Neuroscienza
Gli inibitori in neuroscienze sono composti progettati per modulare l'attività di proteine, enzimi o recettori specifici all'interno del sistema nervoso. Questi inibitori sono cruciali per studiare i meccanismi molecolari alla base della funzione neuronale, della trasmissione sinaptica e delle malattie neurodegenerative. Mirando ai recettori dei neurotrasmettitori, ai canali ionici e alle vie di segnalazione, gli inibitori in neuroscienze aiutano a esplorare la funzione cerebrale e a sviluppare strategie terapeutiche per disturbi neurologici come l'Alzheimer, il Parkinson e l'epilessia. Presso CymitQuimica, offriamo una vasta gamma di inibitori in neuroscienze di alta qualità per supportare la tua ricerca in neurobiologia, neurofarmacologia e scienze cognitive.
Sottocategorie di "Neuroscienza"
- recettore 5-HT(1.025 prodotti)
- ACK(1 prodotti)
- AChR(645 prodotti)
- Citrato liasi ATP(17 prodotti)
- Recettore adrenergico(3.018 prodotti)
- BACE(37 prodotti)
- Beta amiloide(228 prodotti)
- CaMK(73 prodotti)
- COX(600 prodotti)
- Recettore della dopamina(445 prodotti)
- Ricettore GABA(372 prodotti)
- Gamma-secretasi(61 prodotti)
- GluR(265 prodotti)
- GlyT(26 prodotti)
- Recettore dell'istamina(385 prodotti)
- LRRK2(43 prodotti)
- Recettore della melatonina(26 prodotti)
- NMDAR(10 prodotti)
- Recettore OX(41 prodotti)
- Recettore degli oppioidi(327 prodotti)
Mostrare 12 più sottocategorie
Trovati 5530 prodotti di "Neuroscienza"
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UH-AH 37
CAS:UH-AH 37 is a antagonist of human muscarinic acetylcholine receptor.Formula:C21H23Cl2N3O2Purezza:98%Colore e forma:SolidPeso molecolare:420.33NW-1772 free base
CAS:NW-1772 free base is a monoamine oxidase B inhibitor.Formula:C18H16ClNO3Colore e forma:SolidPeso molecolare:329.78Dexetimide HCl
CAS:Dexetimide HCl is a muscarinic antagonist that has been used to treat neuroleptic-induced parkinsonism. Benzetimide is the (-)-enantimorph of dexetimide.Formula:C23H27ClN2O2Colore e forma:SolidPeso molecolare:398.93(E/Z)-VU0029767
CAS:VU0029767 enhances M1 muscarinic receptor function, increasing acetylcholine potency and efficacy.Formula:C21H21N3O3Colore e forma:SolidPeso molecolare:363.41Ciclotizolam
CAS:Ciclotizolam, a thienotriazolodiazepine derivative and partial GABAA receptor agonist, has low efficacy but similar affinity as brotizolam.Formula:C20H18BrClN4SColore e forma:SolidPeso molecolare:461.81AChE/BChE-IN-4
CAS:AChE/BChE-IN-4 (BMC-3) crosses the BBB; IC50: hAChE 792 nM, hBChE 2.2 nM. Dual AChE/BChE inhibitor.Formula:C17H26N2O3Colore e forma:SolidPeso molecolare:306.4Methoxy-PEPy
CAS:Methoxy-PEPy is a potent and selective mGlu5 receptor inhibitor with an IC50 value of 1 nM.Formula:C13H10N2OPurezza:98.66%Colore e forma:SolidPeso molecolare:210.23MRK-623
CAS:MRK-623 (14k) is an oral GABA A agonist with high affinity for α1/α2/α3/α5 subunits and anxiolytic properties.Formula:C20H17FN4OColore e forma:SolidPeso molecolare:348.37Ethybenztropine HBr
CAS:Ethybenztropine HBr is an anticholinergic which is used as an antiparkinsonian agent. Ethybenztropine may also act as a dopamine reuptake inhibitor.Formula:C22H28BrNOColore e forma:SolidPeso molecolare:402.37Eplivanserin hemifumarate
CAS:Eplivanserin is an inverse agonist of 5-HT2A.Formula:C23H25FN2O6Colore e forma:SolidPeso molecolare:444.45Tropatepine
CAS:Tropatepine: oral anticholinergic, treats extrapyramidal symptoms, anti-Parkinson's.Formula:C22H23NSColore e forma:SolidPeso molecolare:333.49Bibn 140
CAS:Bibn 140 is a highly selective M2 antagonist, it is used to treat Alzheimer's disease and other cognitive disorders.Formula:C32H44N4O3Purezza:98%Colore e forma:SolidPeso molecolare:532.72Atropine Oxide Hydrochloride
CAS:Atropine Oxide, a derivative of anticholinergic Atropine, treats poisonings, slow heart rate, and reduces saliva during surgery.Formula:C17H24ClNO4Colore e forma:SolidPeso molecolare:341.83Neostigmine hydroxide
CAS:Neostigmine hydroxide, a cholinesterase inhibitor, treats myasthenia gravis and reverses muscle relaxants; doesn't cross the blood-brain barrier.Formula:C12H20N2O3Colore e forma:SolidPeso molecolare:240.3F-15599 tosylate
CAS:F-15599 tosylate is a selective 5-HT(1A) agonist.Formula:C26H29ClF2N4O4SColore e forma:SolidPeso molecolare:567.05RX 67668
CAS:RX 67668: Muscle relaxant, relieves fatigue; cholinesterase inhibitor (IC50: 5 μM); reverses D-tubocurarine effects.Formula:C16H24ClNPurezza:98%Colore e forma:SolidPeso molecolare:265.82RJR-2403 oxalate
CAS:RJR-2403 oxalate is a highly selective agonist of α4β2 subtype nicotinic receptor.Formula:C14H18N2O4Purezza:98%Colore e forma:SolidPeso molecolare:278.308Levomepromazine Maleate
