
Neuroscienza
Sottocategorie di "Neuroscienza"
- recettore 5-HT(1.025 prodotti)
- ACK(1 prodotti)
- AChR(642 prodotti)
- Citrato liasi ATP(17 prodotti)
- Recettore adrenergico(3.004 prodotti)
- BACE(37 prodotti)
- Beta amiloide(220 prodotti)
- CaMK(73 prodotti)
- COX(598 prodotti)
- Recettore della dopamina(445 prodotti)
- Ricettore GABA(371 prodotti)
- Gamma-secretasi(60 prodotti)
- GluR(265 prodotti)
- GlyT(26 prodotti)
- Recettore dell'istamina(385 prodotti)
- LRRK2(43 prodotti)
- Recettore della melatonina(26 prodotti)
- NMDAR(10 prodotti)
- Recettore OX(41 prodotti)
- Recettore degli oppioidi(326 prodotti)
Trovati 5476 prodotti di "Neuroscienza"
BMY-14802 hydrochloride
CAS:BMY-14802 hydrochloride (BMS 181100 hydrochloride) is a selective antagonist of σ receptor (IC50 = 112 nM) with antipsychotic effects.Formula:C18H23ClF2N4OPurezza:99.97%Colore e forma:SolidPeso molecolare:384.85PNU-282987 free base
CAS:PNU-282987 is an α7 nAChR agonist (EC50=154 nM) and a 5-HT3 antagonist (IC50=4541 nM) for nervous system research.
Formula:C14H17ClN2OPurezza:99.64%Colore e forma:SolidPeso molecolare:264.75NS-2710
CAS:NS-2710, a GABA receptor agonist, is used potentially for the treatment of anxiety.Formula:C22H20N4OPurezza:99.7% - 99.82%Colore e forma:SolidPeso molecolare:356.42McN-A 343
CAS:McN-A 343: Selective M1 muscarinic agonist; reduces inflammation in colitis models.Formula:C14H18Cl2N2O2Purezza:99.65%Colore e forma:SolidPeso molecolare:317.21Oxotremorine M iodide
CAS:Oxotremorine M iodide (Oxotremorine methiodide) is an agonist of mAChR and potentiates NMDA receptors.Formula:C11H19IN2OPurezza:99.57%Colore e forma:SolidPeso molecolare:322.19ATC 0175
CAS:ATC 0175 hydrochloride is an orally active melanocyte concentrating hormone 1 receptor antagonist that is potent and selective.Formula:C23H26ClF2N5OPurezza:99.98%Colore e forma:SolidPeso molecolare:461.93BL-1020 Mesylate
CAS:BL-1020 Mesylate (CYP-1020 Mesylate) is a GABA A receptor agonist and D2 antagonist used in studies of neurodegeneration.Formula:C28H45ClN4O11S4Purezza:>99.99%Colore e forma:SolidPeso molecolare:777.39Ensaculin
CAS:Ensaculin, a benzopyrone-piperazine compound, enhances memory, protects neurons, and may treat dementia.Formula:C26H32N2O5Purezza:99.56% - 99.81%Colore e forma:SolidPeso molecolare:452.54Itasetron
CAS:Itasetron, a 5-HT3 antagonist, prevents memory loss in rats and has antiemetic effects in cancer treatments.
Formula:C16H20N4O2Purezza:98.58% - 99.33%Colore e forma:SolidPeso molecolare:300.36Faxeladol
CAS:Faxeladol: adrenergic, serotonin inhibitor & opioid agonist for neurological studies.Formula:C15H23NOPurezza:98.77% - 99.67%Colore e forma:SolidPeso molecolare:233.35Golexanolone
CAS:Golexanolone can be used to study neurological diseases.Formula:C21H31NO2Purezza:99.90% - 99.99%Colore e forma:SolidPeso molecolare:329.48LY 272015 hydrochloride
CAS:LY 272015 hydrochloride is a 5-HT2B receptor antagonist.Formula:C21H25ClN2O2Purezza:99.47%Colore e forma:SolidPeso molecolare:372.89CP 96021
CAS:"CP 96021 is an antagonist of 5-HT1/2 receptors, with anti-inflammatory and anti-ulcer effects for treating GI tract and asthma."
