Ricettore GABA
I recettori GABA sono i principali recettori dei neurotrasmettitori inibitori nel sistema nervoso centrale, svolgendo un ruolo cruciale nella regolazione dell'eccitabilità neuronale e nel mantenimento dell'equilibrio tra eccitazione e inibizione. La disfunzione dei recettori GABA è implicata in vari disturbi neurologici e psichiatrici, tra cui epilessia, ansia e depressione. Presso CymitQuimica, offriamo una gamma completa di modulatori dei recettori GABA per supportare la tua ricerca in neurobiologia, salute mentale e sviluppo terapeutico.
Trovati 362 prodotti di "Ricettore GABA"
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Flumazenil
CAS:Flumazenil (Ro 15-1788) antagonizes the benzodiazepine binding site of the gamma-aminobutyric acid (GABA)/benzodiazepine receptor complex in the central nervousFormula:C15H14FN3O3Purezza:99.72% - 99.98%Colore e forma:Less Crystals Colourless CrystalsPeso molecolare:303.29L-Cycloserine
CAS:L-Cycloserine irreversibly inhibits E. coli GABA aminotransferase, raising GABA levels, an inhibitory neurotransmitter.Formula:C3H6N2O2Purezza:99.75% - 99.99%Colore e forma:Crystals White PowderPeso molecolare:102.09Chlormezanone
CAS:<p>Chlormezanone (Trancopal) is a non-benzodiazepine that is used in the management of anxiety. It has been suggested for use in the treatment of muscle spasm.</p>Formula:C11H12ClNO3SPurezza:99.89% - >99.99%Colore e forma:Crystals SolidPeso molecolare:273.74Pivagabine
CAS:<p>Pivagabine (CXB-722), a 4-aminobutyric acid derivative, modulates GABA, CRF, and crosses the rat blood-brain barrier.</p>Formula:C9H17NO3Purezza:99.87%Colore e forma:SolidPeso molecolare:187.24Phenelzine sulfate
CAS:Phenelzine sulfate is a non-selective and irreversible inhibitor of monoamine oxidase (MAOI), and with antidepressant and anxiolytic.Formula:C8H14N2O4SPurezza:98.38% - 99.83%Colore e forma:SolidPeso molecolare:234.27γ-Aminobutyric acid
CAS:γ-Aminobutyric acid (4-Aminobutyric acid) is the most common inhibitory neurotransmitter in the central nervous system.Formula:C4H9NO2Purezza:99.95%Colore e forma:White Or Almost White(According To Quality Test Specification It Can Be White Or Almost White ) Solid PowderPeso molecolare:103.12Etifoxine hydrochloride
CAS:<p>Etifoxine hydrochloride (HOE 36-801 hydrochloride) is an anxiolytic and anticonvulsant drug.</p>Formula:C17H18Cl2N2OPurezza:99.36%Colore e forma:SolidPeso molecolare:337.24Phenibut
CAS:<p>Phenibut (Aminophenylbutyric acid) is a central depressant and derivative of the naturally occurring inhibitory neurotransmitter γ-aminobutyric acid (GABA).</p>Formula:C10H13NO2Purezza:99.55%Colore e forma:SolidPeso molecolare:179.22Baclofen
CAS:Baclofen (Lioresal), a chlorophenyl-butanoic acid derivative, treats spasms from spinal cord injury and MS by mimicking GABA at GABA-B receptors.Formula:C10H12ClNO2Purezza:98% - >99.99%Colore e forma:1992)Peso molecolare:213.66Lotilaner
CAS:<p>Lotilaner is a parasiticide.</p>Formula:C20H14Cl3F6N3O3SPurezza:99.56%Colore e forma:SolidPeso molecolare:596.763,4,5-Trimethoxycinnamic acid
CAS:3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) (TMCA) is one of the constituents of Polygalae Radix and may exert anti-seizure activity by acting at theFormula:C12H14O5Purezza:98.91%Colore e forma:SolidPeso molecolare:238.24Vigabatrin
CAS:<p>Vigabatrin (Sabril), an analogue of gamma-aminobutyric acid, is an irreversible inhibitor of 4-aminobutyrate Transaminase responsible for the catabolism of γ-</p>Formula:C6H11NO2Purezza:99.47% - 99.88%Colore e forma:SolidPeso molecolare:129.16Pentetrazol
CAS:Pentylenetetrazol is a GABA(A) receptor antagonist, that displays activity as a central nervous system and respiratory stimulant.Formula:C6H10N4Purezza:99.67% - 99.90%Colore e forma:Bitter Taste Aqueous Solutions Neutral To Litmus (Ntp 1992)Peso molecolare:138.17Bemegride
CAS:<p>Bemegride (3-Ethyl-3-methylglutarimide), a central nervous system stimulant, serves as an antidote for barbiturate poisoning.</p>Formula:C8H13NO2Purezza:99.89%Colore e forma:Physical Description White Crystalline Solid Sublimes At 212°F And 200 Mm Pressure (Ntp 1992)Peso molecolare:155.19Afoxolaner
CAS:<p>Afoxolaner is an isoxazoline insecticide/acaricide against Ixodes scapularis in dogs.</p>Formula:C26H17ClF9N3O3Purezza:99.1% - 99.38%Colore e forma:SolidPeso molecolare:625.87Fluxametamide
CAS:Fluxametamide, an isoxazoline insecticide, targets insect chloride channels with IC50s of 1.95 nM (GABA) and 225 nM (glutamate).Formula:C20H16Cl2F3N3O3Purezza:99.49%Colore e forma:SolidPeso molecolare:474.26Nikethamide
CAS:Nikethamide is a stimulant which mainly influences the respiratory cycle. Widely known by its former sales name of Coramine, it was used in the mid-twentieth century as a medical countermeasure against tranquilizer overtreatments, before the advent of endFormula:C10H14N2OPurezza:99.42%Colore e forma:Followed By A Faint Sensation Of The Warmth (Ntp 1992)Peso molecolare:178.23Nefiracetam
CAS:Nefiracetam (DM9384), in Phase 2 trials, enhances GABA, choline, monoamine systems, and treats Ro 5-4864 convulsions.Formula:C14H18N2O2Purezza:97.37%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:246.3GET73
CAS:<p>GET73 (Gamma hydroxybutyric acid analogue) is an negative allosteric modulator of mGluR5.</p>Formula:C13H16F3NO2Purezza:99.54%Colore e forma:SolidPeso molecolare:275.27Domperidone EP Impurity A
CAS:Domperidone EP Impurity A is used as pharmaceutical intermediates.Formula:C12H14ClN3OPurezza:99.97%Colore e forma:SolidPeso molecolare:251.71Oxiracetam