CAS:Levomepromazine Maleate: TCA and SNRI with antihistamine, antiadrenergic, and anticholinergic properties.Formula:C23H28N2O5SColore e forma:SolidPeso molecolare:444.546Belaperidone
CAS:Belaperidone, an antipsychotic, resembles clozapine, binds D(4) and 5-HT(2A) receptors, minimally extends Q-T without causing arrhythmias.Formula:C22H22FN3O2Colore e forma:SolidPeso molecolare:379.43Almoxatone
CAS:Almoxatone, also known as MD 780236, is a monoamine oxidase (MAO) inhibitor.Formula:C18H19ClN2O3Colore e forma:SolidPeso molecolare:346.81MD 780236
CAS:MD 780236 is a monoamine oxidase-B inhibitor.Formula:C18H19ClN2O3Colore e forma:SolidPeso molecolare:346.81Tribendimidine
CAS:Tribendimidine: broad-spectrum oral anthelmintic, nAChR agonist, effective against A. lumbricoides and N. americanus.Formula:C28H32N6Purezza:≥98%Colore e forma:SolidPeso molecolare:452.59W-9 hydrochloride
CAS:W-9 hydrochloride is a calmodulin antagonist.Formula:C16H22Cl2N2O2SPurezza:98.9%Colore e forma:SolidPeso molecolare:377.33Ref: TM-T23525
1mg34,00€2mg42,00€5mg60,00€10mg90,00€25mg173,00€50mg269,00€100mg389,00€500mgPrezzo su richiesta1mL*10mM (DMSO)66,00€Ensaculin
CAS:Ensaculin, a benzopyrone-piperazine compound, enhances memory, protects neurons, and may treat dementia.Formula:C26H32N2O5Purezza:99.56% - 99.81%Colore e forma:SolidPeso molecolare:452.54LY-2300559
CAS:LY-2300559 is an agonist of metabotropic glutamate receptor 2 (mGluR2) and can be used in studies about the treatment of migraine.Formula:C26H26O6Purezza:99.22%Colore e forma:SolidPeso molecolare:434.48Ref: TM-T27932
1mg315,00€5mg745,00€10mg1.018,00€25mg1.431,00€50mg1.783,00€100mg2.250,00€500mg4.410,00€VU 0285683
CAS:VU 0285683 is a specific negative allosteric modulator of mGluR5 with a high affinity for the MPEP binding site. VU 0285683 shows anxiolytic-like activity.Formula:C14H7FN4OPurezza:99.98%Colore e forma:SolidPeso molecolare:266.23Ref: TM-T23509
2mg42,00€5mg64,00€10mg79,00€25mg118,00€50mg170,00€100mg235,00€200mg319,00€1mL*10mM (DMSO)71,00€(E/Z)-SIB-1893
CAS:(E/Z)-SIB-1893 (SIB 1893) is the racemate of (E)-SIB-1893 and (Z)-SIB-1893.Formula:C14H13NPurezza:99.96%Colore e forma:SolidPeso molecolare:195.26Agomelatine hydrochloride
CAS:Agomelatine HCl is a MT1/MT2 receptor agonist (Ki: 0.1-0.27 nM) and a 5-HT2C antagonist (pKi: 6.2-6.4).Formula:C15H18ClNO2Purezza:99.57%Colore e forma:SolidPeso molecolare:279.76Riluzole hydrochloride
CAS:Riluzole hydrochloride, an anticonvulsant Na+ channel blocker, inhibits GABA uptake (IC50: 43 µM).Formula:C8H6ClF3N2OSPurezza:99.76%Colore e forma:SolidPeso molecolare:270.66Suriclone
CAS:Suriclone (RP 31264), a cyclic pyrrolidone for anxiety, modulates GABA-A receptors without major sedation.Formula:C20H20ClN5O3S2Purezza:99.21% - 99.73%Colore e forma:SolidPeso molecolare:477.99NS-2710
CAS:NS-2710, a GABA receptor agonist, is used potentially for the treatment of anxiety.Formula:C22H20N4OPurezza:99.7% - 99.82%Colore e forma:SolidPeso molecolare:356.42Golexanolone
CAS:Golexanolone can be used to study neurological diseases.Formula:C21H31NO2Purezza:99.90% - 99.99%Colore e forma:SolidPeso molecolare:329.48GR 46611
CAS:GR 46611 is a selective 5-HT1B and 5-HT1D receptor agonist and can be used in studies about the treatment of epilepsy.Formula:C23H27N3O2Purezza:99.75%Colore e forma:SolidPeso molecolare:377.48Ecopipam
CAS:Ecopipam: orally active, selective dopamine D1/D5 antagonist (Ki: 1.2 nM/2.0 nM). 40x more selective over D2/D4/5-HT/α2a. For schizophrenia, obesity research.Formula:C19H20ClNOPurezza:99.68%Colore e forma:SolidPeso molecolare:313.82AZD6538
CAS:AZD6538 is an mGluR5 negative allosteric modulator used in the study of CNS-related diseases such as Alzheimer's disease.Formula:C15H6FN5OPurezza:98.68%Colore e forma:SolidPeso molecolare:291.24Femoxetine hydrochloride
CAS:Femoxetine hydrochloride is a selective 5-hydroxytryptamine reuptake inhibitor used in the study of migraine, depression and eating disorders.Formula:C20H26ClNO2Purezza:99.63%Colore e forma:SolidPeso molecolare:347.88Ricasetron
CAS:Ricasetron (Brl 46470) is a 5-HT3 receptor antagonist with pro-axonal lysing properties and is used in the study of anxiety disorders and anxiety disorders.Formula:C19H27N3OPurezza:99.52%Colore e forma:SolidPeso molecolare:313.44Ru-32514
CAS:Ru-32514 is a benzodiazepine receptor agonist.Formula:C18H17N3O2Purezza:99.21%Colore e forma:SolidPeso molecolare:307.35Divaplon
CAS:Divaplon is a GABA receptor agonist (IC50: 0.056 µM) that displays non-sedating anxiolytic behavioral characteristics in a rat model of anxiety.Formula:C17H17N3O2Purezza:97.44% - 98.25%Colore e forma:SolidPeso molecolare:295.345-HT2 antagonist 1
CAS:5-HT2 antagonist 1 is a potent 5-HT2 receptor antagonist, has weak α1 adrenoceptor blocking activity.Formula:C22H29FN4O2Purezza:99.76%Colore e forma:SolidPeso molecolare:400.49Ref: TM-T12597
