Neuroscienza
Gli inibitori in neuroscienze sono composti progettati per modulare l'attività di proteine, enzimi o recettori specifici all'interno del sistema nervoso. Questi inibitori sono cruciali per studiare i meccanismi molecolari alla base della funzione neuronale, della trasmissione sinaptica e delle malattie neurodegenerative. Mirando ai recettori dei neurotrasmettitori, ai canali ionici e alle vie di segnalazione, gli inibitori in neuroscienze aiutano a esplorare la funzione cerebrale e a sviluppare strategie terapeutiche per disturbi neurologici come l'Alzheimer, il Parkinson e l'epilessia. Presso CymitQuimica, offriamo una vasta gamma di inibitori in neuroscienze di alta qualità per supportare la tua ricerca in neurobiologia, neurofarmacologia e scienze cognitive.
Sottocategorie di "Neuroscienza"
- recettore 5-HT(1.025 prodotti)
- ACK(1 prodotti)
- AChR(647 prodotti)
- Citrato liasi ATP(17 prodotti)
- Recettore adrenergico(3.024 prodotti)
- BACE(37 prodotti)
- Beta amiloide(230 prodotti)
- CaMK(73 prodotti)
- COX(602 prodotti)
- Recettore della dopamina(445 prodotti)
- Ricettore GABA(373 prodotti)
- Gamma-secretasi(62 prodotti)
- GluR(265 prodotti)
- GlyT(26 prodotti)
- Recettore dell'istamina(385 prodotti)
- LRRK2(43 prodotti)
- Recettore della melatonina(26 prodotti)
- NMDAR(10 prodotti)
- Recettore OX(41 prodotti)
- Recettore degli oppioidi(327 prodotti)
Mostrare 12 più sottocategorie
Trovati 5637 prodotti di "Neuroscienza"
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Citalopram-d6
CAS:Prodotto controllatoApplications Labelled Citalopram (C505000), an inhibitor of serotonin (5-HT) uptake. Used as an antidepressant.
References Christensen, A.V., et al.: Eur. J. Pharmacol., 41, 153 (1977), Keller, M.B., et al.: J. Clin. Psychiatry, 61, 896 (2000), Von Moltke, L.L., et al.: Drug Metab. Dispos., 29, 1102 (2001),Formula:C202H6H15FN2OColore e forma:NeatPeso molecolare:330.43Jatrorrhizine chloride
CAS:Jatrorrhizine chloride (Neprotine chloride) is an alkaloid isolated from Rhizoma coptidis with neuroprotective, antimicrobial, and antiplasmodial activities.Formula:C20H20ClNO4Purezza:99.79%Colore e forma:SolidPeso molecolare:373.8GSK-1034702
CAS:GSK-1034702 is an M1 mAChR agonist that improves cognitive deficits and may be useful in the study of neurologic disorders.Formula:C18H24FN3O2Purezza:99.41%Colore e forma:SolidPeso molecolare:333.4Xanomeline tartrate
CAS:Xanomeline tartrate (LY 246708 tartrate) 是 M1和 M4 mAChR 激动剂，具有抗精神病样活性，可改善认知，可用于研究精神分裂症和阿尔茨海默病。Formula:C18H29N3O7SPurezza:99.19% - 99.99%Colore e forma:SolidPeso molecolare:431.5LP-533401 hydrochloride
CAS:LP-533401 hydrochloride is a peripheral Tph inhibitor that does not cross the BBB and can be used to study periodontal disease and hepatic steatosis.Formula:C27H23ClF4N4O3Purezza:98%Colore e forma:SolidPeso molecolare:562.94S1RA
CAS:S1RA (E-52862)(E-52862) is a potent, selective antagonist of the sigma-1 receptor (σ1R, Ki=17 nM), demonstrating significant selectivity over the sigma-2Formula:C20H23N3O2Purezza:99.45%Colore e forma:SolidPeso molecolare:337.42Rotigotine
CAS:Rotigotine (1-Naphthalenol, 5,6,7,8-tetrahydro-6-[propyl[2-(2-thienyl)ethyl]amino]-) is an antiparkinson agent and dopamine receptor agonist.Formula:C19H25NOSPurezza:99.04% - 99.88%Colore e forma:SolidPeso molecolare:315.47Riluzole
CAS:Riluzole (RP-54274) is an anticonvulsant, glutamate antagonist, and prolongs ALS patient survival.Formula:C8H5F3N2OSPurezza:99.71% - 99.88%Colore e forma:PowderPeso molecolare:234.2(S)-4CPG
CAS:(S)-4CPG ((S)-4-Carboxyphenylglycine) is a competitive mGlu1 receptor antagonist that attenuates nociceptive hypersensitivity and nociceptive abnormalities associated with sciatic nerve constriction injuries in rats, and may be used in the study of neurological disorders.Formula:C9H9NO4Purezza:99.96%Colore e forma:SolidPeso molecolare:195.17Monepantel
CAS:Monepantel (AAD1566) is an organic anthelmintic and an antagonist of nAChRs from roundworms and esophageostomy.Formula:C20H13F6N3O2SPurezza:99.83%Colore e forma:White PowderPeso molecolare:473.39Ref: TM-T16126
1mg93,00€5mg236,00€1mL*10mM (DMSO)259,00€10mg340,00€25mg670,00€50mg964,00€100mg1.378,00€Velufenacin
CAS:Velufenacin is an antagonist of muscarinic receptor[1].Formula:C19H20ClFN2O2Purezza:99.65%Colore e forma:SolidPeso molecolare:362.83Ref: TM-T9771
1mg47,00€5mg96,00€1mL*10mM (DMSO)105,00€10mg156,00€25mg270,00€50mg370,00€100mg522,00€200mg687,00€Syk Inhibitor II
CAS:Syk inhibitor II, a cell-permeable, ATP-competitive, pyrimidine-carboxamide compound, selectively and reversibly inhibits Syk (IC50 = 41 nM).Formula:C14H15F3N6OPurezza:97.63%Colore e forma:SolidPeso molecolare:340.3Chlorpyrifos (diethyl-d10)
CAS:Chlorpyrifos (diethyl-d10) is a deuterated compound of Chlorpyrifos. Chlorpyrifos has a CAS number of 2921-88-2. Chlorpyrifos is an organothiophosphate cholinesterase inhibitor that is used as an insecticide and as an acaricide.Formula:C9H1D10Cl3NO3PSColore e forma:SolidPeso molecolare:360.65Donepezil-d5
CAS:Donepezil-d5 is a deuterated compound of Donepezil. Donepezil has a CAS number of 120014-06-4. Donepezil is a piperidine-based, potent, specific, and reversible inhibitor of acetylcholinesterase (AChE). It can be used for the treatment of mild to moderate dementia of the Alzheimer's type.Formula:C24H24D5NO3Colore e forma:SolidPeso molecolare:384.52Acephate-d3 (acetyl-d3)
CAS:Acephate-d3 (acetyl-d3) is a deuterated compound of Acephate. Acephate has a CAS number of 30560-19-1. Acephate is an anticholinesterase insecticide with a weak inhibitory effect on AChE in rats, but it can effectively inhibit AChE in cockroaches.Formula:C4H7D3NO3PSColore e forma:SolidPeso molecolare:186.18Sulindac EP Impurity C-d3
CAS:Sulindac EP Impurity C-d3 is a deuterated compound of Sulindac EP Impurity C. Sulindac EP Impurity C has a CAS number of 32004-67-4. (E/Z)-Sulindac sulfide is a potent γ-secretase modulator (GSM) that selectively reduces Aβ42 production in favor of shorter Aβ species. (E/Z)-Sulindac sulfide can be used for researching Alzheimer's disease [1].Formula:C20H14D3FO2SColore e forma:SolidPeso molecolare:343.43Pyridostigmine-d6 bromide
CAS:Pyridostigmine D6 bromide is the deuterium labeled Pyridostigmine, which is a parasympathomimetic and a reversible inhibitor of cholinesterase.Formula:C9H13BrN2O2Purezza:98%Colore e forma:SolidPeso molecolare:267.15Fenitrothion-d6 (O,O-dimethyl-d6)
CAS:Fenitrothion-d6 (O,O-dimethyl-d6) is a deuterated compound of Fenitrothion. Fenitrothion has a CAS number of 122-14-5. Fenitrothion is an organothiophosphate cholinesterase inhibitor. Fenitrothion is used as an insecticide.
