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Recettore degli androgeni

Recettore degli androgeni

Il recettore degli androgeni (AR) è un recettore ormonale nucleare che viene attivato dal legame con gli androgeni, come il testosterone e il diidrotestosterone. Questo recettore svolge un ruolo cruciale nello sviluppo e nel mantenimento delle caratteristiche maschili, nonché nella regolazione di diversi processi fisiologici, tra cui la crescita muscolare, la libido e la densità ossea. Gli inibitori del recettore degli androgeni sono ampiamente studiati nel contesto del cancro alla prostata, dove la segnalazione dell'AR è spesso sovraregolata. Presso CymitQuimica, offriamo una gamma di modulatori del recettore degli androgeni di alta qualità per supportare la tua ricerca in endocrinologia, biologia del cancro e regolazione ormonale.

Trovati 229 prodotti di "Recettore degli androgeni"

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  • VPC-14449
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    VPC-14449

    CAS:
    VPC-14449 is a selective androgen receptor DNA-binding domain (AR-DBD) inhibitor, useful in prostate cancer research.
    Formula:C10H10Br2N4OS
    Purezza:99.56%
    Colore e forma:Solid
    Peso molecolare:394.09

    Ref: TM-T24944

  • BMS-564929
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    BMS-564929

    CAS:
    BMS-564929 is an AR agonist that upregulates the expression and activity of fat-producing enzymes, reducing VAT content and lipid levels.
    Formula:C14H12ClN3O3
    Purezza:98.17%
    Colore e forma:Solid
    Peso molecolare:305.72

    Ref: TM-T14675

  • VPC-13789
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    VPC-13789

    CAS:
    VPC-13789: potent, selective oral antiandrogen for CRPC with 0.19 μM IC50 in LNCaP cells.
    Formula:C21H16F3N3O
    Colore e forma:Solid
    Peso molecolare:383.37

    Ref: TM-T61653

  • Androgen receptor antagonist 3
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    Androgen receptor antagonist 3

    CAS:
    Androgen receptor antagonist 3 (Compound C18) has anticancer activities that is an antagonist of androgen receptor (AR) (IC 50 = 2.4 μM) [1].
    Formula:C22H18ClN
    Colore e forma:Solid
    Peso molecolare:331.84

    Ref: TM-T60987

  • (R)-UT-155
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    (R)-UT-155

    CAS:
    (R)-UT-155 is a selective androgen receptor degrader (SARD) ligand.
    Formula:C20H15F4N3O2
    Colore e forma:Solid
    Peso molecolare:405.35

    Ref: TM-T13977

  • Lubabegron fumarate
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    Lubabegron fumarate

    CAS:
    Lubabegron (LY591281, LY488756 fumarate) is a beta-agonist approved in 2018 to lower ammonia in cattle waste, aiding environment and health.
    Formula:C29H29N3O3SC4H4O4
    Colore e forma:Solid
    Peso molecolare:557.66

    Ref: TM-T69306

  • MK-4541
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    MK-4541

    CAS:
    MK-4541: oral, selective AR modulator, blocks 5α-reductase, curbs AR+ prostate cancer growth, effective in mouse model.
    Formula:C22H31F3N2O3
    Colore e forma:Solid
    Peso molecolare:428.49

    Ref: TM-T73410

  • HG122
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    HG122

    CAS:
    HG122 promotes AR degradation via proteasome, inhibiting castration-resistant prostate cancer.
    Formula:C15H13N5O5
    Colore e forma:Solid
    Peso molecolare:343.29

    Ref: TM-T61109

  • LGD-2226
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    LGD-2226

    CAS:
    LGD-2226: selective oral androgen receptor modulator, EC50: 0.2nM, Ki: 1.5nM. Treats muscle loss, osteoporosis, sexual issues.
    Formula:C14H9F9N2O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:392.22

    Ref: TM-T15749

  • Dimethomorph
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    Dimethomorph

    CAS:
    Dimethomorph is a fungicide and sterol biosynthesis inhibitor that inhibits fungal cell wall formation,. inhibits androgen receptor (AR) .
    Formula:C21H22ClNO4
    Purezza:99.20%
    Colore e forma:Solid Crystalline
    Peso molecolare:387.86

    Ref: TM-T41322

  • CSRM617
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    CSRM617

    CAS:
    CSRM617: selective ONECUT2 inhibitor, Kd 7.43 uM, binds OC2-HOX, induces apoptosis, tolerable in mouse prostate cancer model.
    Formula:C10H13N3O5
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:255.23

    Ref: TM-T10896

  • MK-3984
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    MK-3984

    CAS:
    MK-3984 is a selective androgen receptor modulator, used in the study of conditions caused by androgen deficiency.
    Formula:C17H12F7NO2
    Purezza:99.91%
    Colore e forma:Solid
    Peso molecolare:395.27

    Ref: TM-T33433

  • TFM-4AS-1
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    TFM-4AS-1

    CAS:
    androgen receptor modulator
    Formula:C27H33F3N2O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:474.56

    Ref: TM-T23455

  • VPC-3033
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    VPC-3033

    CAS:
    VPC-3033 is an antagonist of the androgen receptor. It acts by inhibiting the LNCaP cell line as well as cell lines with the wild-type androgen receptor.
    Formula:C21H14O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:298.33

    Ref: TM-T26323

  • Topterone
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    Topterone

    CAS:
    Topterone (Win 17,665) is a potent topical antiandrogen that inhibits the stimulation of lumbar organ development by testosterone and dihydrotestosterone in
    Formula:C22H34O2
    Purezza:>99.99%
    Colore e forma:Solid
    Peso molecolare:330.5

    Ref: TM-T13187

  • Ar-V7-IN-1
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    Ar-V7-IN-1

    CAS:
    Ar-V7-IN-1 (compound 47) is a potent inhibitor of Ar-V7,associated with resistance to AR-targeted therapy with desmoplasia-resistant prostate cancer (mCRPC).
    Formula:C10H10Br2N4OS
    Colore e forma:Solid
    Peso molecolare:394.09

    Ref: TM-T61820

  • Carbazole derivative 1
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    Carbazole derivative 1

    CAS:
    Carbazole derivative 1 is used to reduce androgen or oestrogen levels in mammals.
    Formula:C18H13FN2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:276.31

    Ref: TM-T19170

  • Seviteronel
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    Seviteronel

    CAS:
    Seviteronel (VT-464) is a novel CYP17 cleavage enzyme inhibitor and androgen receptor antagonist for the study of breast and prostate cancer.
    Formula:C18H17F4N3O3
    Purezza:99.67% - 99.98%
    Colore e forma:Solid
    Peso molecolare:399.34

    Ref: TM-T13312L

  • BMS-641988
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    BMS-641988

    CAS:
    BMS-641988 is a novel nonsteroidal androgen receptor antagonist for the treatment of prostate cancer.
    Formula:C20H20F3N3O5S
    Purezza:99.3% - 99.92%
    Colore e forma:Soild
    Peso molecolare:471.45

    Ref: TM-T67818

  • Rosolutamide
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    Rosolutamide

    CAS:
    Rosolutamide (ALZ-003) is a curcumin analog, an Nrf1 and Nrf2 activator.
    Formula:C28H32O6
    Purezza:95.48% - 99.15%
    Colore e forma:Solid
    Peso molecolare:464.55

    Ref: TM-T71552