
Neuroscienza
Gli inibitori in neuroscienze sono composti progettati per modulare l'attività di proteine, enzimi o recettori specifici all'interno del sistema nervoso. Questi inibitori sono cruciali per studiare i meccanismi molecolari alla base della funzione neuronale, della trasmissione sinaptica e delle malattie neurodegenerative. Mirando ai recettori dei neurotrasmettitori, ai canali ionici e alle vie di segnalazione, gli inibitori in neuroscienze aiutano a esplorare la funzione cerebrale e a sviluppare strategie terapeutiche per disturbi neurologici come l'Alzheimer, il Parkinson e l'epilessia. Presso CymitQuimica, offriamo una vasta gamma di inibitori in neuroscienze di alta qualità per supportare la tua ricerca in neurobiologia, neurofarmacologia e scienze cognitive.
Sottocategorie di "Neuroscienza"
- recettore 5-HT(1.025 prodotti)
- ACK(1 prodotti)
- AChR(646 prodotti)
- Citrato liasi ATP(17 prodotti)
- Recettore adrenergico(3.022 prodotti)
- BACE(37 prodotti)
- Beta amiloide(228 prodotti)
- CaMK(73 prodotti)
- COX(600 prodotti)
- Recettore della dopamina(445 prodotti)
- Ricettore GABA(373 prodotti)
- Gamma-secretasi(61 prodotti)
- GluR(265 prodotti)
- GlyT(26 prodotti)
- Recettore dell'istamina(385 prodotti)
- LRRK2(43 prodotti)
- Recettore della melatonina(26 prodotti)
- NMDAR(10 prodotti)
- Recettore OX(41 prodotti)
- Recettore degli oppioidi(327 prodotti)
Mostrare 12 più sottocategorie
Trovati 5584 prodotti di "Neuroscienza"
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Org-12962
CAS:Org-12962: 5-HT2C agonist (pEC50: 7.01), anti-panic in rats, affects 5-HT2A/B (pEC50: 6.38/6.28).Formula:C10H11ClF3N3Purezza:98.34%Colore e forma:SolidPeso molecolare:265.66(R)-Baclofen hydrochloride
CAS:Arbaclofen HCl, a GABA-B agonist, treats spasticity from spinal injury by reducing excitatory transmission.Formula:C10H13Cl2NO2Purezza:98%Colore e forma:SolidPeso molecolare:250.12MSOP
CAS:MSOP is a selective antagonist of group III metabotropic glutamate receptor (KD of 51 μM for the L-AP4-sensitive presynaptic mGluR).Formula:C4H10NO6PPurezza:98%Colore e forma:SolidPeso molecolare:199.1Repinotan HCl
CAS:Repinotan HCl (Bay-x-3702) is a 5-HT1A receptor agonist with potent neuroprotective effects for the study of ischemic stroke and traumatic brain injury.
Formula:C21H25ClN2O4SPurezza:99.57%Colore e forma:SolidPeso molecolare:436.95EMDT
CAS:EMDT oxalate is a selective 5-HT6 agonist, and has antidepressant effects.Formula:C15H22N2OPurezza:97.66% - 99.78%Colore e forma:SolidPeso molecolare:246.35Ref: TM-T11183
1mg87,00€2mg118,00€1mL*10mM (DMSO)166,00€5mg167,00€10mg202,00€25mg449,00€50mg652,00€100mg888,00€500mg1.783,00€Methoxy-PEPy
CAS:Methoxy-PEPy is a potent and selective mGlu5 receptor inhibitor with an IC50 value of 1 nM.Formula:C13H10N2OPurezza:98.66%Colore e forma:SolidPeso molecolare:210.23Bifenazate
CAS:Bifenazate is a positive allosteric modulator of GABA receptor. Bifenazate is an acaricide that controls 100% of mites at a concentration of 25 ppm.Formula:C17H20N2O3Purezza:99.62%Colore e forma:Solid CrystallinePeso molecolare:300.35Eplivanserin
CAS:Eplivanserin (SR-46349) is an effective and selective antagonist of 5-HT2A receptor with a Kd of 1.14 nM and an IC50 value of 5.8 nM in rat cortical membrane.Formula:C19H21FN2O2Purezza:97.04%Colore e forma:SolidPeso molecolare:328.38Pridefine
CAS:Pridefine: antidepressant, balances serotonin, dopamine, norepinephrine reuptake, weakly releases them.Formula:C19H21NPurezza:99.15% - 99.66%Colore e forma:SolidPeso molecolare:263.38CJ 033466
CAS:CJ 033466 is a selective partial agonist of 5-HT4 receptor (EC50 = 9 nM) with gastroprokinetic effect.Formula:C19H28ClN5OPurezza:99.72%Colore e forma:SolidPeso molecolare:377.91E-3620
CAS:E-3620 is a potent antagonist of the 5-HT3 receptor and can be used to study dyskinesia and gastrointestinal dysfunction.Formula:C20H27Cl2N3O2Purezza:98.88% - 98.88%Colore e forma:SolidPeso molecolare:412.35TG41
CAS:TG41 is a GABAA receptors positive modulator.Formula:C18H13BrCl2N2O2Purezza:98%Colore e forma:SolidPeso molecolare:440.12CP-457920
CAS:CP-457920 is a selective α5 GABAA receptor inverse agonist that is suitable for investigating dementia in Alzheimer's disease.Formula:C18H17N3O3Purezza:99.06% - 99.74%Colore e forma:SolidPeso molecolare:323.35FR-188582
CAS:FR-188582 is a highly selective cyclooxygenase (COX)-2 inhibitor (IC50: 17 nM).Formula:C16H13ClN2O2SPurezza:98%Colore e forma:SolidPeso molecolare:332.8AVN-322
CAS:AVN-322 is a 5-HT6 receptor antagonist. 5-HT6R antagonists improves cognition in animal models of cognitive impairment.Formula:C17H20ClN5O2SPurezza:>99.99%Colore e forma:SolidPeso molecolare:393.89Pentolinium Tartrate
CAS:Pentolinium Tartrate (Pendine) is a nicotinic antagonist that has been used as a ganglionic blocking agent in hypertension.Formula:C15H32N2·2C4H5O6Purezza:98%Colore e forma:SolidPeso molecolare:538.6SCH 50911 hydrochloride
