Caseina chinasi
Le caseina chinasi sono una famiglia di proteine chinasi serina/treonina che regolano vari processi cellulari, tra cui la riparazione del DNA, i ritmi circadiani e la trasduzione del segnale. Queste chinasi sono coinvolte nella fosforilazione di numerose proteine e sono implicate in malattie come il cancro, i disturbi neurodegenerativi e le sindromi metaboliche. Presso CymitQuimica, offriamo una selezione di inibitori della caseina chinasi per supportare la tua ricerca nella trasduzione del segnale, nella regolazione del ciclo cellulare e nello sviluppo terapeutico.
Trovati 143 prodotti per "Caseina chinasi".
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PF-4800567
CAS:PF-4800567 is a selective inhibitor of casein kinase 1ε (CK1ε; IC50 = 32 nM) with greater than 20-fold selectivity over CK1δ.Formula:C17H18ClN5O2Purezza:99.74% - 99.76%Colore e forma:White SolidPeso molecolare:359.81LH846
CAS:LH846 is a selective inhibitor of CK1δ (IC50 values are 290 nM, 1.3 uM and 2.5 uM for CK1δ, ε and α); exhibits no inhibitory activity at CK2.Formula:C16H13ClN2OSPurezza:90% - 98.26%Colore e forma:SolidPeso molecolare:316.81TBB
CAS:TBB (NSC-231634)(NSC-231634) is a highly selective, ATP/GTP-competitive inhibitor of casein kinase-2 (CK2).Formula:C6HBr4N3Purezza:98.51% - 99.45%Colore e forma:SolidPeso molecolare:434.708NCC007
CAS:NCC007 is a novel CKIα and CKIδ dual inhibitors by structural modification of N9 and C2 position of longdaysin.Formula:C22H28F3N7Purezza:98.88%Colore e forma:SolidPeso molecolare:447.5Umbralisib hydrochloride
CAS:Umbralisib hydrochloride: PI3Kδ inhibitor; IC50=22.2 nM, EC50=24.3 nM; active vs CK1ε, EC50=6.0 μM.Formula:C31H25ClF3N5O3Purezza:98%Colore e forma:SolidPeso molecolare:608.01SR-3029
CAS:SR-3029 is a potent and highly specific CK1δ/CK1ε inhibitor.Formula:C23H19F3N8OPurezza:99.64%Colore e forma:SolidPeso molecolare:480.45(E/Z)-GO289
CAS:(E/Z)-GO289, which strongly lengthened circadian period, is a potent and selective inhibitor of CK2.Formula:C17H15BrN4O2SPurezza:98.1%Colore e forma:SolidPeso molecolare:419.3Ref: TM-T9356
2mg34,00€5mg52,00€1mL*10mM (DMSO)54,00€10mg86,00€25mg170,00€50mg250,00€100mg354,00€200mg482,00€AS-252424
CAS:AS-252424 is a potent and selective inhibitor of PI3Kγ with IC50 of 33 nM; >10 fold selectivity for PI3Kγ versus PI3Kα.Formula:C14H8FNO4SPurezza:99.06% - 99.09%Colore e forma:Orange SolidPeso molecolare:305.28Ref: TM-T6208
1mg37,00€2mg52,00€5mg77,00€1mL*10mM (DMSO)84,00€10mg128,00€25mg205,00€50mg309,00€100mg447,00€500mg973,00€IWP-2
CAS:IWP-2 is a Wnt pathway inhibitor and an ATP-competitive CK1δ inhibitor. IWP-2 inhibits self-renewal of embryonic stem cells. Cost effective and quality assured.Formula:C22H18N4O2S3Purezza:96.1% - 99.49%Colore e forma:White SolidPeso molecolare:466.6Umbralisib
CAS:Umbralisib (TGR 1202) is a PI3Kδ inhibitor.Formula:C31H24F3N5O3Purezza:99.56% - 99.56%Colore e forma:White SolidPeso molecolare:571.55Ref: TM-T4976
1mg46,00€2mg62,00€5mg90,00€1mL*10mM (DMSO)114,00€10mg166,00€25mg324,00€50mg425,00€100mg623,00€DMAT
CAS:DMAT (Casein kinase II Inhibitor) is a potent and specific inhibitor of CK2(IC50 value of 130 nM).Formula:C9H7Br4N3Purezza:99.48%Colore e forma:White SolidPeso molecolare:476.79Epiblastin A
CAS:Epiblastin A inhibits CK1, targets its isoenzymes, and converts EpiSCs to cESCs.Formula:C12H10ClN7Purezza:99.45%Colore e forma:SolidPeso molecolare:287.71TTP 22
CAS:TTP 22: ATP-competitive CK2 inhibitor; IC50/Ki: 0.1 μM/40 nM; >250x selective over JNK3, ROCK1, MET.Formula:C16H14N2O2S2Purezza:97.08% - 97.78%Colore e forma:SolidPeso molecolare:330.42LY-364947
CAS:LY-364947 (HTS466284) is a potent ATP-competitive inhibitor of TGFβR-I.Formula:C17H12N4Purezza:99.65% - 99.96%Colore e forma:Yellow SolidPeso molecolare:272.3Ref: TM-T2048
5mg62,00€1mL*10mM (DMSO)69,00€10mg78,00€25mg136,00€50mg241,00€100mg354,00€200mg530,00€500mg830,00€LY294002
CAS:LY294002 (SF 1101) is a broad-spectrum inhibitor of PI3K, inhibiting PI3Kα, PI3Kδ, and PI3Kβ (IC50=0.5/0.57/0.97 μM).Formula:C19H17NO3Purezza:98% - 99.96%Colore e forma:White SolidPeso molecolare:307.34CK1-IN-1
CAS:CK1-IN-1, a CK1 inhibitor with IC50: 15nM CK1δ, 16nM CK1ε, 73nM p38σ; patent WO2015119579A1.Formula:C24H15F2N3Purezza:98.79%Colore e forma:White SolidPeso molecolare:383.39Ref: TM-T5393
1mg47,00€2mg62,00€5mg92,00€1mL*10mM (DMSO)101,00€10mg152,00€25mg289,00€50mg447,00€100mg670,00€D4476
CAS:D4476 (Casein Kinase I Inhibitor) is an effective, selective, and cell-permeant CK1 (casein kinase 1) inhibitor( IC50=300 nM in a cell-free assay).Formula:C23H18N4O3Purezza:99.7% - 99.96%Colore e forma:SolidPeso molecolare:398.41TA-01
CAS:TA-01 is a potent CK1 and p38 MAPK inhibitor, with IC50s of 6.4 nM, 6.8 nM, 6.7 nM for CK1ε, CK1δ and p38 MAPK, respectively.Formula:C20H12F3N3Purezza:99.55% - 99.94%Colore e forma:SolidPeso molecolare:351.32Ref: TM-T4645
2mg34,00€5mg50,00€1mL*10mM (DMSO)67,00€10mg80,00€25mg147,00€50mg224,00€100mg313,00€200mg439,00€Silmitasertib
CAS:Silmitasertib (CX-4945) is a potent, orally bioavailable inhibitor of casein kinase 2 (CK2; Ki: 0.38 nM).Formula:C19H12ClN3O2Purezza:98% - 99.90%Colore e forma:SolidPeso molecolare:349.77Ref: TM-T2259
1mg38,00€2mg49,00€5mg80,00€1mL*10mM (DMSO)88,00€10mg118,00€25mg197,00€50mg313,00€100mg492,00€500mg1.054,00€
