
Neuroscienza
Gli inibitori in neuroscienze sono composti progettati per modulare l'attività di proteine, enzimi o recettori specifici all'interno del sistema nervoso. Questi inibitori sono cruciali per studiare i meccanismi molecolari alla base della funzione neuronale, della trasmissione sinaptica e delle malattie neurodegenerative. Mirando ai recettori dei neurotrasmettitori, ai canali ionici e alle vie di segnalazione, gli inibitori in neuroscienze aiutano a esplorare la funzione cerebrale e a sviluppare strategie terapeutiche per disturbi neurologici come l'Alzheimer, il Parkinson e l'epilessia. Presso CymitQuimica, offriamo una vasta gamma di inibitori in neuroscienze di alta qualità per supportare la tua ricerca in neurobiologia, neurofarmacologia e scienze cognitive.
Sottocategorie di "Neuroscienza"
- recettore 5-HT(1.025 prodotti)
- ACK(1 prodotti)
- AChR(641 prodotti)
- Citrato liasi ATP(17 prodotti)
- Recettore adrenergico(2.997 prodotti)
- BACE(37 prodotti)
- Beta amiloide(217 prodotti)
- CaMK(73 prodotti)
- COX(598 prodotti)
- Recettore della dopamina(445 prodotti)
- Ricettore GABA(370 prodotti)
- Gamma-secretasi(57 prodotti)
- GluR(265 prodotti)
- GlyT(26 prodotti)
- Recettore dell'istamina(385 prodotti)
- LRRK2(43 prodotti)
- Recettore della melatonina(26 prodotti)
- NMDAR(10 prodotti)
- Recettore OX(40 prodotti)
- Recettore degli oppioidi(325 prodotti)
Mostrare 12 più sottocategorie
Trovati 5450 prodotti di "Neuroscienza"
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Talsaclidine
CAS:Talsaclidine: full M1 agonist, partial M2/M3 agonist with neuron-stimulating effects.Formula:C10H15NOPurezza:98%Colore e forma:SolidPeso molecolare:165.23Deramciclane fumarate
CAS:Deramciclane fumarate is a 5-HT(2A/C) antagonist with putative anxiolytic activity.Formula:C24H35NO5Colore e forma:SolidPeso molecolare:417.54Penbutolol
CAS:Penbutolol is a nonselective beta-blocker utilized as an antihypertensive and an antianginal.Formula:C18H29NO2Purezza:98%Colore e forma:SolidPeso molecolare:291.43GABAA receptor modulator-2
CAS:Compound 20: Selective, oral α5-GABAAR inhibitor, Ki: 4.1 nM. High stability, CNS safe.Formula:C22H22FN3O5SColore e forma:SolidPeso molecolare:459.49WAY-361789
CAS:WAY-361789 is an agonist of alpha7 nicotinic acetylcholine receptor.Formula:C22H31N5O3Colore e forma:SolidPeso molecolare:413.51VU0400195
CAS:VU0400195 is a oral effective, positive allosteric modulator of the metabotropic glutamate receptor 4 (mGlu(4)).Formula:C21H16ClN3O3Purezza:98%Colore e forma:SolidPeso molecolare:393.82Beperidium iodide
CAS:Beperidium iodide is a competitive antagonist of the acetylcholine receptor (pA2: 7.93).Formula:C23H34IN3O3Colore e forma:SolidPeso molecolare:527.44Muscarine iodide
CAS:Muscarinic acetylcholine receptor agonistFormula:C9H20INO2Purezza:98%Colore e forma:SolidPeso molecolare:301.17LY-411575 isomer 1
CAS:LY-411575 isomer 1 is a potent γ-secretase inhibitor. LY-411575 isomer 1 is an isomer of LY411575.Formula:C26H23F2N3O4Purezza:98%Colore e forma:SolidPeso molecolare:479.48Thiobencarb
CAS:Thiobencarb (Siacarb), a thiocarbamate herbicide, is a cholinesterase inhibitor.Formula:C12H16ClNOSPurezza:99.63%Colore e forma:Clear Colorless Liquid Thiobencarb Is A Pale Yellow To Brownish Yellow Liquid Non Corrosive Used As An HerbicidePeso molecolare:257.78E-3620