CAS:SCH 50911 hydrochloride is a selective, orally-active and competitive antagonist of γ-Aminobutyric acid B GABA(B) receptor(IC50 : 1.1 μM).Formula:C8H16ClNO3Purezza:98%Colore e forma:SolidPeso molecolare:209.67VU 0469650
CAS:VU 0469650 is a potent and selective negative allosteric modulator of mGluR1 (IC50 = 99 nM).Formula:C22H28N4OPurezza:98.03%Colore e forma:SolidPeso molecolare:364.48Ref: TM-T29118
1mg42,00€5mg79,00€1mL*10mM (DMSO)90,00€10mg108,00€25mg210,00€50mg313,00€100mg464,00€200mg640,00€Pancopride
CAS:Pancopride(LAS 30451) is a novel, orally available, long-acting, selective 5-HT3 receptor antagonist that blocks nitrogen mustard and dacarbazine-inducedFormula:C18H24ClN3O2Purezza:93.64%Colore e forma:SolidPeso molecolare:349.86γ-secretase modulator 1
CAS:gamma-secretase modulator 1 is a modulator of γ secretase and can be used in studies about the treatment of Alzheimer's disease.Formula:C24H24N4OSPurezza:99.75% - 99.96%Colore e forma:SolidPeso molecolare:416.54GTS-21
CAS:GTS-21 (DMXB-A) is an α7 nAChR agonist. GTS-21 suppresses inflammation associated with rheumatoid arthritis by inhibiting RA Th1 cell differentiation.Formula:C19H20N2O2Purezza:98%Colore e forma:SolidPeso molecolare:308.375-HT3 antagonist 2
CAS:5-HT3 antagonist 2 is an antagonist of 5-HT3 receptor.Formula:C18H21N3OPurezza:98%Colore e forma:SolidPeso molecolare:295.38Trelanserin
CAS:Trelanserin (SL-650472) is an antagonist of the serotonin receptor.Formula:C24H24FN5O2SColore e forma:SolidPeso molecolare:465.54BTA-1
CAS:BTA-1 is an uncharged derivative of thioflavin-T that has high affinity for Aβ fibrils and shows very good brain entry and clearance [1].Formula:C14H12N2SColore e forma:SolidPeso molecolare:240.32SB 714786
CAS:SB 714786 is a selective antagonist of 5-HT1D.Formula:C26H28N4OPurezza:98%Colore e forma:SolidPeso molecolare:412.53Benzoctamine
CAS:Benzoctamine: oral psychoactive with tranquillizing effects; boosts catecholamine turnover; enhances rat heart [3H]noradrenaline uptake.Formula:C18H19NColore e forma:SolidPeso molecolare:249.35R-PSOP
CAS:R-PSOP, a selective NMUR2 antagonist, binds human/rat receptors with 52/32 nM affinity, useful for CNS-related disorders.Formula:C20H22N4O2Colore e forma:SolidPeso molecolare:350.41Nialamide monohydrochloride
CAS:Nialamide monohydrochloride, a withdrawn MAOI antidepressant, poses hepatotoxicity risk.Formula:C16H19ClN4O2Colore e forma:SolidPeso molecolare:334.8hiCE inhibitor-1
CAS:Sulfonamide-derived hiCE inhibitor-1 selectively targets human intestinal enzyme, Ki 53.3 nM, mitigates Irinotecan-induced diarrhea.Formula:C18H14Cl2N2O4S2Colore e forma:SolidPeso molecolare:457.35(R)-DOI hydrochloride
CAS:(R)-DOI hydrochloride is the salt form of 2,5-Dimethoxy-4-iodoamphetamine (DOI), a potent 5-HT2A and 5-HT2C receptor agonist, orally active and hallucinogenic.Formula:C11H17ClINO2Purezza:99.88% - >99.99%Colore e forma:SolidPeso molecolare:357.62DCB
CAS:DCB is an mGluR5 allosteric ligand that blocks mGluR modulation, countering DMeOB and DFB effects.Formula:C14H10Cl2N2Purezza:99.12% - 99.9%Colore e forma:SolidPeso molecolare:277.15Esoxybutynin Chloride
CAS:(S)-oxybutynin, with antimuscarinic effects, is being developed for urinary incontinence.Formula:C22H32ClNO3Colore e forma:SolidPeso molecolare:393.95PF-184298
CAS:PF-184298 is a serotonin and norepinephrine monoamine reuptake inhibitor (SNRI) that inhibits dopamine reuptake.Formula:C15H20Cl2N2OPurezza:98.67%Colore e forma:SolidPeso molecolare:315.24Isamoltane
CAS:Isamoltane is a serotonin 5-HT1 Receptor AntagonistFormula:C16H23ClN2O2Colore e forma:SolidPeso molecolare:310.82Ro 63-0563
CAS:Ro 63-0563 is a potent, 5-HT6 receptors selective antagonist.Formula:C13H17N5O2SPurezza:98%Colore e forma:SolidPeso molecolare:307.37KDS2010 mesylate
CAS:KDS2010: potent, reversible MAO-B inhibitor with 12,500x selectivity vs. MAO-A; enhances memory in APP/PS1 mice.Formula:C18H21F3N2O4SColore e forma:SolidPeso molecolare:418.432-Methyl-5-HT maleate
CAS:2-Methyl-5-HT maleate, a selective 5-HT3 agonist, shows anti-depressive effects.Formula:C15H18N2O5Purezza:98%Colore e forma:SolidPeso molecolare:306.31PF-4522654
CAS:PF-4522654 is a potent and selective 5-HT2C receptor agonist.Formula:C16H18F2N4Colore e forma:SolidPeso molecolare:304.34Pozanicline
CAS:Pozanicline, a selective α4β2 nAChR partial agonist (Ki=16 nM), may treat nicotine addiction by reversing cognitive deficits.Formula:C11H16N2OPurezza:98%Colore e forma:SolidPeso molecolare:192.26CDD0102
CAS:CDD0102 is a potent agonist of M1 Muscarinic receptor.Formula:C8H12N4OPurezza:98%Colore e forma:SolidPeso molecolare:180.21FK-1052 HCl
CAS:FK-1052 HCl is a serotonin 3 & 4 dual receptor antagonist.Formula:C18H20ClN3OColore e forma:SolidPeso molecolare:329.83Pralidoxime mesylate
CAS:Pralidoxime mesylate is a Cholinesterase ReactivatorFormula:C8H12N2O4SColore e forma:SolidPeso molecolare:232.25ELN318463 racemate
