Cromatina/Epigenetica
Gli inibitori della cromatina/epigenetica sono composti che modulano la struttura e la funzione della cromatina o interferiscono con le modificazioni epigenetiche, come la metilazione del DNA e la modifica degli istoni. Questi inibitori sono strumenti essenziali per studiare la regolazione dell'espressione genica e il ruolo dell'epigenetica in malattie come il cancro, i disturbi neurologici e le anomalie dello sviluppo. Mirando ai processi epigenetici, questi inibitori possono alterare i modelli di espressione genica e offrire nuove opportunità terapeutiche. Presso CymitQuimica, offriamo un'ampia selezione di inibitori della cromatina/epigenetica di alta qualità per supportare le tue ricerche in biologia molecolare, genetica ed epigenetica.
Sottocategorie di "Cromatina/Epigenetica"
Trovati 2613 prodotti di "Cromatina/Epigenetica"
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1-benzyl-2-ethyl-4,5,6,7-tetrahydro-1H-indol-4-one
CAS:1-benzyl-2-ethyl-4,5,6,7-tetrahydro-1H-indol-4-one is an inhibitor Bromodomain-containing protein 4 (human).Formula:C17H19NOPurezza:99.08%Colore e forma:SolidPeso molecolare:253.34Ref: TM-T8601
1mg58,00€1mL*10mM (DMSO)109,00€5mg116,00€10mg172,00€25mg281,00€50mg396,00€100mg537,00€200mg712,00€GSK620
CAS:GSK620, a selective pan-BD2 inhibitor, has anti-inflammatory properties and favorable oral pharmacokinetics.Formula:C18H19N3O3Purezza:99.42% - 99.88%Colore e forma:SolidPeso molecolare:325.36Ref: TM-T9020
2mg34,00€5mg49,00€10mg73,00€1mL*10mM (DMSO)87,00€25mg136,00€50mg212,00€100mg314,00€200mg467,00€Talazoparib
CAS:Talazoparib (LT-673) is a new-type PARP inhibitor (IC50: 0.58 nM), It similarly binds to PARP1/2 (Kis: 1.2/0.85 nM).Formula:C19H14F2N6OPurezza:97.02% - 99.92%Colore e forma:SolidPeso molecolare:380.35Ref: TM-T6253
2mg42,00€5mg62,00€1mL*10mM (DMSO)67,00€10mg88,00€25mg135,00€50mg187,00€100mg311,00€200mg429,00€500mg697,00€Solcitinib
CAS:Solcitinib (GLPG-0778), a JAK1 inhibitor, may treat psoriasis, ulcerative colitis, and lupus.
Formula:C22H23N5O2Purezza:99.61% - 99.82%Colore e forma:SolidPeso molecolare:389.45Dbet57
CAS:dBET57: PROTAC-based BRD4BD1 degrader, DC50/5h at 500 nM, ineffective on BRD4BD2.Formula:C34H31ClN8O5SPurezza:99.36% - 99.52%Colore e forma:SolidPeso molecolare:699.18Ref: TM-T5440
1mg47,00€5mg92,00€10mg147,00€1mL*10mM (DMSO)166,00€25mg264,00€50mg409,00€100mg592,00€500mg1.224,00€MAT2A inhibitor 4
CAS:MAT2A Inhibitor 4 acts as an inhibitor targeting the catalytic subunit of methionine S-adenosyltransferase-2 (MAT2A), offering potential utility in cancerFormula:C16H15ClFNPurezza:99.17%Colore e forma:SolidPeso molecolare:275.75Ref: TM-T9262
1mg40,00€1mL*10mM (DMSO)89,00€5mg90,00€10mg131,00€25mg220,00€50mg314,00€100mg426,00€200mg575,00€Mivebresib
CAS:Mivebresib (ABBV-075) is a potent BET inhibitor with antitumor effects, disrupting gene expression and MYC, TMPRSS2-ETS proteins.Formula:C22H19F2N3O4SPurezza:98.74% - 99.32%Colore e forma:SolidPeso molecolare:459.47Ref: TM-T3712
1mg55,00€2mg78,00€5mg92,00€1mL*10mM (DMSO)94,00€10mg150,00€25mg244,00€50mg437,00€100mg625,00€PHA-680632
CAS:PHA-680632 is potent inhibitor of Aurora A, Aurora B and Aurora C with IC50 of 27 nM, 135 nM and 120 nM, respectively.Formula:C28H35N7O2Purezza:98.2%Colore e forma:SolidPeso molecolare:501.623-Aminobenzamide
