
Neuroscienza
Gli inibitori in neuroscienze sono composti progettati per modulare l'attività di proteine, enzimi o recettori specifici all'interno del sistema nervoso. Questi inibitori sono cruciali per studiare i meccanismi molecolari alla base della funzione neuronale, della trasmissione sinaptica e delle malattie neurodegenerative. Mirando ai recettori dei neurotrasmettitori, ai canali ionici e alle vie di segnalazione, gli inibitori in neuroscienze aiutano a esplorare la funzione cerebrale e a sviluppare strategie terapeutiche per disturbi neurologici come l'Alzheimer, il Parkinson e l'epilessia. Presso CymitQuimica, offriamo una vasta gamma di inibitori in neuroscienze di alta qualità per supportare la tua ricerca in neurobiologia, neurofarmacologia e scienze cognitive.
Sottocategorie di "Neuroscienza"
- recettore 5-HT(1.025 prodotti)
- ACK(1 prodotti)
- AChR(641 prodotti)
- Citrato liasi ATP(17 prodotti)
- Recettore adrenergico(2.997 prodotti)
- BACE(37 prodotti)
- Beta amiloide(217 prodotti)
- CaMK(73 prodotti)
- COX(598 prodotti)
- Recettore della dopamina(445 prodotti)
- Ricettore GABA(370 prodotti)
- Gamma-secretasi(57 prodotti)
- GluR(265 prodotti)
- GlyT(26 prodotti)
- Recettore dell'istamina(385 prodotti)
- LRRK2(43 prodotti)
- Recettore della melatonina(26 prodotti)
- NMDAR(10 prodotti)
- Recettore OX(40 prodotti)
- Recettore degli oppioidi(325 prodotti)
Mostrare 12 più sottocategorie
Trovati 5450 prodotti di "Neuroscienza"
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Methoxy-PEPy
CAS:Methoxy-PEPy is a potent and selective mGlu5 receptor inhibitor with an IC50 value of 1 nM.Formula:C13H10N2OPurezza:98.66%Colore e forma:SolidPeso molecolare:210.23Zamifenacin
CAS:Zamifenacin obviously decreases colonic motility in irritable bowel syndrome. Zamifenacin is an effective gut-selective muscarinic M3 receptor antagonist.Formula:C27H29NO3Purezza:98%Colore e forma:SolidPeso molecolare:415.52RR-11a
CAS:RR-11a is a synthetic enzyme Legumain inhibitor.
Formula:C24H28N6O10Purezza:98%Colore e forma:SolidPeso molecolare:560.51Bifeprunox
CAS:Bifeprunox: potent antipsychotic, partial agonist at D2-like/5-HT1A receptors; treats schizophrenia.Formula:C24H23N3O2Purezza:98%Colore e forma:SolidPeso molecolare:385.46LY487379 hydrochloride
CAS:Positive allosteric modulator of mGlu2 receptorsFormula:C21H20ClF3N2O4SPurezza:98%Colore e forma:SolidPeso molecolare:488.91EMDT
CAS:EMDT oxalate is a selective 5-HT6 agonist, and has antidepressant effects.Formula:C15H22N2OPurezza:97.66% - 99.78%Colore e forma:SolidPeso molecolare:246.35Ref: TM-T11183
1mg87,00€2mg118,00€5mg167,00€10mg202,00€25mg449,00€50mg652,00€100mg888,00€500mg1.783,00€1mL*10mM (DMSO)166,00€Pancopride
CAS:Pancopride(LAS 30451) is a novel, orally available, long-acting, selective 5-HT3 receptor antagonist that blocks nitrogen mustard and dacarbazine-inducedFormula:C18H24ClN3O2Purezza:93.64%Colore e forma:SolidPeso molecolare:349.86Repinotan HCl
CAS:Repinotan HCl (Bay-x-3702) is a 5-HT1A receptor agonist with potent neuroprotective effects for the study of ischemic stroke and traumatic brain injury.