CAS:E-3620 is a potent antagonist of the 5-HT3 receptor and can be used to study dyskinesia and gastrointestinal dysfunction.Formula:C20H27Cl2N3O2Purezza:98.88% - 98.88%Colore e forma:SolidPeso molecolare:412.35Melatonin receptor agonist 1
CAS:Melatonin receptor agonist 1 (compound 20c) is a potent agonist of melatonin receptor (MT) with Ki values of 108 nM for MT2 and 1140 nM for MT 1 [1].Formula:C15H19N3O2Colore e forma:SolidPeso molecolare:273.33Tacitin
CAS:Tacitin (Benzoctamine Hydrochloride) shows sedative and anti-anxiety properties. Tacitin blocks the central postsynaptic serotonin receptors.Formula:C18H20ClNPurezza:98%Colore e forma:SolidPeso molecolare:285.81TC 1698 dihydrochloride
CAS:nicotinic α7 receptor agonistFormula:C13H18N2Purezza:98%Colore e forma:SolidPeso molecolare:202.3CGS8216
CAS:CGS8216 shows analgesic activity at high doses, has anxiolytic activity, and can be used to study immune system disorders.Formula:C16H11N3OPurezza:98.53%Colore e forma:SolidPeso molecolare:261.28M1 ligand 1
CAS:Compound 3b-b: N-desmethyl arecoline derivative, muscarinic M1 ligand, potential PET radiotracer.Formula:C20H21NO2Colore e forma:SolidPeso molecolare:307.39(1S,3R)-ACPD
CAS:(1S,3R)-ACPD is a group I and II mGlu receptor agonist.Formula:C7H11NO4Purezza:98%Colore e forma:SolidPeso molecolare:173.17DS2
CAS:Positive allosteric modulator of δ-subunit containing GABAA receptorsFormula:C18H12ClN3OSPurezza:98%Colore e forma:SolidPeso molecolare:353.83Ciclotizolam
CAS:Ciclotizolam, a thienotriazolodiazepine derivative and partial GABAA receptor agonist, has low efficacy but similar affinity as brotizolam.Formula:C20H18BrClN4SColore e forma:SolidPeso molecolare:461.81Foliglurax monohydrochloride
CAS:Foliglurax monohydrochloride, an antiparkinsonian, is a selective brain-penetrant mGluR4 PAM with an EC50 of 79 nM.Formula:C23H24ClN3O3SColore e forma:SolidPeso molecolare:457.9717-PA
CAS:17-PA is a GABAA receptor antagonist.Formula:C25H34OPurezza:98%Colore e forma:SolidPeso molecolare:350.54Prenylamine lactate
CAS:Prenylamine lactate, an ex-angina drug, depletes heart catecholamines and blocks calcium channels.Formula:C27H33NO3Purezza:98%Colore e forma:SolidPeso molecolare:419.56UCSF678
CAS:UCSF678: selective 42 nM partial agonist at 5-HT5AR, fewer off-target effects, and lower assay risks than SB-699551.Formula:C15H18N2O2SColore e forma:SolidPeso molecolare:290.38Desmethyl-YM 298198
CAS:mGlu1-selective antagonistFormula:C17H21ClN4OSPurezza:98%Colore e forma:SolidPeso molecolare:364.89CGP11952
CAS:CGP11952 is same the benzodiazepines in its pharmacological action and it also is an experimental benzodiazepine derivative.Formula:C21H21Cl2N5O2Purezza:98%Colore e forma:SolidPeso molecolare:446.33AChE/MAO-IN-2
Potent AChE/MAO-B inhibitor; IC50: AChE 0.0224 μM, MAO-B 0.0412 μM, MAO-A 0.1116 μM. Antioxidant, anti-β-amyloid, for AD research.Formula:C23H26N2O3Colore e forma:SolidPeso molecolare:378.46SX-3228
CAS:SX-3228 is a selective agonist of benzodiazepine1 (BZ1) receptor(IC50 of 17 nM).Formula:C18H18N4O3Purezza:98%Colore e forma:SolidPeso molecolare:338.36Itameline