CAS:ELN318463 racemate (ELN 318463 racemate) is the racemate of ELN318463 which is an amyloid precursor protein (APP) selective γ-secretase inhibitor.Formula:C19H20BrClN2O3SPurezza:99.69%Colore e forma:SolidPeso molecolare:471.8Ref: TM-T11178L
1mg154,00€5mg370,00€1mL*10mM (DMSO)424,00€10mg583,00€25mg858,00€50mg1.170,00€100mg1.575,00€Radequinil
CAS:Radequinil is a benzodiazepine receptor partial inverse agonist. Rade quinil binds to GABA(-) and GABA(+) ligand (Kis: 5.15 and 6.11 nM, respectively).Formula:C18H14N4O3Purezza:98%Colore e forma:SolidPeso molecolare:334.33Adinazolam Mesylate
CAS:Adinazolam Mesylate is an anxiolytic and antidepressant agent. Adinazolam Mesylate binds to peripheral-type benzodiazepine receptors that interact allosterically with GABA receptors as an agonist to produce inhibitory effects.Formula:C20H22ClN5O3SPurezza:98%Colore e forma:SolidPeso molecolare:447.94Ro 14-7437
CAS:Ro 14-7437 is an antagonist of GABA-benzodiazepine receptor.Formula:C15H15N3O3Colore e forma:SolidPeso molecolare:285.3Profadol hydrochloride
CAS:Profadol hydrochloride acts as a mixed agonist-antagonist of the μ-opioid receptor with analgesic activity.Formula:C14H22ClNOPurezza:98%Colore e forma:SolidPeso molecolare:255.78SCH-50910 free base
CAS:SCH-50910 is an antagonist of GABAB receptor.Formula:C8H15NO3Colore e forma:SolidPeso molecolare:173.21(R)-Duloxetine Hydrochloride
CAS:(R)-Duloxetine Hydrochloride, naphthalenyloxy amine, binds human serum albumin, less effective than (S)-enantiomer as SNRI.Formula:C18H20ClNOSColore e forma:SolidPeso molecolare:333.87Elzasonan
CAS:Elzasonan is a selective 5-hydroxytryptamine 1B receptor antagonist used to treat patients with major depressive disorder and obsessive compulsive disorder.Formula:C22H23Cl2N3OSColore e forma:SolidPeso molecolare:448.41BChE-IN-8
CAS:BChE-IN-8, compound 20, is a potent oral BChE inhibitor effective on eqBChE and hBChE, crosses blood-brain barrier, and may help in Alzheimer's research.Formula:C18H12BrN7O2Colore e forma:SolidPeso molecolare:438.24(S)-MCPG
CAS:(S)-MCPG is the active isomer of (RS)-MCPG, non-selective group I/group II metabotropic glutamate receptor antagonist.Formula:C10H11NO4Purezza:98.72%Colore e forma:SolidPeso molecolare:209.20Ro 15-1310
CAS:Ro 15-3505, a benzodiazepine receptor partial inverse agonist, has shown the ability to improve impaired recent memory of aged mice.Formula:C15H14ClN3O3Colore e forma:SolidPeso molecolare:319.74MAO-B-IN-23
CAS:MAO-B-IN-23, also known as Compound 11f, is a reversible and competitive monoamine oxidase B (MAO-B) inhibitor with an IC50 value of 1.44 μM and a Ki of 0.51 μMFormula:C19H18BrNOPurezza:98%Colore e forma:SolidPeso molecolare:356.26Bitopertin (R enantiomer)
CAS:Bitopertin R enantiomer (RG1678 R enantiomer) is the R-enantiomer of Bitopertin.Formula:C21H20F7N3O4SPurezza:98%Colore e forma:SolidPeso molecolare:543.46Anxiolytic/nonsedative agent-1
CAS:TCS 1205: Selective GABAA agonist, BzR affinity in bovine brain (Kis: 14-239 nM), α2 efficacy in vitro, anxioselective in vivo.Formula:C18H15N3O4Purezza:98.61%Colore e forma:SolidPeso molecolare:337.33Ref: TM-T23445
1mg64,00€2mg96,00€5mg115,00€10mg150,00€25mg330,00€50mg472,00€100mg655,00€500mg1.293,00€PNU-142633
CAS:PNU-142633: anti-migraine, selective 5-HT1D agonist, Ki=6 nM; >18,000 nM for 5-HT1B.Formula:C24H30N4O3Purezza:98%Colore e forma:SolidPeso molecolare:422.52Glutaminyl Cyclase Inhibitor 5
Glutaminyl Cyclase Inhibitor 5 is a potent, selective inhibitor of human glutaminyl cyclase (hQC), demonstrating an inhibition concentration half-max (IC 50) ofFormula:C22H30N6OColore e forma:SolidPeso molecolare:394.51YM-58790
CAS:YM-58790 is a potent mAChR blocker with Ki values of 28 nM (M1), 260 nM (M2), 15 nM (M3), and reduces bladder contractions in rats.Formula:C27H31N3O2Purezza:99.87%Colore e forma:SoildPeso molecolare:429.55LC kinetic stabilizer-2
CAS:LC Kinetic Stabilizer-2 is a powerful stabilizer for amyloidogenic immunoglobulin light chains (LC), demonstrating significant efficacy with an EC50 of 24 nM.Formula:C28H31N3O3Colore e forma:SolidPeso molecolare:457.56A-850002
CAS:A-850002 is a bioactive chemical.Formula:C18H16N4OSColore e forma:SolidPeso molecolare:336.41Asoxime dichloride
CAS:Asoxime dichloride (HI-6) blocks AChRs, including α7 nAChR, and boosts vaccination in the nervous system.Formula:C14H16Cl2N4O3Purezza:99.75% - 99.86%Colore e forma:SolidPeso molecolare:359.21Thiothixene hydrochloride
CAS:Thiothixene hydrochloride is an antipsychotic agent that can be used in the study of schizophrenia and bipolar mania.Formula:C23H30ClN3O2S2Colore e forma:SolidPeso molecolare:480.08Almoxatone
CAS:Almoxatone, also known as MD 780236, is a monoamine oxidase (MAO) inhibitor.Formula:C18H19ClN2O3Colore e forma:SolidPeso molecolare:346.81F-15599 tosylate
CAS:F-15599 tosylate is a selective 5-HT(1A) agonist.Formula:C26H29ClF2N4O4SColore e forma:SolidPeso molecolare:567.05(E/Z)-VU0029767
CAS:VU0029767 enhances M1 muscarinic receptor function, increasing acetylcholine potency and efficacy.Formula:C21H21N3O3Colore e forma:SolidPeso molecolare:363.41Dexetimide HCl