Formula:C29H21FN4OSPurezza:97.81% - 99.62%Colore e forma:SoildPeso molecolare:492.57Xanomeline
CAS:Xanomeline: orally active, M1/M4 selective activator for neurological disorders; promising in trials, crosses blood-brain barrier, liver metabolized.Formula:C14H23N3OSPurezza:99.61%Colore e forma:SolidPeso molecolare:281.42RS 67333 hydrochloride
CAS:RS 67333 hydrochloride is a selective 5-HT4R partial agonist (pKi=8.7) with neuroprotective properties for Alzheimer's research.Formula:C19H30Cl2N2O2Purezza:98.78%Colore e forma:SolidPeso molecolare:389.36LY-2624803
CAS:LY-2624803 is a 5-HT2A receptor antagonist and histamine receptor inverse agonist that can be used to improve slow wave sleep.Formula:C22H25N3O3Purezza:99.78% - 99.97%Colore e forma:SolidPeso molecolare:379.45Otenzepad
CAS:Otenzepad (AF-DX 116) is a selective antagonist of M2 mAChR with IC50s of 386 nM and 640 nM for rat heart and rabbit peripheral lung.Formula:C24H31N5O2Purezza:99.79%Colore e forma:SolidPeso molecolare:421.54Ref: TM-T16411
1mg47,00€5mg84,00€10mg120,00€25mg235,00€50mg376,00€100mg603,00€200mg848,00€1mL*10mM (DMSO)92,00€Tedatioxetine
CAS:Tedatioxetine (Lu AA24530) is a serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI) with antidepressant properties.Formula:C18H21NSPurezza:99.76% - >99.99%Colore e forma:SolidPeso molecolare:283.43AQW051
CAS:AQW051 (VQW-765) is an oral α7-nAChR activator for cognitive impairments, used in anxiety disorder studies.Formula:C19H22N2OPurezza:99.94%Colore e forma:SolidPeso molecolare:294.39Ref: TM-T26646
1mg34,00€2mg46,00€5mg66,00€10mg99,00€25mg205,00€50mg313,00€100mg439,00€500mg954,00€1mL*10mM (DMSO)67,00€Ricasetron
CAS:Ricasetron (Brl 46470) is a 5-HT3 receptor antagonist with pro-axonal lysing properties and is used in the study of anxiety disorders and anxiety disorders.Formula:C19H27N3OPurezza:99.52%Colore e forma:SolidPeso molecolare:313.44Progabide
CAS:Progabide (SL 76002) is an agonist of the gamma-aminobutyric acid receptor.Formula:C17H16ClFN2O2Purezza:99.68%Colore e forma:SolidPeso molecolare:334.77Cilansetron
CAS:Cilansetron is an effective and selective 5-HT3 receptor antagonist that can be used for related diseases caused by colitis.Formula:C20H21N3OPurezza:99.82% - 99.98%Colore e forma:SolidPeso molecolare:319.4BI-1408
CAS:BI-1408 is a modulator potent of γ secretase (IC50: 0.04 μM for Aβ42).Formula:C22H23FN6Purezza:99.63%Colore e forma:SolidPeso molecolare:390.46Adoprazine
CAS:Adoprazine (SLV313) is a potential atypical antipsychotic bearing potent D2 receptor antagonist and 5-HT1A receptor agonist properties.
Formula:C24H24FN3O2Purezza:99.83%Colore e forma:SolidPeso molecolare:405.46Saripidem
CAS:Saripidem (SL-85.0274) is a compound with anxiolytic activity.Formula:C19H20ClN3OPurezza:98.42%Colore e forma:SolidPeso molecolare:341.83Viloxazine
CAS:Viloxazine (Viloxazin) (Viloxazin) is a dual-action compound that functions as a norepinephrine reuptake inhibitor and exhibits potent agonistic activityFormula:C13H19NO3Purezza:99.65%Colore e forma:SolidPeso molecolare:237.29Cirsimaritin
CAS:Cirsimaritin has anti-bacterial, anti-inflammatory, anti-tumor, antioxidant effects, and protects kidneys; it weakly targets GABAA receptors.