CAS:<p>Oxiracetam (ISF2522), a cyclic derivative of gamma-aminobutyric acid (GABA), is utilized for the treatment of cognitive impairments.</p>Formula:C6H10N2O3Purezza:99.67%Colore e forma:White Crystalline PowderPeso molecolare:158.16NEO 376
CAS:<p>NEO 376 (SPI-376) is a selective 5-HT1 receptor, GABA receptor and dopamine receptor modulator, showing anti-psychotic actively.</p>Formula:C20H24ClN3OPurezza:99.56%Colore e forma:SolidPeso molecolare:357.88Emamectin Benzoate
CAS:<p>Emamectin Benzoate (MK-244), by binding gamma-aminobutyric acid (GABA) receptor and glutamate-gated chloride channels disrupting nerve signals within arthropods</p>Formula:C56H81NO15Purezza:98.68%Colore e forma:SolidPeso molecolare:1008.256Clomethiazole
CAS:Clomethiazole (Distraneurin) is an orally active GABAA agonist and it is an anticonvulsant agent. It has potential for treating convulsive status epilepticus.Formula:C6H8ClNSPurezza:99.06%Colore e forma:SolidPeso molecolare:161.65Topiramate
CAS:<p>Topiramate (RWJ 17021) is a unique antiseizure medication that is used in the treatment of partial and generalized seizures.</p>Formula:C12H21NO8SPurezza:99.79% - 99.92%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:339.36Broflanilide
CAS:<p>Broflanilide metabolite desmethyl-broflanilide blocks GABA receptor in dieldrin-resistant insects, inhibiting S. litura at IC50 1.3 nM.</p>Formula:C25H14BrF11N2O2Purezza:99.82%Colore e forma:SolidPeso molecolare:663.29GABAA receptor agent 1
CAS:<p>GABAA receptor agent 1 has strong anticonvulsant activity and is a high affinity ligand of GABAA receptor.</p>Formula:C13H8ClN3O2Purezza:99.31%Colore e forma:SolidPeso molecolare:273.67Isoguvacine hydrochloride
CAS:<p>Isoguvacine hydrochloride (1,2,3,6-tetrahydro-4-pyridinecarboxylic acid hydrochloride) is a GABA receptor agonist.</p>Formula:C6H10ClNO2Purezza:99.59%Colore e forma:SolidPeso molecolare:163.6LAU159
CAS:<p>LAU159 is a functionally selective positive α1β3 GABA(A) receptor modulator(EC50 : 2.2 μM).</p>Formula:C17H12ClN3O2Purezza:98.7% - 99.38%Colore e forma:SolidPeso molecolare:325.75FG 7142
CAS:<p>FG 7142 (LSU-65), a benzodiazepine inverse agonist, targets α1 subunit GABAA receptors (EC50=137 nM, Ki=91 nM) and upregulates β-adrenoceptors.</p>Formula:C13H11N3OPurezza:98.75%Colore e forma:SolidPeso molecolare:225.25Neurotransmitter Receptor Compound Library
<p>A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening；</p>Colore e forma:Odour SolidCinazepam
CAS:Cinazepam is a GABAA receptor partial agonist and a benzodiazepine derivative with anxiolytic and sedative properties. Cinazepam can be utilized in research related to sleep disorders.Formula:C19H14BrClN2O5Colore e forma:SolidPeso molecolare:465.68Azocarnil
<p>Azocarnil is a GABAergic agonist-enhancer used in neurological system research.</p>Colore e forma:Odour SolidMIDD0301
CAS:<p>MIDD0301 is a potent positive allosteric α5β3γ selective GABAA receptor (GABAAR) ligand with EC50 of 17 nM.</p>Formula:C19H13BrFN3O2Purezza:98%Colore e forma:SolidPeso molecolare:414.23Anisatin
<p>Anisatin is a useful organic compound for research related to life sciences and the catalog number is T124719.</p>Formula:C15H20O8Colore e forma:SolidPeso molecolare:328.317DAA-1106
CAS:DAA-1106 is a potent and selective ligand for PBR, acting as a potent and selective agonist at the peripheral benzodiazepine receptor.Formula:C23H22FNO4Purezza:99.54%Colore e forma:SolidPeso molecolare:395.42Nipecotic acid
CAS:<p>Compound PDK0243, with CAS No. 498-95-3, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0243 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.</p>Formula:C6H11NO2Colore e forma:Off-White To Pale Yellow-Beige PowderPeso molecolare:129.16Endosulfan I
CAS:<p>Endosulfan I is one of the two major stereoisomers of the broad-spectrum insecticide Endosulfan inhibi the GABA/benzodiazepine/picrotoxin complex</p>Formula:C9H6Cl6O3SPurezza:99.86%Colore e forma:SolidPeso molecolare:406.93Furosemide
CAS:Furosemide is a potent NKCC2 (Na-K-2Cl symporter) inhibitor, used for edema and chronic renal insufficiency.Formula:C12H11ClN2O5SPurezza:99.32% - 99.89%Colore e forma:Crystals From Aqueous Ethanol Tasteless (Ntp 1992)Peso molecolare:330.744Inaperisone
CAS:Inaperisone: a novel muscle relaxant that indirectly inhibits voiding reflex via brainstem GABAB receptors.Formula:C16H23NOPurezza:98.83%Colore e forma:SolidPeso molecolare:245.36Brexanolone caprilcerbate
CAS:Brexanolone caprilcerbate is an effective positive allosteric modulator of the GABAA receptor.Formula:C48H78O12Colore e forma:SolidPeso molecolare:847.13CGP 35348
CAS:CGP 35348 是 GABAB 受体的选择性拮抗剂 (EC50 = 34 μM)。 CGP 35348 可用于研究白化新生小鼠脑损伤后的神经肌肉协调和空间学习。Formula:C8H20NO4PPurezza:≥98%Colore e forma:SolidPeso molecolare:225.22Furosemide sodium
CAS:<p>Furosemide sodium: potent NKCC inhibitor, loop diuretic, treats heart failure, hypertension, edema, selective GABAA antagonist.</p>Formula:C12H10ClN2NaO5SPurezza:99.52% - >99.99%Colore e forma:SolidPeso molecolare:352.7312,14-Dichlorodehydroabietic acid
CAS:12,14-Dichlorodehydroabietic acid activates BK channels, blocks GABA A receptors, and increases calcium and neurotransmitter release.Formula:C20H26Cl2O2Colore e forma:SolidPeso molecolare:369.33Fipronil sulfone
CAS:Fipronil sulfone is an insecticide fipronil. Its metabolite fipronil sulphone is an inhibitor of rat ɑ1β2γ2L GABA(A) receptor.Formula:C12H4Cl2F6N4O2SPurezza:98%Colore e forma:SolidPeso molecolare:453.14Chrodrimanin B