Formula:C9H6D6NO5PSColore e forma:SolidPeso molecolare:283.27R 59-022
CAS:R 59-022 (DKGI-I) is a DGK inhibitor and a 5-HT Receptor antagonist that blocks filovirus internalization in host cells.Formula:C27H26FN3OSPurezza:98.55%Colore e forma:SolidPeso molecolare:459.58Ref: TM-T16709
1mg35,00€5mg74,00€1mL*10mM (DMSO)75,00€10mg119,00€25mg269,00€50mg447,00€100mg733,00€200mg973,00€Varenicline
CAS:Varenicline (CP 526555) is a selective partial agonist of the α4β2 nAChR and a full agonist of the α3β4 nAChR and α7 nAChR.Formula:C13H13N3Purezza:99.76%Colore e forma:SolidPeso molecolare:211.26Ref: TM-T4246L
2mg34,00€5mg50,00€1mL*10mM (DMSO)55,00€10mg75,00€25mg137,00€50mg200,00€100mg313,00€200mg464,00€Cyproheptadine hydrochloride
CAS:Cyproheptadine hydrochloride (Periactin hydrochloride) is a hydrochloride salt form of cyproheptadine which is a histamine receptor antagonist.Formula:C21H21N·HClPurezza:99.88% - 99.97%Colore e forma:SolidPeso molecolare:323.86Anatabine dicitrate
Anatabine dicitrate is a tobacco alkaloid that can cross the blood-brain barrier.Formula:C22H28N2O14Purezza:98%Colore e forma:SolidPeso molecolare:544.46Dilpacimab
CAS:Dilpacimab (ABT165) is a dual-variable antibody that targets DLL4 and VEGF pathways, showing potential in cancer research by blocking angiogenesis and Notch.Purezza:95% - 97.7% (SDS-PAGE); 95.6% (SEC-HPLC)Colore e forma:LiquideeAChE/eqBuChE-IN-1
CAS:eeAChE/eqBuChE-IN-1 (compound 3F) serves as a reversible dual inhibitor of eeAChE/eqBuChE, exhibiting IC50 values of 1.3 μM and 0.81 μM, respectively. In addition, this compound demonstrates anti-inflammatory properties and provides neuroprotective effects against Aβ25-35-induced injury in PC12 cells [1].Formula:C14H16N2O2Colore e forma:SolidPeso molecolare:244.29Arazasetron HCl
CAS:Arazasetron is an antiemetic which acts as a 5-HT3 receptor antagonist, pKi = 9.27.Formula:C17H20ClN3O3Purezza:98%Colore e forma:SolidPeso molecolare:349.81Monoamine Oxidase B inhibitor 4
CAS:Monoamine Oxidase B Inhibitor 4 (compound 1l), with a potent IC50 value of 8.3 nM, is a selective human monoamine oxidase-B (hMAO-B) inhibitor. This compound demonstrates anti-neuroinflammatory properties and exhibits low neurotoxicity. It effectively inhibits the release of NO, TNF-α, and IL-1β induced by LPS and Aβ1-42, and additionally mitigates the cytotoxic effects triggered by Aβ(1-42) .Formula:C15H11Cl2NO3Colore e forma:SolidPeso molecolare:324.16Atropine hydrobromide
CAS:Atropine hydrobromide is a biochemical.Formula:C17H24BrNO3Colore e forma:SolidPeso molecolare:370.28BChE-IN-25
CAS:BChE-IN-25 (compound 4I) acts as a selective inhibitor of BChE, demonstrating an IC 50 of 3.77μM and exhibiting 22-fold greater selectivity towards BChE over AChE [1].Formula:C17H23NO2Colore e forma:SolidPeso molecolare:273.37Risperidone Mesylate
CAS:Risperidone Mesylate is a selective serotonin 5-HT2 receptor and dopamine D2 receptor blocker.Formula:C24H31FN4O5SPurezza:98%Colore e forma:SolidPeso molecolare:506.59Benmoxin
CAS:Benmoxin is a monoamine oxidase inhibitor (MAOI) that is irreversible and nonselective.Formula:C15H16N2OPurezza:98%Colore e forma:SolidPeso molecolare:240.30Unasnemab
CAS:Unasnemab (MT-3921) binds RGMa, promoting neuroregeneration and locomotor function, showing potential for spinal cord injury and regenerative research.Purezza:95% - 97.4% (SDS-PAGE); 98.3% (SEC-HPLC)Colore e forma:LiquidPeso molecolare:144.90 kDaKeto Ziprasidone
CAS:Ziprasidone, an antipsychotic agent, functions as a dual antagonist of 5-HT (serotonin) and dopamine receptors.Formula:C21H19ClN4O2SPurezza:98%Colore e forma:SolidPeso molecolare:426.92Bapineuzumab
CAS:Bapineuzumab (AAB-001) is a humanised monoclonal antibody targeting amyloid-beta (Aβ), soluble and oligomeric forms of amyloid β, Alzheimer's disease (AD).Purezza:95%Colore e forma:LiquidPeso molecolare:145.86 kDaRocatinlimab
CAS:Rocatinlimab (AMG 451) (KHK4083) is a fully human, non-fucosylated IgG1 anti-OX40 monoclonal antibody indicated for atopic dermatitis (AD) research [1].Colore e forma:LiquidRemternetug
CAS:Remternetug (LY3372993) is a humanised monoclonal antibody targeting N3pG-Aβ, recognising pyroglutamated Aβ within amyloid plaques, Alzheimer's disease.Purezza:95% - 97.6% (SDS-PAGE); 98.7% (SEC-HPLC)Colore e forma:LiquidPeso molecolare:144.87 kDaEscitalopram
CAS:Escitalopram (Seroplex), a serotonin inhibitor for depression, curbs alcohol intake and is favored over tricyclics for tardive dyskinesia.Formula:C20H21FN2OPurezza:99.82%Colore e forma:White Or White Crystalline PowderPeso molecolare:324.39Tarextumab
CAS:Tarextumab is an anti-Notch2/3 mAb, a promising candidate for breast, lung, ovarian, and pancreatic cancers.Purezza:95%Colore e forma:LiquidPeso molecolare:~150 kDaAChE-IN-65
CAS:AChE-IN-65 (Compound DABA_1) serves as a mixed inhibitor of acetylcholinesterase (AChE), exhibiting a Ki of 556.4 μM against Electrophorus electricus AChE.Formula:C15H8N2O6Colore e forma:SolidPeso molecolare:312.23Dezamizumab
CAS:Dezamizumab is a humanized antibody targeting the serum amyloid P component (SAP) to clear amyloid fibrils via macrophage phagocytosis, for research in systemic amyloid diseases.Purezza:95% - 98.2% (SDS-PAGE); 98.7% (SEC-HPLC)Colore e forma:LiquidPeso molecolare:145.82 kDaN-Methyl amisulpride
CAS:N-Methyl amisulpride (Amisulpride impurity H) is a 5-HT7 receptor, D2 receptor, and D3 receptor antagonist used in the study of acute schizophrenia.Formula:C18H29N3O4SColore e forma:SolidPeso molecolare:383.51(+)-Tomoxetine hydrochloride