CAS:3-Aminobenzamide (PARP-IN-1) is an effective inhibitor of PARP (IC50<50 nM in CHO cells) and a mediator of oxidant-induced myocyte dysfunction duringFormula:C7H8N2OPurezza:98.4% - 99.5%Colore e forma:White To Off-White PowderPeso molecolare:136.15SF2523
CAS:SF2523 is a highly selective and potent inhibitor.Formula:C19H17NO5SPurezza:99.1% - 99.51%Colore e forma:SolidPeso molecolare:371.41Ref: TM-T3986
1mg34,00€5mg74,00€1mL*10mM (DMSO)82,00€10mg113,00€25mg260,00€50mg409,00€100mg605,00€500mg1.288,00€JNJ-64619178
CAS:JNJ-64619178: selective, oral, pseudo-irreversible PRMT5 inhibitor (IC50: 0.14 nM), effective in lung cancer.Formula:C22H23BrN6O2Purezza:98.86% - 99.98%Colore e forma:SolidPeso molecolare:483.36Ref: TM-T15624
1mg84,00€5mg167,00€1mL*10mM (DMSO)172,00€10mg260,00€25mg537,00€50mg893,00€100mg1.571,00€GeA-69
CAS:GeA-69 (GeA69) is a selective and allosteric PARP14 macrodomain 2 (MD2) inhibitor (Kd: 0.86 μM in ITC assays).Formula:C20H16N2OPurezza:99.85%Colore e forma:SolidPeso molecolare:300.35TTK21
CAS:TTK21 is an activator of CBP/p300 histone acetyltransferase activity.Formula:C17H15ClF3NO2Purezza:98.43%Colore e forma:SolidPeso molecolare:357.75Ref: TM-T8778
1mg57,00€5mg105,00€1mL*10mM (DMSO)114,00€10mg158,00€25mg308,00€50mg462,00€100mg692,00€500mg1.404,00€PX-478
CAS:PX-478 is a HIF-1α inhibitor with selectivity, oral activity, and blood-brain barrier permeability.Formula:C13H20Cl4N2O3Purezza:97% - 99.79%Colore e forma:SolidPeso molecolare:394.12Ref: TM-T6961
1mg39,00€5mg84,00€1mL*10mM (DMSO)84,00€10mg130,00€25mg193,00€50mg261,00€100mg411,00€200mg605,00€LW6
CAS:LW6 (HIF-1α inhibitor) is a novel HIF-1 inhibitor.Formula:C26H29NO5Purezza:98.1% - 98.22%Colore e forma:SolidPeso molecolare:435.51Ref: TM-T3494
2mg44,00€5mg65,00€1mL*10mM (DMSO)65,00€10mg94,00€25mg173,00€50mg281,00€100mg424,00€500mg888,00€Ref: TM-T5S2358
1mg49,00€2mg69,00€5mg105,00€1mL*10mM (DMSO)116,00€10mg137,00€25mg197,00€50mg295,00€100mg447,00€Belzutifan
CAS:"Belzutifan (MK-6482) is an oral HIF-2α inhibitor for ccRCC, with enhanced potency (IC50: 9 nM)."Formula:C17H12F3NO4SPurezza:99.34% - 99.88%Colore e forma:SolidPeso molecolare:383.34Ref: TM-T16679
1mg66,00€5mg144,00€1mL*10mM (DMSO)158,00€10mg205,00€25mg389,00€50mg625,00€100mg888,00€200mg1.198,00€I-BET151
CAS:I-BET151 (GSK1210151A) (GSK1210151A) is a specific BET inhibitor for BRD2/3/4 (IC50: 0.5/0.25/0.79 μM, in cell-free assays).Formula:C23H21N5O3Purezza:97.34% - 99.63%Colore e forma:SolidPeso molecolare:415.44Ref: TM-T2120
1mg48,00€2mg65,00€5mg96,00€1mL*10mM (DMSO)105,00€10mg115,00€25mg202,00€50mg339,00€100mg507,00€500mg1.130,00€Veliparib
CAS:Veliparib (ABT-888) (ABT-888) is an orally bioavailable inhibitor of PARP (Kis: 5.2/2.9 nM for PARP1/2). It enhances apoptosis and autophagy.Formula:C13H16N4OPurezza:98.66% - 99%Colore e forma:SolidPeso molecolare:244.29Ref: TM-T2591
5mg54,00€1mL*10mM (DMSO)60,00€10mg77,00€25mg120,00€50mg195,00€100mg314,00€200mg512,00€500mg807,00€Tranylcypromine hemisulfate
CAS:Tranylcypromine hemisulfate (Tranylcypromine Sulfate) is an inhibitor of monoamine oxidase (MAO) and lysine-specific demethylase 1 (LSD1) with a rapid onset ofFormula:C9H11N1H2SO4Purezza:98% - 99.96%Colore e forma:SolidPeso molecolare:182.23