CAS:<p>Chrodrimanin B is a useful organic compound for research related to life sciences. The catalog number is T126052 and the CAS number is 132196-54-4.</p>Formula:C27H32O8Colore e forma:SolidPeso molecolare:484.545KGP-25
KGP-25 is an inhibitor of the voltage-gated sodium channel 1.8 (Nav1.8), utilized for analgesia by targeting the peripheral nervous system (PNS). Additionally, it targets the γ-aminobutyric acid subtype A receptor (GABAA) in the central nervous system (CNS) for use as a general anesthetic.3-Hydroxy desalkylflurazepam
CAS:3-Hydroxy desalkylflurazepam is a benzodiazepine compound with potential sedative and anxiolytic effects.Formula:C15H10ClFN2O2Colore e forma:SolidPeso molecolare:304.7γ-Acetylenic GABA hydrochloride
CAS:γ-Acetylenic GABA hydrochloride is a GABA transaminase inhibitor.Formula:C6H10ClNO2Purezza:97.83% - 99.28%Colore e forma:SolidPeso molecolare:163.6GABA-A Receptor Ligand-1
GABA-A Receptor Ligand-1 (Compound 4) is a ligand for the GABA-A receptor with a pKi of 7.27. It alleviates mitochondrial dysfunction, promotes neurite outgrowth and neuronal regeneration, and demonstrates neuroprotective effects in a rat ischemic stroke model.Formula:C20H20FN3OColore e forma:SolidPeso molecolare:337.3915α-Androst-16-en-3α-ol
CAS:5α-Androst-16-en-3α-ol is a steroid pheromone that has been found in boar testes and human male axillary sweat and has diverse biological activities.1,2ItFormula:C19H30OColore e forma:SolidPeso molecolare:274.448Riluzole-13C,15N2
CAS:<p>Riluzole-13C,15N2 (PK 26124-13C,15N2) is a 13C and 15N labeled form of Riluzole, a glutamate antagonist with anticonvulsant activity, inhibiting GABA uptake.</p>Formula:CC7H5F3OS15N2Colore e forma:SolidPeso molecolare:237.18GABA-IN-1
GABA-IN-1 (Compound 6), a GABA inhibitor, exhibits larvicidal and insecticidal properties, achieving a mortality rate of 93% at a concentration of 50 mg/L [1].Colore e forma:Odour SolidDesalkylgidazepam
CAS:Desalkylgidazepam, a benzodiazepine compound, is a metabolite of gidazepam. It is capable of activating both GABA A-type receptors and the translocator protein (TSPO).Formula:C15H11BrN2OColore e forma:SolidPeso molecolare:315.17AHN-683
CAS:AHN-683 is a fluorescent ligand. It was used for peripheral-type benzodiazepine receptors.Formula:C42H32FN3O7Purezza:98%Colore e forma:SolidPeso molecolare:709.72RuBi-GABA
CAS:Ruthenium-bipyridine-triphenylphosphine caged GABAFormula:C42H39F6N5O2P2RuPurezza:98%Colore e forma:SolidPeso molecolare:922.83-(4-Chlorophenyl)-4-hydroxybutyric Acid (sodium salt)
CAS:3-(4-Chlorophenyl)-4-hydroxybutyric Acid (sodium salt) can be used in related research in the field of life sciences.Formula:C10H10ClNaO3Colore e forma:SolidPeso molecolare:236.63α5-GABAA receptor modulator 1
α5-GABAA receptor modulator 1 (Compound A-4) is a selective silent allosteric modulator (SAM) targeting the α5 subunit of GABAA receptors, useful for research into central nervous system (CNS) disorders.Formula:C21H20FN3O4Colore e forma:SolidPeso molecolare:397.4S-8510 free base
CAS:S-8510 is a GABA-A receptor inverse agonist enhancing memory, LTP, and neurotransmitters in rats.Formula:C12H10N4O2Colore e forma:SolidPeso molecolare:242.23Anticonvulsant agent 8
Anticonvulsant agent 8 (compound D4) is a chemical used in treating epilepsy by inhibiting GABAA currents. In mouse models, its ED50 values are 2.23 mg/kg for the maximal electroshock (MES) test and 24.60 mg/kg for the pentylenetetrazol (PTZ) test.Formula:C15H11N5OColore e forma:SolidPeso molecolare:277.28GABAA receptor modulator-3
GABAA receptor modulator-3 (compound 3b) is a positive allosteric modulator (PAM). It inhibits the peak current and steady-state current of α1β3γ2 GABAAR with IC50 values of 671 μM and 64 μM, respectively.Formula:C18H22O2Colore e forma:SolidPeso molecolare:270.37Anticonvulsant agent 9
<p>Anticonvulsant agent 9 (compound 4f) is an activator of the α1β2γ2GABA_A receptor, with an EC50 value of 1.24 μM. It inhibits the inactivation of Nav1.2 channels and exhibits significant anticonvulsant activity.</p>Formula:C22H24N4O2Colore e forma:SolidPeso molecolare:376.45Sandaracopimaric acid
CAS:Sandaracopimaric acid, an anti-inflammatory diterpene, relaxes pulmonary arteries with an EC50 of 43.93 μM.Formula:C20H30O2Colore e forma:SolidPeso molecolare:302.45GABAA receptor modulator-4
<p>GABAA receptor modulator-4 (Compound 4) acts as a negative allosteric modulator of the GABAA receptor. It inhibits the peak and steady-state currents mediated by the α1β3γ2 GABAA receptors, with an IC50 of 10 μM for both.</p>Formula:C15H17BrO4SColore e forma:SolidPeso molecolare:373.26LU-32-176B
CAS:LU32-176B is a bioactive chemical.Formula:C23H24F2N2O2Colore e forma:SolidPeso molecolare:398.453-Aminopropylphosphinic acid
CAS:<p>3-Aminopropylphosphinic acid (3-APPA) is a phosphonic analog of gamma-aminobutyric acid (GABA).</p>Formula:C3H10NO2PColore e forma:SolidPeso molecolare:123.092(Iso)-Atagabalin HCl
CAS:<p>(Iso)-Atagabalin HCl(isomer-Atagabalin HCl) is an alpha -2- delta ligand that can be used to treat non-restorative sleep.</p>Formula:C10H20ClNO2Purezza:99.26% - >99.99%Colore e forma:SoildPeso molecolare:221.72FGIN-1-43
CAS:FGIN-1-43 is a potent and specific ligand for the mitochondrial DBI receptor.Formula:C28H36Cl2N2OPurezza:99.57%Colore e forma:SolidPeso molecolare:487.5Imagabalin
CAS:Imagabalin is an active compound used in the study of neurological diseases.Formula:C9H19NO2Colore e forma:SolidPeso molecolare:173.25Flufiprole