CAS:(+)-Tomoxetine hydrochloride is a bioactive chemical.Formula:C17H22ClNOPurezza:98%Colore e forma:SolidPeso molecolare:291.821,2-Dimyristoyl-sn-glycero-3-phospho-rac-(1-glycerol) Sodium Salt
CAS:Formula:C34H66NaO10PPurezza:>98.0%(T)Colore e forma:White to Almost white powder to crystalPeso molecolare:688.86Pipamperone
CAS:Formula:C21H30FN3O2Purezza:>98.0%(HPLC)Colore e forma:White to Light yellow to Light orange powder to crystalPeso molecolare:375.49Gestrinone
CAS:Formula:C21H24O2Purezza:>98.0%(T)Colore e forma:Light yellow to Yellow powder to crystalPeso molecolare:308.42KB-R 7943
CAS:Formula:C16H17N3O3S·CH4O3SPurezza:>98.0%(HPLC)Colore e forma:White to Yellow to Green powder to crystalPeso molecolare:427.49Ruthenium(II) Nitrosyl Chloride
CAS:Formula:RuCl3NOPurezza:>97.0%(T)Colore e forma:Yellow to Amber to Dark red powder to crystalPeso molecolare:255.45Tyrphostin AG 494
CAS:Formula:C16H12N2O3Purezza:>98.0%(HPLC)(N)Colore e forma:Light yellow to Amber to Dark green powder to crystalPeso molecolare:280.28Hyodeoxycholic Acid
CAS:Formula:C24H40O4Purezza:>98.0%(T)Colore e forma:White to Orange to Green powder to crystalPeso molecolare:392.58Medroxyprogesterone
CAS:Formula:C22H32O3Purezza:>98.0%(HPLC)Colore e forma:White to Almost white powder to crystalPeso molecolare:344.504,5,6,7-Tetrabromobenzotriazole
CAS:Formula:C6HBr4N3Purezza:>97.0%(T)(HPLC)Colore e forma:White to Light yellow powder to crystalPeso molecolare:434.71Serotonin Creatinine Sulfate Monohydrate
CAS:Formula:C14H19N5O2·H2SO4·H2OPurezza:>98.0%(T)Colore e forma:White to Light yellow powder to crystalPeso molecolare:405.43(-)-Deguelin
CAS:Formula:C23H22O6Purezza:>95.0%(HPLC)Colore e forma:White to Yellow to Green powder to crystalPeso molecolare:394.42Lubiprostone
CAS:Formula:C20H32F2O5Purezza:>97.0%(HPLC)Colore e forma:White to Light yellow powder to crystalPeso molecolare:390.47Prostaglandin F2α
CAS:Formula:C20H34O5Purezza:>95.0%(T)Colore e forma:White or Colorless to Almost white or Almost colorless powder to lump to clear liquidPeso molecolare:354.49Tomatine from Tomato
CAS:Formula:C50H83NO21Purezza:>80.0%(HPLC)Colore e forma:White to Yellow to Orange powder to crystalPeso molecolare:1,034.20Tetrasodium 1,2-Bis(2-aminophenoxy)ethane-N,N,N',N'-tetraacetate
CAS:Formula:C22H20N2Na4O10Purezza:>98.0%(T)Colore e forma:White to Almost white powder to crystalPeso molecolare:564.37Homotaurine-d6
CAS:Homotaurine-d6 is a deuterated compound of Homotaurine. Homotaurine has a CAS number of 3687-18-1. Because of its similarity in structure to the neurotransmitter gamma-aminobutyric acid (GABA), it has GABAergic effects and may be useful as an anticonvulsant. Homotaurine has also been investigated as a potential treatment for Alzheimer's disease. It binds to soluble amyloid beta and inhibits the formation of neurotoxic aggregates that lead to amyloid plaque deposition in the brain. However, clinical trials failed to show improvement compared to placebo.Formula:C3D6H3NO3SColore e forma:SolidPeso molecolare:145.21Amitriptyline-d6 Hydrochloride
CAS:Amitriptyline-d6 Hydrochloride is a deuterated compound of Amitriptyline Hydrochloride. Amitriptyline Hydrochloride has a CAS number of 549-18-8. Amitriptyline Hydrochloride is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptive activities.Formula:C20H18D6ClNColore e forma:SolidPeso molecolare:319.90Brexpiprazole-d8
CAS:Brexpiprazole D8 is a deuterium-modified partial agonist of 5-HT1A and dopamine receptors, with Ki values of 0.12 nM and 0.3 nM respectively.Formula:C25H27N3O2SPurezza:98%Colore e forma:SolidPeso molecolare:441.62Milnacipran-d10 Hydrochloride
CAS:Milnacipran-d10 Hydrochloride is a deuterated compound of Milnacipran Hydrochloride. Milnacipran Hydrochloride has a CAS number of 101152-94-7. Levomilnacipran is a serotonin and norepinephrine reuptake inhibitor used to treat major depressive disorders. Levomilnacipran is an enantiomer of milnacipran, which is used to treat fibromyalgia. Levomilnacipran and milnacipran have been associated with a low rate of transient elevations in serum aminotransferase levels during treatment and with rare instances of clinically apparent acute liver injury with jaundice.Formula:C15H13D10ClN2OColore e forma:SolidPeso molecolare:292.87Mirtazapine D3
CAS:Mirtazapine D3 is a deuterium labeled Mirtazapine. Mirtazapine is an inhibitor of 5-HT receptor .Formula:C17H19N3Purezza:98%Colore e forma:SolidPeso molecolare:268.37N-Biotinyl p-aminophenyl arsenic acid
CAS:N-Biotinyl p-aminophenyl arsenic acid is a bifunctional reagent that binds to streptavidin and disulfide compounds. It diminishes the binding sites of rbungarotoxin on reduced nicotinic receptors with an IC50 ranging from 10-300 nM, thus shielding the receptors from irreversible alkylation by bromoacetylcholine.Formula:C16H22AsN3O4SColore e forma:SolidPeso molecolare:427.35Catestatin
CAS:Non-competitive inhibitor of nicotinic receptors; blocks cationic signalling and catecholamine release; stimulates histamine release. IC50 ~200-250nM.Formula:C107H173N37O26SPurezza:98%Colore e forma:SolidPeso molecolare:2425.84Hydroxy ziprasidone
CAS:Hydroxy ziprasidone is an impurity of Ziprasidone. Ziprasidone, an antipsychotic agent, is a 5-HT and dopamine receptor antagonist.Formula:C21H21ClN4O2SPurezza:98%Colore e forma:SolidPeso molecolare:428.94Penbutolol sulfate
CAS:Penbutolol sulfate ((-)-Terbuclomine) is able to bind to both β2-adrenergic receptor and β1-adrenergic receptor, thus making it a non-selective β blocker.Formula:C18H29NO2H2O4SPurezza:99.95%Colore e forma:SolidPeso molecolare:340.47Phenglutarimide hydrochloride
