Neuroscienza
Gli inibitori in neuroscienze sono composti progettati per modulare l'attività di proteine, enzimi o recettori specifici all'interno del sistema nervoso. Questi inibitori sono cruciali per studiare i meccanismi molecolari alla base della funzione neuronale, della trasmissione sinaptica e delle malattie neurodegenerative. Mirando ai recettori dei neurotrasmettitori, ai canali ionici e alle vie di segnalazione, gli inibitori in neuroscienze aiutano a esplorare la funzione cerebrale e a sviluppare strategie terapeutiche per disturbi neurologici come l'Alzheimer, il Parkinson e l'epilessia. Presso CymitQuimica, offriamo una vasta gamma di inibitori in neuroscienze di alta qualità per supportare la tua ricerca in neurobiologia, neurofarmacologia e scienze cognitive.
Sottocategorie di "Neuroscienza"
- recettore 5-HT(1.025 prodotti)
- ACK(1 prodotti)
- AChR(642 prodotti)
- Citrato liasi ATP(17 prodotti)
- Recettore adrenergico(2.999 prodotti)
- BACE(37 prodotti)
- Beta amiloide(217 prodotti)
- CaMK(73 prodotti)
- COX(598 prodotti)
- Recettore della dopamina(445 prodotti)
- Ricettore GABA(370 prodotti)
- Gamma-secretasi(57 prodotti)
- GluR(265 prodotti)
- GlyT(26 prodotti)
- Recettore dell'istamina(385 prodotti)
- LRRK2(43 prodotti)
- Recettore della melatonina(26 prodotti)
- NMDAR(10 prodotti)
- Recettore OX(40 prodotti)
- Recettore degli oppioidi(325 prodotti)
Mostrare 12 più sottocategorie
Trovati 5445 prodotti di "Neuroscienza"
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COR659
CAS:COR659: suppresses alcohol/chocolate intake in rats; enhances GABAB receptor, blocks CB1 receptor.Formula:C16H16ClNO3SPurezza:99.75%Colore e forma:SolidPeso molecolare:337.82Ref: TM-T36520
1mg38,00€5mg86,00€10mg123,00€25mg215,00€50mg299,00€100mg411,00€200mg560,00€1mL*10mM (DMSO)94,00€VU0029251
CAS:VU0029251 serves as a partial antagonist of mGluR5, exhibiting a binding affinity with a K i of 1.07 μM.Formula:C10H11N3S2Colore e forma:SolidPeso molecolare:237.34Wf-516
CAS:Wf-516 is a 5-HT reuptake inhibitor (Kis: 5 nM and 40 nM for 5-HT1A receptor and 5-HT2A receptor in humans, respectively), and with potent antidepressantFormula:C25H25Cl2N3O4Purezza:98%Colore e forma:SolidPeso molecolare:502.39Robalzotan
CAS:Robalzotan is a selective 5-HT1A receptor antagonist.Formula:C18H23FN2O2Purezza:98%Colore e forma:SolidPeso molecolare:318.395-HT2A&5-HT2C agonist-1
CAS:5-HT2A&5-HT2C agonist-1 (Example 2) is a dual-acting agent targeting the 5-HT2A and 5-HT2C receptors with respective IC50 values of 196 nM and 0.9 nM.