CAS:Flufiprole is used as a phenylpyrazole pesticide. It has enantioselective metabolism in human and rat liver microsomes.Formula:C16H10Cl2F6N4OSColore e forma:SolidPeso molecolare:491.24(1S,3R)-3-Aminocyclopentane carboxylic acid
CAS:<p>(1S,3R)-3-Aminocyclopentane carboxylic acid exhibits activity on GABAA receptors.</p>Formula:C6H11NO2Colore e forma:SolidPeso molecolare:129.16Antidepressant agent 3
Agent 3: orally active, antidepressant, anxiolytic, boosts performance and cognition.Formula:C17H30ClN5O2SColore e forma:SolidPeso molecolare:403.97Nitrazolam
CAS:Nitrazolam is a benzodiazepine compound that may exhibit central nervous system depressant properties similar to traditional benzodiazepine drugs by acting on the GABA receptors (GABA receptor). These effects include sedation, hypnosis, anxiolytic, and anticonvulsant activities.Formula:C17H13N5O2Colore e forma:SolidPeso molecolare:319.32Withasomniferolide B
CAS:<p>Withasomniferolide B, a withanolide from Withania somnifera root, activates GABAA receptors.</p>Formula:C28H36O4Colore e forma:SolidPeso molecolare:436.58Antidepressant agent 4
Antidepressant agent 4: orally active, has antidepressant, anxiolytic, and nootropic effects.Formula:C19H38ClN5O2SColore e forma:SolidPeso molecolare:436.06Lesogaberan napadisylate
CAS:Lesogaberan (AZD-3355) is a selective GABAB agonist with EC50 of 8.6 nM, Ki of 5.1 nM in rats, and acts peripherally on the esophageal sphincter.Formula:C13H17FNO5PSColore e forma:SolidPeso molecolare:349.31epi-Aszonalenin A
CAS:epi-Aszonalenin A: a psychoactive benzodiazepine from Aspergillus novofumigatus.Formula:C25H25N3O3Colore e forma:SolidPeso molecolare:415.48Rilmazolam
CAS:Rilmazolam is a triazolobenzodiazepine compound and serves as the active metabolite of Rilmazafone.Formula:C19H15Cl2N5OColore e forma:SolidPeso molecolare:400.266,7-dimethylisatin
CAS:6,7-Dimethylisatin (6,7-dimethyl-1H-indole-2,3-dione) inhibits hGAT3 with IC50 of 108 μM. 6,7-Dimethylisatin also inhibits hBGT1, hGAT2.Formula:C10H9NO2Purezza:98.98%Colore e forma:SolidPeso molecolare:175.18Pyrazolam
CAS:Pyrazolam is a psychoactive benzodiazepine compound serving as a central nervous system depressant. [Pyrazolam] can lead to psychomotor impairment.Formula:C16H12BrN5Colore e forma:SolidPeso molecolare:354.2α-Casozepine
CAS:<p>α-Casozepine,Bioactive peptide from milk α-S1 casein. Binds GABA receptors. Anti-anxiety effects.</p>Formula:C60H94N14O16Colore e forma:SolidPeso molecolare:1267.47GABA receptor Antagonist 1
GABA receptor Antagonist 1 (compound 7w) effectively inhibits the Px RDL1 GABAR at an IC50 of 7.08 nmol/L and demonstrates insecticidal efficacy against P.Purezza:98%Colore e forma:Odour SolidTET-13
<p>TET-13 is a positive allosteric modulator of the GABAA receptor with an EC50 of 5.65 μM, which is more potent than Etomidate (EC50: 9.29 μM). It exhibits strong anesthetic effects in both mice and rats, with an ED50 of 0.48 mg/kg in mice and 0.69 mg/kg in rats.</p>Formula:C15H16N2O3SColore e forma:SolidPeso molecolare:304.36Guvacine hydrobromide
CAS:<p>Guvacine hydrobromide, an alkaloid derived from the Areca catechu nut, serves as a potent inhibitor of GABA (GABA uptakp) uptake.</p>Formula:C6H10BrNO2Purezza:98%Colore e forma:SolidPeso molecolare:208.053-Aminopropylphosphonic Acid
CAS:<p>3-aminopropylphosphonic acid (3-APPA) is a phosphonic analog of GABA that acts as a partial agonist of GABAB receptors (IC50 = 1.5 μM in a radioligand binding</p>Formula:C3H10NO3PPurezza:99.84%Colore e forma:Light Yellow LiquidPeso molecolare:139.09Emamectin B1a
CAS:<p>Emamectin B1a can be used in relevant research in the life sciences. Its product number is T37663 and CAS number is 121124-29-6.</p>Formula:C49H75NO13Colore e forma:SolidPeso molecolare:886.133Ion Channel Targeted Library
<p>A unique collection of 931 compounds targeting ion channels for research in ion channels-related diseases and ion channel drug discovery;</p>Colore e forma:Odour SolidAtagabalin
CAS:Atagabalin (PD 0200390), a gabamimetic for insomnia treatment and related to gabapentin, was halted due to poor trial outcomes.Formula:C10H19NO2Colore e forma:SolidPeso molecolare:185.26Furosemide-d5
CAS:Furosemide-d5 is a deuterium marker for Furosemide and used in isotope tracer experiments. orally active inhibitor of Na+/K+/2Cl- (NKCC) diuretic reagent.Formula:C12H11ClN2O5SColore e forma:SolidPeso molecolare:335.78Propanidid
CAS:Propanidid (Sombrevin) is a gamma-aminobutyric acid type A receptor (GABAA) agonist and an intravenous anesthetic that lowers arterial blood pressure.Formula:C18H27NO5Purezza:99.64%Colore e forma:SolidPeso molecolare:337.41(-)-α-Pinene
CAS:(-)-α-Pinene ((1S)-(-)-Alpha-Pinene) enhances the quantity of NREMS without affecting the intensity of NREMS by prolonging GABAergic synaptic transmission,Formula:C10H16Purezza:98.02% - 98.60%Colore e forma:Colourless LiquidPeso molecolare:136.23MRK-016
CAS:MRK-016 is a selective GABAA α5 receptor inverse agonist/ negative allosteric modulator, orally available and penetrating the BBB. MRK-016 is antidepressant.Formula:C17H20N8O2Purezza:99.76%Colore e forma:SolidPeso molecolare:368.39Dipropofol
CAS:<p>Dipropofol (4,4-Bis(2,6-di-isopropylphenol)) is a small molecule GABAA receptor agonist that can be used to study epilepsy.</p>Formula:C24H34O2Purezza:99.51%Colore e forma:SolidPeso molecolare:354.53Padsevonil