CAS:Dexetimide HCl is a muscarinic antagonist that has been used to treat neuroleptic-induced parkinsonism. Benzetimide is the (-)-enantimorph of dexetimide.Formula:C23H27ClN2O2Colore e forma:SolidPeso molecolare:398.93Fonazine hydrochloride
CAS:Fonazine hydrochloride is a phenothiazine drug used for the treatment of migraine. It is a serotonin antagonist and histamine antagonist.Formula:C19H26ClN3O2S2Colore e forma:SolidPeso molecolare:428.01KL8604166
CAS:KL8604166 (UCB-11056) is a potential puzzle compound.UCB-11056 amplifies the formation of inducible cyclic AMP in rat brain tissue.Formula:C12H21N5O2Purezza:99.21%Colore e forma:SolidPeso molecolare:267.33Ref: TM-T29038
1mg264,00€1mL*10mM (DMSO)590,00€5mg650,00€10mg888,00€25mg1.369,00€50mg1.783,00€100mg2.250,00€PD 118717
CAS:PD 118717: a piperazinyl benzopyranone dopamine agonist with potential antipsychotic properties and no neurological side effects in tests.Formula:C20H22N4O3Purezza:98%Colore e forma:SolidPeso molecolare:366.41mAChr-in-1
CAS:mAChR-IN-1 is muscarinic cholinergic receptor(mAChR) antagonist (IC50=17 nM).Formula:C23H25IN2O2Purezza:98%Colore e forma:SolidPeso molecolare:488.36NRA-0160
CAS:NRA-0160 is a selective antagonist of dopamine D4 receptor(Ki of 0.48 nM)Formula:C24H23F2N3OSPurezza:98%Colore e forma:SolidPeso molecolare:439.52PNU-107484A
CAS:PNU-107484A is a unique GABA(A) receptor ligand.Formula:C18H23ClN6Purezza:98%Colore e forma:SolidPeso molecolare:358.87SB 272183
CAS:SB 272183 is a highly potent dual 5-HT1A and 5-HT1B antagonists as potential antidepressant drug.Formula:C29H28ClN5OPurezza:98%Colore e forma:SolidPeso molecolare:498.02LRE1
CAS:LRE1 is a specific and allosteric soluble adenylyl cyclase inhibitor.Formula:C12H13ClN4SPurezza:>99.99%Colore e forma:SolidPeso molecolare:280.78Methiothepin maleate
CAS:Methiothepin maleate (Metitepine) is a 5-HT1, 5-HT6, 5-HT7 serotonin receptor antagonist, which blocks serotonin autoreceptors.Formula:C24H28N2O4S2Purezza:98%Colore e forma:SolidPeso molecolare:472.62DAA-1097
CAS:DAA-1097 is a novel ligand of peripheral benzodiazepine receptor.Formula:C24H24ClNO3Purezza:98%Colore e forma:SolidPeso molecolare:409.91Anisopirol
CAS:Anisopirol is an antipsychotic drug. Studies have shown that it can target dopamine receptors (DA), N-methyl-d-aspartate receptors (NMDA).Formula:C21H27FN2O2Colore e forma:SolidPeso molecolare:358.45DBO-83
CAS:DBO-83, an agonist of nicotinic acetylcholine receptors (nAChRs), has anti-amnesic and antinociceptive activities.Formula:C10H15Cl3N4Purezza:98%Colore e forma:SolidPeso molecolare:297.61ABP-700
CAS:ABP-700 is a positive allosteric modulator of the GABAA receptor.Formula:C17H18N2O4Purezza:98%Colore e forma:SolidPeso molecolare:314.34Suclofenide
CAS:Suclofenide: a benzenesulfonamide anticonvulsant, effective in mouse seizure models, with side effects like lethargy and diarrhea.Formula:C16H13ClN2O4SPurezza:98%Colore e forma:SolidPeso molecolare:364.8RS-0466
CAS:RS-0466 is an β-amyloid-induced cytotoxicity inhibitor.Formula:C17H17N5O2Purezza:98%Colore e forma:SolidPeso molecolare:323.35JY-XHe-053
CAS:JY-XHe-053 is a selective modulator of GABAA receptors.Formula:C22H16FN3O2Purezza:98%Colore e forma:SolidPeso molecolare:373.38W-5 hydrochloride
CAS:W-5 hydrochloride (N-(6-Aminohexyl)-1-naphthalenesulfonamide HCl) is a potent calmodulin antagonist.Formula:C16H23ClN2O2SPurezza:99.35%Colore e forma:Off-White Crystalline SolidPeso molecolare:342.88MDL 73005EF hydrochloride
CAS:5-HT1A receptor antagonistFormula:C20H27ClN2O4Purezza:98%Colore e forma:SolidPeso molecolare:394.89S16961
CAS:S16961 (S169611) is an agonist of nicotinic receptor.Formula:C41H71NO6Purezza:99.69%Colore e forma:SolidPeso molecolare:674.01Afacifenacin
CAS:Afacifenacin (SMP-986) fumarate is an M3-selective antagonist for ischemic heart disease and urinary disorders.Formula:C27H26F3N3O2Purezza:99.83%Colore e forma:SolidPeso molecolare:481.51AR-R 17779 hydrochloride
CAS:AR-R17779 hydrochloride: potent α7 nAChR agonist; K i : 92 nM (α7), 16,000 nM (α4β2); enhances rat cognition; anxiolytic; anti-inflammatory.Formula:C9H15ClN2O2Colore e forma:SolidPeso molecolare:218.68LP44 hydrochloride
CAS:LP44 hydrochloride is a 5-HT7 agonist with analgesic effects on formalin-induced orofacial pain in mice and can be used to study neuroinflammation.Formula:C27H38ClN3OSPurezza:98.06%Colore e forma:SolidPeso molecolare:488.13CB-7921220
CAS:CB-7921220 (6-[2-(4-Aminophenyl)vinyl]-2-pyridinecarboxylic acid) is an inhibitor of adenylate cyclase.Formula:C14H12N2O2Purezza:99.59%Colore e forma:SolidPeso molecolare:240.26VU6001376
CAS:VU6001376 is an effective and selective positive allosteric modulator of the metabotropic glutamate receptor 4 (EC50: 50.1 nM).Formula:C18H14F2N6OSPurezza:98%Colore e forma:SolidPeso molecolare:400.41DFMTI
CAS:DFMTI can completely block the rmGlu1 L757V glutamate response.Formula:C20H18F2N4OColore e forma:SolidPeso molecolare:368.38PRX933 hydrochloride