Formula:C17H14O6Purezza:99.9%Colore e forma:SolidPeso molecolare:314.29Divaplon
CAS:Divaplon is a GABA receptor agonist (IC50: 0.056 µM) that displays non-sedating anxiolytic behavioral characteristics in a rat model of anxiety.Formula:C17H17N3O2Purezza:97.44% - 98.25%Colore e forma:SolidPeso molecolare:295.34E6801
CAS:E6801: selective 5-HT6 agonist for research in dementia, Parkinson's, depression, obesity, epilepsy, anxiety, etc.Formula:C17H18ClN5O2S2Purezza:96.32% - 97.24%Colore e forma:SolidPeso molecolare:423.94W-9 hydrochloride
CAS:W-9 hydrochloride is a calmodulin antagonist.Formula:C16H22Cl2N2O2SPurezza:98.9%Colore e forma:SolidPeso molecolare:377.33Ref: TM-T23525
1mg34,00€2mg42,00€5mg60,00€10mg90,00€25mg173,00€50mg269,00€100mg389,00€500mgPrezzo su richiesta1mL*10mM (DMSO)66,00€2-BFI hydrochloride
CAS:2-BFI hydrochloride: High-affinity I2 agonist; used in researching stroke and immune disease protection.Formula:C11H11ClN2OPurezza:99.94%Colore e forma:SolidPeso molecolare:222.67Ticalopride
CAS:Ticalopride: 5-HT3 agonist for digestive, orofacial, ENT disorders, and bulimia, GERD, IBS research.Formula:C14H20ClN3O3Purezza:99.51%Colore e forma:SolidPeso molecolare:313.78NB001
CAS:NB001 (HTS 09836) is an inhibitor of adenyl cyclase 1 exhibiting effects on neural and non-neural pain.Formula:C12H20N6OPurezza:99.69%Colore e forma:Off-White To Pale Pink SolidPeso molecolare:264.33Ref: TM-T16275
1mg74,00€5mg200,00€10mg295,00€25mg497,00€50mg710,00€100mg964,00€500mg1.935,00€1mL*10mM (DMSO)173,00€AZD 9272
CAS:AZD 9272 is a brain-permeable mGluR5 antagonist for the study of gastroesophageal reflux.Formula:C14H6F2N4OPurezza:98.29%Colore e forma:SolidPeso molecolare:284.22DA-6886
CAS:DA-6886 is a 5-HT4 agonist, relaxes rat oesophagus, with 1000x selectivity over hERG channels, pIC50: 4.3.Formula:C19H28Cl2N6O2Purezza:99.91% - 99.99%Colore e forma:SolidPeso molecolare:443.37R 59-022 hydrochloride
CAS:R 59-022 hydrochloride is a 5-HT antagonist, PKC activator, DGK inhibitor (IC50: 2.8 µM), and modulates lipid production in platelets and neutrophils.
Formula:C27H27ClFN3OSPurezza:97.7%Colore e forma:SolidPeso molecolare:496.04Nexopamil
CAS:Nexopamil (LU-49938) is a dual calcium channel and 5-HT2A receptor antagonist that inhibits cell contraction and growth.