CAS:Padsevonil (UCB-0942) is a potential GABA A receptor orthosteric modulator with antiepileptic activity for the treatment of epilepsy.Formula:C14H14ClF5N4O2SPurezza:99.63%Colore e forma:SolidPeso molecolare:432.80CGP 36742
CAS:CGP 36742 blocks GABAB receptor, crosses blood-brain barrier, aids depression treatment (IC50: 32 μM).Formula:C7H18NO2PColore e forma:SolidPeso molecolare:179.2Vigabatrin Hydrochloride
CAS:Vigabatrin Hydrochloride (γ-Vinyl-GABA hydrochloride) is a structural analog of the GABA, irreversibly inhibiting the catabolism of GABA by GABA transaminase.Formula:C6H11NO2·HClPurezza:98%Colore e forma:SolidPeso molecolare:165.62L-655708
CAS:L-655708 is a selective and highly potent GABAA receptor reverse agonist with a Ki value of 0.45 nM.Formula:C18H19N3O4Purezza:99.36%Colore e forma:PowderPeso molecolare:341.36Valnoctamide
CAS:Valnoctamide (Valmethamide) has antiepileptic and anticonvulsant activity and may be used in the study of neurological disorders.Formula:C8H17NOPurezza:98%Colore e forma:SolidPeso molecolare:143.23Etifoxine
CAS:Etifoxine targets β2/β3 GABAA receptors, is anxiolytic in humans/rodents, boosts GABAA, binds TSPO, aids axon regeneration, no sedative effects.Formula:C17H17ClN2OPurezza:98%Colore e forma:SolidPeso molecolare:300.78Primidone (Standard)
CAS:Primidone (Standard) is the standard substance of Primidone, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Primidone (NCI-C56360) is a potent anticonvulsant agent. It is a neuronal voltage-gated sodium channel blocker and has value in the study of epilepsy, essential tremor, and psychiatric disorders.Formula:C12H14N2O2Peso molecolare:218.25Fipronil
CAS:Fipronil (Fluocyanobenpyrazole) is a broad-use insecticide that belongs to the phenylpyrazole chemical family.Formula:C12H4Cl2F6N4OSPurezza:97.21%Colore e forma:Solid PowderPeso molecolare:437.15Acamprosate calcium
CAS:Acamprosate calcium (Campral EC) is a GABA receptor agonist and modulator of glutamatergic systems, used for treating alcohol dependence.Formula:C10H20CaN2O8S2Purezza:98% - 99.93%Colore e forma:White Odorless Or Nearly Odorless PowderPeso molecolare:400.48Acetoxyvalerensre
CAS:<p>Acetoxyvalerensre (acetylvalerenolic acid) (acetylvalerenolic acid) is a derivative of valerenic acid, which is a a GABAA receptor modulator.</p>Formula:C17H24O4Purezza:98.22%Colore e forma:SolidPeso molecolare:292.37Piperazine citrate
CAS:<p>Piperazine citrate, an organic compound, consists of a six-membered ring, containing two nitrogen atoms at opposite positions in the ring.</p>Formula:C24H46N6O14Purezza:99.8%Colore e forma:Crystals IndicationPeso molecolare:642.65AZD7325
CAS:<p>AZD7325 (AZD-7325) is a GABA-Aα2,3 -selective receptor modulator.</p>Formula:C19H19FN4O2Purezza:99.83%Colore e forma:SolidPeso molecolare:354.38Ginkgolide A
CAS:<p>Ginkgolide A (BN-52020), from Ginkgo biloba leaves, is an active PAF antagonist with potential in treating inflammation and immune disorders.</p>Formula:C20H24O9Purezza:98.76% - 99.81%Colore e forma:White PowderPeso molecolare:408.4Guvacine hydrochloride
CAS:<p>Guvacine hydrochloride is an inhibits of GABA uptake (IC50 : 10 μM)</p>Formula:C6H10ClNO2Purezza:98.42%Colore e forma:SolidPeso molecolare:163.602CL 218872
CAS:CL 218872: selective α1 GABAA receptor agonist, anxiolytic, and anticonvulsant; Ki=130 nM for α1, less potent for α2-α6.Formula:C13H9F3N4Purezza:99.92%Colore e forma:SolidPeso molecolare:278.23Pipequaline hydrochloride
CAS:<p>Pipequaline hydrochloride (PK-8165 hydrochloride) is an anticonflict & anticonvulsant quinoline derivative.</p>Formula:C22H25ClN2Purezza:99.46%Colore e forma:SolidPeso molecolare:352.9Arecaidine hydrochloride
CAS:Arecaidine hydrochloride may have carcinogenesis.Formula:C7H12ClNO2Purezza:99.69% - ≥95%Colore e forma:SolidPeso molecolare:177.63(R)-baclofen
CAS:<p>(R)-baclofen (STX209), a derivative of gamma-aminobutyric acid, is commonly utilized for the treatment of spasticity.</p>Formula:C10H12ClNO2Purezza:97.20% - 98.94%Colore e forma:SolidPeso molecolare:213.66Ocinaplon
CAS:<p>Ocinaplon (DOV 273547) is a GABAA receptors modulator.</p>Formula:C17H11N5OPurezza:99.81%Colore e forma:SolidPeso molecolare:301.3L-DABA
CAS:<p>L-DABA (L-2,4-Diaminobutyric acid) is an inhibitor of GABA transaminase (IC50 > 500 μM).</p>Formula:C4H10N2O2Purezza:99.32%Colore e forma:SolidPeso molecolare:118.13Kavain
CAS:<p>Kavain, a compound extracted from the Kava plant, Piper methysticum, is found to be involved in TNF-α expression in human and mouse cells via regulation of</p>Formula:C14H14O3Purezza:99.93% - ≥95%Colore e forma:SolidPeso molecolare:230.26Songorine
CAS:Songorine (Napellonine) shows anti-tumor activity in preliminary pharmacological verification trials including cell proliferation and molecular docking assays.Formula:C22H31NO3Purezza:98% - 99.92%Colore e forma:SolidPeso molecolare:357.49AZD-6280
CAS:AZD6280 is a novel, subtype-selective GABAAα2/3 receptor positive modulators, used for treatment of generalized anxiety disorder.Formula:C20H22N4O3Purezza:98.99%Colore e forma:SolidPeso molecolare:366.41Cholesterol myristate
CAS:<p>Cholesterol myristate, a natural steroid in Chinese medicine, affects GABAA, nicotinic receptors, and potassium channels.</p>Formula:C41H72O2Purezza:99.65%Colore e forma:SolidPeso molecolare:597.01α-Thujone
CAS:α-Thujone is an inhibitor of ACh with an IC50 value of 24.7μM.Formula:C10H16OPurezza:97.02% - 98.41%Colore e forma:Less Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996) Colorless Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996)Peso molecolare:152.23(2S)-6-Prenylnaringenin