CAS:PRX933 hydrochloride (GW876167 hydrochloride) is an agonist of 5-HT2C receptor and can be used in studies about hypertension acute treatment.Formula:C16H22ClN5O2Purezza:99.51% - 99.89%Colore e forma:SolidPeso molecolare:351.84Ref: TM-T12565
1mg338,00€5mg538,00€1mL*10mM (DMSO)618,00€10mg858,00€25mg1.269,00€50mg1.720,00€100mg2.305,00€HOCPCA
CAS:HOCPCA: potent, selective GHB site ligand; 27x higher affinity than GHB; crosses blood-brain barrier.Formula:C6H8O3Purezza:98%Colore e forma:SolidPeso molecolare:128.13Hyoscyamine hydrobromide
CAS:Hyoscyamine hydrobromide is an agent of anticholinergic.Formula:C17H24BrNO3Purezza:98%Colore e forma:SolidPeso molecolare:370.28Epibatidine 2HCl
CAS:Epibatidine 2HCl is a potent nicotinic agonist.Formula:C11H15Cl3N2Purezza:98%Colore e forma:SolidPeso molecolare:281.61CPP-115
CAS:CPP-115 is a GABA-aminotransferase inhibitor and a high-affinity vigabatrin analogue.Formula:C7H9F2NO2Colore e forma:SolidPeso molecolare:177.15Btm 1042
CAS:Btm 1042 is an antispasmodic drug. It has been found to depress twitch responses in the ileum of guinea pigs.Formula:C21H26ClN3OSColore e forma:SolidPeso molecolare:403.97SDZ 205-557 hydrochloride
CAS:5-HT3/5-HT4 receptor antagonistFormula:C14H22Cl2N2O3Purezza:98%Colore e forma:SolidPeso molecolare:337.245-Nonyloxytryptamine oxalate
CAS:5-HT1B agonistFormula:C21H32N2O5Purezza:98%Colore e forma:SolidPeso molecolare:392.49RGH 1756
CAS:RGH 1756 is an atypical antipsychotic with high affinity to dopamine D(3) receptors that leads to c-Fos induction in a unique pattern.Formula:C26H30N4O2SPurezza:98%Colore e forma:SolidPeso molecolare:462.61AZ4800
CAS:AZD4800 is a gamma secretase modulators.Formula:C24H29N5O3Colore e forma:SolidPeso molecolare:435.52Palonosetron
CAS:Palonosetron, a 5-HT3 antagonist with Ki of 0.17 nM, is used in the prevention and treatment of chemotherapy-induced nausea and vomiting (CINV).Formula:C19H24N2OPurezza:98%Colore e forma:SolidPeso molecolare:296.41N,N-Dipropyldopamine (hydrobromide)
CAS:N,N-Dipropyldopamine is a dopamine agonist reducing DOPA and locomotion in rats and mice, reversible by spiroperidol.Formula:C14H24BrNO2Colore e forma:SolidPeso molecolare:318.255Astrophloxine
CAS:Astrophloxine is a fluorescent imaging probe that targets antiparallel dimers.Astrophloxine can be used to detect aggregated Aβ in brain tissue andFormula:C27H33IN2Purezza:99.89%Colore e forma:SolidPeso molecolare:512.47Mirisetron
CAS:Mirisetron (WAY-100579, SEC-579) is a 5-HT3 receptor antagonist, cognitive-enhancing effects. counteracts learning deficits.Formula:C24H31N3O2Purezza:99.88%Colore e forma:SolidPeso molecolare:393.52Sulfoxaflor
CAS:Sulfoxaflor (GF 2032) is an agonist of nAChR1 and nAChR2 subtypes and a systemic insecticide. Cost-effective and quality-assured.Formula:C10H10F3N3OSPurezza:99.56% - 99.98%Colore e forma:SolidPeso molecolare:277.27Ref: TM-T19940
1mg100,00€1mL*10mM (DMSO)245,00€5mg275,00€10mg384,00€25mg572,00€50mg780,00€100mg1.018,00€250mg2.080,00€S 24795
CAS:S 24795 (Catestatin acetate(142211-96-9 free base)) is an α7 nAChR partial agonist.Formula:C14H13BrINOPurezza:99.934%Colore e forma:SolidPeso molecolare:418.07Ref: TM-T23286
5mg44,00€1mL*10mM (DMSO)48,00€10mg66,00€25mg138,00€50mg215,00€100mg338,00€200mg480,00€Protriptyline
CAS:Protriptyline: Antidepressant, AChE inhibitor (IC50 0.06 mM), prevents Aβ aggregation; potential for depression and Alzheimer's.Formula:C19H21NColore e forma:SolidPeso molecolare:263.38Naronapride
CAS:Naronapride (ATI-7505) is a potent agonist of the prokinetic 5-HT4receptor and can be used to study gastrointestinal disorders.Formula:C27H41ClN4O5Colore e forma:SolidPeso molecolare:537.09BChE-IN-9
CAS:BChE-IN-9 (Azepano-11-deoxo-glycyrrhetol) is a hybrid BChE inhibitor (Ki: 0.21 μM).Formula:C30H51NOColore e forma:SolidPeso molecolare:441.73(±)-Muscarine chloride
CAS:(±)-Muscarine chloride is the racemate of Muscarine chloride. Muscarine is a prototypical agonist for the muscarinic acetylcholine receptor [1] [2].Formula:C9H20ClNO2Colore e forma:SolidPeso molecolare:209.71(Rac)-SEP-363856
CAS:(Rac)-SEP-363856 is the racemate of SEP-363856. SEP-363856 is an orally active and CNS active psychotropic agent with a uniqueFormula:C9H13NOSPurezza:98%Colore e forma:SolidPeso molecolare:183.27AChE/BChE-IN-5
CAS:AChE/BChE-IN-5 (BMC-16) crosses BBB; IC50: hAChE 266 nM, hBChE 10.6 nM. Dual AChE/BChE inhibitor.Formula:C17H26N2O3Colore e forma:SolidPeso molecolare:306.4S-15535
CAS:S-15535 is a potent, orally active, partial 5-HT1A receptor agonist.Formula:C21H24N2O2Purezza:98%Colore e forma:SolidPeso molecolare:336.43OSU 6162 hydrochloride
CAS:Dopamine stabilizerFormula:C15H24ClNO2SPurezza:98%Colore e forma:SolidPeso molecolare:317.88mGluR2 modulator 2
CAS:mGluR2 modulator 2: potent, selective, oral, EC50 = 0.13 μM, for antipsychotic research.Formula:C20H22FN3Colore e forma:SolidPeso molecolare:323.41PF-06455943