Formula:C21H25ClN2O4SPurezza:99.57%Colore e forma:SolidPeso molecolare:436.95S16961
CAS:S16961 (S169611) is an agonist of nicotinic receptor.Formula:C41H71NO6Purezza:99.69%Colore e forma:SolidPeso molecolare:674.01MSOP
CAS:MSOP is a selective antagonist of group III metabotropic glutamate receptor (KD of 51 μM for the L-AP4-sensitive presynaptic mGluR).Formula:C4H10NO6PPurezza:98%Colore e forma:SolidPeso molecolare:199.1(R)-Baclofen hydrochloride
CAS:Arbaclofen HCl, a GABA-B agonist, treats spasticity from spinal injury by reducing excitatory transmission.Formula:C10H13Cl2NO2Purezza:98%Colore e forma:SolidPeso molecolare:250.12Ampreloxetine
CAS:Ampreloxetine (TD-9855) is a norepinephrine reuptake inhibitor used to study neurological diseases.Formula:C18H18F3NOPurezza:98%Colore e forma:SolidPeso molecolare:321.34PF-4479745
CAS:PF-4479745 ia a potent and selective agonist of 5-HT2C receptor.Formula:C17H22N4Purezza:98%Colore e forma:SolidPeso molecolare:282.38Clovoxamine
CAS:Clovoxamine fumarate (DU 23811 fumarate) is a 5-HT reuptake, serotonin and norepinephrine inhibitor with antidepressant and anticonvulsant activity.Formula:C14H21ClN2O2Purezza:99.44% - 99.75%Colore e forma:SolidPeso molecolare:284.78BuChE-IN-1
CAS:BuChE-IN-1 is a potent BBB-permeable, low-toxic BuChE inhibitor with potential for AD research.Formula:C23H23FN2O4SColore e forma:SolidPeso molecolare:442.5NNC052090
CAS:NNC052090 inhibits GABA uptake, favoring hBGT-1 (Ki=1.4μM), affects α1/D2 receptors (IC50=266/1632nM).Formula:C27H30N2O2Colore e forma:SolidPeso molecolare:414.54(Rac)-SEP-363856
CAS:(Rac)-SEP-363856 is the racemate of SEP-363856. SEP-363856 is an orally active and CNS active psychotropic agent with a uniqueFormula:C9H13NOSPurezza:98%Colore e forma:SolidPeso molecolare:183.27γ-Secretase modulator 12
CAS:γ-Secretase modulator 12 (Compound 1a) is a selective compound that effectively reduces amyloid-β42 (Aβ42) levels with an IC50 of 0.39 μM.Formula:C25H23N3O2Colore e forma:SolidPeso molecolare:397.47hMAO-B-IN-2
CAS:hMAO-B-IN-2: selective oral hMAO-B inhibitor, crosses BBB, IC50=4 nM, potential for Alzheimer's research, neuroprotective, low toxicity.Formula:C18H23NO3Colore e forma:SolidPeso molecolare:301.38SGS518 oxalate
CAS:SGS518 oxalate is a 5-HT6 antagonist.Formula:C23H24F2N2O7SPurezza:98%Colore e forma:SolidPeso molecolare:510.51Pipazethate
CAS:Pipipyrazine is a nonnarcotic oral cough suppressant, cough suppressant.Formula:C21H25N3O3SColore e forma:SolidPeso molecolare:399.51TCS 1105
CAS:TCS 1105 is a GABAA BZR ligand, blocking Sema3A and altering mouse anxiety, aggression, and social dominance.Formula:C17H13FN2O2Purezza:99.75%Colore e forma:SolidPeso molecolare:296.3VU0418506
CAS:VU0418506 is a positive allosteric modulator (PAM) of the metabotropic glutamate receptor 4 (mGlu4).Formula:C12H8ClFN4Purezza:98%Colore e forma:SolidPeso molecolare:262.67Pirenzepine