CAS:RU 47213 can be used to inhibit scopolamine-induced working memory impairment in rats.Formula:C14H15ClN2O3Purezza:99.98%Colore e forma:SolidPeso molecolare:294.73Dual AChE-MAO B-IN-2
CAS:Potent Dual AChE-MAO B-IN-2 inhibits AChE (0.12 μM) & MAO B (0.01 μM); promising for Alzheimer's research.Formula:C26H25NO4Colore e forma:SolidPeso molecolare:415.48CGS 20625
CAS:partial agonist for the benzodiazepine binding site of the GABAA receptorFormula:C18H19N3O2Purezza:99.61%Colore e forma:SolidPeso molecolare:309.36Tridihexethyl chloride
CAS:Tridihexethyl is an anticholinergic, antimuscarinic, and antispasmolytic drug, which can be used to treat acquired nystagmus or peptic ulcer disease.Formula:C21H36ClNOColore e forma:SolidPeso molecolare:353.97DV 7028 hydrochloride
CAS:DV 7028 hydrochloride is a 5-HT2A receptor antagonist.Formula:C21H26ClFN4O3Purezza:98%Colore e forma:SolidPeso molecolare:436.91S20928
CAS:S20928 is an antagonist of melatonin receptor.Formula:C17H19NOColore e forma:SolidPeso molecolare:253.34AChE/MAO-IN-1
AChE/MAO-IN-1 is a potent inhibitor of human acetylcholinesterase (AChE), monoamine oxidase A (MAO-A), and monoamine oxidase B (MAO-B), demonstrating inhibitoryFormula:C23H26N2O3Colore e forma:SolidPeso molecolare:378.46NW-1772 free base
CAS:NW-1772 free base is a monoamine oxidase B inhibitor.Formula:C18H16ClNO3Colore e forma:SolidPeso molecolare:329.78NW-1772
CAS:NW-1772 is a highly potent and orally active inhibitor of monoamine oxidase B.Formula:C19H20ClNO6SPurezza:98%Colore e forma:SolidPeso molecolare:425.88Org 24598
CAS:Potent GlyT1b inhibitor, IC50 = 6.9 nM; little effect on GlyT-2, adrenoceptors, dopamine, 5HT receptors, GABA transporters.Formula:C19H20F3NO3Colore e forma:SolidPeso molecolare:367.36PXS-6302
CAS:PXS-6302: irreversible lysyl oxidase inhibitor, skin-penetrating, reduces scar collagen; IC50: 0.3-3.7 μM. May treat various fibrotic diseases.Formula:C10H10F3NO2SColore e forma:SolidPeso molecolare:265.25Chrysamine G
CAS:Chrysamine G, Congo red analog, blocks Aβ toxicity, probes Alzheimer's amyloid.Formula:C26H16N4Na2O6Colore e forma:SolidPeso molecolare:526.416UH-AH 37
CAS:UH-AH 37 is a antagonist of human muscarinic acetylcholine receptor.Formula:C21H23Cl2N3O2Purezza:98%Colore e forma:SolidPeso molecolare:420.33Lintopride
CAS:Lintopride is an antagonist of 5HT4. It has moderate 5HT3 antagonist properties.Formula:C14H19ClN4O2Purezza:98%Colore e forma:SolidPeso molecolare:310.78Ro 60-0175 fumarate
CAS:5-HT2 receptor agonistFormula:C15H16ClFN2O4Purezza:98%Colore e forma:SolidPeso molecolare:342.75Nerispirdine HCl
CAS:Nerispirdine enhances acetylcholine, blocks Na+ channels (IC50 11.9µM) and K(v) 1.1/1.2 channels (IC50 3.6/3.7µM).Formula:C17H19ClFN3Purezza:98%Colore e forma:SolidPeso molecolare:319.8AC260584
CAS:AC260584 is an M1 muscarinic receptor allosteric agonist (pEC50: 7.6).Formula:C20H29FN2O2Colore e forma:SolidPeso molecolare:348.45LY487379 hydrochloride
CAS:Positive allosteric modulator of mGlu2 receptorsFormula:C21H20ClF3N2O4SPurezza:98%Colore e forma:SolidPeso molecolare:488.91PF-4479745
CAS:PF-4479745 ia a potent and selective agonist of 5-HT2C receptor.Formula:C17H22N4Purezza:98%Colore e forma:SolidPeso molecolare:282.38hMAO-B-IN-2