Formula:C14H20N2OPurezza:98%Colore e forma:SolidPeso molecolare:232.32Bisnorcymserine
CAS:Bisnorcymserine reversibly inhibits butyrylcholinesterase, binding Ser(200) and His(440) non-covalently and stacking with Trp(84).Formula:C21H25N3O2Purezza:98%Colore e forma:SolidPeso molecolare:351.44YM348
CAS:YM348 is an effective and orally active 5-HT2C receptor agonist. YM348 also shows a high affinity for the cloned human 5-HT2C receptor (Ki: 0.89 nM).Formula:C14H17N3OPurezza:98%Colore e forma:SolidPeso molecolare:243.3Lanabecestat
CAS:Lanabecestat (AZD3293) is a BACE1 inhibitor (Ki: 0.4 nM), Lanabecestat is used in the study of neurological diseases like Alzheimer's disease.Formula:C26H28N4OPurezza:98.55%Colore e forma:SolidPeso molecolare:412.53PNU109291
CAS:PNU109291, a potent and selective agonist of the 5-HT1D receptor, effectively mitigates dural plasma extravasation induced by trigeminal ganglion stimulation.Formula:C24H31N3O3Purezza:98%Colore e forma:SolidPeso molecolare:409.52C3
CAS:C3 functions as a selective inhibitor of monoamine oxidase B (MAO-B; IC50= 0.021 µM), demonstrating preference over monoamine oxidase A (MAO-A; IC50= 26.8 µM). This compound, at dosages of 0.1, 1, and 3 mg/kg, effectively counters MPTP-induced reductions in dopamine levels within the mouse brain.Formula:C18H19FN2O2Colore e forma:SolidPeso molecolare:314.35Facinicline hydrochloride
CAS:Facinicline hydrochloride (RG3487) is both a novel nicotinic alpha-7 receptor (alpha7nAChR) partial agonist (Ki = 6 nM) and an antagonist of 5-HT3(Ki = 1.2 nM).Formula:C15H19ClN4OPurezza:98.70%Colore e forma:SolidPeso molecolare:306.79Cyanopindolol fumarate
CAS:Cyanopindolol fumarate is a 5-HT receptor antagonist [1].Formula:C16H21N3O2C4H4O4Colore e forma:SolidPeso molecolare:345.4PZ-1190
CAS:PZ-1190, a multitarget ligand for serotonin and dopamine receptors, exhibits potential antipsychotic activity in rodents [1].Formula:C27H30N4O2S2Purezza:98%Colore e forma:SolidPeso molecolare:506.68Biphenylindanone A
CAS:Biphenylindanone A is a selective potentiator of human mGluR2 (hmGluR2),and for the treatment of neurological disorders.Formula:C30H30O4Purezza:98%Colore e forma:SolidPeso molecolare:454.56Octahydroaminoacridine succinate
CAS:Octahydroaminoacridine succinate, an acetylcholinesterase inhibitor, is used potentially for the treatment of Alzheimer's disease.Formula:C17H24N2O4Purezza:99.91%Colore e forma:SolidPeso molecolare:320.38Fosthiazate
CAS:Fosthiazate is a broad-spectrum nematicide that combats a range of plant parasitic nematodes such as Meloidogyne spp., Globodera spp., and Pratylenchus spp., byFormula:C9H18NO3PS2Purezza:97.78%Colore e forma:SolidPeso molecolare:283.35VU 0255035
CAS:VU 0255035 is a highly selective, competitive and brain penetrant muscarinic M1 receptor antagonist with an IC50 of 130 nM.
Formula:C18H20N6O3S2Purezza:98.09% - 98.1%Colore e forma:SolidPeso molecolare:432.52BMT-124110
CAS:BMT-124110: AAK1 inhibitor, IC50=0.9 nM, pain relief. BMT-090605: BIKE inhibitor, IC50=17 nM; GAK inhibitor, IC50=99 nM.Formula:C21H27N3O3Purezza:98.07%Colore e forma:SolidPeso molecolare:369.46AAK1-IN-3
CAS:AAK1-IN-3: Brain-penetrant AAK1 inhibitor for neuropathic pain research; IC50=11 nM.Formula:C20H20N4Colore e forma:SolidPeso molecolare:316.4AChE-IN-31
CAS:AChE-IN-31 (compound 1), a non-competitive acetylcholinesterase (AChE) inhibitor, exhibits potential for Alzheimer's disease research [1].Formula:C27H44Na2O9S2Colore e forma:SolidPeso molecolare:622.74AAK1-IN-4