1mg642,00€5mg1.288,00€10mg1.738,00€25mg2.583,00€50mg3.484,00€100mg4.708,00€1mL*10mM (DMSO)1.521,00€LRRK2-IN-7
CAS:LRRK2-IN-7: potent, selective CNS-active LRRK2 inhibitor, IC50 0.9 nM, >1000x selectivity vs kinases/channels/CYPs.Formula:C24H26N6OPurezza:99.26%Colore e forma:SolidPeso molecolare:414.5SCH-900271
CAS:SCH-900271 treats dyslipidemia by targeting nicotinic acid receptors, addressing hyperlipidaemia.Formula:C14H16N2O4Purezza:98.82% - 99.93%Colore e forma:SolidPeso molecolare:276.29Ref: TM-T34573
1mg112,00€5mg261,00€10mg396,00€25mg655,00€50mg888,00€100mg1.251,00€500mg2.493,00€1mL*10mM (DMSO)249,00€Valiglurax
CAS:Valiglurax (VU2957), potent mGlu4 PAM, crosses blood-brain barrier, orally available; promising for Parkinson's treatment.Formula:C16H10F3N5Purezza:98.29%Colore e forma:SolidPeso molecolare:329.28CBiPES hydrochloride
CAS:CBiPES hydrochloride (CBiPES HCl) is an orthosteric modulator of the mGlu2 receptor and is used to study neurological disorders like epilepsy.Formula:C21H20ClN3O2SPurezza:99.66%Colore e forma:SolidPeso molecolare:413.92Xanomeline oxalate
CAS:Xanomeline oxalate (LY246708), a potent SMRA, boosts phosphoinositide hydrolysis; key for Alzheimer's research.Formula:C16H25N3O5SPurezza:99.1%Colore e forma:SolidPeso molecolare:371.45Ref: TM-T13353
5mg35,00€10mg55,00€25mg100,00€50mg159,00€100mg245,00€200mg353,00€1mL*10mM (DMSO)39,00€Litoxetine
CAS:Litoxetine: a selective 5-HT inhibitor & 5-HT3 antagonist, used as an antidepressant with antiemetic effects, Ki=85 nM.Formula:C16H19NOPurezza:99.68%Colore e forma:SolidPeso molecolare:241.33Ref: TM-T67956
1mg92,00€5mg207,00€10mg309,00€25mg527,00€50mg755,00€100mg1.044,00€500mg2.088,00€1mL*10mM (DMSO)178,00€Cirsimaritin
CAS:Cirsimaritin has anti-bacterial, anti-inflammatory, anti-tumor, antioxidant effects, and protects kidneys; it weakly targets GABAA receptors.
Formula:C17H14O6Purezza:99.9%Colore e forma:SolidPeso molecolare:314.29Muscimol HBr
CAS:Muscimol HBr (Agarin HBr) is an agonist of GABAA receptor.Formula:C4H7BrN2O2Purezza:98.13%Colore e forma:Off-White PowderPeso molecolare:195.01Ref: TM-T20657
1mg113,00€2mg169,00€5mg240,00€10mg385,00€25mg622,00€50mg898,00€100mg1.198,00€500mg2.422,00€1mL*10mM (DMSO)205,00€Progabide
CAS:Progabide (SL 76002) is an agonist of the gamma-aminobutyric acid receptor.Formula:C17H16ClFN2O2Purezza:99.68%Colore e forma:SolidPeso molecolare:334.77Fananserin
CAS:Fananserin: Oral 5-HT2A antagonist (Ki=0.37 nM, rat), blocks human D4 receptor (Ki=2.93 nM).Formula:C23H24FN3O2SPurezza:99.88%Colore e forma:SolidPeso molecolare:425.52Ref: TM-T15270
2mg39,00€5mg52,00€10mg77,00€25mg110,00€50mg166,00€100mg236,00€200mg349,00€1mL*10mM (DMSO)58,00€Dipraglurant
CAS:Dipraglurant: a blood-brain permeable mGluR5 NAM, orally active, selective, IC50 = 21 nM, treats PD-LID.Formula:C16H12FN3Purezza:98.7%Colore e forma:SolidPeso molecolare:265.29Ref: TM-T15134
1mg92,00€5mg215,00€10mg313,00€25mg685,00€50mg1.009,00€100mg1.341,00€1mL*10mM (DMSO)260,00€Masupirdine free base
CAS:Masupirdine free base (SUVN-502 free base) is a 5-HT6 receptor antagonist that can be used to study neurological disorders like Alzheimer's disease.Formula:C21H24BrN3O3SPurezza:98.36% - 99.65%Colore e forma:SolidPeso molecolare:478.4PHA 543613
CAS:PHA 543613 is a specific agonist of α7 nAChR (Ki = 8.8 nM) and can be used in studies about the cognitive deficits of Alzheimer's disease and schizophrenia.Formula:C15H17N3O2Purezza:99.43% - 99.96%Colore e forma:SolidPeso molecolare:271.31Ref: TM-T23145
1mg52,00€5mg102,00€10mg166,00€25mg358,00€50mg610,00€100mg895,00€500mg1.945,00€1mL*10mM (DMSO)100,00€R 59-022 hydrochloride
CAS:R 59-022 hydrochloride is a 5-HT antagonist, PKC activator, DGK inhibitor (IC50: 2.8 µM), and modulates lipid production in platelets and neutrophils.
Formula:C27H27ClFN3OSPurezza:97.7%Colore e forma:SolidPeso molecolare:496.04RS 42358-197
CAS:RS 42358-197 (RS 25259-007) is a competitive 5-HT3 receptor antagonist.Formula:C19H23ClN2OPurezza:99.70%Colore e forma:SolidPeso molecolare:330.85Ref: TM-T20739
1mg158,00€5mg351,00€10mg527,00€25mg783,00€50mg1.054,00€100mg1.414,00€200mg1.908,00€1mL*10mM (DMSO)349,00€Tedatioxetine
CAS:Tedatioxetine (Lu AA24530) is a serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI) with antidepressant properties.Formula:C18H21NSPurezza:99.76% - >99.99%Colore e forma:SolidPeso molecolare:283.43Glutaminyl Cyclase Inhibitor 1
CAS:Glutaminyl Cyclase Inhibitor 1 is a glutaminyl cyclase inhibitor (IC50: 0.5 μM) that can be used to study neurological disorders.Formula:C21H24FN3O2Purezza:99.81%Colore e forma:SolidPeso molecolare:369.43Lecozotan HCl
CAS:Lecozotan HCl is a selective 5-HT antagonist boosting glutamate and acetylcholine release without causing 5-HT(1A) tolerance.