CAS:hMAO-B-IN-2: selective oral hMAO-B inhibitor, crosses BBB, IC50=4 nM, potential for Alzheimer's research, neuroprotective, low toxicity.Formula:C18H23NO3Colore e forma:SolidPeso molecolare:301.38LY 2365109 hydrochloride
CAS:glycine transporter 1 (GlyT1) inhibitorFormula:C22H27NO5Purezza:98%Colore e forma:SolidPeso molecolare:385.45Alaproclate (hydrochloride)
CAS:Alaproclate, an SSRI, enhances serotonin and SIRT1, hinders NMDA and K+ currents in neurons, and shows antidepressant-like effects in rats.Formula:C13H19Cl2NO2Colore e forma:SolidPeso molecolare:292.2MPDC
CAS:MPDC acts as a competitive inhibitor against the Na+-dependent high-affinity glutamate transporter within forebrain synaptosomes.Formula:C7H9NO4Purezza:98%Colore e forma:SolidPeso molecolare:171.15Levemopamil HCl
CAS:Levemopamil HCl is used as a calcium channel blocker.Formula:C23H31ClN2Purezza:98%Colore e forma:SolidPeso molecolare:370.96SB 206553 hydrochloride
CAS:SB 206553 hydrochloride is a 5-HT2C inverse agonist and a 5-HT2C/5-HT2B receptor antagonist with anxiolytic activity, useful for studying neurological disordersFormula:C17H17ClN4OPurezza:99.56%Colore e forma:SolidPeso molecolare:328.8Ro 19-4603
CAS:Benzodiazepine inverse agonistFormula:C15H17N3O3SPurezza:98%Colore e forma:SolidPeso molecolare:319.38CC4
CAS:Selective α6β2/α4β2 partial agonist; Ki: 12/26nM (rat); poor α3β4/α7 affinity; stimulates dopamine release; reduces nicotine self-admin in rats.Formula:C24H30N4O2Colore e forma:SolidPeso molecolare:406.52AR-A 2
CAS:AR-A 2, a selective 5-HT1B antagonist; high guinea pig 5-HT1B/1D affinity (Ki: 0.24, 0.47 nM); 10x less for 5-HT1D (Ki: 5 nM).Formula:C27H36N4O2Purezza:98%Colore e forma:SolidPeso molecolare:448.6Telenzepine
CAS:Telenzepine is a potent and selective M1 antimuscarinic.Formula:C19H22N4O2SPurezza:98%Colore e forma:SolidPeso molecolare:370.47BChE-IN-14
CAS:BChE-IN-14 reverses cognitive decline, is safe for primary cells, crosses the blood-brain barrier, and selectively inhibits BChE (IC50: 0.011 μM for hBChE).Formula:C24H29NColore e forma:SolidPeso molecolare:331.49BNC375
CAS:BNC375 is a α7 nAChRs type I positive allosteric modulator (EC50: 1.9 μM).Formula:C19H23ClN2O3SPurezza:98%Colore e forma:SolidPeso molecolare:394.92NCS-382
CAS:γ-Hydroxybutyric acid antagonistFormula:C13H14O3Purezza:98%Colore e forma:SolidPeso molecolare:218.25Pregabalin arenacarbil
CAS:Pregabalin arenacarbil is a gabamimetic.Formula:C15H27NO6Colore e forma:SolidPeso molecolare:317.38HZ166
CAS:HZ-166 is a positive GABAA receptor modulator and a GABAA receptor subtype-selective benzodiazepine site ligand.Formula:C21H16N4O2Purezza:98%Colore e forma:SolidPeso molecolare:356.38VU0410425
CAS:VU0410425 is a metabotropic glutamate receptor subtype 1 negative allosteric modulator.Formula:C19H16ClN3O3Purezza:98%Colore e forma:SolidPeso molecolare:369.8T 82
CAS:T 82 is an antagonist of 5-HT3 and inhibitor of acetylcholinesterase (AChE) and used for the treatment of Alzheimer's Disease.Formula:C56H62N6O8Purezza:98%Colore e forma:SolidPeso molecolare:947.146GR 128107
CAS:GR 128107 is an antagonist of melatonin receptor.Formula:C16H20N2O2Colore e forma:SolidPeso molecolare:272.34γ-secretase modulator 2
