Endocrinologia/Ormoni
Gli inibitori dell'endocrinologia/oromone sono composti che bloccano l'azione degli ormoni o interferiscono con le vie di segnalazione ormonale. Questi inibitori sono fondamentali per studiare la regolazione dei sistemi endocrini e per sviluppare trattamenti per malattie correlate agli ormoni, come il diabete, i disturbi della tiroide e i tumori ormono-dipendenti. Modulando l'attività ormonale, questi inibitori possono aiutare a chiarire le complesse interazioni all'interno del sistema endocrino. Presso CymitQuimica, offriamo un'ampia gamma di inibitori di alta qualità per endocrinologia/oromone per supportare le tue ricerche in endocrinologia, farmacologia e scienze mediche.
Sottocategorie di "Endocrinologia/Ormoni"
- Recettore degli androgeni(229 prodotti)
- Annessina A(16 prodotti)
- Aromatasi(22 prodotti)
- Recettore degli estrogeni/progestogeni(57 prodotti)
- GPR(1 prodotti)
- Recettore dei glucocorticoidi(166 prodotti)
- LHRH(1 prodotti)
- Recettore degli oppioidi(326 prodotti)
- Recettore della prostaglandina(122 prodotti)
- RAAS(90 prodotti)
- Riduttasi(50 prodotti)
- Somatostatina(57 prodotti)
- Recettore dell'ormone tiroideo (THR)(32 prodotti)
- Recettore della vasopressina(48 prodotti)
Mostrare 6 più sottocategorie
Trovati 3371 prodotti di "Endocrinologia/Ormoni"
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Dynorphin A (1-8)
CAS:Dynorphin (1-8) is an opioid octapeptide from the porcine hypothalamus. It comprises the N-terminal eight residues of dynorphin.Formula:C46H72N14O10Purezza:98%Colore e forma:SolidPeso molecolare:981.151-Methyl-2-[(4Z,7Z)-4,7-tridecadienyl]-4(1H)-quinolone
CAS:1-Methyl-quinolone alkaloid inhibits DAG acyltransferase, blocks angiotensin II receptor (IC50s: 20.1 & 34.1 μM), and fights H. pylori (MIC: 10 μg/mL).Formula:C23H31NOColore e forma:SolidPeso molecolare:337.5Raloxifene 4'-glucuronide
CAS:<p>Raloxifene 4'-glucuronide is a primary metabolite of Raloxifene.</p>Formula:C34H35NO10SPurezza:98%Colore e forma:SolidPeso molecolare:649.71[Nphe1]Nociceptin(1-13)NH2
CAS:<p>Competitive nociceptin receptor antagonist with pKi=8.4; no agonist activity; blocks nociceptin effects in vitro/in vivo.</p>Formula:C61H100N22O15Purezza:98%Colore e forma:SolidPeso molecolare:1381.6ET receptor antagonist 3
"ET receptor antagonist 3 (compound 17d) is an orally active ET receptor antagonist with an IC50 of 0.26 nM, utilized for pulmonary arterial hypertension (PAH)Formula:C27H28N6O5SPurezza:98%Colore e forma:SolidPeso molecolare:548.61Olmesartan medoxomil impurity C
CAS:Impurity C of Olmesartan medoxomil is a selective AT1 inhibitor with an IC50 of 66.2 μM.Formula:C29H28N6O5Colore e forma:SolidPeso molecolare:540.57ET receptor antagonist 1
ET Receptor Antagonist 1 (compound 16h), with an IC50 value of 0.18 nM, is an orally active agent that can be utilized for pulmonary arterial hypertension (PAHFormula:C21H25N5O5SPurezza:98%Colore e forma:SolidPeso molecolare:459.52Azilsartan Medoxomil Potassium
