Caseina chinasi
Le caseina chinasi sono una famiglia di proteine chinasi serina/treonina che regolano vari processi cellulari, tra cui la riparazione del DNA, i ritmi circadiani e la trasduzione del segnale. Queste chinasi sono coinvolte nella fosforilazione di numerose proteine e sono implicate in malattie come il cancro, i disturbi neurodegenerativi e le sindromi metaboliche. Presso CymitQuimica, offriamo una selezione di inibitori della caseina chinasi per supportare la tua ricerca nella trasduzione del segnale, nella regolazione del ciclo cellulare e nello sviluppo terapeutico.
Trovati 138 prodotti di "Caseina chinasi"
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Epiblastin A
CAS:Epiblastin A inhibits CK1, targets its isoenzymes, and converts EpiSCs to cESCs.Formula:C12H10ClN7Purezza:99.45%Colore e forma:SolidPeso molecolare:287.71Longdaysin
CAS:Longdaysin is an inhibitor of CK1α and CK1δ (IC50s: 5.6/8.8 μM). It also can inhibit ERK2 (IC50: 52 μM).Formula:C16H16F3N5Purezza:99.97%Colore e forma:SolidPeso molecolare:335.33PF-670462
CAS:PF-670462 is a potent (IC50 = 7.7 ± 2.2 nM) and selective (>30-fold with respect to 42 additional kinases) inhibitor of CK1ε in isolated enzyme preparations.Formula:C19H22Cl2FN5Purezza:99.42% - 99.72%Colore e forma:SolidPeso molecolare:410.32XL413
CAS:XL-413 is an oral CDC7 kinase inhibitor, potentially blocking DNA replication, mitosis, and cancer cell growth.Formula:C14H12ClN3O2Purezza:98.40% - 99.94%Colore e forma:SolidPeso molecolare:289.72SSTC3
CAS:SSTC3 is a casein kinase 1α (CK1α) activator with potential antitumor activity that inhibits WNT signaling.Formula:C23H17F3N4O3S2Purezza:98.65% - 99.94%Colore e forma:SolidPeso molecolare:518.53AMG-548
CAS:AMG-548, oral p38α inhibitor (Ki=0.5 nM), >1000x selectivity over p38γ/δ, blocks TNFα (IC50=3 nM), also inhibits Wnt/Casein kinase 1δ/ε.Formula:C29H27N5OPurezza:99.91%Colore e forma:SolidPeso molecolare:461.56SR-1277
CAS:SR-1277 is a potent, highly selective and ATP-competitive CK1δ/ε inhibitor, regulating Wee1 activity at the G2/M cell-cycle interface, and antiproliferative.Formula:C21H19N9O3SColore e forma:SolidPeso molecolare:477.5CK2/PIM1-IN-1
CAS:CK2/PIM1-IN-1 inhibits CK2 & PIM1 (IC50s: 3.787 & 4.327 μM), aimed for cancer research.Formula:C15H9NO4S2Purezza:98%Colore e forma:SolidPeso molecolare:331.374,5,6,7-Tetrabromobenzimidazole
CAS:4,5,6,7-Tetrabromobenzimidazole is a selective and ATP-competitive inhibitor of protein kinase CK2 [1].Formula:C7H2Br4N2Colore e forma:SolidPeso molecolare:433.72CK2-IN-9
CAS:CK2-IN-9, a potent and selective CK2 kinase inhibitor, exhibits an inhibitory concentration (IC50) of 3 nM against its target enzyme and hampers Wnt reporterFormula:C23H29N9OColore e forma:SolidPeso molecolare:447.54Quinalizarin
CAS:Quinalizarin, the most selective CK2 inhibitor, is superior to CX-4945 which is the first-in-class CK2 inhibitor.Formula:C14H8O6Purezza:98%Colore e forma:SolidPeso molecolare:272.21Tyrphostin AG 1112
CAS:Tyrphostin AG 1112 is a Bcr-Abl kinase blocker. It can activate the terminal differentiation of K562 cells and the purging of Ph+ cells.Formula:C15H10N6Colore e forma:SolidPeso molecolare:274.28PF 4800567 hydrochloride
CAS:casein kinase 1ε inhibitorFormula:C17H19Cl2N5O2Purezza:98%Colore e forma:SolidPeso molecolare:396.27IQA
CAS:IQA is a casein kinase 2 (CK2) inhibitor.Formula:C17H12N2O3Colore e forma:SolidPeso molecolare:292.29(R)-DRF053 dihydrochloride
CAS:cdk/CK1 inhibitor,potent and ATP-competitiveFormula:C23H29Cl2N7OPurezza:98%Colore e forma:SolidPeso molecolare:490.43TMCB
CAS:CK2 and ERK8 inhibitorFormula:C11H9Br4N3O2Purezza:98%Colore e forma:SolidPeso molecolare:534.82CK2-IN-6
CAS:CK2-IN-6: Potent CK2 inhibitor for cancer, inflammation, pain, and immune research.Formula:C19H16ClN7O2Colore e forma:SolidPeso molecolare:409.83SRPIN-803
CAS:SRPIN-803 is a selective dual SRPK1 and CK2 inhibitor.Formula:C14H9F3N4O3SPurezza:98%Colore e forma:SolidPeso molecolare:370.31Umbralisib sulfate
CAS:Umbralisib sulfate, an oral dual PI3Kδ/CK1ε inhibitor (EC50: 22.2 nM/6.0 μM), targets CLL T cells for blood cancer research.Formula:C31H26F3N5O7SColore e forma:SolidPeso molecolare:669.63Umbralisib tosylate
CAS:Umbralisib tosylate, an oral PI3Kδ/CK1ε inhibitor (EC50: 22.2 nM/6.0 μM), shows promise for CLL research.Formula:C38H32F3N5O6SColore e forma:SolidPeso molecolare:743.75