Formula:C28H30ClN5O3Purezza:99.04%Colore e forma:SolidPeso molecolare:520.02MK-3328
CAS:MK-3328, a potential Alzheimer's drug, binds β-Amyloid with strong affinity (IC50:10.5 nM) and may serve as a PET ligand to gauge plaque load.Formula:C14H9FN4OPurezza:99.77% - >99.99%Colore e forma:SolidPeso molecolare:268.25Ref: TM-T16094
1mg315,00€5mg745,00€10mg1.018,00€25mg1.431,00€50mg1.783,00€100mg2.250,00€500mg4.410,00€2-BFI hydrochloride
CAS:2-BFI hydrochloride: High-affinity I2 agonist; used in researching stroke and immune disease protection.Formula:C11H11ClN2OPurezza:99.94%Colore e forma:SolidPeso molecolare:222.67NKY80
CAS:NKY80 regulates the adenylyl cyclase catalytic activity in heart and lung tissues.Formula:C12H11N3O2Purezza:99.88%Colore e forma:SolidPeso molecolare:229.23Ref: TM-T16333
2mg44,00€5mg64,00€10mg90,00€25mg177,00€50mg309,00€100mg470,00€200mg677,00€1mL*10mM (DMSO)100,00€RS 67333 hydrochloride
CAS:RS 67333 hydrochloride is a selective 5-HT4R partial agonist (pKi=8.7) with neuroprotective properties for Alzheimer's research.Formula:C19H30Cl2N2O2Purezza:98.78%Colore e forma:SolidPeso molecolare:389.36Goxalapladib
CAS:Goxalapladib（GSK 677116） is a small molecule compound that can be used to treat cardiovascular risks associated with atherosclerosis.Formula:C40H39F5N4O3Purezza:99.64% - 99.93%Colore e forma:SolidPeso molecolare:718.75Teniloxazine
CAS:Teniloxazine is an orally available antidepressant compound with anti-hypoxic properties.Formula:C16H19NO2SPurezza:99.29%Colore e forma:SolidPeso molecolare:289.39CP-810123
CAS:CP-810123 is an α7 nAChR agonist used to treat cognitive deficits associated with psychiatric or neurological disorders such as schizophrenia.Formula:C14H18N4OPurezza:98.63% - 99.60%Colore e forma:SolidPeso molecolare:258.32Itasetron
CAS:Itasetron, a 5-HT3 antagonist, prevents memory loss in rats and has antiemetic effects in cancer treatments.
Formula:C16H20N4O2Purezza:98.58% - 99.33%Colore e forma:SolidPeso molecolare:300.36Ezeprogind disulfate
CAS:Ezeprogind disulfate: neurotrophic inducer targeting neurodegeneration causes like Abeta, tau; for neurological disorder research.Formula:C25H48N6O8S2Purezza:99.72%Colore e forma:SolidPeso molecolare:624.81NNC 05-711
CAS:NNC 05-711 (NO-711 hydrochloride) is a potent and selective inhibitor of GAT-1 (GABA transporter 1), exerting anticonvulsant and analgesic effects.Formula:C21H23ClN2O3Purezza:99.92%Colore e forma:SolidPeso molecolare:386.87CT-179
CAS:CT-179 is a potent and selective inhibitor of OLIG2, reduces tumor cell proliferation and induces apoptosis, fpr medulloblastoma and glioblastoma.Formula:C17H22Cl2N6OPurezza:98.67%Colore e forma:SolidPeso molecolare:397.3BL-1020 Mesylate
CAS:BL-1020 Mesylate (CYP-1020 Mesylate) is a GABA A receptor agonist and D2 antagonist used in studies of neurodegeneration.Formula:C28H45ClN4O11S4Purezza:>99.99%Colore e forma:SolidPeso molecolare:777.39Desformylflustrabromine hydrochloride
CAS:Desformylflustrabromine hydrochloride (dFBr hydrochloride) is a selective agonist of nicotinic acetylcholine receptor (nAChR) in α4β2 neurons, with pEC50 of 6.Formula:C17H12INO5Purezza:99.79%Colore e forma:SolidPeso molecolare:437.19Ref: TM-T11004
2mg34,00€5mg50,00€10mg80,00€25mg145,00€50mg225,00€100mg353,00€200mg550,00€1mL*10mM (DMSO)57,00€Adoprazine
CAS:Adoprazine (SLV313) is a potential atypical antipsychotic bearing potent D2 receptor antagonist and 5-HT1A receptor agonist properties.
Formula:C24H24FN3O2Purezza:99.83%Colore e forma:SolidPeso molecolare:405.46Aceclidine
CAS:Aceclidine (1-azabicyclo[2.2.2]octan-3-yl acetate) is a modulator of M3 mAChR and can be used in studies about treating glaucoma by reducing intraocularFormula:C9H15NO2Purezza:>99.99%Colore e forma:SolidPeso molecolare:169.22E6801
CAS:E6801: selective 5-HT6 agonist for research in dementia, Parkinson's, depression, obesity, epilepsy, anxiety, etc.Formula:C17H18ClN5O2S2Purezza:96.32% - 97.24%Colore e forma:SolidPeso molecolare:423.94DMCM hydrochloride
CAS:DMCM hydrochloride is a non-selective fully inverse agonist of benzodiazepine.Formula:C17H19ClN2O4Purezza:99.56%Colore e forma:SolidPeso molecolare:350.8Ref: TM-T11061
1mg34,00€2mg50,00€5mg80,00€10mg105,00€25mg236,00€50mg439,00€100mg620,00€1mL*10mM (DMSO)88,00€Cilansetron
CAS:Cilansetron is an effective and selective 5-HT3 receptor antagonist that can be used for related diseases caused by colitis.Formula:C20H21N3OPurezza:99.82% - 99.98%Colore e forma:SolidPeso molecolare:319.4DSP-0565
CAS:DSP-0565 is a broad-spectrum anti-epileptic with a high safety margin and effectiveness in several convulsant models.Formula:C14H12FNOPurezza:99.51% - 99.56%Colore e forma:SolidPeso molecolare:229.25Ref: TM-T11106
1mg109,00€2mg163,00€5mg241,00€10mg354,00€25mg532,00€50mg745,00€100mg1.018,00€500mg2.035,00€1mL*10mM (DMSO)208,00€Lirequinil
CAS:Lirequinil (Ro 41-3696) is a small molecule GABAA receptor agonist used to study neurological disorders.Formula:C26H25ClN2O3Purezza:98.54%Colore e forma:SolidPeso molecolare:448.94Ticalopride