CAS:Phenglutarimide hydrochloride is an anticholinergic. It is used as an antiparkinsonian agent.Formula:C17H25ClN2O2Colore e forma:SolidPeso molecolare:324.857-Acetoxy-1-methylquinolinium iodide
CAS:7-Acetoxy-1-methylquinolinium iodide (AMQI) is a cholinesterase substrate for inhibitor detection with 320 nm Ex and 410 nm Em.Formula:C12H12INO2Colore e forma:SolidPeso molecolare:329.13Ketanserinol
CAS:Ketanserinol is a metabolite of the antihypertensive drug ketanserin, which blocks 5-HT2 receptors to treat protamine-induced pulmonary hypertension.Formula:C22H24FN3O3Colore e forma:SolidPeso molecolare:397.44Aprofene
CAS:Aprofene blocks acetylcholine receptors, used for peptic ulcers, endarteritis, cholecystitis, and colitis.Formula:C21H27NO2Colore e forma:SolidPeso molecolare:325.44Aftin-5
CAS:Aftin-5 is an inducer of amyloid beta protein 42 (Aβ42). It functions by modifying the ultrastructure of mitochondria, leading to an upregulation of Aβ42 and a downregulation of Aβ38 through a β-secretase and γ-secretase-dependent mechanism. Aftin-5 exhibits mild cytotoxicity in SH-SY5Y, HT22, N2a, and N2a-AβPP695 cells, with IC50 values of 180, 194, 178, and 150 μM, respectively.Formula:C19H26N6OColore e forma:SolidPeso molecolare:354.45VU0477886
CAS:VU0477886: Potent mGlu4 PAM, effective in preclinical Parkinson's model HIC.Formula:C20H13ClN4O3Purezza:98%Colore e forma:SolidPeso molecolare:392.80AN317
CAS:AN317 is a selective agonist for the nicotinic acetylcholine receptor (nAChR) containing α6β2, with dissociation constants (Ki) of 6.2 nM and 4.1 nM for the α6/α3β2β3 and α4β2 receptor subtypes, respectively. It induces dopamine release in rat striatal synaptosomes, enhances the activity of dopaminergic neurons in the substantia nigra, and exhibits protective effects against the dopaminergic neurotoxin MPP+ in rat neurons. AN317 also demonstrates favorable pharmacokinetic properties in rats and permeability across the blood-brain barrier (BB).Formula:C13H19N3Colore e forma:SolidPeso molecolare:217.31MCI-225 dehydratase
CAS:MCI-225 dehydratase is an oral, selective inhibitor of noradrenaline reuptake, and functions as a 5-HT3 antagonist, exhibiting antidepressant effects in vivo .Formula:C17H18ClFN4SColore e forma:SolidPeso molecolare:364.87Nicardipine pyridine metabolite II
CAS:Nicardipine pyridine metabolite II is a biaoctive chemical.Formula:C26H27N3O6Colore e forma:SolidPeso molecolare:477.51Biperiden lactate
CAS:Biperiden lactate is a biochemical.Formula:C24H35NO4Colore e forma:SolidPeso molecolare:401.54Aβ1-42 aggregation inhibitor 1
CAS:Aβ1-42 aggregation inhibitor 1 effectively inhibits acetylcholinesterase (AChE) and butyrylcholinesterase (BuChE), demonstrating IC50 values of 2.64 μM and 1.29Formula:C29H32N4SColore e forma:SolidPeso molecolare:468.66SB 271046 hydrochloride
CAS:SB 271046 hydrochloride (SB 271046A) is selective, orally active 5-HT6 antagonist and is > 200-fold selective over 55 other receptors, enzymes and ion channels.Formula:C20H22ClN3O3S2·HClPurezza:99.77%Colore e forma:SolidPeso molecolare:488.45Diclofensine
CAS:Diclofensine (Ro 8-4650) inhibits the uptake of serotonin, noradrenaline and dopamine.Formula:C17H17Cl2NOPurezza:97.01% - 98.13%Colore e forma:SolidPeso molecolare:322.236-hydroxy Buspirone
CAS:6-Hydroxy Buspirone, an active metabolite of the anxiolytic compound buspirone, is produced via the cytochrome P450 (CYP) isoform CYP3A4.Formula:C21H31N5O3Colore e forma:SolidPeso molecolare:401.50Dianicline dihydrochloride
CAS:Dianicline dihydrochloride is a partial agonist of α4β2 nicotinic acetylcholine receptor. It increases cessation rates in a dose-dependent manner.Formula:C13H16N2OPurezza:98%Colore e forma:SolidPeso molecolare:216.285-Methyltryptamine hydrochloride
CAS:5-Methyltryptamine hydrochloride is a high-affinity 5-HT1C receptor ligand and a partial agonist of 5-HT. 5-Methyltryptamine hydrochloride protects mice subjected to burn, tourniquet and endotoxin shock.Formula:C11H15ClN2Purezza:99.45%Colore e forma:SolidPeso molecolare:210.703Eprodisate
CAS:Eprodisate disrupts protein-glycosaminoglycan binding, halting amyloid fibril formation, potentially delaying AA amyloidosis progression.Formula:C3H8O6S2Colore e forma:SolidPeso molecolare:204.22VU0029767
CAS:VU0029767 is an allosteric enhancer of the M1 muscarinic receptor, capable of modulating the receptor's activity. This compound enhances M1 receptor activity by increasing agonist affinity. However, VU0029767 demonstrates distinct characteristics from other compounds, particularly under varying experimental conditions such as its interaction with mutated M1 receptors and its effects on downstream signaling pathways.
Formula:C21H21N3O3Colore e forma:SolidPeso molecolare:363.417-Desmethyl-3-hydroxyagomelatine
CAS:7-Desmethyl-3-hydroxyagomelatine, less active than parent drug Agomelatine, is a melatonergic agonist and 5-HT2C antagonist.Formula:C14H15NO3Purezza:98%Colore e forma:SolidPeso molecolare:245.27Pardoprunox
CAS:Pardoprunox (SLV-308) is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties.Formula:C12H15N3O2Purezza:98%Colore e forma:SolidPeso molecolare:233.274-(6-Bromo-2-benzothiazolyl)-N-methylbenzenamine
CAS:4-(6-Bromo-2-benzothiazolyl)-N-methylbenzenamine is a potent amyloid imaging agent that binds to Amyloid-β (1-40) (KD: 1.7 nM).Formula:C14H11BrN2SPurezza:98%Colore e forma:SolidPeso molecolare:319.22(4-Hydroxy-3-methoxyphenyl)acetic-2,2-d2 Acid
CAS:Prodotto controllatoApplications (4-Hydroxy-3-methoxyphenyl)acetic-2,2-d2 Acid (CAS# 53587-33-0) is a useful isotopically labeled research compound.