CAS:Pirenzepine targets M1 mAChR, curbs acid secretion, eases spasms, and has anti-cancer properties.Formula:C19H21N5O2Colore e forma:SolidPeso molecolare:351.4SSAO inhibitor-2
CAS:SSAO inhibitor-2 targets human SSAO (<10 nM) and MAO-A (10-100 μM); useful in various diseases research.Formula:C14H21FN4O2Colore e forma:SolidPeso molecolare:296.34ATC0065 HCl
CAS:ATC0065 dihydrochloride is a novel nonpeptidic and potent melanin-concentrating hormone receptor 1 (MCHR1) selective antagonist.Formula:C25H31BrCl2F3N5OColore e forma:SolidPeso molecolare:625.35Oxybutynin R-isomer HCl
CAS:Aroxybutynin, R-isomer of oxybutynin, is a muscarinic antagonist with antispasmodic effects on bladder muscle, weaker than atropine.Formula:C22H32ClNO3Colore e forma:SolidPeso molecolare:393.95Etbicyphat
CAS:Etbicyphat: potent GABA(A) antagonist, induces epileptiform activity, binds to GABA/benzodiazepine receptors.Formula:C6H11O4PColore e forma:SolidPeso molecolare:178.12UCSF686
CAS:UCSF686, a UCSF678 analog, lacks 5-HT5A potency but keeps affinity for 5-HT1A, 5-HT2B, 5-HT7, and serves as a control.Formula:C14H19N3O2SColore e forma:SolidPeso molecolare:293.38AChE/BChE-IN-5
CAS:AChE/BChE-IN-5 (BMC-16) crosses BBB; IC50: hAChE 266 nM, hBChE 10.6 nM. Dual AChE/BChE inhibitor.Formula:C17H26N2O3Colore e forma:SolidPeso molecolare:306.4Safrazine
CAS:Safrazine is an irreversible, non-specific and orally active monoamine oxidase (MAO) inhibitor. Safrazine can be used in depression research[1].Formula:C11H16N2O2Colore e forma:SolidPeso molecolare:208.26GR-55562 dihydrobromide
CAS:GR-55562 dihydrobromide is a antagonist of 5-HT1B/5-HT1D serotonin receptor.Formula:C23H26ClN3O2Purezza:98%Colore e forma:SolidPeso molecolare:411.93CBP501
CAS:CBP501 peptide inhibits kinases like MAPKAP-K2/C-Tak1/CHK1, preventing Cdc25C function and blocking the entry into mitosis.Formula:C86H122F5N29O17Colore e forma:SolidPeso molecolare:1929.06DREADD agonist 21 dihydrochloride
CAS:DREADD agonist 21 dihydrochloride is a potent human muscarinic acetylcholine M3 receptors ( hM3Dq ) agonist with EC 50 of 1.7 nM [1].Formula:C17H20Cl2N4Purezza:98%Colore e forma:SolidPeso molecolare:351.27Bradanicline HCl
CAS:Bradanicline(TC-5619) is the agonist of Alpha-7 Nicotinic Receptor.Formula:C22H24ClN3O2Colore e forma:SolidPeso molecolare:397.9AChE/MAO-B-IN-3
AChE/MAO-B-IN-3: dual inhibitor for AChE (IC50 = 0.0257 µM) and MAO-B (IC50 = 0.0456 µM), researched for Alzheimer's.Formula:C24H28N2O4Colore e forma:SolidPeso molecolare:408.49S-15535
CAS:S-15535 is a potent, orally active, partial 5-HT1A receptor agonist.Formula:C21H24N2O2Purezza:98%Colore e forma:SolidPeso molecolare:336.43Org-12962
CAS:Org-12962: 5-HT2C agonist (pEC50: 7.01), anti-panic in rats, affects 5-HT2A/B (pEC50: 6.38/6.28).Formula:C10H11ClF3N3Purezza:98.34%Colore e forma:SolidPeso molecolare:265.66OSU 6162 hydrochloride