CAS:Ticalopride: 5-HT3 agonist for digestive, orofacial, ENT disorders, and bulimia, GERD, IBS research.Formula:C14H20ClN3O3Purezza:99.51%Colore e forma:SolidPeso molecolare:313.78DA-6886
CAS:DA-6886 is a 5-HT4 agonist, relaxes rat oesophagus, with 1000x selectivity over hERG channels, pIC50: 4.3.Formula:C19H28Cl2N6O2Purezza:99.91% - 99.99%Colore e forma:SolidPeso molecolare:443.37L-838417
CAS:L-838417 is a GABAA receptor subtype-selective benzodiazepine site-selective ligand and GABAA receptor-positive modulator used in the study of anxiety disordersFormula:C19H19F2N7OPurezza:98.12% - 99.70%Colore e forma:SolidPeso molecolare:399.4Saripidem
CAS:Saripidem (SL-85.0274) is a compound with anxiolytic activity.Formula:C19H20ClN3OPurezza:98.42%Colore e forma:SolidPeso molecolare:341.83Alpidem
CAS:Alpidem (Ananxyl), a non-sedative imidazopyridine anxiolytic, treats anxiety with high benzodiazepine receptor affinity.Formula:C21H23Cl2N3OPurezza:99.56% - 99.97%Colore e forma:White To Off-White SolidPeso molecolare:404.33Ref: TM-T26600
1mg58,00€5mg137,00€10mg207,00€25mg371,00€50mg522,00€100mg747,00€500mg1.513,00€1mL*10mM (DMSO)122,00€CPCCOEt
CAS:CPCCOEt is a low affinity, selective, non-competitive and reversible antagonist of mGluR1bFormula:C13H13NO4Purezza:99.91%Colore e forma:SolidPeso molecolare:247.25AZD 9272
CAS:AZD 9272 is a brain-permeable mGluR5 antagonist for the study of gastroesophageal reflux.Formula:C14H6F2N4OPurezza:98.29%Colore e forma:SolidPeso molecolare:284.22amyloid P-IN-1
CAS:amyloid P-IN-1 can be used in studies about diseases with depletion of serum amyloid P components such as Alzheimer's disease, amyloidosis, osteoarthritis, andFormula:C30H44N2O14Purezza:99.76%Colore e forma:SolidPeso molecolare:656.68McN-A 343
CAS:McN-A 343: Selective M1 muscarinic agonist; reduces inflammation in colitis models.Formula:C14H18Cl2N2O2Purezza:99.65%Colore e forma:SolidPeso molecolare:317.21Aβ-IN-1
CAS:Aβ-IN-1 is a novel, potent and orally active γ-secretase modulator (GSM).Formula:C35H49NPurezza:99.1%Colore e forma:SoildPeso molecolare:483.77(Z)-Thiothixene
CAS:(Z)-Thiothixene (Thiothixene) is an antagonist of serotonergic receptor.
Formula:C23H29N3O2S2Purezza:99.21%Colore e forma:Yellow To Yellow With A Tan Cast PowderPeso molecolare:443.63PPI-1019
CAS:PPI-1019 is an APP (β-amyloid A4) inhibitor for the treatment of neurological disorders and the study of Alzheimer's disease (AD).Formula:C36H54N6O5Purezza:95.16% - 98.16%Colore e forma:SolidPeso molecolare:650.85LY266097 hydrochloride
CAS:LY266097 hydrochloride is a 5-HT2 antagonist with pKi of 7.7/9.8/7.6 for 5-HT2A/B/C, used in depression research.
Formula:C21H24Cl2N2O2Purezza:98.58%Colore e forma:SolidPeso molecolare:407.33CP 96021
CAS:"CP 96021 is an antagonist of 5-HT1/2 receptors, with anti-inflammatory and anti-ulcer effects for treating GI tract and asthma."
Formula:C29H21FN4OSPurezza:97.81% - 99.62%Colore e forma:SoildPeso molecolare:492.57MNI 137
CAS:MNI 137 is a negative allosteric modulator of mGlu2. MNI 137 inhibits glutamate-induced calcium mobilization with IC50s of 8.3 and 12.6 nM for human and rat.Formula:C15H9BrN4OPurezza:97.49%Colore e forma:SolidPeso molecolare:341.16Xanomeline
CAS:Xanomeline: orally active, M1/M4 selective activator for neurological disorders; promising in trials, crosses blood-brain barrier, liver metabolized.Formula:C14H23N3OSPurezza:99.61%Colore e forma:SolidPeso molecolare:281.42Otenzepad
CAS:Otenzepad (AF-DX 116) is a selective antagonist of M2 mAChR with IC50s of 386 nM and 640 nM for rat heart and rabbit peripheral lung.Formula:C24H31N5O2Purezza:99.79%Colore e forma:SolidPeso molecolare:421.54Ref: TM-T16411
1mg44,00€5mg79,00€10mg114,00€25mg222,00€50mg356,00€100mg572,00€200mg803,00€1mL*10mM (DMSO)87,00€Oxotremorine M iodide
CAS:Oxotremorine M iodide (Oxotremorine methiodide) is an agonist of mAChR and potentiates NMDA receptors.Formula:C11H19IN2OPurezza:99.57%Colore e forma:SolidPeso molecolare:322.19ASM-024
CAS:ASM-024, a synthetic piperazine, activates nicotinic and β2-adrenergic receptors for potential asthma and bronchitis treatment with anti-inflammatory effects.Formula:C15H25N2Purezza:99.74%Colore e forma:SolidPeso molecolare:233.37Panadiplon
CAS:Panadiplon (FG 10571) is a selective gamma-aminobutyric acid receptor agonist and partial agonist of 5GABAA, a benzodiazepine receptor, used in the treatment ofFormula:C18H17N5O2Purezza:98.30% - 98.94%Colore e forma:SolidPeso molecolare:335.36Faxeladol
CAS:Faxeladol: adrenergic, serotonin inhibitor & opioid agonist for neurological studies.Formula:C15H23NOPurezza:98.77% - 99.67%Colore e forma:SolidPeso molecolare:233.35ADR-851 free base
CAS:ADR-851 free base is an antagonist of the HT3 receptor.Formula:C14H18ClN3O2Purezza:97.88% - 98.39%Colore e forma:SolidPeso molecolare:295.77BI-1408
CAS:BI-1408 is a modulator potent of γ secretase (IC50: 0.04 μM for Aβ42).Formula:C22H23FN6Purezza:99.63%Colore e forma:SolidPeso molecolare:390.46RWJ-51204
CAS:RWJ-51204: potent adenosine A2A blocker, GABA(A) partial agonist (IC50: 0.2-2 nM), neuroprotective, may treat Parkinson's.