CAS:Azilsartan Medoxomil Potassium (TAK-491 Potassium) is an orally administered angiotensin II receptor type 1 antagonist with IC50 of 0.62 nM, which used in the treatment of adults with essential hypertension.Formula:C30H23N4O8·KPurezza:99.99%Colore e forma:SolidPeso molecolare:606.62Anticancer agent 135
<p>Anticancer agent 135 (compound 26h) acts as a potent androgen receptor (AR) antagonist, effectively blocking AR nuclear translocation and inhibiting AR/AR-V7</p>Formula:C23H21F3N4OSPurezza:98%Colore e forma:SolidPeso molecolare:458.5ACTH (6-24) (human)
CAS:Adrenocorticotropic hormone (6-24) (ACTH (6-24) (human)) is a fragment of ACTH that acts as a competitive inhibitor of steroidogenesis prompted by full-lengthFormula:C111H175N35O21Peso molecolare:2335.8Hydrocortisone sodium succinate
CAS:Hydrocortisone sodium succinate is a glucocorticoid which is used to alleviate allergic reactions, particularly those of the skin and gums.Formula:C25H34NaO8Colore e forma:SolidPeso molecolare:485.529L 363564
CAS:L 363564 is a kidney renin inhibitor.Formula:C54H76N12O10Colore e forma:SolidPeso molecolare:1053.276Androgen receptor antagonist 9
CAS:Androgen Receptor Antagonist 9 (compound 28) serves as an antagonist to the androgen receptor [1].Formula:C19H14F3N3O2SPurezza:98%Colore e forma:SolidPeso molecolare:405.39ST-CY14
ST-CY14 is an inhibitor of the Nur77-PPARγ interaction with an EC50 of 3.15 μM. It binds to Nur77 (Kd=32 nM) to prevent its ubiquitination and degradation by PPARγ, reducing fatty acid uptake and mitochondrial respiration, and inhibiting the transcription of CD36 and FABP4. ST-CY14 suppresses proliferation and migration of MCF7 and MDA-MB-231 cancer cells and impedes tumor growth and bone metastasis in mouse models.Formula:C139H237N57O31S2Colore e forma:SolidPeso molecolare:3266.86PTP1B/AKR1B1-IN-2
PTP1B/AKR1B1-IN-2 (Compound 7f) is a potent inhibitor targeting both PTP1B and AKR1B1 with IC50 values of 3.2 and 2.1 μM, respectively, and K i values of 4.0Formula:C23H23NO4S2Purezza:98%Colore e forma:SolidPeso molecolare:441.56AZ 1729
CAS:<p>FFA2 modulator; inhibits cAMP, enhances 35SGTPγS binding (pEC50: 6.9, 7.23); alters Gi/Gq signaling; affects lipolysis, neutrophil migration.</p>Formula:C18H16FN5OSColore e forma:SolidPeso molecolare:369.42Estrogen receptor modulator 6
CAS:<p>ER modulator 6 (3a) is a potent ERβ agonist with a K i of 0.44 nM; 19x more selective for ERβ than ERα.</p>Formula:C18H16F2O3Colore e forma:SolidPeso molecolare:318.32WCA-814
<p>WCA-814, an androgen receptor (AR) antagonist-Hsp90 inhibitor conjugate, induces degradation of both full-length and AR-V7, exhibiting cytotoxic effects in</p>Formula:C46H53ClN10O5Purezza:98%Colore e forma:SolidPeso molecolare:861.43Ro 64-6198
CAS:Ro 64-6198: Nonpeptide, selective NOP agonist, high brain uptake, EC50=25.6 nM, 100x NOP>opioid affinity.Formula:C26H31N3OPurezza:98%Colore e forma:SolidPeso molecolare:401.5414-3-3σ/ERα stabilizer-1
Compound 181, also known as 14-3-3σ/ERα Stabilizer-1, is a covalent stabilizer targeting the 14-3-3σ/ERα proteins.Formula:C25H35Cl2N3O3Purezza:98%Colore e forma:SolidPeso molecolare:496.47
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