CAS:(2S)-6-Prenylnaringenin (6-Prenylnaringenin) is an isomer of the potent phytoestrogen, 8-prenylnaringenin.Formula:C20H20O5Purezza:99.47%Colore e forma:SolidPeso molecolare:340.37Temgicoluril
CAS:<p>Temgicoluril (mebikar) acts on GABA Receptor.</p>Formula:C8H14N4O2Purezza:99.8%Colore e forma:SolidPeso molecolare:198.226-Aminonicotinic acid
CAS:<p>6-Aminonicotinic acid is a natural product.</p>Formula:C6H6N2O2Purezza:99.94%Colore e forma:SoildPeso molecolare:138.1238rac-BHFF
CAS:<p>rac-BHFF, a GABA B receptor modulator, boosts GABA potency >15x, efficacy >149%, has anxiolytic effects, and is orally active.</p>Formula:C17H21F3O3Purezza:99.69% - >99.99%Colore e forma:SolidPeso molecolare:330.34α-Asarone
CAS:<p>alpha-Asarone (trans-Asarone) is a psychoactive compound with antidepressant-like activity in mice.</p>Formula:C12H16O3Purezza:99.64% - 99.64%Colore e forma:Monoclinic Needles From Water Monoclinic Needles From WaterPeso molecolare:208.25Thiocolchicoside
CAS:<p>Thiocolchicoside, a muscle relaxant, has anti-inflammatory and analgesic properties; not for seizure-prone people.</p>Formula:C27H33NO10SPurezza:99.11% - 99.39%Colore e forma:SolidPeso molecolare:563.62γ-Acetylenic GABA
CAS:<p>γ-Acetylenic GABA (4-Aminohex-5-ynoic acid) is a potent, irreversible inhibitor of GABA-transaminase.</p>Formula:C6H9NO2Colore e forma:SolidPeso molecolare:127.143Tiagabine hydrochloride
CAS:<p>Tiagabine hydrochloride, a nipecotic acid derivative, is an anticonvulsant and selective GABA reuptake inhibitor.</p>Formula:C20H25NO2S2·HClPurezza:99.09% - 99.77%Colore e forma:White To Off-White SolidPeso molecolare:412.01Gabazine free base
CAS:Gabazine free base is a specific antagonist of the GABA receptor. It does not affect GABA-transaminase or glutamate-decarboxylase activities.Formula:C15H17N3O3Colore e forma:SolidPeso molecolare:287.31Lorediplon
CAS:Lorediplon is a novel hypnotic drug acting as a GABAA receptor modulator, differentially active at the α1-subunit, associated with promoting sleep.Formula:C20H15FN4O2SPurezza:99.12% - 99.19%Colore e forma:SolidPeso molecolare:394.42Loreclezole hydrochloride
CAS:Loreclezole hydrochloride is an antiepileptic, enhancing GABA A receptors with β2/β3 subunits.Formula:C10H7Cl4N3Colore e forma:SolidPeso molecolare:310.99Tiagabine hydrochloride hydrate
CAS:Tiagabine HCl hydrate, IC50: 67-446 nM, selectively inhibits GABA uptake, acts as an anticonvulsant.Formula:C20H28ClNO3S2Colore e forma:SolidPeso molecolare:430.022'MeO6MF
CAS:2'MeO6MF is a brain-penetrant positive allosteric modulator at α2β1γ2L and all α1-containing GABAA receptors.It offers neuroprotection and improved functionalFormula:C17H14O3Purezza:99.28% - 99.63%Colore e forma:SolidPeso molecolare:266.29Piperazine
CAS:Piperazine (1,4-Diazacyclohexane), a gamma-aminobutyric acid (GABA) agonist, serves as a crucial building block and core component in a wide range of marketed drugs known for their varied pharmacological activities.Formula:C4H10N2Colore e forma:SolidPeso molecolare:86.14Pikamilone
CAS:Pikamilone (Picamilon) is an intelligent medicine.Formula:C10H12N2O3Purezza:99.38%Colore e forma:White Crystalline PowderPeso molecolare:208.21(+)-Kavain
CAS:(+)-Kavain ((R)-KAWAIN) is one of the six major kavalactones found in the Piper methysticum (kava) plant; reversible inhibitor of MAO-B.Formula:C14H14O3Purezza:97% - ≥95%Colore e forma:White Fine PowderPeso molecolare:230.26(-)-Securinine
CAS:<p>(-)-Securinine (Securinine) is plant-derived alkaloid and also a GABAA receptor antagonist.</p>Formula:C13H15NO2Purezza:99.58% - 99.87%Colore e forma:SolidPeso molecolare:217.26Isonipecotic acid
CAS:Isonipecotic acid (4-Piperidinecarboxylic acid) is a heterocyclic compound. Isonipecotic acid mainly characterized as a GABAA receptor partial agonist.Formula:C6H11NO2Purezza:99.82%Colore e forma:White To Faint Pink-Beige PowderPeso molecolare:129.16SKF89976A hydrochloride
CAS:<p>SKF89976A hydrochloride (d,l-SKF89976A hydrochloride) is a selective inhibitor GABA transporter such as GAT-1 (IC50s = 0.28 μM), GAT-2 (IC50s = 137.34 μM) and</p>Formula:C22H26ClNO2Purezza:98.02%Colore e forma:SolidPeso molecolare:371.9Miltirone
CAS:Miltirone is a CYPs inhibitor, it has been characterized as a low-affinity ligand for central benzodiazepine receptors.Formula:C19H22O2Purezza:99.22% - 99.66%Colore e forma:SolidPeso molecolare:282.38Phenibut (hydrochloride)
CAS:Phenibut hydrochloride (3-Amino-4-phenylbutyric acid hydrochloride) is a GABA mimetic that acts as an agonist at GABAB receptors.Formula:C10H14ClNO2Purezza:99.93%Colore e forma:White Crystalline PowderPeso molecolare:215.684-Acetamidobutanoic acid
CAS:4-Acetamidobutanoic acid, a GABA derivative in eukaryotes, found in blood, feces, urine, and human prostate.Formula:C6H11NO3Purezza:98.51%Colore e forma:SolidPeso molecolare:145.16CGP52432
CAS:CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM).Formula:C15H24Cl2NO4PPurezza:98.75%Colore e forma:SolidPeso molecolare:384.24(E)-3,4,5-Trimethoxycinnamic acid
CAS:<p>(E)-3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) is a natural product from the roots and rhizomes of Notopterygium incisum.</p>Formula:C12H14O5Purezza:99.83%Colore e forma:SolidPeso molecolare:238.24Imidazenil
CAS:<p>Imidazenil is an modulator of GABA-A that blocks the sedative effects without lowering the convulsion threshold.</p>Formula:C18H12BrFN4OPurezza:98.4%Colore e forma:SolidPeso molecolare:399.22Isoflurane