CAS:Dopamine stabilizerFormula:C15H24ClNO2SPurezza:98%Colore e forma:SolidPeso molecolare:317.88CGP 36216 hydrochloride
CAS:CGP 36216 hydrochloride is a potent and selective antagonist of GABAB receptors (IC50: 43 μM).Formula:C5H14NO2PPurezza:98%Colore e forma:SolidPeso molecolare:151.14RG-12915
CAS:RG-12915 is a selective antagonist of 5-HT3(IC50 value of 0.16 nM).Formula:C20H25ClN2O2Purezza:98%Colore e forma:SolidPeso molecolare:360.88MK-212
CAS:MK-212 is a 5HT2C agonist; boosts corticosterone and lowers activity at 0.5-1mg/kg; reduces anxiety without affecting movement at 0.1-0.2mg/kg in mice.Formula:C8H11ClN4Colore e forma:SolidPeso molecolare:198.65Cinitapride Hydrogen Tartrate
CAS:Cinitapride Hydrogen Tartrate is a gastroprokinetic agent that acts as an antagonist of the 5-HT2 receptors and as an agonist of the 5-HT1 and 5-HT4 receptorsFormula:C25H36N4O10Purezza:98%Colore e forma:SolidPeso molecolare:552.581AT-1001
CAS:AT-1001 is an α3β4 nAChR partial agonist reducing nicotine relapse and withdrawal with negligible impact on food response and dopamine release.Formula:C15H21BrN2Colore e forma:SolidPeso molecolare:309.24Indisetron Dihydrochloride
CAS:Indisetron Dihydrochloride is a 5-HT(3) and 5-HT(4) receptor antagonist. Indisetron reduces 2-methyl-5-serotonin (HT)-induced bradycardia.Formula:C17H24ClN5OColore e forma:SolidPeso molecolare:349.86Cyclopenin
CAS:Cyclopenin is an inhibitor of acetylcholinesterase (AChE; IC50 = 2.04 μM for human recombinant AChE).Formula:C17H14N2O3Colore e forma:SolidPeso molecolare:294.35-HT4 antagonist 1
CAS:5-HT4 antagonist 1 is an antagonist of 5-HT4 (pKi = 9.6).Formula:C23H36N4O5SPurezza:99.75%Colore e forma:SolidPeso molecolare:480.62PNU-282987 S enantiomer hydrochloride
CAS:(S)-PNU-282987, selective α7 nAChR agonist; Ki=26 nM (rat), weak on other receptors except 5-HT3; Ki=930 nM.Formula:C14H18Cl2N2OPurezza:98%Colore e forma:SolidPeso molecolare:301.21Vinconate
CAS:Vinconate is an indolonaphthyridine derivative and can stimulate the muscarinic acetylcholine receptor.Formula:C18H20N2O2Purezza:98%Colore e forma:SolidPeso molecolare:296.36Z-Cyclopentyl-AP4
CAS:Group III mGlu receptor agonistFormula:C6H12NO5PPurezza:98%Colore e forma:SolidPeso molecolare:209.14Mazaticol
CAS:Mazaticol: an anticholinergic, blocks muscarinic receptors, inhibits dopamine uptake, used in Parkinson's research.Formula:C21H27NO3S2Colore e forma:SolidPeso molecolare:405.57BuChE-IN-4
CAS:BuChE-IN-4 is a potent inhibitor of BuChE (IC50: 7.7 nM) and exhibits mild antioxidant capacity, non-toxicity, lipophilicity and neuroprotective effects.Formula:C21H21BrFN3O4SColore e forma:SolidPeso molecolare:510.38Sultroponium
CAS:Sultroponium may be used as an anticholinergic agent or antispasmodic.Formula:C20H29NO6SColore e forma:SolidPeso molecolare:411.51LY 2365109 hydrochloride
CAS:glycine transporter 1 (GlyT1) inhibitorFormula:C22H27NO5Purezza:98%Colore e forma:SolidPeso molecolare:385.45Alvameline maleate