CAS:AAK1-IN-4 selectively inhibits AAK1 with IC50 of 4.6 nM; penetrates CNS, oral bioactive, potential for studying neuropathic pain.Formula:C20H28N4O3Colore e forma:SolidPeso molecolare:372.46mGAT3/4-IN-2
CAS:mGAT3/4-IN-2 are potent inhibitors of mGAT3/mGAT4 with their pIC50 values of 5.44 and 5.25, respectively.Formula:C26H32ClN3OS2Colore e forma:SolidPeso molecolare:502.13AAK1-IN-5
CAS:AAK1-IN-5: Potent, selective AAK1 inhibitor; CNS-penetrant; oral; IC50: 1.2 nM; Ki: 0.05 nM; cell IC50: 0.5 nM. Useful in neuropathic pain research.Formula:C19H23F4N3OColore e forma:SolidPeso molecolare:385.4Quinolactacin A1
CAS:Quinolactacin A1, a strong AChE inhibitor from Penicillium citrinum, aids Alzheimer's research.Formula:C16H18N2O2Colore e forma:SolidPeso molecolare:270.33QM-FN-SO3
CAS:QM-FN-SO3 is a blood-brain barrier (BBB)-penetrable, near-infrared (NIR) probe with aggregation-induced emission (AIE) activity, specifically designed for the detection of Aβ plaques. It exhibits ultra-high signal-to-noise (S/N) ratio, binding affinity, and high-performance NIR emission, making it suitable for in vivo detection of Aβ plaques [1].Formula:C29H25N4NaO3S2Colore e forma:SolidPeso molecolare:564.65NAS-181 free base
CAS:NAS-181 free base is a 5-HT(1B) receptor antagonist.Formula:C19H26N2O4Colore e forma:SolidPeso molecolare:346.42MAO-B-IN-13
CAS:MAO-B-IN-13: a potent, reversible MAO-B inhibitor with BBB penetration, neuroprotective effects; used in Parkinson’s research (IC50=10nM).Formula:C18H19NO3Colore e forma:SolidPeso molecolare:297.35Tolterodine Dimer
CAS:Tolterodine Dimer is a derivative of Tolterodine -- a muscarinic receptor antagonist that is used to treat patients with overactive bladder.Formula:C35H41NO2Colore e forma:SolidPeso molecolare:507.71L-822179
CAS:L-822179 (α5IA) is a selective inverse agonist for the Α5 subtype of GABAA receptor with higher intrinsic activity at the A5 subtype than other drugs.Formula:C17H14N8O2Purezza:98.5% - 99.61%Colore e forma:SolidPeso molecolare:362.35AChE-IN-30
CAS:AChE-IN-30 is an acetylcholinesterase inhibitor (IC50 4.4 μM) that reduces oxidative stress and apoptosis, useful for Alzheimer’s disease research models.Formula:C22H24N4O2Purezza:99.96%Colore e forma:SolidPeso molecolare:376.45AAK1-IN-2
CAS:AAK1-IN-2, a potent (IC50=5.8 nM) AAK1 inhibitor, selective & brain-penetrant, is used for neuropathic pain studies.Formula:C20H20N4Colore e forma:SolidPeso molecolare:316.4Gepirone
CAS:Gepirone is a 5-HT1A receptor agonist belonging to the buspirone family. Gepirone HCl possesses greater selectivity for the 5-HT1A receptor than SSRIs.Formula:C19H29N5O2Purezza:99.35% - 99.89%Colore e forma:SolidPeso molecolare:359.473β-Hydroxy-lup-20(29)-en-16-one
CAS:3β-Hydroxy-lup-20(29)-en-16-one (compound 9) serves as a dual inhibitor of both AChE and BChE, displaying a preference for BChE with an IC50 of 28.9 μM [1].Formula:C30H48O2Colore e forma:SolidPeso molecolare:440.7Pomaglumetad methionil hydrochloride
CAS:LY2140023 hydrochloride: oral methionine prodrug of LY404039, a selective mGlu2/3 agonist, studied for schizophrenia.Formula:C12H19ClN2O7S2Purezza:98.57%Colore e forma:SolidPeso molecolare:402.87Diproqualone
CAS:Diproqualone, analogous to methaqualone, exhibits sedative, anxiolytic, anti-inflammatory, and analgesic properties [1].Formula:C12H14N2O3Colore e forma:SolidPeso molecolare:234.255CAY10649