Formula:C24H40N2O3Purezza:97.87% - >99.99%Colore e forma:SolidPeso molecolare:404.59Perphenazine dihydrochloride
CAS:Perphenazine dihydrochloride: Oral dopamine, histamine-1 antagonist; targets D2, D3, 5-HT2A, Alpha-1A; may treat psychiatric disorders, cancer.Formula:C21H28Cl3N3OSPurezza:99.67%Colore e forma:SolidPeso molecolare:476.89Femoxetine hydrochloride
CAS:Femoxetine hydrochloride is a selective 5-hydroxytryptamine reuptake inhibitor used in the study of migraine, depression and eating disorders.Formula:C20H26ClNO2Purezza:99.63%Colore e forma:SolidPeso molecolare:347.88Cyamemazine
CAS:Cyamemazine is an antipsychotic compound with sedative and anxiolytic activity.Cyamemazine is a 5-HT3, 5-HT2A, and 5-HT2C receptor antagonist.Formula:C19H21N3SPurezza:97.01%Colore e forma:SolidPeso molecolare:323.46Buntanetap
CAS:Buntanetap ((+)-Phenserine) is an inhibitor of TINAPs used in the study of neurological disorders, endocrine and metabolic disorders, and cardiovascular diseaseFormula:C20H23N3O2Purezza:98.2%Colore e forma:SolidPeso molecolare:337.42Ref: TM-T17312
1mg177,00€5mg447,00€10mg713,00€25mg1.333,00€50mg1.935,00€100mg2.520,00€1mL*10mM (DMSO)492,00€Cianopramine
CAS:Cianopramine (Ro 112465) is a selective 5-hydroxytryptamine uptake inhibitor and a tricyclic antidepressant used in the study of neurological disorders.Formula:C20H23N3Purezza:99.92% - 99.92%Colore e forma:SolidPeso molecolare:305.42Ezeprogind disulfate
CAS:Ezeprogind disulfate: neurotrophic inducer targeting neurodegeneration causes like Abeta, tau; for neurological disorder research.Formula:C25H48N6O8S2Purezza:99.72%Colore e forma:SolidPeso molecolare:624.81Sudoxicam
CAS:Sudoxicam (4-Hydroxy-2-methyl-N-2-thiazolyl-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxide) is a reversible antagonist of COX with anti-inflammatory, anti-edema
Formula:C13H11N3O4S2Purezza:99.93%Colore e forma:SolidPeso molecolare:337.37Suriclone
CAS:Suriclone (RP 31264), a cyclic pyrrolidone for anxiety, modulates GABA-A receptors without major sedation.Formula:C20H20ClN5O3S2Purezza:99.21% - 99.73%Colore e forma:SolidPeso molecolare:477.99Dipraglurant
CAS:Dipraglurant: a blood-brain permeable mGluR5 NAM, orally active, selective, IC50 = 21 nM, treats PD-LID.Formula:C16H12FN3Purezza:98.7%Colore e forma:SolidPeso molecolare:265.29Ref: TM-T15134
1mg92,00€5mg215,00€10mg313,00€25mg685,00€50mg1.009,00€100mg1.341,00€1mL*10mM (DMSO)260,00€Lirequinil
CAS:Lirequinil (Ro 41-3696) is a small molecule GABAA receptor agonist used to study neurological disorders.Formula:C26H25ClN2O3Purezza:98.54%Colore e forma:SolidPeso molecolare:448.94Masupirdine free base
CAS:Masupirdine free base (SUVN-502 free base) is a 5-HT6 receptor antagonist that can be used to study neurological disorders like Alzheimer's disease.Formula:C21H24BrN3O3SPurezza:98.36% - 99.65%Colore e forma:SolidPeso molecolare:478.4Felcisetrag
CAS:Felcisetrag (TD-8954), an oral 5-HT4 agonist with GI prokinetic effects, has a high affinity (pKi 9.4) for h5-HT4(c) receptors.Formula:C25H37N5O3Purezza:99.99%Colore e forma:SolidPeso molecolare:455.59Ref: TM-T28934
1mg87,00€5mg215,00€10mg318,00€25mg510,00€50mg692,00€100mg928,00€200mg1.251,00€1mL*10mM (DMSO)235,00€(Z)-Thiothixene
CAS:(Z)-Thiothixene (Thiothixene) is an antagonist of serotonergic receptor.