Formula:C9H8D2O4Colore e forma:NeatPeso molecolare:184.192-(4-Chlorophenyl)-2-(methylamino)cyclohexanone Hydrochloride
CAS:Prodotto controllatoFormula:C13H17Cl2NOColore e forma:NeatPeso molecolare:274.196S-Nalfurafine
CAS:Prodotto controllatoApplications 6S-Nalfurafine is a stereoisomer of Nalfurafine (N255600), a on-narcotic opioid drug for intractable itch caused by hemodialysis. It showed significant opioid κ-agonist activity and induced neither aversion nor preference in rats on the CPP (Conditioned Place Preference) test. Nalfurafine is a new therapeutic agent for the treatment of uremic pruritus in hemodialysis patients.
References Fujii, H., et al.: Bioorg. Med. Chem., 12, 4133 (2004); Mori, T., et al.: Life Sci., 75, 2433 (2004); Fujii, H., et al.: Curr. Med. Chem., 13, 1109 (2006); Nagase, H., et al.: Bioorg. Med. Chem. Lett., 20, 6302 (2010)Formula:C28H32N2O5Colore e forma:NeatPeso molecolare:476.562-(3-Chlorophenyl)-2-(methylamino)cyclohexanone Hydrochloride
CAS:Prodotto controllatoFormula:C13H17Cl2NOColore e forma:NeatPeso molecolare:274.192Z-Nalfurafine
CAS:Prodotto controllatoApplications 2Z-Nalfurafine is a geometric isomer of Nalfurafine (N255600), a on-narcotic opioid drug for intractable itch caused by hemodialysis. It showed significant opioid κ-agonist activity and induced neither aversion nor preference in rats on the CPP (Conditioned Place Preference) test. Nalfurafine is a new therapeutic agent for the treatment of uremic pruritus in hemodialysis patients.
References Fujii, H., et al.: Bioorg. Med. Chem., 12, 4133 (2004); Mori, T., et al.: Life Sci., 75, 2433 (2004); Fujii, H., et al.: Curr. Med. Chem., 13, 1109 (2006); Nagase, H., et al.: Bioorg. Med. Chem. Lett., 20, 6302 (2010)Formula:C28H32N2O5Colore e forma:NeatPeso molecolare:476.56Dolasetron Mesylate
CAS:Dolasetron Mesylate (MDL-73147EF) is an antagonist of the 5-HT3 receptor and can be used in research on the treatment of vomiting and nausea followingFormula:C20H24N2O6SPurezza:99.05%Colore e forma:White PowderPeso molecolare:420.48LY 344864
CAS:LY 344864, a specifc receptor agonist, is an affinity of 6 nM (Ki) at the recently cloned 5-HT1F receptor.Formula:C21H22FN3OPurezza:98%Colore e forma:SolidPeso molecolare:351.42Paroxetine hydrochloride hemihydrate
CAS:Paroxetine hydrochloride hemihydrate (Paxil) is an effective and selective serotonin reuptake inhibitor (SSRI).Formula:C38H44Cl2F2N2O7Purezza:99.949%Colore e forma:SolidPeso molecolare:749.67GTS-21
CAS:GTS-21 (DMXB-A) is an α7 nAChR agonist. GTS-21 suppresses inflammation associated with rheumatoid arthritis by inhibiting RA Th1 cell differentiation.Formula:C19H20N2O2Purezza:98%Colore e forma:SolidPeso molecolare:308.375-HT2A receptor agonist-2
CAS:Potent 5-HT2A receptor agonist-2 targets 5-HT2A/B/C with EC50 1.7, 0.58, 0.50 nM.Formula:C20H21ClN2O3Colore e forma:SolidPeso molecolare:372.85Nelonicline citrate
CAS:Nelonicline citrate (ABT-126) is a selective α7 nAChR agonist with a Ki of 12.3 nM, studied for schizophrenia and Alzheimer's.Formula:C23H27N3O8SColore e forma:SolidPeso molecolare:505.54AP-521 (Free base)
CAS:AP-521, a 5-HT1A receptor antagonist, is used potentially for the treatment of anxiety.Formula:C20H18N2O3SColore e forma:SolidPeso molecolare:366.43Territrem B
CAS:Territrem B: A mycotoxin that irreversibly blocks AChE, causes tremors in mice at 0.21 mg/kg.Formula:C29H34O9Colore e forma:SolidPeso molecolare:526.57AChE-IN-20
CAS:AChE-IN-20: AChE inhibitor (IC50: 397.32 nM), hCA-I/II blocker (IC50: ~77 nM avg), α GLY suppressor (IC50: 52.08 nM).Formula:C22H20N8O6S2Colore e forma:SolidPeso molecolare:556.57AChE/BChE/MAO-B-IN-3
AChE/BChE/MAO-B-IN-3: potent MAO-B, AChE & BChE inhibitor; IC50: 0.0359μM (MAO-B), 0.0473/0.0782μM (AChE/BChE); possible Alzheimer's research use.Formula:C25H31N3O3Colore e forma:SolidPeso molecolare:421.53Ambutonium bromide
CAS:Ambutonium bromide is an antagonist of acetylcholine.Formula:C20H27BrN2OPurezza:98%Colore e forma:SolidPeso molecolare:391.35MAO-B-IN-15
CAS:MAO-B-IN-15 selectively inhibits MAO-B, targeting Tyr 326 (IC50 = 13.5 μM), useful for Parkinson's research.Formula:C17H18FNO2Colore e forma:SolidPeso molecolare:287.33SV5
CAS:SV5: potent anti-Alzheimer's, protects SHSY-5Y from Aβ1-42 death, stable with optimal pharmacology in plasma, antioxidant, neuroprotective.Formula:C21H30N2O4S2Colore e forma:SolidPeso molecolare:438.6Bopindolol (malonate)
CAS:Bopindolol is a non-selective β-adrenergic receptor antagonist.Formula:C26H32N2O7Colore e forma:SolidPeso molecolare:484.549CJ 033466
CAS:CJ 033466 is a selective partial agonist of 5-HT4 receptor (EC50 = 9 nM) with gastroprokinetic effect.Formula:C19H28ClN5OPurezza:99.72%Colore e forma:SolidPeso molecolare:377.91SB 207710
CAS:SB 207710 is a selective and high affinity antagonist of 5-HT4 receptor.Formula:C19H27IN2O4Colore e forma:SolidPeso molecolare:474.33Bornaprine
CAS:Bornaprine is an anticholinergic drug used to treat Parkinson's disease due to inhibition of muscarinic or nicotinic transmission.Formula:C21H31NO2Colore e forma:SolidPeso molecolare:329.48Naronapride
CAS:Naronapride (ATI-7505) is a potent agonist of the prokinetic 5-HT4receptor and can be used to study gastrointestinal disorders.Formula:C27H41ClN4O5Colore e forma:SolidPeso molecolare:537.09LOX-IN-3
CAS:LOX-IN-3, an orally active inhibitor of lysyl oxidase (LOX), holds potential application in the fields of fibrosis, cancer, and angiogenesis research[1].Formula:C13H13FN2O2SColore e forma:SolidPeso molecolare:280.32SSAO inhibitor-3