CAS:1CAY10649, a thiazolinone compound, directly inhibits 5-lipoxygenase (5-LO) product formation in intact polymorphonuclear leukocytes (PMNL) with an IC50 value of 0.28 μM and in a soluble fraction of an S100 PMNL cell lysate with an IC50 value of 0.09 μM, following stimulation by calcium and arachidonic acid. This activity highlights its potential in mitigating inflammatory responses by targeting the biosynthesis of leukotrienes, substances implicated in various inflammatory processes such as neutrophil chemotaxis, increased vascular permeability, and smooth muscle contraction.Formula:C17H12ClNO2SColore e forma:SolidPeso molecolare:329.8BACE1-IN-10
CAS:BACE1-IN-10 is a potent inhibitor of BACE1, demonstrating sub-micromolar activity against recombinant BACE1 (rBACE1) [1].Formula:C33H49N5O8SPurezza:98%Colore e forma:SolidPeso molecolare:675.84SCS
CAS:SCS is a GABAA receptor antagonist.Formula:C14H12N2O3Purezza:99.73%Colore e forma:SolidPeso molecolare:256.26ELND007
CAS:ELND007 is a Gamma secretase inhibitor.Formula:C19H14F4N4O2SColore e forma:SolidPeso molecolare:438.4AMG-8718
CAS:AMG-8718, an oral BACE1 blocker (IC50: 0.0007 μM), also inhibits BACE2 (IC50: 0.005 μM), lowering CSF and Aβ40 brain levels.Formula:C25H19FN4O3Colore e forma:SolidPeso molecolare:442.44UNC9994
CAS:UNC9994 is a β-arrestin-biased dopamine D₂ receptor agonist (β-arrestin EC50 = 50 nM; Emax = 97%) with robust in vivo antipsychotic drug-like activities.Formula:C21H22Cl2N2OSColore e forma:SolidPeso molecolare:421.38NAS-181
CAS:NAS-181 is a potent and selective rat 5-hydroxytryptamine 1B (r5-HT1B) antagonist (Ki: 47 nM).NAS-181 enhances the accumulation of 5-HTP in rat brain regions.Formula:C20H30N2O7SColore e forma:SolidPeso molecolare:442.53CGP 55845 hydrochloride
CAS:CGP55845 hydrochloride is a potent and selective GABAB receptor antagonist with an IC 50 of 6 nM which can be used in neurological research [1] [2].Formula:C18H23Cl3NO3PColore e forma:SolidPeso molecolare:438.71RPC425 free base
CAS:RPC425 is a noncompetitive inhibitors of the Betaine-γ-Aminobutyric Acid Transporter 1 (BGT1).Formula:C22H27NO2S2Purezza:98%Colore e forma:SolidPeso molecolare:401.59N-Demethyl MK-6884
CAS:N-Demethyl MK-6884 (compound 34) is an M4 mAChR modulator for Alzheimer's and related disease research.Formula:C24H23N5OColore e forma:SolidPeso molecolare:397.47Zaldaride (free base)
CAS:Zaldaride (free base) is a calmodulin antagonist.Formula:C26H28N4O2Colore e forma:SolidPeso molecolare:428.53L-AP4
CAS:L-APB is an effective and specific agonist for the group III mGluRs (EC50s: 0.13, 0.29, 1.0, 249 μM for mGlu4, mGlu8, mGlu6, and mGlu7 receptors, respectively).Formula:C4H10NO5PPurezza:98%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:183.1SB 649915
CAS:SB 649915 is a serotonin reuptake inhibitor and 5-HT1A and 5-HT1B receptor antagonist.Formula:C26H29N3O3Colore e forma:SolidPeso molecolare:431.535-HT3-In-1
CAS:5-HT3-In-1 (compound example 8) exhabits with 5-HT3 inhibition activity.Formula:C16H21ClN4O3Purezza:98%Colore e forma:SolidPeso molecolare:352.82FPPQ
CAS:FPPQ blocks 5-HT3 and 5-HT6 receptors (Ki: 0.9 & 3 nM) and may improve psychosis and cognition.Formula:C21H19FN4O2SColore e forma:SolidPeso molecolare:410.46Zamifenacin fumarate
CAS:Zamifenacin fumarate (UK-76654 fumarate) is a potent and gut-selective antagonist of muscarinic M3 receptor.Formula:C31H33NO7Purezza:99.88%Colore e forma:SolidPeso molecolare:531.6Ref: TM-T13385
2mg34,00€5mg50,00€10mg75,00€25mg128,00€50mg200,00€100mg304,00€200mg424,00€1mL*10mM (DMSO)58,00€BMS 433796
CAS:BMS 433796 is a γ-secretase inhibitor that demonstrates Aβ-lowering activity within a transgenic mouse model of Alzheimer's disease.