Formula:C23H29N3O2S2Purezza:99.21%Colore e forma:Yellow To Yellow With A Tan Cast PowderPeso molecolare:443.63SPD-473 citrate
CAS:SPD-473 citrate is an inhibitior of serotonin/dopamine/norepinephrine reuptake.Formula:C23H31Cl2NO8SPurezza:99.37%Colore e forma:SolidPeso molecolare:552.47RS 42358-197
CAS:RS 42358-197 (RS 25259-007) is a competitive 5-HT3 receptor antagonist.Formula:C19H23ClN2OPurezza:99.70%Colore e forma:SolidPeso molecolare:330.85Ref: TM-T20739
1mg158,00€5mg351,00€10mg527,00€25mg783,00€50mg1.054,00€100mg1.414,00€200mg1.908,00€1mL*10mM (DMSO)349,00€Litoxetine
CAS:Litoxetine: a selective 5-HT inhibitor & 5-HT3 antagonist, used as an antidepressant with antiemetic effects, Ki=85 nM.Formula:C16H19NOPurezza:99.68%Colore e forma:SolidPeso molecolare:241.33Ref: TM-T67956
1mg92,00€5mg207,00€10mg309,00€25mg527,00€50mg755,00€100mg1.044,00€500mg2.088,00€1mL*10mM (DMSO)178,00€Aβ-IN-1
CAS:Aβ-IN-1 is a novel, potent and orally active γ-secretase modulator (GSM).Formula:C35H49NPurezza:99.1%Colore e forma:SoildPeso molecolare:483.77Lesopitron
CAS:Lesopitron: anxiolytic, 5-HT1A agonist, treats rodent anxiety, counters benzodiazepine withdrawal, low toxicity, no alcohol/barbiturate interaction.Formula:C15H21ClN6Purezza:99.33% - 99.46%Colore e forma:SolidPeso molecolare:320.82Ref: TM-T25672
1mg133,00€5mg324,00€10mg477,00€25mg773,00€50mg1.063,00€100mg1.431,00€500mg2.872,00€1mL*10mM (DMSO)323,00€BPDBA
CAS:BPDBA is an effective, selective, and non-competitive inhibitor of the betaine/GABA transporter (BGT-1), displaying inhibitory activity against human BGT-1 andFormula:C19H20Cl2N2OPurezza:99.43% - 99.95%Colore e forma:SolidPeso molecolare:363.28ABP688
CAS:ABP688 is a non-competitive and selective mGluR5 antagonist(Ki = 1.7 nM). ABP688 can be used as a PET tracer for clinical imaging.Formula:C15H16N2OPurezza:98.63%Colore e forma:SolidPeso molecolare:240.3NNC 05-711
CAS:NNC 05-711 (NO-711 hydrochloride) is a potent and selective inhibitor of GAT-1 (GABA transporter 1), exerting anticonvulsant and analgesic effects.Formula:C21H23ClN2O3Purezza:99.92%Colore e forma:SolidPeso molecolare:386.87Iperoxo
CAS:Iperoxo (Iperoxo iodide) is an agonist of Muscarinic AChR and can be used to probe activation-related conformational transitions of muscarinic receptors.Formula:C10H17IN2O2Purezza:99.81%Colore e forma:SolidPeso molecolare:324.16Ref: TM-T25538
1mg50,00€5mg106,00€10mg168,00€25mg339,00€50mg512,00€100mg748,00€200mg1.026,00€1mL*10mM (DMSO)117,00€CT-179
CAS:CT-179 is a potent and selective inhibitor of OLIG2, reduces tumor cell proliferation and induces apoptosis, fpr medulloblastoma and glioblastoma.Formula:C17H22Cl2N6OPurezza:98.67%Colore e forma:SolidPeso molecolare:397.3Sarizotan HCl
CAS:Sarizotan HCl (EMD 128130 HCl) is a 5-HT1A receptor and dopamine receptor agonist and an hERG channel inhibitor used in Parkinson;s disease research.Formula:C22H22ClFN2OPurezza:96%Colore e forma:SolidPeso molecolare:384.87GSK233705
CAS:GSK233705, a muscarinic antagonist, is used to prevent/treat COPD and asthma.Formula:C24H29BrN2Purezza:99.87% - 99.98%Colore e forma:SolidPeso molecolare:425.4Roxindole
CAS:Roxindole: dopamine agonist, serotonin reuptake inhibitor, 5-HT1A agonist, developed for schizophrenia.Formula:C23H26N2OPurezza:98.03% - 98.93%Colore e forma:SolidPeso molecolare:346.47PPI-1019
CAS:PPI-1019 is an APP (β-amyloid A4) inhibitor for the treatment of neurological disorders and the study of Alzheimer's disease (AD).Formula:C36H54N6O5Purezza:95.16% - 98.16%Colore e forma:SolidPeso molecolare:650.85RWJ-51204
CAS:RWJ-51204: potent adenosine A2A blocker, GABA(A) partial agonist (IC50: 0.2-2 nM), neuroprotective, may treat Parkinson's.