CAS:Alvameline maleate is used as a Partial M1 Agonist and M2/M3 Antagonist.Formula:C13H19N5O4Colore e forma:SolidPeso molecolare:309.32BACE1-IN-12
CAS:BACE1-IN-12: potent BACE1 and BuChE inhibitor, IC50s - 8.9 μM and 3.2 μM, blood-brain barrier permeable, anti-Alzheimer's potential.Formula:C29H28Cl2N6OColore e forma:SolidPeso molecolare:547.48PF-06371900
CAS:PF-06371900 is a potent and highly selective inhibitor of leucine-rich repeat kinase 2 (LRRK2).Formula:C17H16N6O2SColore e forma:SolidPeso molecolare:368.41Darenzepine
CAS:Darenzepine is a muscarinic receptor inhibitor.Formula:C21H21N3O2Purezza:99.87%Colore e forma:SolidPeso molecolare:347.41Ref: TM-T10961
1mg215,00€5mg426,00€10mg598,00€25mg889,00€50mg1.188,00€100mg1.605,00€1mL*10mM (DMSO)472,00€Alaproclate (hydrochloride)
CAS:Alaproclate, an SSRI, enhances serotonin and SIRT1, hinders NMDA and K+ currents in neurons, and shows antidepressant-like effects in rats.Formula:C13H19Cl2NO2Colore e forma:SolidPeso molecolare:292.2Bopindolol
CAS:Bopindolol: oral β1/β2-ARs antagonist and partial agonist; prodrug of pindolol for hypertension research.Formula:C23H28N2O3Colore e forma:SolidPeso molecolare:380.48Edivoxetine hydrochloride
CAS:Edivoxetine HCl, a potent NERI, treats depression and ADHD.Formula:C18H27ClFNO4Colore e forma:SolidPeso molecolare:375.87sEH/AChE-IN-2
CAS:sEH/AChE-IN-2 targets sEH & AChE, may reduce neuroinflammation & memory loss, potential in Alzheimer's research.Formula:C30H33ClF3N5O3Colore e forma:SolidPeso molecolare:604.06Metixene hydrochloride
CAS:Metixene hydrochloride is an anticholinergic antiparkinsonian agent.Formula:C20H24ClNSPurezza:98%Colore e forma:SolidPeso molecolare:345.93MPDC
CAS:MPDC acts as a competitive inhibitor against the Na+-dependent high-affinity glutamate transporter within forebrain synaptosomes.Formula:C7H9NO4Purezza:98%Colore e forma:SolidPeso molecolare:171.15J 104129 fumarate
CAS:M3 muscarinic receptor antagonistFormula:C24H36N2O2Purezza:98%Colore e forma:SolidPeso molecolare:384.55Levemopamil HCl
CAS:Levemopamil HCl is used as a calcium channel blocker.Formula:C23H31ClN2Purezza:98%Colore e forma:SolidPeso molecolare:370.96Befloxatone
CAS:Befloxatone is a potent, selective and reversible inhibitor of monoamine oxidase A.Formula:C15H18F3NO5Colore e forma:SolidPeso molecolare:349.3mGluR2 modulator 2
CAS:mGluR2 modulator 2: potent, selective, oral, EC50 = 0.13 μM, for antipsychotic research.Formula:C20H22FN3Colore e forma:SolidPeso molecolare:323.41PF-06455943
CAS:PF-06455943: LRRK2 inhibitor, IC50=3nM, PET radioligand, used for ADME/neuro PK & Parkinson's research.Formula:C17H14FN5OColore e forma:SolidPeso molecolare:323.32Talaglumetad hydrochloride
CAS:Talaglumetad hydrochloride, a prodrug of Eglumegad, targets mGluR2/3 to treat psychiatric disorders.Formula:C11H17ClN2O5Colore e forma:SolidPeso molecolare:292.72AZD 0328