Formula:C21H20F2N4O4Purezza:99.17%Colore e forma:SolidPeso molecolare:430.4A-424274
CAS:A-424274 is a positive allosteric modulator of α4β2 neuronal nicotinic receptor.Formula:C14H15N3Purezza:98%Colore e forma:SolidPeso molecolare:225.29L 687306
CAS:L 687306 is a partial agonist of muscarinic M1 receptors. It is also a highly competitive antagonist at cardiac M2 receptors and ileal M3 muscarinic receptors.Formula:C11H15N3OColore e forma:SolidPeso molecolare:205.26Cyclophostin
CAS:Cyclophostin is an irreversible inhibitor of acetylcholinesterase (AChE).Formula:C8H11O6PPurezza:98%Colore e forma:SolidPeso molecolare:234.14Capeserod HCl
CAS:Capeserod HCl, a 5-hydroxytriptamine 4 (5-HT4) receptor agonist, is used potentially for the treatment of Alzheimer's disease.Formula:C23H26Cl2N4O4Purezza:98%Colore e forma:SolidPeso molecolare:493.38Indeloxazine hydrochloride
CAS:Indeloxazine HCl: Serotonin releaser, NE reuptake inhibitor, NMDA antagonist; antidepressant that boosts acetylcholine in rats.Formula:C14H18ClNO2Purezza:98%Colore e forma:SolidPeso molecolare:267.75LY 53857
CAS:LY 53857 is a potent and selective antagonist of 5-HT2 serotonin receptor.Formula:C27H36N2O7Colore e forma:SolidPeso molecolare:500.592Frovatriptan
CAS:Frovatriptan, potent 5-HT 1B/D agonist, shows high cerebroselectivity and efficacy for migraine with aura.Formula:C14H17N3OPurezza:100%Colore e forma:SolidPeso molecolare:243.3Ref: TM-T60345
1mgPrezzo su richiesta5mgPrezzo su richiesta10mgPrezzo su richiesta25mg1.369,00€50mg1.783,00€100mg2.250,00€VU6007477
CAS:VU6007477 is a brain-penetrant M1 muscarinic receptor PAM (EC50 230 nM) used for research on CNS exposure and seizure-related models.Formula:C24H26N6O2Purezza:99.67%Colore e forma:SolidPeso molecolare:430.5MRK-560
CAS:MRK-560 is an effective and brain-penetrant inhibitor of γ-secretase.Formula:C19H17ClF5NO4S2Purezza:98.87%Colore e forma:SolidPeso molecolare:517.92FGIN-1-27
CAS:FGIN-1-27 is a high-affinity agonist of the translocator protein and a specific peripheral benzodiazepine receptor (PBR) ligand(Ki = 5.0 nM).Formula:C28H37FN2OPurezza:99.86%Colore e forma:SolidPeso molecolare:436.6RAGE/SERT-IN-1
CAS:RAGE/SERT-IN-1 is a potent, orally active inhibitor of advanced glycation end products (RAGE) and serotonin transporter (SERT), with IC50 values of 8.26 μM andFormula:C38H41ClN4OSColore e forma:SolidPeso molecolare:637.28BMS-933043
CAS:BMS-933043: α7 nAChR partial agonist, binds rat (Ki=3.3 nM) & human (Ki=8.1 nM), agonist with EC50=23.4 nM (calcium assay), 0.14-0.29 μM (electrophysiology).Formula:C16H19N7OPurezza:98%Colore e forma:SolidPeso molecolare:325.37PZ-II-029
CAS:PZ-II-029 is a modulator of α6β3γ2-selective GABAA channel.Formula:C18H15N3O3Purezza:99.79%Colore e forma:SolidPeso molecolare:321.33Ref: TM-T28479
1mg52,00€5mg111,00€10mg170,00€25mg305,00€50mg472,00€100mg723,00€500mg1.454,00€1mL*10mM (DMSO)202,00€GR 127935 hydrochloride
CAS:5-HT1B/1D receptor antagonistFormula:C29H32ClN5O3Purezza:98%Colore e forma:SolidPeso molecolare:534.05KBR 2822
CAS:KBR 2822 is an inhibitor of esterase.Formula:C9H15ClF3O3PSPurezza:98%Colore e forma:SolidPeso molecolare:326.7NAD 299 hydrochloride
CAS:Selective, high affinity 5-HT1A receptor antagonistFormula:C18H24ClFN2O2Purezza:98%Colore e forma:SolidPeso molecolare:354.85NO-711ME