CAS:PF-06455943: LRRK2 inhibitor, IC50=3nM, PET radioligand, used for ADME/neuro PK & Parkinson's research.Formula:C17H14FN5OColore e forma:SolidPeso molecolare:323.32Talaglumetad hydrochloride
CAS:Talaglumetad hydrochloride, a prodrug of Eglumegad, targets mGluR2/3 to treat psychiatric disorders.Formula:C11H17ClN2O5Colore e forma:SolidPeso molecolare:292.72AZD 0328
CAS:AZD 0328 is a nicotinic receptor agonist for α7 neurons.Formula:C13H16N2OColore e forma:SolidPeso molecolare:216.28AChE/BChE/MAO-B-IN-4
AChE/BChE/MAO-B-IN-4 inhibits MAO-B (IC50: 0.0393 µM), AChE (IC50: 0.0458 µM), BChE (IC50: 0.075 µM), and fights AD with antioxidant action.Formula:C26H33N3O4Colore e forma:SolidPeso molecolare:451.56RS 23597-190 hydrochloride
CAS:RS 23597-190 hydrochloride is a 5-HT4 receptor antagonist.Formula:C16H24Cl2N2O3Purezza:98%Colore e forma:SolidPeso molecolare:363.28AChE/BChE-IN-4
CAS:AChE/BChE-IN-4 (BMC-3) crosses the BBB; IC50: hAChE 792 nM, hBChE 2.2 nM. Dual AChE/BChE inhibitor.Formula:C17H26N2O3Colore e forma:SolidPeso molecolare:306.4Bibn 140
CAS:Bibn 140 is a highly selective M2 antagonist, it is used to treat Alzheimer's disease and other cognitive disorders.Formula:C32H44N4O3Purezza:98%Colore e forma:SolidPeso molecolare:532.72RX 67668
CAS:RX 67668: Muscle relaxant, relieves fatigue; cholinesterase inhibitor (IC50: 5 μM); reverses D-tubocurarine effects.Formula:C16H24ClNPurezza:98%Colore e forma:SolidPeso molecolare:265.82RO5488608
CAS:RO5488608 is a new type of high-efficiency mGlu2/3 NAM.Formula:C23H17F3N2O4SColore e forma:SolidPeso molecolare:474.45Aβ-IN-5
CAS:Aβ-IN-5 (Compound e12) is an orally active Aβ aggregation inhibitor that also inhibits AChE and BuChE with IC50 values of 21.29 μM and 1.32 μM, respectively.Formula:C21H20N2O3Colore e forma:SolidPeso molecolare:348.4A 841720
CAS:Potent, selective mGlu1 antagonist A-841720; IC50: 10 nM; 34x selectivity vs mGlu5; analgesic potential.Formula:C17H21N5OSColore e forma:SolidPeso molecolare:343.45BChE-IN-11
CAS:BChE-IN-11: potent, selective, non-competitive BChE inhibitor; IC50=2.1μM; used in AD research.Formula:C22H18O4Colore e forma:SolidPeso molecolare:346.38NPEC-caged-LY379268
CAS:NPEC-caged-LY379268 is a type II mGluR agonist [1].Formula:C16H16N2O9Colore e forma:SolidPeso molecolare:380.31Anabasine hydrochloride
CAS:neuronal nicotinic ACh receptor partial agonistFormula:C10H15ClN2Purezza:98%Colore e forma:White To Off-White SolidPeso molecolare:198.693Pheniprazine
CAS:Pheniprazine, a potent and long-acting monoamine oxidase inhibitor, shows promise for depression research.Formula:C9H14N2Colore e forma:SolidPeso molecolare:150.22Ethybenztropine
CAS:Ethybenztropine is an anticholinergic used as an antiparkinsonian agent and may also act as a dopamine reuptake inhibitor.Formula:C22H27NOPurezza:98%Colore e forma:SolidPeso molecolare:321.46Zicronapine
CAS:Zicronapine (LU 31-130), an atypical antipsychotic with monoaminergic action, targets dopamine D1/D2 and serotonin 5HT2A.Formula:C22H27ClN2Colore e forma:SolidPeso molecolare:354.925-HT7 agonist 2
CAS:Potent 5-HT7 agonist with 28.7 nM IC50; promising for CNS disorder research.Formula:C23H29N3OColore e forma:SolidPeso molecolare:363.5Memoquin
CAS:Memoquin is a multi-target-directed ligand for the therapy of Alzheimer's disease.Formula:C38H56N4O4Colore e forma:SolidPeso molecolare:632.88Bornaprine
CAS:Bornaprine is an anticholinergic drug used to treat Parkinson's disease due to inhibition of muscarinic or nicotinic transmission.Formula:C21H31NO2Colore e forma:SolidPeso molecolare:329.48CP-809101
CAS:CP-809101 is an effective and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).Formula:C15H17ClN4OPurezza:98%Colore e forma:SolidPeso molecolare:304.77Antioxidant agent-2
CAS:Antioxidant agent-2 (3c), BBB-permeable, selectively chelates metals; shows neuroprotection, fights liver damage in Alzheimer's research.Formula:C23H26N2O7Colore e forma:SolidPeso molecolare:442.46VU0455691
CAS:VU0455691 is a selective M1 Muscarinic Receptor Allosteric Modulators.Formula:C24H25N5O3SPurezza:98%Colore e forma:SolidPeso molecolare:463.55LY314228
CAS:LY314228 is an antagonist of 5-HT2A receptor.Formula:C20H24N4O3Colore e forma:SolidPeso molecolare:368.43Dihydro Donepezil
CAS:Dihydro Donepezil (Dihydro E2020), a Donepezil metabolite, is a potent AChE inhibitor (IC50: hAChE 11.6 nM, bAChE 8.12 nM).Formula:C24H31NO3Colore e forma:SolidPeso molecolare:381.51NAP-1
CAS:NAP-1 is an anesthetic that enhances CA1 brain inhibition in rats and causes tadpole sedation (EC50 = 0.53 μM).Formula:C20H18ClNO2Colore e forma:SolidPeso molecolare:339.82BACE2-IN-1
CAS:BACE2-IN-1, a potent BACE2 inhibitor characterized by its exceptional selectivity and a Ki value of 1.6 nM, is utilized in the investigation of Type 2 Diabetes.Formula:C36H38F3N3O3Colore e forma:SolidPeso molecolare:617.7LSP4-2022
CAS:LSP4-2022, a mGlu4 selective agonist, increases behavioral despair in mouse models of antidepressant action.Formula:C13H18NO8PPurezza:100%Colore e forma:SolidPeso molecolare:347.26Trimedoxime bromide
