and cell-active inhibitor of the methyltransferase activity of SETD7 (IC50: 2 nM),Formula:C23H26ClF4N3O3SPurezza:99.31% - 99.91%Colore e forma:SolidPeso molecolare:535.98Ref: TM-T4583
1mg38,00€2mg49,00€5mg80,00€10mg111,00€25mg200,00€50mg358,00€100mg523,00€500mg1.108,00€1mL*10mM (DMSO)122,00€4-amino-1,8-Naphthalimide
CAS:4-amino-1,8-Naphthalimide (4-ANI) is a PARP inhibitor with IC50 of 180 nMFormula:C12H8N2O2Purezza:95.13%Colore e forma:Yellow Solid PowderPeso molecolare:212.2AMPK activator 2
CAS:AMPK activator 2, a chloroformin derivative, may boost cancer treatment by enhancing AMPK and inhibiting mTOR pathways, and cancer cell growth.Formula:C13H18F3N5Purezza:99.86%Colore e forma:SolidPeso molecolare:301.31BMS-P5 free base
CAS:BMS-P5 free base is a specific and orally active peptidylarginine deiminase 4 (PAD4) inhibitor.Formula:C27H32N6O2Purezza:99.88%Colore e forma:SolidPeso molecolare:472.58Niraparib tosylate monohyrate
CAS:Niraparib (MK-4827), a PARP inhibitor, boosts DNA breaks to trigger genomic instability and apoptosis, offering anti-cancer effects.Formula:C26H30N4O5SPurezza:97.7% - 99.99%Colore e forma:SolidPeso molecolare:510.61Ref: TM-T9497
5mg57,00€10mg82,00€25mg111,00€50mg137,00€100mg205,00€200mg309,00€500mg515,00€1mL*10mM (DMSO)66,00€Fucosterol
CAS:Fucosterol, from E. stolonifera, has anti-diabetic, anti-adipogenic, anti-cancer properties; it affects PPARα and C/EBPα to control fat cell formation.Formula:C29H48OPurezza:98.39% - 99.68%Colore e forma:White PowderPeso molecolare:412.69BAY 87-2243
CAS:BAY 87-2243 is a potent and selective inhibitor of hypoxia-inducible factor-1 (HIF-1).Formula:C26H26F3N7O2Purezza:98% - 99.95%Colore e forma:SolidPeso molecolare:525.53Ref: TM-T2488
1mg35,00€2mg43,00€5mg63,00€10mg101,00€25mg212,00€50mg351,00€100mg588,00€1mL*10mM (DMSO)73,00€ML324
CAS:ML324(IC50=920 nM) is a specific inhibitor of jumonji histone demethylase (JMJD2).Formula:C21H23N3O2Purezza:98.22% - 98.57%Colore e forma:SolidPeso molecolare:349.43Ref: TM-T6593
2mg35,00€5mg51,00€10mg79,00€25mg128,00€50mg216,00€100mg354,00€200mg520,00€1mL*10mM (DMSO)84,00€Amifostine sodium
CAS:Amifostine sodium is a phosphorothioate proposed as a radiation-protective agent. It causes splenic vasodilation and may block autonomic ganglia.Formula:C5H15N2NaO3PSColore e forma:SolidPeso molecolare:237.21IOX2
CAS:IOX2 is a selective HIF PHD inhibitor, active in cells with 21 nM IC50 for PHD2/ELGN-1, not inhibiting FIH at 20uM.Formula:C19H16N2O5Purezza:98% - 99.59%Colore e forma:SolidPeso molecolare:352.34HNHA
CAS:HNHA is an inhibitor of HDAC.Formula:C17H21NO2SPurezza:98.04%Colore e forma:SolidPeso molecolare:303.42Ref: TM-T21806
1mg44,00€5mg84,00€10mg135,00€25mg279,00€50mg445,00€100mg640,00€200mg879,00€1mL*10mM (DMSO)90,00€Senaparib hydrochloride
CAS:Senaparib hydrochloride is a potent and selective oral PARP1/2 inhibitor with strong antitumor activity.Formula:C24H21ClF2N6O3Colore e forma:SolidPeso molecolare:514.92Eicosapentaenoic Acid sodium
CAS:EPA sodium, an oral omega-3, demethylates DNA, reactivates tumor suppressors, and induces vasodilation.Formula:C20H29NaO2Colore e forma:SolidPeso molecolare:324.43OTS186935 hydrochloride
OTS186935 HCl inhibits SUV39H2 (IC50 6.49 nM), curbs tumor growth in mice, and modulates γ-H2AX in cancer cells.Formula:C25H27Cl2N5O2Colore e forma:SolidPeso molecolare:522.31TIQ-A
CAS:TIQ-A blocks PARP1 to prevent excessive DNA damage response, implicated in ischemia, asthma, and atherosclerosis.Formula:C11H7NOSPurezza:99.75%Colore e forma:SolidPeso molecolare:201.24Ref: TM-T50098
1mg52,00€5mg92,00€10mg161,00€25mg290,00€50mg414,00€100mg532,00€200mg737,00€1mL*10mM (DMSO)96,00€