CAS:NO-711ME (N-O711 Methyl ester) is a prodrug of NO-711. It also is a potent and selective GABA uptake inhibitor.Formula:C22H24N2O3Purezza:99.54%Colore e forma:SolidPeso molecolare:364.44Ref: TM-T24540
1mg64,00€5mg129,00€10mg188,00€25mg299,00€50mg427,00€100mg575,00€200mg767,00€1mL*10mM (DMSO)138,00€LY-426965
CAS:LY-426965 is a selective, potent, orally bioavailable 5-HT1A antagonist.Formula:C28H38N2O2Colore e forma:SolidPeso molecolare:434.61BACE1-IN-1
CAS:BACE1-IN-1 is a high brain penetrant BACE1 inhibitor (IC50s: 32 and 47 nM for human BACE1 and BACE2).Formula:C18H14F3N5O2Purezza:98%Colore e forma:SolidPeso molecolare:389.33ABT-418 hydrochloride
CAS:ABT-418 HCl enhances cognition and reduces anxiety as a selective nAChRs agonist, researched for Alzheimer's.Formula:C9H15ClN2OColore e forma:SolidPeso molecolare:202.68Dothiepin
CAS:Dothiepin (Dosulepin; Dothep), an antidepressant with sedative/anxiolytic properties, preferentially inhibits noradrenaline over serotonin uptake, enhancingFormula:C19H21NSPurezza:98%Colore e forma:SolidPeso molecolare:295.44Thioflosulide
CAS:Thioflosulide (L-745337) is a selective and potent COX2 inhibitor (IC50: 2.3 nM) with anti-inflammatory activity for the study of gastric ulcers.
Formula:C16H13F2NO3S2Purezza:>99.99%Colore e forma:SolidPeso molecolare:369.41LY108742
CAS:LY108742 is an antagonist of 5-HT2.Formula:C21H28N2O3Purezza:98%Colore e forma:SolidPeso molecolare:356.46Befiradol
CAS:Befiradol (NLX-112) is an agonist of 5-HT1A receptor.Formula:C20H22ClF2N3OColore e forma:SolidPeso molecolare:393.86Muscarine tosylate
CAS:Muscarine ((+)-Muscarine) tosylate, a prototype mAChR agonist, serves as a parasympathetic nervous system stimulant and is recognized for its toxic properties [1] [2].Formula:C16H27NO5SColore e forma:SolidPeso molecolare:345.45L 663581
CAS:L 663581 is the benzodiazepine receptor partial agonist.Formula:C17H16ClN5O2Purezza:98%Colore e forma:SolidPeso molecolare:357.79Des-4-fluorobenzyl Mosapride
CAS:Des-4-fluorobenzyl Mosapride, the main metabolite of mosapride, acts as a gastroprokinetic agent improving upper gastrointestinal (GI) motility by stimulating the serotonin receptor 4 (5-HT4; EC50= 74.2 nM, in guinea pig ileal longitudinal muscle myenteric plexus). It has been shown to increase colonic motility in dogs, horses, and guinea pigs in vivo. Mosapride, including this metabolite, is utilized in human and veterinary medicine to mitigate post-surgical and Parkinson's-induced constipation.Formula:C14H20ClN3O3Colore e forma:SolidPeso molecolare:313.78mAChR antagonist 1
CAS:Compound 4a, a mAChR antagonist, exhibits K i values of 255 nM for M1 and M5 subtypes, and lower values of 121 nM and 158 nM for M3 and M4 subtypes,Formula:C19H22N2O2Colore e forma:SolidPeso molecolare:310.39(2R,4R)-APDC
CAS:(2R,4R)-APDC is a selective group II metabotropic glutamate receptors (mGluRs) agonist. It has anticonvulsant and neuroprotective effects.Formula:C6H10N2O4Purezza:98%Colore e forma:SolidPeso molecolare:174.15UNC9994 hydrochloride
CAS:UNC9994 hydrochloride is a selective β-arrestin-biased D2R agonist, Ki of 79 nM, that stimulates β-arrestin and modulates cAMP.Formula:C21H23Cl3N2OSColore e forma:SolidPeso molecolare:457.84Nemonapride