CAS:Isoflurane (Forane) is a stable, non-explosive inhalation anesthetic that has been reported to induce caspase-3 activation.Formula:C3H2ClF5OPurezza:98%Colore e forma:Clear Colorless Liquid LiquidPeso molecolare:184.49Cyclothiazide
CAS:<p>Cyclothiazide enhances AMPA receptors, prevents desensitization, and boosts glutamic acid response (EC50 = 3.8µM).</p>Formula:C14H16ClN3O4S2Purezza:98.23% - 99.49%Colore e forma:Crystals From Dilute Alcohol SolidPeso molecolare:389.88SSD114 HCl
CAS:<p>SSD114 is a novel GABAB receptor positive allosteric modulator.</p>Formula:C18H21ClF3N3OPurezza:99.03% - 99.95%Colore e forma:SolidPeso molecolare:387.83p-Hydroxybenzaldehyde
CAS:1.Formula:C7H6O2Purezza:99.05% - 99.86%Colore e forma:SolidPeso molecolare:122.12Aminooxyacetic acid hemihydrochloride
CAS:Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABAFormula:C2H5NO3·5HClPurezza:98.03%Colore e forma:Light Beige Crystalline PowderPeso molecolare:109.3Amentoflavone
CAS:Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications.Formula:C30H18O10Purezza:98.21% - 99.22%Colore e forma:Odourless Whitish SolidPeso molecolare:538.46Tiagabine
CAS:Tiagabine (NO050328) is an Anti-epileptic Agent.Formula:C20H25NO2S2Purezza:99.25% - 99.67%Colore e forma:White To Off-White Crystalline SolidPeso molecolare:375.55Gaboxadol hydrochloride
CAS:Gaboxadol (hydrochloride) is a GABAA receptor agonist.Formula:C6H9ClN2O2Purezza:99.39%Peso molecolare:176.601SKF89976A HCl
CAS:SKF89976A: GABA uptake inhibitor, selective for GAT-1, passes blood-brain barrier, active in vivo (IC50: 0.13 μM hGAT-1).Formula:C22H25NO2Colore e forma:SolidPeso molecolare:335.44Gabazine
CAS:Gabazine (SR95531) is an antagonist of GABAA receptors (Ki : 74-150 nM)Formula:C15H18BrN3O3Purezza:98.51% - 99.24%Colore e forma:SolidPeso molecolare:368.236-(4-Methoxyphenyl)-3-pyridazinamine
CAS:6-(4-Methoxyphenyl)-3-pyridazinamine is a GABAA receptor antagonistFormula:C11H11N3OPurezza:99.03%Colore e forma:SolidPeso molecolare:201.222'-O-Methylisoliquiritigenin
CAS:2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-Formula:C16H14O4Purezza:98.75%Colore e forma:SolidPeso molecolare:270.28Baclofen hydrochloride
CAS:Baclofen HCL, a GABA-B agonist, treats muscle spasticity by reducing excitatory transmission.Formula:C10H13Cl2NO2Purezza:99.55%Colore e forma:SolidPeso molecolare:250.1226-Methylflavone
CAS:6-Methylflavone is an activator of α1β2γ2L and α1β2 GABAA receptors.Formula:C16H12O2Purezza:99.69%Colore e forma:SolidPeso molecolare:236.27DL-Menthol
CAS:DL-Menthol ((±)-Menthol) is a racemic mixture of the monoterpene alcohols (–)-menthol and (+)-menthod, which have been found in Cannabis.Formula:C10H20OPurezza:99.74%Colore e forma:White Crystals /89-78-1/ Physical Description White Crystalline Solid With A Peppermint Odor And Taste (Ntp 1992)Peso molecolare:156.27Saclofen
CAS:<p>Saclofen is a GABA analog and GABAB receptor antagonist, useful for studying inhibitory brain signals. IC50: 7.8 μM.</p>Formula:C9H12ClNO3SPurezza:99.17%Colore e forma:White Crystalline SolidPeso molecolare:249.71Imepitoin
CAS:<p>Imepitoin (AWD 131-138), a new low-affinity partial benzodiazepine receptor agonist, shows potent anticonvulsant and anxiolytic properties in rodent models.</p>Formula:C13H14ClN3O2Purezza:99.82%Colore e forma:SolidPeso molecolare:279.72U93631
CAS:GABAA antagonist; binds picrotoxin site, stabilizes inactive channel. Speeds GABA-induced Cl- decay, minor peak effect. Inhibits 5-HT3A receptors.Formula:C17H21N3O2Purezza:99.65% - 99.76%Colore e forma:SolidPeso molecolare:299.37Fluralaner
CAS:Fluralaner (A1443) is an isoxazoline ectoparasiticide.Formula:C22H17Cl2F6N3O3Purezza:99.72% - 99.99%Colore e forma:Solid PowderPeso molecolare:556.29Ginsenoside Rc
CAS:<p>Ginsenoside Rc (Panaxoside Rc) is one of the ginsenosides from Panax ginseng, inhibits the expression of TNF-α and IL-1β.</p>Formula:C53H90O22Purezza:98.83% - 99.56%Colore e forma:White PowderPeso molecolare:1079.27NS11394
CAS:<p>NS11394 is a effective and subtype-selective GABA(A) receptor-positive modulator; possesses a functional efficacy selectivity profile of α(5) > α(3) > α(2) > α(</p>Formula:C23H19N3OPurezza:99.44% - 99.86%Colore e forma:SolidPeso molecolare:353.42ONO-8590580
CAS:ONO-8590580 (CS-2894) is a negative allosteric modulator of GABAA α5.Formula:C21H21FN6Purezza:99.43%Colore e forma:SolidPeso molecolare:376.43Jujuboside A
CAS:Jujuboside A: glycoside from Semen Ziziphi Spinosae, may treat Alzheimer's, has neuro-inhibitory effects.Formula:C58H94O26Purezza:98% - >99.99%Colore e forma:SolidPeso molecolare:1207.35Suritozole
CAS:<p>Suritozole (MDL-26479) is a negative modulator at the gamma-aminobutyric acidA (GABAA) receptor</p>Formula:C10H10FN3SPurezza:99.25%Colore e forma:SolidPeso molecolare:223.27Basmisanil
CAS:Basmisanil (RG1662) is a negative allosteric modulator/inverse agonist of GABAAα5 receptors.Formulations containing basmisanil are in clinical trials for theFormula:C21H20FN3O5SPurezza:99.21% - 99.42%Colore e forma:SolidPeso molecolare:445.46Dihydroergotoxine mesylate
CAS:Dihydroergotoxine mesylate (Ergoloid mesylates) is mainly used to improve symptoms and physical symptoms of mental degeneration related to aging.Formula:C20H29N3O5SPurezza:99.39% - ≥95%Colore e forma:SolidPeso molecolare:423.53Bicuculline
CAS:Bicuculline, a plant-derived GABAA receptor antagonist, identified in 1932, reacts to light.Formula:C20H17NO6Purezza:98% - 99.99%Colore e forma:Light Yellow PowderPeso molecolare:367.35Loreclezole