Formula:C21H19F2N3O3Purezza:99.57% - 99.95%Colore e forma:SolidPeso molecolare:399.39Ref: TM-T16811
1mg333,00€5mg787,00€10mg1.074,00€25mg1.510,00€50mg1.882,00€100mg2.375,00€500mg4.655,00€Cianopramine
CAS:Cianopramine (Ro 112465) is a selective 5-hydroxytryptamine uptake inhibitor and a tricyclic antidepressant used in the study of neurological disorders.Formula:C20H23N3Purezza:99.92% - 99.92%Colore e forma:SolidPeso molecolare:305.42LY-2624803
CAS:LY-2624803 is a 5-HT2A receptor antagonist and histamine receptor inverse agonist that can be used to improve slow wave sleep.Formula:C22H25N3O3Purezza:99.78% - 99.97%Colore e forma:SolidPeso molecolare:379.45Quinupramine
CAS:Quinupramine: an oral antidepressant targeting the serotonin system; penetrates CNS; doesn’t affect β-adrenergic system.Formula:C21H24N2Purezza:99.77%Colore e forma:SolidPeso molecolare:304.43ELB-139
CAS:ELB-139 is a GABA A receptor agonist. ELB139 increases 5-HT in the striatum and prefrontal cortex of rats.Formula:C14H16ClN3OPurezza:>99.99%Colore e forma:SolidPeso molecolare:277.75cis-Urocanic acid
CAS:cis-Urocanic acid ((E)-Urocanic acid) is a 5-HT2A receptor agonist (Kd: 4.6 nM).Formula:C6H6N2O2Purezza:99.81%Colore e forma:SolidPeso molecolare:138.12AQW051
CAS:AQW051 (VQW-765) is an oral α7-nAChR activator for cognitive impairments, used in anxiety disorder studies.Formula:C19H22N2OPurezza:99.94%Colore e forma:SolidPeso molecolare:294.39Ref: TM-T26646
1mg34,00€2mg46,00€5mg66,00€10mg99,00€25mg205,00€50mg313,00€100mg439,00€500mg954,00€1mL*10mM (DMSO)67,00€8-OH-Dpat
CAS:8-OH-Dpat (8-Hydroxy-DPAT) is a serotonin 1A-receptor agonist that is used experimentally to test the effects of serotonin.Formula:C16H25NOPurezza:98%Colore e forma:SolidPeso molecolare:247.38SB-215505
CAS:SB215505: potent 5-HT2B/2C blocker, enhances rat wakefulness/motor activity. (pKi: 5-HT2B - 8.3, 5-HT2C - 7.66, 5-HT2A - 6.77).Formula:C19H16ClN3OPurezza:98.33%Colore e forma:SolidPeso molecolare:337.8Piromelatine
CAS:Piromelatine is an agonist of melatonin MT1/MT2 receptors, 5-HT1A and 5-HT1D, and an antagonist of 5-HT2B.Piromelatine has antinociceptive activity withFormula:C17H16N2O4Purezza:99.83%Colore e forma:SolidPeso molecolare:312.32Ref: TM-T34081
1mg60,00€5mg130,00€10mg178,00€25mg334,00€50mg522,00€100mg713,00€1mL*10mM (DMSO)142,00€ML 10302 hydrochloride
CAS:ML 10302 hydrochloride is a specific agonist 5-HT4 and binds 5-HT receptors with Kis of 1.07 nM and 782 nM for 5-HT4 and 5-HT3.Formula:C15H22Cl2N2O3Purezza:99.99%Colore e forma:SolidPeso molecolare:349.25Buntanetap
CAS:Buntanetap ((+)-Phenserine) is an inhibitor of TINAPs used in the study of neurological disorders, endocrine and metabolic disorders, and cardiovascular diseaseFormula:C20H23N3O2Purezza:98.2%Colore e forma:SolidPeso molecolare:337.42Ref: TM-T17312
1mg177,00€5mg447,00€10mg713,00€25mg1.333,00€50mg1.935,00€100mg2.520,00€1mL*10mM (DMSO)492,00€Viloxazine
CAS:Viloxazine (Viloxazin) (Viloxazin) is a dual-action compound that functions as a norepinephrine reuptake inhibitor and exhibits potent agonistic activityFormula:C13H19NO3Purezza:99.65%Colore e forma:SolidPeso molecolare:237.295-HT6/7 antagonist 1
CAS:5-HT6/7 antagonist 1 is a dual 5-HT6/7/2A and D2 receptor antagonist for the study of dementia and Alzheimer's disease.
Formula:C22H20FN3O3Purezza:98.78% - 99.26%Colore e forma:SolidPeso molecolare:393.41Roxindole
CAS:Roxindole: dopamine agonist, serotonin reuptake inhibitor, 5-HT1A agonist, developed for schizophrenia.Formula:C23H26N2OPurezza:98.03% - 98.93%Colore e forma:SolidPeso molecolare:346.47SB228357
CAS:SB228357 is a potent and selective antagonist of the 5-HT receptor with pKis of 6.9, 8.0, and 9.0 for 5-HT2A, 5-HT2B, and 5-HT2C, respectively.Formula:C22H17F4N3O2Purezza:99.82%Colore e forma:SolidPeso molecolare:431.38Fengabine
CAS:Fengabine (SL-79229) is a GABA receptor agonist with antidepressant activity and is used to treat depression.Formula:C17H17Cl2NOPurezza:99.37%Colore e forma:SolidPeso molecolare:322.235HT6-ligand-1
CAS:5HT6-ligand-1 is an orally active ligand of 5-HT6 receptor (Ki = 1.43 nM).Formula:C20H22BrN3O2SPurezza:99.24% - 99.93%Colore e forma:SolidPeso molecolare:448.38Cyamemazine
CAS:Cyamemazine is an antipsychotic compound with sedative and anxiolytic activity.Cyamemazine is a 5-HT3, 5-HT2A, and 5-HT2C receptor antagonist.Formula:C19H21N3SPurezza:97.01%Colore e forma:SolidPeso molecolare:323.46Tiospirone
CAS:Tiospirone (BMY 13859-1 free base) is a 5-HT2 receptor antagonist and a dopamine blocker used in the study of neurological disorders such as schizophrenia.Formula:C24H32N4O2SPurezza:99.74%Colore e forma:SolidPeso molecolare:440.6Ref: TM-T24885
1mg123,00€5mg293,00€10mg537,00€25mg863,00€50mg1.161,00€100mg1.558,00€1mL*10mM (DMSO)354,00€Perphenazine dihydrochloride