CAS:Nemonapride is a dopamine D2-like receptor antagonist.Formula:C21H26ClN3O2Purezza:98%Colore e forma:SolidPeso molecolare:387.9U 89843A
CAS:U 89843A is a positive allosteric modulator of gamma-aminobutyric acid (GABA)A receptors.Formula:C16H23N5Purezza:99.62%Colore e forma:SolidPeso molecolare:285.39(±)-Fabesetron hydrochloride
CAS:FK1052 hydrochloride is a potent 5-HT3 and 5-HT4 receptor dual antagonist.Formula:C18H20ClN3OPurezza:98%Colore e forma:SolidPeso molecolare:329.82NAS181
CAS:rat 5-HT1B receptor antagonistFormula:C21H34N2O10S2Purezza:98%Colore e forma:SolidPeso molecolare:538.63GABAA receptor agent 2 TFA
CAS:Potent GABAA antagonist; IC50: 24 nM (α1β2γ2), Ki: 28 nM (rat); inactive on human GABA transporters.Formula:C22H22F3N3O3Colore e forma:SolidPeso molecolare:433.42Mesembrine
CAS:Mesembrine is an alkaloid, a 5-HT transporter inhibitor (K i 1.4 nM), and inhibits PDE4B (IC50 7.8 μM).Formula:C17H23NO3Colore e forma:SolidPeso molecolare:289.37MAO-B-IN-1
CAS:MAO-B-IN-1 is a monoamine oxidase B inhibitor and can be used for the research of neurological diseases.Formula:C16H14F3N3O2SPurezza:98%Colore e forma:SolidPeso molecolare:369.36GYKI-46903 HCl
CAS:GYKI-46903 is a noncompetitive 5-HT3 receptor antagonist.Formula:C17H21ClFNO2Colore e forma:SolidPeso molecolare:325.81LY3202626
CAS:LY3202626, an amyloid precursor protein secretase (BACE protein) inhibitor, is used for the treatment of Alzheimer's disease.Formula:C22H20F2N8O2SPurezza:98%Colore e forma:SolidPeso molecolare:498.51VU6005649
CAS:VU6005649 is an agonist of CNS penetrant mGlu7/8 receptor (EC50s: 0.65 μM and 2.6 μM for mGlu7 receptor and mGlu8 receptor, respectively).Formula:C16H12F5N3OPurezza:99.87%Colore e forma:SolidPeso molecolare:357.28Brasofensine sulfate
CAS:Brasofensine sulfate is a dopamine reuptake inhibitor.Formula:C16H22Cl2N2O5SColore e forma:SolidPeso molecolare:425.33rel-HDMP 28 hydrochloride
CAS:Rel-HDMP-28 hydrochloride (Compound 2g) is an analogue of methylphenidate, exhibiting selective affinity for the serotonin transporter (SERT) with a binding constant (Ki) of 105 nM [1].Formula:C18H22ClNO2Colore e forma:SolidPeso molecolare:319.83Gentisein
CAS:Gentisein (NSC-329491), a primary metabolite of Mangiferin, exhibits significant inhibition of serotonin uptake, demonstrating potency with an IC50 value of 4.7Formula:C13H8O5Purezza:96.89%Colore e forma:SolidPeso molecolare:244.2MFZ 10-7
CAS:MFZ 10-7 is anegative allosteric modulator of the mGluR5.Formula:C15H9FN2Purezza:99.80%Colore e forma:SolidPeso molecolare:236.24(+)-Bicuculline methiodide
CAS:(+)-Bicuculline methiodide is a GABAA receptor blocker that blocks epileptogens and may be used in the study of neurological disorders.Formula:C21H20INO6Purezza:99.24%Colore e forma:SolidPeso molecolare:509.29JM-1232
CAS:JM-1232 is a sedative and hypnotic drug being researched as a potential anesthetic.Formula:C24H27N3O2Colore e forma:SolidPeso molecolare:389.49CGP-54626 free base
CAS:CGP-54626 is a selective antagonist of the GABAB receptor (IC50 = 4 nM ).Formula:C18H28Cl2NO3PPurezza:98%Colore e forma:SolidPeso molecolare:408.3L-772,405
CAS:L-772,405 is a highly selective agonists of h5-HT(1D) receptor.Formula:C26H31FN6OPurezza:98%Colore e forma:SolidPeso molecolare:462.56