Formula:C21H19F2N3O3Purezza:99.57% - 99.95%Colore e forma:SolidPeso molecolare:399.39Ref: TM-T16811
1mg333,00€5mg787,00€10mg1.074,00€25mg1.510,00€50mg1.882,00€100mg2.375,00€500mg4.655,00€Alpidem
CAS:Alpidem (Ananxyl), a non-sedative imidazopyridine anxiolytic, treats anxiety with high benzodiazepine receptor affinity.Formula:C21H23Cl2N3OPurezza:99.56% - 99.97%Colore e forma:White To Off-White SolidPeso molecolare:404.33Ref: TM-T26600
1mg58,00€5mg137,00€10mg207,00€25mg371,00€50mg522,00€100mg747,00€500mg1.513,00€1mL*10mM (DMSO)122,00€5-HT6/7 antagonist 1
CAS:5-HT6/7 antagonist 1 is a dual 5-HT6/7/2A and D2 receptor antagonist for the study of dementia and Alzheimer's disease.
Formula:C22H20FN3O3Purezza:98.78% - 99.26%Colore e forma:SolidPeso molecolare:393.41Nerisopam
CAS:Nerisopam is an agonist of gamma-aminobutyric acid (GABA) receptor.Formula:C18H19N3O2Purezza:98.52%Colore e forma:SolidPeso molecolare:309.36Ref: TM-T28159
1mg88,00€5mg190,00€10mg286,00€25mg464,00€50mg672,00€100mg945,00€200mg1.279,00€1mL*10mM (DMSO)256,00€Anpirtoline hydrochloride
CAS:Anpirtoline hydrochloride (D-16949 hydrochloride) is a 5-HT1B receptor agonist and 5-HT3 receptor antagonist used in the study of dyskinesia.Formula:C10H14Cl2N2SPurezza:>99.99% - >99.99%Colore e forma:SolidPeso molecolare:265.20Ecopipam
CAS:Ecopipam: orally active, selective dopamine D1/D5 antagonist (Ki: 1.2 nM/2.0 nM). 40x more selective over D2/D4/5-HT/α2a. For schizophrenia, obesity research.Formula:C19H20ClNOPurezza:99.68%Colore e forma:SolidPeso molecolare:313.82Muscimol HBr
CAS:Muscimol HBr (Agarin HBr) is an agonist of GABAA receptor.Formula:C4H7BrN2O2Purezza:98.13%Colore e forma:Off-White PowderPeso molecolare:195.01Ref: TM-T20657
1mg113,00€2mg169,00€5mg240,00€10mg385,00€25mg622,00€50mg898,00€100mg1.198,00€500mg2.422,00€1mL*10mM (DMSO)205,00€ADR-851 free base
CAS:ADR-851 free base is an antagonist of the HT3 receptor.Formula:C14H18ClN3O2Purezza:97.88% - 98.39%Colore e forma:SolidPeso molecolare:295.77Aplindore Fumarate
CAS:Aplindore Fumarate (DAB-452), a selective dopamine D2/D3 partial agonist, is used in Parkinson's and schizophrenia research.Formula:C22H22N2O7Purezza:99.66%Colore e forma:SolidPeso molecolare:426.42Teniloxazine
CAS:Teniloxazine is an orally available antidepressant compound with anti-hypoxic properties.Formula:C16H19NO2SPurezza:99.29%Colore e forma:SolidPeso molecolare:289.39Rilapine
CAS:Rilapine (Rilapinum) is an antipsychotic compound that shows high affinity for 5-HT6 receptors and can be used to study neurological disorders.Formula:C22H20ClN3Purezza:97.76% - 99.20%Colore e forma:SolidPeso molecolare:361.87Agomelatine hydrochloride
CAS:Agomelatine HCl is a MT1/MT2 receptor agonist (Ki: 0.1-0.27 nM) and a 5-HT2C antagonist (pKi: 6.2-6.4).Formula:C15H18ClNO2Purezza:99.57%Colore e forma:SolidPeso molecolare:279.76Eltenac
CAS:Eltenac, a cyclooxygenase (COX) inhibitor, is used potentially for the treatment of pain.
