
Cromatina/Epigenetica
Gli inibitori della cromatina/epigenetica sono composti che modulano la struttura e la funzione della cromatina o interferiscono con le modificazioni epigenetiche, come la metilazione del DNA e la modifica degli istoni. Questi inibitori sono strumenti essenziali per studiare la regolazione dell'espressione genica e il ruolo dell'epigenetica in malattie come il cancro, i disturbi neurologici e le anomalie dello sviluppo. Mirando ai processi epigenetici, questi inibitori possono alterare i modelli di espressione genica e offrire nuove opportunità terapeutiche. Presso CymitQuimica, offriamo un'ampia selezione di inibitori della cromatina/epigenetica di alta qualità per supportare le tue ricerche in biologia molecolare, genetica ed epigenetica.
Sottocategorie di "Cromatina/Epigenetica"
Trovati 2613 prodotti di "Cromatina/Epigenetica"
Ordinare per
Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
SGI-1027
CAS:SGI-1027 (DNA Methyltransferase Inhibitor II) is an effective and selective inhibitor of DNA methyltransferase (DNMT).Formula:C27H23N7OPurezza:99.45% - 99.78%Colore e forma:SolidPeso molecolare:461.52Ref: TM-T1904
5mg58,00€10mg94,00€25mg163,00€50mg296,00€100mg467,00€500mg1.035,00€1mL*10mM (DMSO)74,00€GSK467
CAS:GSK467 is a potent and selective inhibitor of KDM5 (JARID1)(Ki : 10 nM).Formula:C17H13N5O2Purezza:99.55% - 99.85%Colore e forma:SolidPeso molecolare:319.32MG 149
CAS:MG 149 (Tip60 HAT inhibitor) is a selective and potent Tip60 inhibitor with IC50 of 74 uM, similar potentcy for MOF(IC50= 47 uM).Formula:C22H28O3Purezza:98.69% - 99.86%Colore e forma:SolidPeso molecolare:340.46Ref: TM-T6584
1mg50,00€2mg71,00€5mg90,00€10mg167,00€25mg308,00€50mg492,00€100mg708,00€1mL*10mM (DMSO)108,00€UNC3866
CAS:UNC3866 is a potent antagonist of the CBX7-H3 interaction as determined by AlphaScreen.Formula:C43H66N6O8Purezza:88.06% - 99.62%Colore e forma:SolidPeso molecolare:795.02GW779439X
CAS:GW779439X is an inhibitor of CDK.Formula:C22H21F3N8Purezza:97.87%Colore e forma:SolidPeso molecolare:454.45Ref: TM-T8866
1mg58,00€2mg82,00€5mg113,00€10mg178,00€25mg404,00€50mg592,00€100mg845,00€1mL*10mM (DMSO)124,00€CCT241736
CAS:CCT241736 is an orally bioavailable dual FLT3/Aurora kinase inhibitor that also inhibits clinically relevant FLT3-resistant mutants including FLT3-ITD and FLT3Formula:C22H23Cl2N7Purezza:96.2% - 99.81%Colore e forma:SolidPeso molecolare:456.37G244-LM
CAS:G244-LM is a potent and specific inhibitor of tankyrase 1/2. G244-LM inhibits Wnt signaling.Formula:C18H22N4O3S2Purezza:98.46%Colore e forma:SolidPeso molecolare:406.52AMG 900
CAS:AMG 900 is a potent and highly selective pan-Aurora kinases inhibitor for Aurora A/B/C with IC50 of 5 nM/4 nM /1 nM.Formula:C28H21N7OSPurezza:98.4% - 99.51%Colore e forma:SolidPeso molecolare:503.58Ref: TM-T6380
1mg49,00€5mg92,00€10mg158,00€25mg286,00€50mg442,00€100mg645,00€500mg1.341,00€1mL*10mM (DMSO)100,00€3-Methoxybenzamide
CAS:3-Methoxybenzamide (3-MBA) is a competitive inhibitor of poly(ADP-ribose) synthetase.Formula:C8H9NO2Purezza:98.52%Colore e forma:SolidPeso molecolare:151.16Amifostine trihydrate