CAS:Loreclezole is a selective GABAA receptor modulator and acts as a positive allosteric modulator of β2 or β3-subunit-containing receptors.Formula:C10H6Cl3N3Purezza:99.78%Colore e forma:SolidPeso molecolare:274.53Afloqualone
CAS:<p>Afloqualone (HQ-495) is a GABA Receptor agonist with sedative and muscle-relaxant properties.</p>Formula:C16H14FN3OPurezza:99.72%Colore e forma:SolidPeso molecolare:283.3Riluzole
CAS:<p>Riluzole (RP-54274) is an anticonvulsant, glutamate antagonist, and prolongs ALS patient survival.</p>Formula:C8H5F3N2OSPurezza:99.71% - 99.88%Colore e forma:PowderPeso molecolare:234.2Darigabat
CAS:Darigabat (PF-06372865) is a GABAA receptor modulator with anxiolytic activity that inhibits α2, α1 PAM, and α2 PAM.Formula:C22H21FN4O3SPurezza:98.42% - 99.29%Colore e forma:SolidPeso molecolare:440.49AZD 3043
CAS:AZD 3043 (THRX 918661) is a modulator of the gamma-aminobutyric acid type A receptor, a novel sedative-hypnotic, and a potential short-acting anesthetic.Formula:C19H29NO5Purezza:98.19% - 99.55%Colore e forma:SolidPeso molecolare:351.44(R)-Baclofen hydrochloride
CAS:Arbaclofen HCl, a GABA-B agonist, treats spasticity from spinal injury by reducing excitatory transmission.Formula:C10H13Cl2NO2Purezza:98%Colore e forma:SolidPeso molecolare:250.12NO 711
CAS:NO 711（NNC-711 free acid） is a selective inhibitor of GAT-1, which enhances non-rapid eye movement sleep, and prevents paclitaxel-induced neuropathic pain.Formula:C21H22N2O3Purezza:99.70%Colore e forma:SolidPeso molecolare:350.41Ro 15-1310
CAS:Ro 15-3505, a benzodiazepine receptor partial inverse agonist, has shown the ability to improve impaired recent memory of aged mice.Formula:C15H14ClN3O3Colore e forma:SolidPeso molecolare:319.74CP-457920
CAS:CP-457920 is a selective α5 GABAA receptor inverse agonist that is suitable for investigating dementia in Alzheimer's disease.Formula:C18H17N3O3Purezza:99.06% - 99.74%Colore e forma:SolidPeso molecolare:323.35CGP 7930
CAS:Positive allosteric modulator of GABAB receptorsFormula:C19H32O2Purezza:98%Colore e forma:SolidPeso molecolare:292.46NCS-382
CAS:γ-Hydroxybutyric acid antagonistFormula:C13H14O3Purezza:98%Colore e forma:SolidPeso molecolare:218.25Etbicyphat
CAS:Etbicyphat: potent GABA(A) antagonist, induces epileptiform activity, binds to GABA/benzodiazepine receptors.Formula:C6H11O4PColore e forma:SolidPeso molecolare:178.12CGP 36216 hydrochloride
CAS:CGP 36216 hydrochloride is a potent and selective antagonist of GABAB receptors (IC50: 43 μM).Formula:C5H14NO2PPurezza:98%Colore e forma:SolidPeso molecolare:151.14BHF-177
CAS:BHF-177 is a positive allosteric modulator of the GABAB receptor. BHF-177 reduces self-administration of nicotine in animal studies.Formula:C19H20F3N3Colore e forma:SolidPeso molecolare:347.38CGS8216
CAS:CGS8216 shows analgesic activity at high doses, has anxiolytic activity, and can be used to study immune system disorders.Formula:C16H11N3OPurezza:98.53%Colore e forma:SolidPeso molecolare:261.28SCH 50911 hydrochloride
CAS:SCH 50911 hydrochloride is a selective, orally-active and competitive antagonist of γ-Aminobutyric acid B GABA(B) receptor(IC50 : 1.1 μM).Formula:C8H16ClNO3Purezza:98%Colore e forma:SolidPeso molecolare:209.67DS2
CAS:Positive allosteric modulator of δ-subunit containing GABAA receptorsFormula:C18H12ClN3OSPurezza:98%Colore e forma:SolidPeso molecolare:353.83(±)-Homoproline Hydrochloride
CAS:(±)-Homoproline Hydrochloride. Affordable Excellence: Reliable Quality You Can TrustFormula:C6H12ClNO2Purezza:99.69%Colore e forma:SolidPeso molecolare:165.62MK-0343
CAS:MK0343 is an orally bioavailable GABAA receptor subtype-selective partial agonist and is a non-sedating anxiolytic.Formula:C19H17F2N7OPurezza:98%Colore e forma:SolidPeso molecolare:397.38GABAA receptor agent 5
CAS:Compound 018 is a potent γ-GABAAR antagonist, Ki of 0.020 μM, with low membrane permeability.Formula:C21H25N3O2SPurezza:99.39%Colore e forma:SolidPeso molecolare:383.5117-PA
CAS:17-PA is a GABAA receptor antagonist.Formula:C25H34OPurezza:98%Colore e forma:SolidPeso molecolare:350.54CGP 46381
CAS:CGP 46381 is a GABAB receptor antagonist.Formula:C10H22NO2PPurezza:98%Colore e forma:White SolidPeso molecolare:219.26Bifenazate
CAS:<p>Bifenazate is a positive allosteric modulator of GABA receptor. Bifenazate is an acaricide that controls 100% of mites at a concentration of 25 ppm.</p>Formula:C17H20N2O3Purezza:99.62%Colore e forma:Solid CrystallinePeso molecolare:300.35RO 4938581
CAS:RO 4938581: potent GABAA α5 inverse agonist (Ki 4.6 nM); lower affinity for α1β3γ2a, α2β3γ2a, α3β3γ2a (Ki: 174, 185, 80 nM).Formula:C13H8BrF2N5Purezza:98%Colore e forma:SolidPeso molecolare:352.14CGP11952
CAS:CGP11952 is same the benzodiazepines in its pharmacological action and it also is an experimental benzodiazepine derivative.Formula:C21H21Cl2N5O2Purezza:98%Colore e forma:SolidPeso molecolare:446.33E2730
CAS:E2730 is a non-competitive GABA transporter 1 (GAT1) inhibitor with anti-epileptic activity, useful in studying neurological disorders.Formula:C9H8F4N2O2SPurezza:98.22% - 98.54%Colore e forma:SolidPeso molecolare:284.23U-89843A
CAS:U-89843A is an allosteric modulator of the GABA_A receptor, known to enhance GABA-induced Cl^- currents [1].Formula:C16H24ClN5Purezza:98%Colore e forma:SolidPeso molecolare:321.85MRK-623
CAS:MRK-623 (14k) is an oral GABA A agonist with high affinity for α1/α2/α3/α5 subunits and anxiolytic properties.Formula:C20H17FN4OColore e forma:SolidPeso molecolare:348.37