CAS:AZD 0328 is a nicotinic receptor agonist for α7 neurons.Formula:C13H16N2OColore e forma:SolidPeso molecolare:216.28SD-6
CAS:SD-6, oral hAChE/hBChE inhibitor (IC50: 0.907/1.579 µM), crosses BBB, non-toxic, for Alzheimer's research.Formula:C20H22N4OSColore e forma:SolidPeso molecolare:366.48TIM-063
CAS:TIM-063: ATP-competitive CaMKKα/β inhibitor, cell-permeable, Ki: 0.35/0.2 μM, IC50: 0.63/0.96 μM.Formula:C18H9N3O4Colore e forma:SolidPeso molecolare:331.28Brofaromine Hydrochloride
CAS:Brofaromine hydrochloride treats depression/anxiety, inhibits MAO-A, affects serotonin/dopamine.Formula:C14H17BrClNO2Colore e forma:SolidPeso molecolare:346.655-HT6/5-HT2A receptor ligand-2
CAS:Compound 42: brain-penetrant, dual 5-HT6/5-HT2A antagonist, Ki of 25 nM/32 nM, pro-cognitive.Formula:C20H18FN3O2Colore e forma:SolidPeso molecolare:351.37UB 165 fumarate
CAS:UB 165 fumarate is a nAChR agonist, α4β2 partial, α3β2 full, with a 0.27 nM Ki for [3H]-nicotine in rat brain.Formula:C17H19ClN2O4Purezza:99.72%Colore e forma:SolidPeso molecolare:350.8SB 206553 hydrochloride
CAS:SB 206553 hydrochloride is a 5-HT2C inverse agonist and a 5-HT2C/5-HT2B receptor antagonist with anxiolytic activity, useful for studying neurological disordersFormula:C17H17ClN4OPurezza:99.56%Colore e forma:SolidPeso molecolare:328.8AChE/BChE/MAO-B-IN-4
AChE/BChE/MAO-B-IN-4 inhibits MAO-B (IC50: 0.0393 µM), AChE (IC50: 0.0458 µM), BChE (IC50: 0.075 µM), and fights AD with antioxidant action.Formula:C26H33N3O4Colore e forma:SolidPeso molecolare:451.56Ambenonium dichloride
CAS:AChE inhibitorFormula:C28H42Cl3N4O2Purezza:98%Colore e forma:SolidPeso molecolare:573.02RS 23597-190 hydrochloride
CAS:RS 23597-190 hydrochloride is a 5-HT4 receptor antagonist.Formula:C16H24Cl2N2O3Purezza:98%Colore e forma:SolidPeso molecolare:363.28EMD 56551
CAS:EMD 56551 is a selective small molecule 5-HT1A receptor agonist with anxiolytic activity for the study of anxiety disorders.Formula:C24H31N3O2Purezza:95.64% - 99.39%Colore e forma:SolidPeso molecolare:393.522PRX-08066 Maleic acid
CAS:PRX-08066 Maleic acid is the salt form of PRX-08066.PRX-08066 is a 5-HT receptor 2B antagonist that induces selective vasodilation of the pulmonary artery.Formula:C23H21ClFN5O4SPurezza:97.59%Colore e forma:SolidPeso molecolare:517.96Ref: TM-T6959
1mg79,00€5mg168,00€10mg220,00€25mg398,00€50mg587,00€100mg835,00€200mg1.134,00€1mL*10mM (DMSO)380,00€Ro 19-4603
CAS:Benzodiazepine inverse agonistFormula:C15H17N3O3SPurezza:98%Colore e forma:SolidPeso molecolare:319.38AChE/BChE-IN-4
CAS:AChE/BChE-IN-4 (BMC-3) crosses the BBB; IC50: hAChE 792 nM, hBChE 2.2 nM. Dual AChE/BChE inhibitor.Formula:C17H26N2O3Colore e forma:SolidPeso molecolare:306.4LP44 hydrochloride
CAS:LP44 hydrochloride is a 5-HT7 agonist with analgesic effects on formalin-induced orofacial pain in mice and can be used to study neuroinflammation.Formula:C27H38ClN3OSPurezza:98.06%Colore e forma:SolidPeso molecolare:488.13Iprindole