CAS:Gamma-secretase modulator 2 selectively targets Alzheimer's by reducing Aβ(1-42), aiding in prevention and treatment.Formula:C25H22F4N6O2Purezza:98%Colore e forma:SolidPeso molecolare:514.47SKF-83566 hydrobromide
CAS:D1-like dopamine receptor antagonistFormula:C17H19BrClNOPurezza:98%Colore e forma:SolidPeso molecolare:368.7MS 245 oxalate
CAS:MS 245 oxalate is a 5-HT6 antagonist.Formula:C21H24N2O7SPurezza:98%Colore e forma:SolidPeso molecolare:448.49S-22153
CAS:S22153 is an antagonist of melatonin receptor.Formula:C14H17NOSColore e forma:SolidPeso molecolare:247.36(+/-)-Marmesin
CAS:Marmesin is a novel angiogenesis inhibitor.Formula:C14H14O4Purezza:98.00% - 98.00%Colore e forma:SolidPeso molecolare:246.26DCG-IV
CAS:DCG-IV: Class II mGluR agonist; anticonvulsant; neuroprotective; EC50: mGlu2R-0.35μM, mGlu3R-0.09μM; antagonizes Group I/III mGluRs.Formula:C7H9NO6Purezza:98%Colore e forma:SolidPeso molecolare:203.15Fonazine hydrochloride
CAS:Fonazine hydrochloride is a phenothiazine drug used for the treatment of migraine. It is a serotonin antagonist and histamine antagonist.Formula:C19H26ClN3O2S2Colore e forma:SolidPeso molecolare:428.01Thiochrome
CAS:Thiochrome is a selective enhancer of M4 muscarinic receptor of acetylcholine (ACh) affinity.Formula:C12H14N4OSPurezza:98%Colore e forma:SolidPeso molecolare:262.33Pd 158771
CAS:Pd 158771 is a D2 and 5-HT1A agonist.Formula:C22H31N5Colore e forma:SolidPeso molecolare:365.52DH97
CAS:MT2 melatonin receptor antagonistFormula:C22H26N2OPurezza:98%Colore e forma:SolidPeso molecolare:334.45AChE-IN-21
CAS:AChE-IN-21 (I-8), potent, selective AChE inhibitor, IC50: 2.66 nM, good BBB permeability.Formula:C24H29NO4Colore e forma:SolidPeso molecolare:395.49VU0090157
CAS:VU0090157, a novel allosteric potentiators of M1 muscarinic receptor, may provide novel treatments for schizophrenia and Alzheimer's disease.Formula:C19H21N3O7Purezza:98%Colore e forma:SolidPeso molecolare:403.39PF-0713
CAS:PF 0713, a GABAA receptor agonist, is used as an intravenous sedative-hypnotic for general anaesthesia, ICU sedation, procedural sedation, chemotherapy.Formula:C14H22OPurezza:98%Colore e forma:SolidPeso molecolare:206.32Ro 41-3290
CAS:Ro 41-3290 is the desethylated derivative of Ro 41-3696, which is an agonist of nonbenzodiazepine partial at the benzodiazepine receptor.Formula:C24H21ClN2O3Purezza:98%Colore e forma:SolidPeso molecolare:420.89Zamifenacin
CAS:Zamifenacin obviously decreases colonic motility in irritable bowel syndrome. Zamifenacin is an effective gut-selective muscarinic M3 receptor antagonist.Formula:C27H29NO3Purezza:98%Colore e forma:SolidPeso molecolare:415.52PD-102807
CAS:PD-102807 is a selective and competitive M4 muscarinic receptor antagonist for Parkinson's disease research, inhibit airway smooth muscle (ASM) contraction.Formula:C23H24N2O4Purezza:98.90%Colore e forma:SolidPeso molecolare:392.45JNJ-40418677
CAS:JNJ-40418677 is a γ-secretase modulator that selectively blocks γ-site cleavage of the APP without affecting the processing of Notch.Formula:C26H22F6O2Purezza:98%Colore e forma:SolidPeso molecolare:480.44VU0431316
CAS:VU0431316 is a negative mGlu5 allosteric modulator. It has activity in a mouse model of anxiety.Formula:C14H9ClN6O2Purezza:98%Colore e forma:SolidPeso molecolare:328.71L-775,606