CAS:Perphenazine dihydrochloride: Oral dopamine, histamine-1 antagonist; targets D2, D3, 5-HT2A, Alpha-1A; may treat psychiatric disorders, cancer.Formula:C21H28Cl3N3OSPurezza:99.67%Colore e forma:SolidPeso molecolare:476.89GSK233705
CAS:GSK233705, a muscarinic antagonist, is used to prevent/treat COPD and asthma.Formula:C24H29BrN2Purezza:99.87% - 99.98%Colore e forma:SolidPeso molecolare:425.4Liafensine
CAS:Liafensine(BMS-820836): Selective inhibitor for serotonin, norepinephrine, dopamine reuptake; targets major depression, CNS disorders.Formula:C24H22N4Purezza:99.91%Colore e forma:SolidPeso molecolare:366.46NB001
CAS:NB001 (HTS 09836) is an inhibitor of adenyl cyclase 1 exhibiting effects on neural and non-neural pain.Formula:C12H20N6OPurezza:99.69%Colore e forma:Off-White To Pale Pink SolidPeso molecolare:264.33Ref: TM-T16275
1mg74,00€5mg200,00€10mg295,00€25mg497,00€50mg710,00€100mg964,00€500mg1.935,00€1mL*10mM (DMSO)173,00€Iperoxo
CAS:Iperoxo (Iperoxo iodide) is an agonist of Muscarinic AChR and can be used to probe activation-related conformational transitions of muscarinic receptors.Formula:C10H17IN2O2Purezza:99.81%Colore e forma:SolidPeso molecolare:324.16Ref: TM-T25538
1mg50,00€5mg106,00€10mg168,00€25mg339,00€50mg512,00€100mg748,00€200mg1.026,00€1mL*10mM (DMSO)117,00€SPD-473 citrate
CAS:SPD-473 citrate is an inhibitior of serotonin/dopamine/norepinephrine reuptake.Formula:C23H31Cl2NO8SPurezza:99.37%Colore e forma:SolidPeso molecolare:552.47ATC 0175
CAS:ATC 0175 hydrochloride is an orally active melanocyte concentrating hormone 1 receptor antagonist that is potent and selective.Formula:C23H26ClF2N5OPurezza:99.98%Colore e forma:SolidPeso molecolare:461.93ALX-1393
CAS:ALX-1393 is a selective GlyT2 inhibitor that effectively reduces neuronal action potential activity in a concentration-dependent manner and inhibits theFormula:C23H22FNO4Purezza:99.83%Colore e forma:SolidPeso molecolare:395.42Ref: TM-T14198
1mg1.243,00€5mg2.520,00€10mg3.402,00€25mg5.059,00€50mg6.832,00€100mg8.883,00€1mL*10mM (DMSO)2.592,00€BPDBA
CAS:BPDBA is an effective, selective, and non-competitive inhibitor of the betaine/GABA transporter (BGT-1), displaying inhibitory activity against human BGT-1 andFormula:C19H20Cl2N2OPurezza:99.43% - 99.95%Colore e forma:SolidPeso molecolare:363.28Nexopamil
CAS:Nexopamil (LU-49938) is a dual calcium channel and 5-HT2A receptor antagonist that inhibits cell contraction and growth.
Formula:C24H40N2O3Purezza:97.87% - >99.99%Colore e forma:SolidPeso molecolare:404.59BMY-14802 hydrochloride
CAS:BMY-14802 hydrochloride (BMS 181100 hydrochloride) is a selective antagonist of σ receptor (IC50 = 112 nM) with antipsychotic effects.Formula:C18H23ClF2N4OPurezza:99.97%Colore e forma:SolidPeso molecolare:384.85Nerisopam
CAS:Nerisopam is an agonist of gamma-aminobutyric acid (GABA) receptor.Formula:C18H19N3O2Purezza:98.52%Colore e forma:SolidPeso molecolare:309.36Ref: TM-T28159
1mg88,00€5mg190,00€10mg286,00€25mg464,00€50mg672,00€100mg945,00€200mg1.279,00€1mL*10mM (DMSO)256,00€Aplindore Fumarate
CAS:Aplindore Fumarate (DAB-452), a selective dopamine D2/D3 partial agonist, is used in Parkinson's and schizophrenia research.Formula:C22H22N2O7Purezza:99.66%Colore e forma:SolidPeso molecolare:426.42Pimethixene maleate
CAS:Pimethixene maleate (Pimetixene maleate) is a 5-HT2B receptor antagonist with sedative activity that can be used to study dry cough in children.Formula:C23H23NO4SPurezza:99.55%Colore e forma:SolidPeso molecolare:409.55-HT1A modulator 1
CAS:5-HT1A modulator 1 displays very high affinities for the 5-HT1A, α1-adrenergic receptor, and D2 receptor (IC50s = 2 nM, 10 nM, and 40 nM).Formula:C21H25N3O2SPurezza:99.68%Colore e forma:SolidPeso molecolare:383.51Sudoxicam
CAS:Sudoxicam (4-Hydroxy-2-methyl-N-2-thiazolyl-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxide) is a reversible antagonist of COX with anti-inflammatory, anti-edema
Formula:C13H11N3O4S2Purezza:99.93%Colore e forma:SolidPeso molecolare:337.37LSN2463359
CAS:LSN2463359 is a positive allosteric modulators of the mGlu5 receptor.Formula:C16H15N3OPurezza:99.26%Colore e forma:SolidPeso molecolare:265.31Ref: TM-T27854
2mg34,00€5mg50,00€10mg80,00€25mg161,00€50mg245,00€100mg363,00€200mg515,00€1mL*10mM (DMSO)55,00€H-9 dihydrochloride
CAS:H-9 dihydrochloride: Strong PKA inhibitor, curbs 5-HT response and EGF signaling, affects pharyngeal function.Formula:C11H15Cl2N3O2SPurezza:97.3%Colore e forma:SolidPeso molecolare:324.23SB 699551 dihydrochloride
CAS:SB 699551 dihydrochloride is a 5-ht5a receptor antagonist.Formula:C34H47Cl2N3OPurezza:99.83%Colore e forma:SolidPeso molecolare:584.66Ref: TM-T23325
1mg50,00€5mg105,00€10mg170,00€25mg295,00€50mg424,00€100mg583,00€1mL*10mM (DMSO)142,00€Lensiprazine