CAS:Trimedoxime bromide is a cholinesterase reactivator used as an antidote in alkyl phosphate poisoning.Formula:C15H18Br2N4O2Colore e forma:SolidPeso molecolare:446.14Lidanserin
CAS:Lidanserin is an antagonist of the 5-HT2A and α1-adrenergic receptor.Formula:C26H31FN2O4Purezza:98%Colore e forma:SolidPeso molecolare:454.53UMB68 sodium
CAS:UMB-68 is a GHB receptor ligand with no affinity (IC(50) >100 microM) at GABA(A) or GABA(B) receptors.Formula:C6H12NaO3Colore e forma:SolidPeso molecolare:155.149Fonazine
CAS:Forazine (dimethiazide) is a phenothiazine drug used in the treatment of migraine and is a serotonin antagonist and a histamine antagonist.Formula:C19H25N3O2S2Colore e forma:SolidPeso molecolare:391.55MMPIP
CAS:allosteric mGlu7-selective receptor antagonistFormula:C19H15N3O3Purezza:98%Colore e forma:SolidPeso molecolare:333.34AChE/BChE/MAO-B-IN-2
AChE/BChE/MAO-B-IN-2 inhibits AChE (48.2 nM), BChE (83.9 nM), MAO-B (31.2 nM), has antioxidant activity, and aids Parkinson's research.Formula:C25H31N3O3Colore e forma:SolidPeso molecolare:421.53AChE/BChE/BACE-1-IN-1
CAS:Compound 4k is an oral AChE, BChE, BACE-1 inhibitor with IC50s: 0.058, 0.082, 0.115 μM, crosses blood-brain barrier, and has neuroprotective effects.Formula:C19H21F3N2OColore e forma:SolidPeso molecolare:350.38ZLWH-23
CAS:ZLWH-23: AChE inhibitor (IC50: 0.27μM), GSK-3β (6.78μM), BChE (20.82μM), potential in Alzheimer's research.Formula:C30H32FN5O2Colore e forma:SolidPeso molecolare:513.61Org-25935
CAS:Org-25935, a GlyT-1 inhibitor, is used potentially for the treatment of schizophrenia and alcohol dependence.Formula:C21H26ClNO3Colore e forma:SolidPeso molecolare:375.89Ro4491533
CAS:Ro4491533 is a potent and selective negative allosteric modulator for group II of the metabotropic glutamate receptors (mGluR2/3).Formula:C24H20F3N3OColore e forma:SolidPeso molecolare:423.43MAO-B ligand-1
CAS:MAO-B ligand-1 is a selective MAO-B inhibitor.Formula:C19H19N5O4SColore e forma:SolidPeso molecolare:413.45(RS)-4-Carboxy-3-hydroxyphenylglycine
CAS:broad spectrum EAA agonist/antagonistFormula:C9H9NO5Purezza:98%Colore e forma:SolidPeso molecolare:211.17sEH/AChE-IN-1
CAS:Compound 12a is a dual sEH/AChE inhibitor with potential for treating Alzheimer's-related neuroinflammation and memory loss.Formula:C29H31ClF3N5O3Colore e forma:SolidPeso molecolare:590.04Phenglutarimid
CAS:Phenglutarimid is an anticholinergic. It is used as an antiparkinsonian agent.Formula:C17H24N2O2Purezza:98%Colore e forma:SolidPeso molecolare:288.38ATC0065
CAS:ATC0065 is a melanin-concentrating hormone receptor 1 antagonist with oral activity.Formula:C25H29BrF3N5OColore e forma:SolidPeso molecolare:552.435-HT7 receptor ligand 1
CAS:Compound 5c: 5-HT7 receptor ligand, K i = 8 nM, not hepatotoxic, moderate CYP3A4/CYP2D6 interaction.Formula:C21H23N7Colore e forma:SolidPeso molecolare:373.45PXS-4787
CAS:PXS-4787 selectively inhibits LOX with IC50 values: 2 μM (Bovine), 3.2 μM (LOXL1), 0.6 μM (LOXL2), 1.4 μM (LOXL3), 0.2 μM (LOXL4).Formula:C10H12FNO2SColore e forma:SolidPeso molecolare:229.27WAY-361789
CAS:WAY-361789 is an agonist of alpha7 nicotinic acetylcholine receptor.Formula:C22H31N5O3Colore e forma:SolidPeso molecolare:413.51VU0400195
CAS:VU0400195 is a oral effective, positive allosteric modulator of the metabotropic glutamate receptor 4 (mGlu(4)).Formula:C21H16ClN3O3Purezza:98%Colore e forma:SolidPeso molecolare:393.82ML337
CAS:ML337 is a negative allosteric modulator of mGlu3 with an IC50 of 593 nM.Formula:C21H20FNO3Purezza:99.83%Colore e forma:SolidPeso molecolare:353.39Ref: TM-T23003
100mgPrezzo su richiesta1mg34,00€5mg60,00€1mL*10mM (DMSO)72,00€10mg92,00€25mg195,00€50mg293,00€Piclozotan
CAS:Piclozotan (anhydrous), a 5-HT1A receptor agonist, demonstrated significant neuroprotective activity in a transient middle cerebral artery occlusion (t-MCAO)Formula:C23H24ClN3O2Purezza:98.59%Colore e forma:SolidPeso molecolare:409.91Melatonin receptor agonist 1
CAS:Melatonin receptor agonist 1 (compound 20c) is a potent agonist of melatonin receptor (MT) with Ki values of 108 nM for MT2 and 1140 nM for MT 1 [1].Formula:C15H19N3O2Colore e forma:SolidPeso molecolare:273.33VU0404251
CAS:VU0404251 is a positive allosteric modulator of mGlu5.Formula:C19H23FN2O2Colore e forma:SolidPeso molecolare:330.4Tacitin
CAS:Tacitin (Benzoctamine Hydrochloride) shows sedative and anti-anxiety properties. Tacitin blocks the central postsynaptic serotonin receptors.Formula:C18H20ClNPurezza:98%Colore e forma:SolidPeso molecolare:285.81TC 1698 dihydrochloride
CAS:nicotinic α7 receptor agonistFormula:C13H18N2Purezza:98%Colore e forma:SolidPeso molecolare:202.3BChE-IN-13
CAS:BChE-IN-13 (17c): Oral, potent, selective BChE inhibitor; IC50: eqBChE 0.22μM, hBChE 0.016μM; aids memory, Alzheimer's research.Formula:C24H28N2OColore e forma:SolidPeso molecolare:360.49CGS8216