CAS:SSAO inhibitor-3 targets human AOC1/SSAO in atherosclerosis, diabetes, obesity, CKD, and more, with IC50s of 0.1-10 μM/<10 nM.Formula:C15H23FN4O3Colore e forma:SolidPeso molecolare:326.37TG41
CAS:TG41 is a GABAA receptors positive modulator.Formula:C18H13BrCl2N2O2Purezza:98%Colore e forma:SolidPeso molecolare:440.12Protriptyline
CAS:Protriptyline: Antidepressant, AChE inhibitor (IC50 0.06 mM), prevents Aβ aggregation; potential for depression and Alzheimer's.Formula:C19H21NColore e forma:SolidPeso molecolare:263.38CP-809101
CAS:CP-809101 is an effective and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).Formula:C15H17ClN4OPurezza:98%Colore e forma:SolidPeso molecolare:304.77Bradanicline
CAS:Bradanicline: potent α7 nAChR agonist, EC50=17 nM, Ki=1.4 nM, used in cognitive disorder research.Formula:C22H23N3O2Colore e forma:SolidPeso molecolare:361.44(-)-Donepezil
CAS:(-)-Donepezil is an isomer of Donepezil -- a nootropic acting as an inhibitor of acetylcholinesterase.Formula:C24H29NO3Colore e forma:SolidPeso molecolare:379.49CP-457920
CAS:CP-457920 is a selective α5 GABAA receptor inverse agonist that is suitable for investigating dementia in Alzheimer's disease.Formula:C18H17N3O3Purezza:99.06% - 99.74%Colore e forma:SolidPeso molecolare:323.35Caroxazone
CAS:Caroxazone is an antidepressant drug, monoamine oxidase inhibitor (MAOI) that is irreversible and nonselective meanwhile.Formula:C10H10N2O3Colore e forma:SolidPeso molecolare:206.2(R)-Oxybutynin
CAS:(R)-Oxybutynin: oral muscarinic blocker with antispasmodic effects, used in neurogenic bladder research.Formula:C22H31NO3Colore e forma:SolidPeso molecolare:357.49AChE/BChE-IN-3
CAS:AChE/BChE-IN-3 (BMC-1) dual inhibitor: IC50 of 6.08 μM for elAChE, 0.383 μM for eqBChE.Formula:C15H24N2O3Colore e forma:SolidPeso molecolare:280.36BuChE-IN-6
CAS:BuChE-IN-6 inhibits BuChE (IC50: 0.46 μM eqBuChE, 0.51 μM hBuChE) and prevents Aβ 42 self-aggregation.Formula:C21H26N4O2Colore e forma:SolidPeso molecolare:366.46FR-188582
CAS:FR-188582 is a highly selective cyclooxygenase (COX)-2 inhibitor (IC50: 17 nM).Formula:C16H13ClN2O2SPurezza:98%Colore e forma:SolidPeso molecolare:332.8hMAO-B-IN-6
CAS:Compound 17d (hMAO-B-IN-6) is an effective and selective hMAO-B inhibitor, demonstrating an IC 50 of 67.02 nM. It significantly ameliorates cognitive deficits induced by Scopolamine in Alzheimer's disease (AD) mice [1].Formula:C19H20N2O5Colore e forma:SolidPeso molecolare:356.37Tarafenacin D-tartrate
CAS:Tarafenacin D-tartrate is a highly selective M3 muscarinic receptor antagonist (Ki= 0.19 nM), ~200 fold selectivity over the M2 receptor.Formula:C25H26F4N2O8Purezza:99.86%Colore e forma:SolidPeso molecolare:558.48Pridefine
CAS:Pridefine: antidepressant, balances serotonin, dopamine, norepinephrine reuptake, weakly releases them.Formula:C19H21NPurezza:99.15% - 99.66%Colore e forma:SolidPeso molecolare:263.38S 24795
CAS:S 24795 (Catestatin acetate(142211-96-9 free base)) is an α7 nAChR partial agonist.Formula:C14H13BrINOPurezza:99.934%Colore e forma:SolidPeso molecolare:418.07Ref: TM-T23286
5mg44,00€1mL*10mM (DMSO)48,00€10mg66,00€25mg138,00€50mg215,00€100mg338,00€200mg480,00€CP94253 hydrochloride
CAS:CP94253 hydrochloride: selective 5-HT1B agonist, Ki=2 nM; less active on 5-HT1A/D/C/2 (Ki=89/49/860/1600 nM).Formula:C15H20ClN3OPurezza:99.78%Colore e forma:SolidPeso molecolare:293.79Ref: TM-T22689
5mg66,00€1mL*10mM (DMSO)66,00€10mg90,00€25mg205,00€50mg334,00€100mg537,00€200mg745,00€MAO-B-IN-12
CAS:MAO-B-IN-12 (16c) is a potent MAO-B inhibitor with an IC50 of 1.3 μM and has neuroprotective properties.Formula:C22H30O4Colore e forma:SolidPeso molecolare:358.47W-13 hydrochloride
CAS:W-13 hydrochloride (W-13 HCl) is a calmodulin antagonist.Formula:C14H18Cl2N2O2SPurezza:98.51%Colore e forma:White PowderPeso molecolare:349.28Antioxidant agent-2
CAS:Antioxidant agent-2 (3c), BBB-permeable, selectively chelates metals; shows neuroprotection, fights liver damage in Alzheimer's research.Formula:C23H26N2O7Colore e forma:SolidPeso molecolare:442.46VU0455691
CAS:VU0455691 is a selective M1 Muscarinic Receptor Allosteric Modulators.Formula:C24H25N5O3SPurezza:98%Colore e forma:SolidPeso molecolare:463.55LY314228
CAS:LY314228 is an antagonist of 5-HT2A receptor.Formula:C20H24N4O3Colore e forma:SolidPeso molecolare:368.43Remeglurant
CAS:Remeglurant is used as a selective antagonist of the mGlu5 receptor.Formula:C17H15BrN4OColore e forma:SolidPeso molecolare:371.23(+)-Nipecotic acid
CAS:(+)-Nipecotic acid ((+)-β-Homoproline) is a specific inhibitor of GABA transport and uptake, capable of activating GABAA receptors.Formula:C6H11NO2Purezza:99.38%Colore e forma:SolidPeso molecolare:129.16PF-03463275 2HCl
CAS:PF-03463275 is an orally available, CNS-penetrant inhibitor of SLC6A9, a GlyT1 glycine transporter.Formula:C19H24Cl3FN4OPurezza:98%Colore e forma:SolidPeso molecolare:449.78Tilapertin
CAS:Tilapertin is an oral glycine transporter type-1 inhibitor.Formula:C20H21F3N2O2Purezza:98%Colore e forma:SolidPeso molecolare:378.39Lesopitron dihydrochloride
CAS:Lesopitron dihydrochloride with IC50 of 125 nM in rat hippocampal membranes, is a full and selective 5-HT1A receptor agonist.Formula:C15H23Cl3N6Purezza:98%Colore e forma:SolidPeso molecolare:393.74Dihydro Donepezil
CAS:Dihydro Donepezil (Dihydro E2020), a Donepezil metabolite, is a potent AChE inhibitor (IC50: hAChE 11.6 nM, bAChE 8.12 nM).Formula:C24H31NO3Colore e forma:SolidPeso molecolare:381.51SERT-IN-2
SERT-IN-2, a potent SERT inhibitor (IC 50 = 0.58 nM), exhibits promising efficacy as an anti-depressant.Colore e forma:SolidNAP-1