CAS:Amifostine trihydrate (WR2721) is the first approved radioprotective drug, used to decrease the risk of kidney problems caused by treatment with cisplatin.Formula:C5H15N2O3PS·3H2OPurezza:99.71% - 99.80%Colore e forma:SolidPeso molecolare:268.27Fosifidancitinib
CAS:Fosifidancitinib is a potent inhibitor of JAK 1 and JAK 3.Formula:C21H21FN5O7PPurezza:99.54%Colore e forma:SolidPeso molecolare:505.39Ref: TM-T38624
1mg93,00€2mg117,00€5mg177,00€10mg269,00€25mg429,00€50mg610,00€100mg820,00€200mg1.099,00€ARV-771
CAS:ARV-771 is an effective BET degrader based on PROTAC technology.Cost-effective and quality-assured.Formula:C49H60ClN9O7S2Purezza:99.69%Colore e forma:SolidPeso molecolare:986.64Ref: TM-T5435
1mg57,00€5mg113,00€10mg177,00€25mg354,00€50mg522,00€100mg732,00€200mg973,00€1mL*10mM (DMSO)192,00€Oclacitinib maleate
CAS:Oclacitinib maleate is a selective JAK inhibitor (IC50: 10-99 nM; JAK1 cytokines: 36-249 nM), with no effect on 38 non-JAK kinases.Formula:C15H23N5O2S·C4H4O4Purezza:99.17% - 99.92%Colore e forma:SolidPeso molecolare:453.51Ref: TM-T6914
1mg37,00€2mg52,00€5mg74,00€10mg94,00€25mg166,00€50mg258,00€100mg432,00€1mL*10mM (DMSO)81,00€CPI-169 racemate
CAS:CPI-169 racemate (CPI 169) is a potent, and selective EZH2 inhibitor with IC50 of 0.24 nM, 0.51 nM, and 6.1 nM for EZH2 WT, EZH2 Y641N, and EZH1, respectively.
Formula:C27H36N4O5SPurezza:99.59%Colore e forma:SolidPeso molecolare:528.66BET bromodomain inhibitor
CAS:BET bromodomain inhibitor is a potent BET inhibitor.Formula:C24H20ClN5O2Purezza:98.22% - 99.85%Colore e forma:SolidPeso molecolare:445.9Ref: TM-T2072
1mg35,00€2mg50,00€5mg75,00€10mg114,00€25mg187,00€50mg264,00€100mg416,00€1mL*10mM (DMSO)84,00€ENMD-2076
CAS:ENMD-2076, a multi-targeted kinase inhibitor, has specific activity against Aurora A, Flt3, KDR/VEGFR2, Flt4/VEGFR3, FGFR1, FGFR2, Src, PDGFRα.Formula:C21H25N7Purezza:97.63% - ≥95%Colore e forma:SolidPeso molecolare:375.47(Z)-SMI-4a
CAS:(Z)-SMI-4a (TCS PIM-1 4a) is a selective ATP-competitive Pim-1 kinase inhibitor with an IC50 of 21 nM.Formula:C11H6F3NO2SPurezza:97.66% - 99.93%Colore e forma:SolidPeso molecolare:273.23Oclacitinib
CAS:Oclacitinib (PF-03394197)(PF03394197) is a potent and selective JAKs inhibitor with IC50 of 10-99 nM; not inhibit a panel of 38 non-JAK kinases (IC50 's > 1000Formula:C15H23N5O2SPurezza:98% - 98.45%Colore e forma:White To Off-White SolidPeso molecolare:337.44lutidinic acid
CAS:lutidinic acid (2,4-Dicarboxypyridine) is an in vitro and in cell inhibitor, as well as a known inhibitor of the histone lysine demethylases.
Formula:C7H5NO4Purezza:98.06%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:167.12RG108
CAS:RG108 (N-Phthalyl-L-tryptophan) is an DNA methyltransferase inhibitor(IC50=115 nM).Formula:C19H14N2O4Purezza:98% - 99.43%Colore e forma:SolidPeso molecolare:334.33Ref: TM-T2038
5mg44,00€10mg65,00€25mg111,00€50mg195,00€100mg271,00€200mg380,00€500mg618,00€1mL*10mM (DMSO)52,00€