CAS:CGS8216 shows analgesic activity at high doses, has anxiolytic activity, and can be used to study immune system disorders.Formula:C16H11N3OPurezza:98.53%Colore e forma:SolidPeso molecolare:261.28SB357134
CAS:SB357134 is a potent, selective and orally active antagonist of 5-HT6 receptor and shows nootropic effects in animal studies.Formula:C17H18Br2FN3O3SPurezza:98%Colore e forma:SolidPeso molecolare:523.21M1 ligand 1
CAS:Compound 3b-b: N-desmethyl arecoline derivative, muscarinic M1 ligand, potential PET radiotracer.Formula:C20H21NO2Colore e forma:SolidPeso molecolare:307.39L-CCG-l
CAS:group II metabotropic glutamate receptor agonistFormula:C6H9NO4Purezza:98%Colore e forma:SolidPeso molecolare:159.1417-PA
CAS:17-PA is a GABAA receptor antagonist.Formula:C25H34OPurezza:98%Colore e forma:SolidPeso molecolare:350.54Prenylamine lactate
CAS:Prenylamine lactate, an ex-angina drug, depletes heart catecholamines and blocks calcium channels.Formula:C27H33NO3Purezza:98%Colore e forma:SolidPeso molecolare:419.56UCSF678
CAS:UCSF678: selective 42 nM partial agonist at 5-HT5AR, fewer off-target effects, and lower assay risks than SB-699551.Formula:C15H18N2O2SColore e forma:SolidPeso molecolare:290.38CGP11952
CAS:CGP11952 is same the benzodiazepines in its pharmacological action and it also is an experimental benzodiazepine derivative.Formula:C21H21Cl2N5O2Purezza:98%Colore e forma:SolidPeso molecolare:446.33AChE/MAO-IN-2
Potent AChE/MAO-B inhibitor; IC50: AChE 0.0224 μM, MAO-B 0.0412 μM, MAO-A 0.1116 μM. Antioxidant, anti-β-amyloid, for AD research.Formula:C23H26N2O3Colore e forma:SolidPeso molecolare:378.46Dual AChE-MAO B-IN-2
CAS:Potent Dual AChE-MAO B-IN-2 inhibits AChE (0.12 μM) & MAO B (0.01 μM); promising for Alzheimer's research.Formula:C26H25NO4Colore e forma:SolidPeso molecolare:415.48Tridihexethyl chloride
CAS:Tridihexethyl is an anticholinergic, antimuscarinic, and antispasmolytic drug, which can be used to treat acquired nystagmus or peptic ulcer disease.Formula:C21H36ClNOColore e forma:SolidPeso molecolare:353.97DV 7028 hydrochloride
CAS:DV 7028 hydrochloride is a 5-HT2A receptor antagonist.Formula:C21H26ClFN4O3Purezza:98%Colore e forma:SolidPeso molecolare:436.91S20928
CAS:S20928 is an antagonist of melatonin receptor.Formula:C17H19NOColore e forma:SolidPeso molecolare:253.34NW-1772
CAS:NW-1772 is a highly potent and orally active inhibitor of monoamine oxidase B.Formula:C19H20ClNO6SPurezza:98%Colore e forma:SolidPeso molecolare:425.88GABAA receptor agent 4
CAS:Compound 1e is a potent γ-GABAAR antagonist with a Ki of 0.18 µM, offering immunomodulatory effects on T cell proliferation.Formula:C17H24N2OColore e forma:SolidPeso molecolare:272.39ML169
CAS:ML169 is a selective and brain penetrant M1 positive allosteric modulator (PAM).Formula:C21H17BrFN3O4SPurezza:98%Colore e forma:SolidPeso molecolare:506.34Ro 60-0175 fumarate
CAS:5-HT2 receptor agonistFormula:C15H16ClFN2O4Purezza:98%Colore e forma:SolidPeso molecolare:342.75GRN-529
CAS:GRN-529 is a selective negative allosteric modulator of the mGluR5 receptor.Formula:C22H15F2N3O2Purezza:98%Colore e forma:SolidPeso molecolare:391.37VMY-2-95
CAS:VMY-2-95 is an α4β2 nicotinic acetylcholine receptors (nAChRs) selective desensitizer.Formula:C17H16N2OColore e forma:SolidPeso molecolare:264.32Arecaidine propargyl ester tosylate
CAS:Arecaidine propargyl ester tosylate is a muscarinic receptor agonist.Formula:C17H21NO5SPurezza:98%Colore e forma:SolidPeso molecolare:351.42S-14671
CAS:S-14671: 5-HT1A agonist (pKi 9.3), potent in vivo; 5-HT2A/2C antagonist (pKi 7.8).Formula:C22H25N3O2SColore e forma:SolidPeso molecolare:395.52GABA-AT-IN-1
CAS:GABA-AT-IN-1 (Compound 6) is an inhibitor of γ-aminobutyric acid transaminase (GABA-AT) that crosses the blood-brain barrier.Formula:C23H18N2O6Colore e forma:SolidPeso molecolare:418.4SB-221284
CAS:5-HT2C/2B receptor antagonistFormula:C16H14F3N3OSPurezza:98%Colore e forma:SolidPeso molecolare:353.36S 32212 hydrochloride
CAS:S 32212 hydrochloride is a high-affinity inverse agonist at the 5-HT2C receptor and an antagonist at the α2-adrenergic receptor, which is antidepressant .Formula:C25H29ClN4O2Purezza:97.11% - 99.57%Colore e forma:SolidPeso molecolare:452.98Org-13011 fumarate
CAS:Org-13011 fumarate1 is an agonist of the 5-HT1A receptor and can be used to study neurological disorders.Formula:C22H29F3N4O5Purezza:98.92%Colore e forma:SolidPeso molecolare:486.48Enciprazine
CAS:Enciprazine (D-3112) shows anxiolytic activity, is used to treat anxiety disorders, and can be used to study depression.Formula:C23H32N2O6Purezza:98.63%Colore e forma:SolidPeso molecolare:432.51LY 125180
CAS:LY 125180 is a serotonin antagonist.Formula:C18H24ClNOPurezza:98%Colore e forma:SolidPeso molecolare:305.84PF-4479745
CAS:PF-4479745 ia a potent and selective agonist of 5-HT2C receptor.Formula:C17H22N4Purezza:98%Colore e forma:SolidPeso molecolare:282.38LY 2365109 hydrochloride
CAS:glycine transporter 1 (GlyT1) inhibitorFormula:C22H27NO5Purezza:98%Colore e forma:SolidPeso molecolare:385.45