CAS:NAP-1 is an anesthetic that enhances CA1 brain inhibition in rats and causes tadpole sedation (EC50 = 0.53 μM).Formula:C20H18ClNO2Colore e forma:SolidPeso molecolare:339.82RU-505
CAS:RU-505 is an interaction inhibitor of Aβ-fibrinogen that acts by rescuing altered thrombosis and cognitive decline in Alzheimer's disease mice.Formula:C28H32FN5OPurezza:98%Colore e forma:SolidPeso molecolare:473.58FG-5893
CAS:FG-5893 is a 5-HT1A agonist and 5-HT2 antagonist with potential anxiolytic activity.Formula:C27H29F2N3O2Purezza:98%Colore e forma:SolidPeso molecolare:465.53S 14506 hydrochloride
CAS:S 14506 hydrochloride is a 5-HT1A receptor full agonist.Formula:C24H27ClFN3O2Purezza:99.92%Colore e forma:SolidPeso molecolare:443.94BACE2-IN-1
CAS:BACE2-IN-1, a potent BACE2 inhibitor characterized by its exceptional selectivity and a Ki value of 1.6 nM, is utilized in the investigation of Type 2 Diabetes.Formula:C36H38F3N3O3Colore e forma:SolidPeso molecolare:617.7LSP4-2022
CAS:LSP4-2022, a mGlu4 selective agonist, increases behavioral despair in mouse models of antidepressant action.Formula:C13H18NO8PPurezza:100%Colore e forma:SolidPeso molecolare:347.26Zatosetron maleate
CAS:Zatosetron maleate（LY 277359 maleate） is a potent and selective serotonin 5HT3 receptor antagonist for the study of acute migraine.Formula:C23H29ClN2O6Purezza:98.07%Colore e forma:SolidPeso molecolare:464.94(Rac)-VU 6008667
CAS:(Rac)-VU 6008667 is a selective M5 NAM with IC50 of 1.8 μM, high CNS penetration.Formula:C24H17ClF2N2O2Purezza:99.82%Colore e forma:SolidPeso molecolare:438.85AChE/BuChE-IN-2
CAS:Compound 5f, an oral AChE/BuChE inhibitor, crosses BBB; IC50: 0.72 μM (AChE), 0.16 μM (BuChE), 62.52 μM (Aβ aggregation).Formula:C20H18N2O2Colore e forma:SolidPeso molecolare:318.375-Carboxamidotryptamine maleate
CAS:5-Carboxamidotryptamine maleate (5-CT maleate) (5-CT maleate) is a receptor agonist with antihypertensive and glucose-raising effects.Formula:C15H17N3O5Purezza:99.88%Colore e forma:SolidPeso molecolare:319.31Trimedoxime bromide
CAS:Trimedoxime bromide is a cholinesterase reactivator used as an antidote in alkyl phosphate poisoning.Formula:C15H18Br2N4O2Colore e forma:SolidPeso molecolare:446.14Lidanserin
CAS:Lidanserin is an antagonist of the 5-HT2A and α1-adrenergic receptor.Formula:C26H31FN2O4Purezza:98%Colore e forma:SolidPeso molecolare:454.53(S)-SNAP5114
CAS:(S)-SNAP5114 is a selective inhibitor of GABA transport with IC50s of 5 μM for hGAT-3 and 21 μM for rGAT-2. (S)-SNAP5114 has anticonvulsant properties.Formula:C30H35NO6Purezza:98.20%Colore e forma:SolidPeso molecolare:505.6Ref: TM-T16831
5mg49,00€1mL*10mM (DMSO)49,00€10mg73,00€25mg152,00€50mg213,00€100mg309,00€200mg423,00€Camylofine
CAS:Camylofine (Avacan) is an antimuscarinic, used for relaxing smooth muscle.Formula:C19H32N2O2·2HClPurezza:98%Colore e forma:SolidPeso molecolare:393.4MAO-B-IN-16
CAS:MAO-B-IN-16 selectively inhibits MAO-B with IC50 of 1.55 μM, useful in studying central nervous disorders like Parkinson's.Formula:C18H19NO3Colore e forma:SolidPeso molecolare:297.35Hyoscyamine hydrobromide
CAS:Hyoscyamine hydrobromide is an agent of anticholinergic.Formula:C17H24BrNO3Purezza:98%Colore e forma:SolidPeso molecolare:370.28DAT 582
CAS:DAT 582 is a novel serotonin3 receptor antagonist. It is also an effective and long-lasting antiemetic agentFormula:C22H28ClN5OPurezza:98%Colore e forma:SolidPeso molecolare:413.95CB-6673567
CAS:CB-6673567 is a selective inhibitor of adenylyl cyclase.Formula:C19H14N4O3Colore e forma:SolidPeso molecolare:346.34trans-4-Hydroxycrotonic acid
CAS:trans-4-Hydroxycrotonic acid (T-HCA) is a selective and competitive ligand for the γ-hydroxybutyric acid (GHB) binding site.Formula:C4H6O3Purezza:99.19%Colore e forma:SolidPeso molecolare:102.09LY 81067
CAS:LY 81067, a new anticonvulsant, prevents PTZ- and picrotoxin-induced seizures in mice via picrotoxin site interaction.Formula:C22H24N4OColore e forma:SolidPeso molecolare:360.45RS 45041-190 hydrochloride
CAS:Highly selective I2 imidazoline receptor ligandFormula:C11H13Cl2N3Purezza:98%Colore e forma:SolidPeso molecolare:258.15NPS ALX Compound 4a dihydrochloride
CAS:NPS ALX Compound 4a dihydrochloride is a potent and selective antagonist of 5-HT6 receptor (IC50 of 7.2 nM)Formula:C25H27Cl2N3O2SPurezza:98%Colore e forma:SolidPeso molecolare:504.47Pridinol
CAS:Pridinol is an antispasmodic and muscle relaxant.Formula:C20H25NOPurezza:98%Colore e forma:Crystals SolidPeso molecolare:295.42Benactyzine
CAS:Benactyzine is a centrally acting muscarinic antagonist.Formula:C20H25NO3Purezza:98%Colore e forma:Crystals SolidPeso molecolare:327.42Aganodine
CAS:Aganodine, a guanidine, activates imidazoline receptors to inhibit norepinephrine release.Formula:C9H10Cl2N4Purezza:98%Colore e forma:SolidPeso molecolare:245.11DR-4004
CAS:DR-4004 is a selective serotonin 5-HT7 receptor antagonist.Formula:C26H30N2OColore e forma:SolidPeso molecolare:386.53MDL 73005EF hydrochloride
CAS:5-HT1A receptor antagonistFormula:C20H27ClN2O4Purezza:98%Colore e forma:SolidPeso molecolare:394.89JY-XHe-053
CAS:JY-XHe-053 is a selective modulator of GABAA receptors.Formula:C22H16FN3O2Purezza:98%Colore e forma:SolidPeso molecolare:373.38Fluoroclorgyline
CAS:Fluoroclorgyline is a specific inhibitor of monoamine oxidase A (MAO-A).Formula:C13H15ClFNOPurezza:98%Colore e forma:SolidPeso molecolare:255.72UMB68 sodium
CAS:UMB-68 is a GHB receptor ligand with no affinity (IC(50) >100 microM) at GABA(A) or GABA(B) receptors.Formula:C6H12NaO3Colore e forma:SolidPeso molecolare:155.149(S)-Baclofen