CAS:L-775,606 is a selective agonist of 5-hydroxytryptamine 1D.Formula:C25H29FN6Purezza:98%Colore e forma:SolidPeso molecolare:432.54tCFA15
CAS:tCFA15: A trimethylated long-chain fatty alcohol with a 15-carbon side chain; may regulate Notch signaling and neuron differentiation.Formula:C24H44O2Purezza:98%Colore e forma:SolidPeso molecolare:364.612-Hydroxysaclofen
CAS:2-Hydroxysaclofen is a GABAB receptor antagonist.Formula:C9H12ClNO4SPurezza:98%Colore e forma:White SolidPeso molecolare:265.715-HT3 antagonist 2
CAS:5-HT3 antagonist 2 is an antagonist of 5-HT3 receptor.Formula:C18H21N3OPurezza:98%Colore e forma:SolidPeso molecolare:295.38ML381
CAS:ML381 is a M5-orthosteric antagonist with a high selectivity of muscarinic subtype.Formula:C21H21N3O4Colore e forma:SolidPeso molecolare:379.41(RS)-PPG
CAS:(RS)-PPG: Potent, selective III mGluRs agonist; EC50s: hmGluR4a 5.2μM, hmGluR6 4.7μM, hmGluR7b 185μM, hmGluR8a 0.2μM; neuroprotective, anticonvulsive.Formula:C8H10NO5PPurezza:98%Colore e forma:SolidPeso molecolare:231.145-HT4 antagonist 1
CAS:5-HT4 antagonist 1 is an antagonist of 5-HT4 (pKi = 9.6).Formula:C23H36N4O5SPurezza:99.75%Colore e forma:SolidPeso molecolare:480.62Clovoxamine
CAS:Clovoxamine fumarate (DU 23811 fumarate) is a 5-HT reuptake, serotonin and norepinephrine inhibitor with antidepressant and anticonvulsant activity.Formula:C14H21ClN2O2Purezza:99.44% - 99.75%Colore e forma:SolidPeso molecolare:284.78Bifeprunox
CAS:Bifeprunox: potent antipsychotic, partial agonist at D2-like/5-HT1A receptors; treats schizophrenia.Formula:C24H23N3O2Purezza:98%Colore e forma:SolidPeso molecolare:385.46GR 196429
CAS:GR 196429: MT1-selective melatonin receptor agonist; induces sleep, alters circadian rhythm, stimulates melatonin in mice.Formula:C14H18N2O2Purezza:98%Colore e forma:SolidPeso molecolare:246.3THK-523
CAS:THK-523 selectively binds to tau in Alzheimer's, potent in vitro/vivo. 18F-THK523 excels in tau imaging.Formula:C17H15FN2OColore e forma:SolidPeso molecolare:282.31Trimipramine
CAS:Trimipramine is an antidepressant with an anxiety-reducing sedative component to its action.Formula:C20H26N2Purezza:98%Colore e forma:SolidPeso molecolare:294.43HTL14242
CAS:HTL14242 is a mGlu5 Negative Allosteric Modulator.Formula:C16H8ClFN4Colore e forma:SolidPeso molecolare:310.71Naronapride
CAS:Naronapride (ATI-7505) is a potent agonist of the prokinetic 5-HT4receptor and can be used to study gastrointestinal disorders.Formula:C27H41ClN4O5Colore e forma:SolidPeso molecolare:537.09BuChE-IN-2
CAS:BuChE-IN-2 inhibits BuChE (IC50: 1.28 μM), NO (0.67 μM), Aβ, ROS, chelates Cu2+, penetrates BBB, used in Alzheimer's research.Formula:C28H20F4N6O3Colore e forma:SolidPeso molecolare:564.49Epibatidine 2HCl
CAS:Epibatidine 2HCl is a potent nicotinic agonist.Formula:C11H15Cl3N2Purezza:98%Colore e forma:SolidPeso molecolare:281.61L-CCG-l
CAS:group II metabotropic glutamate receptor agonistFormula:C6H9NO4Purezza:98%Colore e forma:SolidPeso molecolare:159.14Palonosetron
CAS:Palonosetron, a 5-HT3 antagonist with Ki of 0.17 nM, is used in the prevention and treatment of chemotherapy-induced nausea and vomiting (CINV).Formula:C19H24N2OPurezza:98%Colore e forma:SolidPeso molecolare:296.41
