
Canale del sodio
I canali del sodio sono proteine di membrana essenziali che permettono il passaggio degli ioni sodio (Na+) attraverso la membrana cellulare, generando e propagando segnali elettrici nei neuroni, nelle cellule muscolari e in altri tessuti eccitabili. Questi canali sono vitali per l'inizio e la conduzione dei potenziali d'azione, rendendoli cruciali in processi come la trasmissione degli impulsi nervosi, la contrazione muscolare e la funzione cardiaca. La disregolazione dei canali del sodio può portare a disturbi neurologici, aritmie e condizioni di dolore cronico. Presso CymitQuimica, offriamo una varietà di modulatori dei canali del sodio per supportare la tua ricerca in neurobiologia, cardiologia e gestione del dolore.
Trovati 367 prodotti per "Canale del sodio".
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Silperisone HCl
CAS:Silperisone HCl is a muscle relaxant and vasodilator, treating myoclonus, hypertonia, dystonia, and myospasm by blocking Na+ and Ca2+ channels.Formula:C15H25ClFNSiPurezza:99.97%Colore e forma:White SolidPeso molecolare:301.9NHE3-IN-1
CAS:NHE3-IN-1 是钠/质子交换剂 3 (NHE-3) 的抑制剂。Formula:C12H10ClN3SPurezza:99.93%Colore e forma:White SolidPeso molecolare:263.75SLC13A5-IN-1
CAS:SLC13A5-IN-1 is a selective inhibitor of sodium-citrate co-transporter (SLC13A5),completely blocks the uptake of 14C-citrate(IC50 : 0.022 μM in HepG2 cells).Formula:C19H19Cl3N2O3SPurezza:99.67%Colore e forma:White SolidPeso molecolare:461.79Ref: TM-T12931
1mg48,00€5mg92,00€1mL*10mM (DMSO)92,00€10mg152,00€25mg268,00€50mg447,00€100mg623,00€200mg883,00€500mg1.305,00€Co 102862
CAS:Co 102862 is a voltage-gated sodium channel blocker. Co 102862 can be used for anticonvulsant studies.Formula:C14H12FN3O2Purezza:99.82%Colore e forma:SolidPeso molecolare:273.26GDC-0310
CAS:GDC-0310 is a selective, orally available Nav1.7 inhibitor with an IC50 of 0.6 nM for human Nav1.7, suitable for pain research.Formula:C25H29Cl2FN2O4SPurezza:99.87%Colore e forma:White SolidPeso molecolare:543.48Dimethylamiloride
CAS:Dimethylamiloride is a specific inhibitor of antiporters [1].Formula:C8H12ClN7OPurezza:98.90%Colore e forma:Yellow SolidPeso molecolare:257.68(Rac)-AMG8379
CAS:(Rac)-AMG8379 ((Rac)-AMG8380) is a racemate of AMG8379 which is an orally active and selective sulfonamide NaV1.7 antagonist.Formula:C25H16ClF2N3O5SPurezza:99.9%Colore e forma:White SolidPeso molecolare:543.93PF-05150122
CAS:PF-05150122 is a potent and selective human Nav1.7 channel blocker with oral activity for treating acute or chronic pain.Formula:C24H21ClN6O3S2Purezza:99.95%Colore e forma:White SolidPeso molecolare:541.04Sodium Channel inhibitor 4
CAS:Sodium Channel inhibitor 4 is a NaV1.7 inhibitor; IC50=33 nM; analgesic activity; neuropathic pain research.Formula:C19H18ClN3O4S2Purezza:99.89%Colore e forma:White SolidPeso molecolare:451.95Aneratrigine
CAS:Aneratrigine is a blocker of the sodium channel protein type 9 subunit alpha, utilized in research on neuropathic pain diseases [1].Formula:C19H20ClF2N5O2S2Purezza:98%Colore e forma:SolidPeso molecolare:487.97GNE-0439
CAS:GNE-0439 is a Nav1.7-selective inhibitor (IC50 0.34 μM), also targeting Nav1.5 and mutant N1742K channels, valuable for ion channel research.Formula:C21H31NO3Purezza:99.60%Colore e forma:White SolidPeso molecolare:345.48Ref: TM-T11437
1mg154,00€5mg371,00€1mL*10mM (DMSO)409,00€10mg620,00€25mg1.305,00€50mg1.783,00€100mg2.250,00€6-Iodoamiloride
CAS:6-Iodoamiloride is a potent inhibitor of acid-sensing ion channel 1 (ASIC1), exhibiting an IC50 value of 88 nM.Formula:C6H8IN7OPurezza:98%Colore e forma:SolidPeso molecolare:321.08PF 04531083
CAS:PF 04531083 is a selective blocker of the NaV1.8 channel. PF 04531083 can be used for neuropathic and inflammatory pain studies.Formula:C17H16ClN5O2Purezza:99.85%Colore e forma:White SolidPeso molecolare:357.79Funapide
CAS:Funapide (TV 45070) is a potent Nav1.7 inhibitor, potentially treating inflammation and various pains.Formula:C22H14F3NO5Purezza:99.91%Colore e forma:SolidPeso molecolare:429.35Ref: TM-T15358
1mg120,00€5mg289,00€1mL*10mM (DMSO)318,00€10mg439,00€25mg708,00€50mg954,00€100mg1.288,00€Aneratrigine hydrochloride
CAS:Aneratrigine hydrochloride is a Nav 1.9 blocker that may be used to prevent or treat sodium channel blocker-related disorders.Formula:C19H21Cl2F2N5O2S2Purezza:98.90% - 99.11%Colore e forma:SolidPeso molecolare:524.43VGSCs-IN-1
CAS:VGSCs-IN-1, a VGSC inhibitor and Riluzole analog, exhibits good blocking activity on Nav1.4 and can be used to study cellular excitability disorders.Formula:C12H12F3N3OSPurezza:99.92%Colore e forma:SolidPeso molecolare:303.303Nav1.8-IN-5
CAS:Nav1.8-IN-5 (Example 1), a voltage-gated sodium channel Nav1.8 inhibitor, is applicable in the research of Nav1.8-mediated diseases including pain, pain-related disorders, and cardiovascular diseases (such as atrial fibrillation) [1].Formula:C23H15F4N3O2Colore e forma:SolidPeso molecolare:441.38Nav1.8-IN-15
CAS:Nav1.8-IN-15 (compound 6) is a potent inhibitor of Nav1.8. It exhibits analgesic properties and holds potential for research in chronic pain management.Formula:C23H26ClNO4S2Colore e forma:SolidPeso molecolare:480.04Vormatrigine
CAS:Vormatrigine effectively inhibits sodium channels (sodium channel).Formula:C16H12F6N4O2Colore e forma:SolidPeso molecolare:406.28LBA-3
CAS:LBA-3, a selective and orally active inhibitor of the sodium-coupled citrate transporter SLC13A5, exhibits an IC50 of 67 nM. This compound effectively reduces triglyceride and total cholesterol levels in both oleic and palmitic acid (OPA)-stimulated AML12 cells and PCN-stimulated primary mouse hepatocytes, as well as in mouse models, without showing detectable toxicity. Additionally, LBA-3 is permeable to the blood-brain barrier [1].Formula:C18H18O5Colore e forma:SolidPeso molecolare:314.33