CAS:Iprindole, a tricyclic indole antidepressant, is a dual weak inhibitor of noradrenaline and 5-HT uptake [1].Formula:C19H28N2Purezza:99.54%Colore e forma:SolidPeso molecolare:284.44Ref: TM-T37015
2mg34,00€5mg50,00€10mg75,00€25mg145,00€50mg253,00€100mg432,00€200mg618,00€1mL*10mM (DMSO)79,00€LY456066
CAS:LY456066 is a mGluR1 receptor-selective, negative allosteric modulator.Formula:C19H23N3OSPurezza:98%Colore e forma:SolidPeso molecolare:341.47MRK-623
CAS:MRK-623 (14k) is an oral GABA A agonist with high affinity for α1/α2/α3/α5 subunits and anxiolytic properties.Formula:C20H17FN4OColore e forma:SolidPeso molecolare:348.37γ-secretase modulator 1
CAS:gamma-secretase modulator 1 is a modulator of γ secretase and can be used in studies about the treatment of Alzheimer's disease.Formula:C24H24N4OSPurezza:99.75% - 99.96%Colore e forma:SolidPeso molecolare:416.54Irindalone
CAS:IrindaloneIrindalone is a potent serotonin (5-HT2) antagonist.Formula:C24H29FN4OPurezza:98%Colore e forma:SolidPeso molecolare:408.51Eplivanserin hemifumarate
CAS:Eplivanserin is an inverse agonist of 5-HT2A.Formula:C23H25FN2O6Colore e forma:SolidPeso molecolare:444.45Deramciclane
CAS:Deramciclane has high affinity for 5-HT2A and 5-HT2C receptors.Formula:C20H31NOColore e forma:SolidPeso molecolare:301.47BChE-IN-4
CAS:BChE-IN-4, a potent butyrylcholinesterase inhibitor, crosses blood-brain barrier, improves memory in mice; promising for Alzheimer's research.Formula:C24H37N3OColore e forma:SolidPeso molecolare:383.57AR-A 2
CAS:AR-A 2, a selective 5-HT1B antagonist; high guinea pig 5-HT1B/1D affinity (Ki: 0.24, 0.47 nM); 10x less for 5-HT1D (Ki: 5 nM).Formula:C27H36N4O2Purezza:98%Colore e forma:SolidPeso molecolare:448.65-Iodo-A-85380 dihydrochloride
CAS:α4β2 and α6β2 nicotinic acetylcholine receptors agonistFormula:C9H13Cl2IN2OPurezza:98%Colore e forma:SolidPeso molecolare:363.02Telenzepine
CAS:Telenzepine is a potent and selective M1 antimuscarinic.Formula:C19H22N4O2SPurezza:98%Colore e forma:SolidPeso molecolare:370.47VU0652835
CAS:VU0652835 is a negative allosteric modulator of metabotropic glutamate receptor subtype 5 (mGlu5) (IC50: 81 nM).Formula:C16H19N3O3SPurezza:98%Colore e forma:SolidPeso molecolare:333.41BChE-IN-14
CAS:BChE-IN-14 reverses cognitive decline, is safe for primary cells, crosses the blood-brain barrier, and selectively inhibits BChE (IC50: 0.011 μM for hBChE).Formula:C24H29NColore e forma:SolidPeso molecolare:331.49BNC375
CAS:BNC375 is a α7 nAChRs type I positive allosteric modulator (EC50: 1.9 μM).Formula:C19H23ClN2O3SPurezza:98%Colore e forma:SolidPeso molecolare:394.92Bibn 140
CAS:Bibn 140 is a highly selective M2 antagonist, it is used to treat Alzheimer's disease and other cognitive disorders.Formula:C32H44N4O3Purezza:98%Colore e forma:SolidPeso molecolare:532.72