Formula:C12H9Cl2NO2SPurezza:98.53%Colore e forma:SolidPeso molecolare:302.18Lensiprazine
CAS:Lensiprazine (SLV314) is a potent dopamine D(2) receptor antagonist that acts as a serotonin reuptake inhibitor , and can be used to study bipolar disorder andFormula:C24H27FN4O2Purezza:97.86%Colore e forma:SolidPeso molecolare:422.5cis-Urocanic acid
CAS:cis-Urocanic acid ((E)-Urocanic acid) is a 5-HT2A receptor agonist (Kd: 4.6 nM).Formula:C6H6N2O2Purezza:99.81%Colore e forma:SolidPeso molecolare:138.12Glutaminyl Cyclase Inhibitor 1
CAS:Glutaminyl Cyclase Inhibitor 1 is a glutaminyl cyclase inhibitor (IC50: 0.5 μM) that can be used to study neurological disorders.Formula:C21H24FN3O2Purezza:99.81%Colore e forma:SolidPeso molecolare:369.43H-9 dihydrochloride
CAS:H-9 dihydrochloride: Strong PKA inhibitor, curbs 5-HT response and EGF signaling, affects pharyngeal function.Formula:C11H15Cl2N3O2SPurezza:97.3%Colore e forma:SolidPeso molecolare:324.23CBiPES hydrochloride
CAS:CBiPES hydrochloride (CBiPES HCl) is an orthosteric modulator of the mGlu2 receptor and is used to study neurological disorders like epilepsy.Formula:C21H20ClN3O2SPurezza:99.66%Colore e forma:SolidPeso molecolare:413.92SB228357
CAS:SB228357 is a potent and selective antagonist of the 5-HT receptor with pKis of 6.9, 8.0, and 9.0 for 5-HT2A, 5-HT2B, and 5-HT2C, respectively.Formula:C22H17F4N3O2Purezza:99.82%Colore e forma:SolidPeso molecolare:431.38MNI 137
CAS:MNI 137 is a negative allosteric modulator of mGlu2. MNI 137 inhibits glutamate-induced calcium mobilization with IC50s of 8.3 and 12.6 nM for human and rat.
Formula:C15H9BrN4OPurezza:97.49%Colore e forma:SolidPeso molecolare:341.16Selurampanel
CAS:Selurampanel (BGG492), an oral AMPA antagonist for epilepsy, migraine, and tinnitus studies.
Formula:C16H19N5O4SPurezza:99.60% - 99.78%Colore e forma:SolidPeso molecolare:377.42PHA 543613
CAS:PHA 543613 is a specific agonist of α7 nAChR (Ki = 8.8 nM) and can be used in studies about the cognitive deficits of Alzheimer's disease and schizophrenia.Formula:C15H17N3O2Purezza:99.43% - 99.96%Colore e forma:SolidPeso molecolare:271.31Ref: TM-T23145
1mg52,00€5mg102,00€10mg166,00€25mg358,00€50mg610,00€100mg895,00€500mg1.945,00€1mL*10mM (DMSO)100,00€MAO-B-IN-9
CAS:MAO-B-IN-9 is a monoamine oxidase B MAO-B inhibitor (IC50: 0.18 μM) that crosses the blood-brain barrier with potency, selectivity and time-dependence.