CAS:(S)-Baclofen may treat hyperacusis and tinnitus by reducing auditory pathway excitation.Formula:C10H12ClNO2Purezza:98%Colore e forma:SolidPeso molecolare:213.66L 646462
CAS:L 646462 is an antidopaminergic agent.Formula:C27H27N3O4Purezza:98%Colore e forma:SolidPeso molecolare:457.52SB 258585 hydrochloride
CAS:SB 258585 hydrochloride is a 5-HT6 receptor antagonist.Formula:C18H23ClIN3O3SPurezza:98%Colore e forma:SolidPeso molecolare:523.82HIE-124
CAS:HIE-124 is a central cervous system active anticonvulsant and ultra-short acting hypnotic.Formula:C10H12N2O3SPurezza:98%Colore e forma:SolidPeso molecolare:240.28(S)-HexylHIBO
CAS:Group I mGlu receptor antagonistFormula:C12H20N2O4Purezza:98%Colore e forma:SolidPeso molecolare:256.3CUMI-101
CAS:CUMI-101 is an agonist of 5-HT1A receptor.Formula:C19H27N5O3Colore e forma:SolidPeso molecolare:373.45Anisopirol
CAS:Anisopirol is an antipsychotic drug. Studies have shown that it can target dopamine receptors (DA), N-methyl-d-aspartate receptors (NMDA).Formula:C21H27FN2O2Colore e forma:SolidPeso molecolare:358.45RP5063 Hydrochloride
CAS:RP5063 Hydrochloride is a modulator of multimodal serotonin receptors.Formula:C22H26Cl3N3O3Purezza:98%Colore e forma:SolidPeso molecolare:486.82Pentolinium Tartrate
CAS:Pentolinium Tartrate (Pendine) is a nicotinic antagonist that has been used as a ganglionic blocking agent in hypertension.Formula:C15H32N2·2C4H5O6Purezza:98%Colore e forma:SolidPeso molecolare:538.6E55888
CAS:E55888 is a potent and selective full agonist of the 5HT7 serotonin receptor.Formula:C16H23N3Colore e forma:SolidPeso molecolare:257.37Etoperidone hydrochloride
CAS:Etoperidone hydrochloride is an antidepressant agent.Formula:C19H29Cl2N5OColore e forma:SolidPeso molecolare:414.37DAA-1097
CAS:DAA-1097 is a novel ligand of peripheral benzodiazepine receptor.Formula:C24H24ClNO3Purezza:98%Colore e forma:SolidPeso molecolare:409.91BACE1/2-IN-1
CAS:BACE1/2-IN-1 inhibits BACE1/2 with IC50s of 0.01μM/0.0053μM, has better permeability and lower Pgp efflux but reduced metabolic stability.Formula:C21H31N5OSColore e forma:SolidPeso molecolare:401.57(RS)-4-Carboxyphenylglycine
CAS:(RS)-4-Carboxyphenylglycine is a racemic mixture. (S)-4-Carboxyphenylglycine is a selective mGlu1α receptor antagonist.Formula:C9H9NO4Purezza:97.22% - >99.99%Colore e forma:SolidPeso molecolare:195.17LEK 8841
CAS:LEK 8841 is an ergoline derivative that is a potential antipsychotic.Formula:C21H24BrN3O4SPurezza:98%Colore e forma:SolidPeso molecolare:494.4TMPH hydrochloride
CAS:neuronal nicotinic ACh receptors (nAChRs) antagonistFormula:C16H32ClNO2Purezza:98%Colore e forma:SolidPeso molecolare:305.88Lofepramine hydrochloride
CAS:Lofepramine is a serotonin and norepinephrine reuptake inhibitor. Lofepramine is also a psychotropic IMIPRAMINE derivative.Formula:C26H28Cl2N2OPurezza:98%Colore e forma:Off-White SolidPeso molecolare:455.42GW-876167
CAS:GW-876167, a 5-HT2C agonist, is used potentially for the treatment of obesity and glaucoma.Formula:C16H21N5O2Purezza:98%Colore e forma:SolidPeso molecolare:315.37WAY 163909
CAS:WAY 163909 is an effective and selective agonist of the 5-HT(2C) receptor (Ki: 10.5±1.1 nM).Formula:C14H18N2Purezza:98%Colore e forma:SolidPeso molecolare:214.31Hexafluronium Bromide
CAS:Hexafluronium bromide enhances muscle relaxation in surgery by blocking acetylcholine receptors.Formula:C36H42BrN2Colore e forma:SolidPeso molecolare:582.649Mimopezil
CAS:Mimopezil is an acetylcholinesterase (AChE) inhibitor.Formula:C23H23ClN2O3Purezza:98%Colore e forma:SolidPeso molecolare:410.89Tebanicline tosylate
CAS:Tebanicline: synthetic, potent, non-opioid analgesic, less toxic than epibatidine; relieves neuropathic pain, acts on α3β4 and α4β2 nicotinic receptors.Formula:C16H19ClN2O4SPurezza:98%Colore e forma:SolidPeso molecolare:370.85SCH 50911 hydrochloride
CAS:SCH 50911 hydrochloride is a selective, orally-active and competitive antagonist of γ-Aminobutyric acid B GABA(B) receptor(IC50 : 1.1 μM).Formula:C8H16ClNO3Purezza:98%Colore e forma:SolidPeso molecolare:209.67Captodiame
CAS:Captodiame is an antihistamine agent.Formula:C21H29NS2Purezza:98%Colore e forma:SolidPeso molecolare:359.59Rivanicline oxalate
CAS:Rivanicline oxalate is an agonist of neuronal nicotinic receptor, showing high selectivity for the α4β2 subtype (Ki=26 nM).Formula:C12H16N2O4Purezza:98%Colore e forma:SolidPeso molecolare:252.27AVN-322
CAS:AVN-322 is a 5-HT6 receptor antagonist. 5-HT6R antagonists improves cognition in animal models of cognitive impairment.Formula:C17H20ClN5O2SPurezza:>99.99%Colore e forma:SolidPeso molecolare:393.89ENS-163 phosphate
CAS:Ens-163 phosphate is a muscarinic M1 receptor agonist. It is selective.Formula:C11H19N2O5PSPurezza:98%Colore e forma:SolidPeso molecolare:322.32Fonazine
CAS:Forazine (dimethiazide) is a phenothiazine drug used in the treatment of migraine and is a serotonin antagonist and a histamine antagonist.Formula:C19H25N3O2S2Colore e forma:SolidPeso molecolare:391.55MMPIP
CAS:allosteric mGlu7-selective receptor antagonistFormula:C19H15N3O3Purezza:98%Colore e forma:SolidPeso molecolare:333.34Ipsapirone
CAS:Ipsapirone is a partial agonist of 5-HT1A receptor and produces an inhibitory effect on 5-HT2 and the α1-adrenergic function at high doses.
Formula:C19H23N5O3SPurezza:99.51%Colore e forma:SolidPeso molecolare:401.48QF0301B
CAS:QF0301B is a potent α1-adrenergic receptor antagonist with inhibitory effects on α2-adrenergic receptors, 5-HT2A and histamine H1 receptors.Formula:C23H28N2O2Purezza:>99.99%Colore e forma:SolidPeso molecolare:364.48