Formula:C18H24N2O2Purezza:99.93%Colore e forma:SolidPeso molecolare:300.4SB 699551 dihydrochloride
CAS:SB 699551 dihydrochloride is a 5-ht5a receptor antagonist.Formula:C34H47Cl2N3OPurezza:99.83%Colore e forma:SolidPeso molecolare:584.66Ref: TM-T23325
1mg50,00€5mg105,00€10mg170,00€25mg295,00€50mg424,00€100mg583,00€1mL*10mM (DMSO)142,00€Quinupramine
CAS:Quinupramine: an oral antidepressant targeting the serotonin system; penetrates CNS; doesn’t affect β-adrenergic system.Formula:C21H24N2Purezza:99.77%Colore e forma:SolidPeso molecolare:304.43GR 46611
CAS:GR 46611 is a selective 5-HT1B and 5-HT1D receptor agonist and can be used in studies about the treatment of epilepsy.Formula:C23H27N3O2Purezza:99.75%Colore e forma:SolidPeso molecolare:377.48Tiospirone
CAS:Tiospirone (BMY 13859-1 free base) is a 5-HT2 receptor antagonist and a dopamine blocker used in the study of neurological disorders such as schizophrenia.Formula:C24H32N4O2SPurezza:99.74%Colore e forma:SolidPeso molecolare:440.6Ref: TM-T24885
1mg123,00€5mg293,00€10mg537,00€25mg863,00€50mg1.161,00€100mg1.558,00€1mL*10mM (DMSO)354,00€Aceclidine
CAS:Aceclidine (1-azabicyclo[2.2.2]octan-3-yl acetate) is a modulator of M3 mAChR and can be used in studies about treating glaucoma by reducing intraocularFormula:C9H15NO2Purezza:>99.99%Colore e forma:SolidPeso molecolare:169.22GSK-1482160
CAS:GSK-1482160 is a CNS-penetrant negative allosteric modulator of P2X7 receptor with oral activity.
Formula:C14H14ClF3N2O2Purezza:99.57%Colore e forma:SolidPeso molecolare:334.72Ru-32514
CAS:Ru-32514 is a benzodiazepine receptor agonist.Formula:C18H17N3O2Purezza:99.21%Colore e forma:SolidPeso molecolare:307.35NKY80
CAS:NKY80 regulates the adenylyl cyclase catalytic activity in heart and lung tissues.Formula:C12H11N3O2Purezza:99.88%Colore e forma:SolidPeso molecolare:229.23Ref: TM-T16333
2mg47,00€5mg67,00€10mg96,00€25mg187,00€50mg325,00€100mg497,00€200mg715,00€1mL*10mM (DMSO)105,00€Sarmazenil
CAS:Sarmazenil (Ro 15-3505) is a partial inverse agonist at the benzodiazepine receptor and is used in the study of chronic hepatic encephalopathy.Formula:C15H14ClN3O3Purezza:99.46%Colore e forma:SolidPeso molecolare:319.74Piromelatine
CAS:Piromelatine is an agonist of melatonin MT1/MT2 receptors, 5-HT1A and 5-HT1D, and an antagonist of 5-HT2B.Piromelatine has antinociceptive activity withFormula:C17H16N2O4Purezza:99.83%Colore e forma:SolidPeso molecolare:312.32Ref: TM-T34081
1mg60,00€5mg130,00€10mg178,00€25mg334,00€50mg522,00€100mg713,00€1mL*10mM (DMSO)142,00€LRRK2-IN-7
CAS:LRRK2-IN-7: potent, selective CNS-active LRRK2 inhibitor, IC50 0.9 nM, >1000x selectivity vs kinases/channels/CYPs.Formula:C24H26N6OPurezza:99.26%Colore e forma:SolidPeso molecolare:414.55-HT2 antagonist 1
CAS:5-HT2 antagonist 1 is a potent 5-HT2 receptor antagonist, has weak α1 adrenoceptor blocking activity.Formula:C22H29FN4O2Purezza:99.76%Colore e forma:SolidPeso molecolare:400.49Ref: TM-T12597
1mg642,00€5mg1.288,00€10mg1.738,00€25mg2.583,00€50mg3.484,00€100mg4.708,00€1mL*10mM (DMSO)1.521,00€ELB-139
CAS:ELB-139 is a GABA A receptor agonist. ELB139 increases 5-HT in the striatum and prefrontal cortex of rats.Formula:C14H16ClN3OPurezza:>99.99%Colore e forma:SolidPeso molecolare:277.75