CAS:Lensiprazine (SLV314) is a potent dopamine D(2) receptor antagonist that acts as a serotonin reuptake inhibitor , and can be used to study bipolar disorder andFormula:C24H27FN4O2Purezza:97.86%Colore e forma:SolidPeso molecolare:422.5Lesopitron
CAS:Lesopitron: anxiolytic, 5-HT1A agonist, treats rodent anxiety, counters benzodiazepine withdrawal, low toxicity, no alcohol/barbiturate interaction.Formula:C15H21ClN6Purezza:99.33% - 99.46%Colore e forma:SolidPeso molecolare:320.82Ref: TM-T25672
1mg133,00€5mg324,00€10mg477,00€25mg773,00€50mg1.063,00€100mg1.431,00€500mg2.872,00€1mL*10mM (DMSO)323,00€Landipirdine
CAS:Landipirdine (RO-5025181) is a selective 5-HT6R antagonist for the study of central nervous system disorders such as dementia.Formula:C18H19FN2O3SPurezza:97.61% - 99.99%Colore e forma:SolidPeso molecolare:362.42PF-03635659
CAS:PF-03635659: potent M3 antagonist, Ki=0.2 nM, long half-life, potential COPD treatment.Formula:C28H32N2O3Purezza:98.39% - 99.85%Colore e forma:SolidPeso molecolare:444.57Ref: TM-T33941
1mg216,00€5mg532,00€10mg758,00€25mg1.153,00€50mg1.558,00€100mg2.097,00€500mg4.204,00€1mL*10mM (DMSO)605,00€Anpirtoline hydrochloride
CAS:Anpirtoline hydrochloride (D-16949 hydrochloride) is a 5-HT1B receptor agonist and 5-HT3 receptor antagonist used in the study of dyskinesia.Formula:C10H14Cl2N2SPurezza:>99.99% - >99.99%Colore e forma:SolidPeso molecolare:265.20Felcisetrag
CAS:Felcisetrag (TD-8954), an oral 5-HT4 agonist with GI prokinetic effects, has a high affinity (pKi 9.4) for h5-HT4(c) receptors.Formula:C25H37N5O3Purezza:99.99%Colore e forma:SolidPeso molecolare:455.59Ref: TM-T28934
1mg87,00€5mg215,00€10mg318,00€25mg510,00€50mg692,00€100mg928,00€200mg1.251,00€1mL*10mM (DMSO)235,00€Rilapine
CAS:Rilapine (Rilapinum) is an antipsychotic compound that shows high affinity for 5-HT6 receptors and can be used to study neurological disorders.Formula:C22H20ClN3Purezza:97.76% - 99.20%Colore e forma:SolidPeso molecolare:361.87PNU-282987 free base
CAS:PNU-282987 is an α7 nAChR agonist (EC50=154 nM) and a 5-HT3 antagonist (IC50=4541 nM) for nervous system research.
Formula:C14H17ClN2OPurezza:99.64%Colore e forma:SolidPeso molecolare:264.75MM 77 dihydrochloride
CAS:MM 77 dihydrochloride is an effecitve 5-HT1A receptor postsynaptic antagonist with anxiolytic-like activity.Formula:C19H29Cl2N3O3Purezza:99.91%Colore e forma:SolidPeso molecolare:418.36Ref: TM-T23007
1mg86,00€5mg157,00€10mg215,00€25mg472,00€50mg687,00€100mg938,00€500mg1.882,00€1mL*10mM (DMSO)281,00€MAO-B-IN-9
CAS:MAO-B-IN-9 is a monoamine oxidase B MAO-B inhibitor (IC50: 0.18 μM) that crosses the blood-brain barrier with potency, selectivity and time-dependence.Formula:C18H24N2O2Purezza:99.93%Colore e forma:SolidPeso molecolare:300.4Ref: TM-T60671
2mg39,00€5mg58,00€10mg93,00€25mg167,00€50mg260,00€100mg378,00€200mg552,00€1mL*10mM (DMSO)66,00€LY 272015 hydrochloride
CAS:LY 272015 hydrochloride is a 5-HT2B receptor antagonist.Formula:C21H25ClN2O2Purezza:99.47%Colore e forma:SolidPeso molecolare:372.89Sarizotan HCl
CAS:Sarizotan HCl (EMD 128130 HCl) is a 5-HT1A receptor and dopamine receptor agonist and an hERG channel inhibitor used in Parkinson;s disease research.Formula:C22H22ClFN2OPurezza:96%Colore e forma:SolidPeso molecolare:384.87Sarmazenil
CAS:Sarmazenil (Ro 15-3505) is a partial inverse agonist at the benzodiazepine receptor and is used in the study of chronic hepatic encephalopathy.Formula:C15H14ClN3O3Purezza:99.46%Colore e forma:SolidPeso molecolare:319.74Lenumlostat
CAS:Lenumlostat is a lysyl oxidase-like protein 2 (LOXL2) inhibitor with inhibitory effects on hLOXL2, hLOXL3 and LOXL2 for the study of fibrotic diseases.Formula:C18H17F4N3O3Purezza:99.11%Colore e forma:SolidPeso molecolare:399.34Ref: TM-T69913
1mg177,00€5mg447,00€10mg672,00€25mg1.341,00€50mg2.088,00€100mg2.988,00€500mg6.004,00€1mL*10mM (DMSO)492,00€PAT-1251
CAS:PAT-1251 is an inhibitor of LOXL2 with IC50s of 10, 0.12, and 0.16 μM for the mouse, rat, and dog and can be used in studies about fibrotic diseases.Formula:C18H17F4N3O3Purezza:97.27% - 97.30%Colore e forma:SolidPeso molecolare:399.34Ref: TM-T12371L
1mg72,00€5mg158,00€10mg243,00€25mg389,00€50mg542,00€100mg762,00€200mg1.017,00€1mL*10mM (DMSO)167,00€Repinotan
CAS:Repinotan (BAY x 3702 free base) is a 5-HT1A receptor agonist used in acute ischemic stroke studies.Formula:C21H24N2O4SPurezza:99%Colore e forma:SolidPeso molecolare:400.49ABP688
CAS:ABP688 is a non-competitive and selective mGluR5 antagonist(Ki = 1.7 nM). ABP688 can be used as a PET tracer for clinical imaging.Formula:C15H16N2OPurezza:98.63%Colore e forma:SolidPeso molecolare:240.3BMS-983970
CAS:BMS-983970 is an oral inhibitor of pan-Notch, and for the treatment of multiplecancers.Formula:C26H26F4N4O3Colore e forma:SolidPeso molecolare:518.5YM348
CAS:YM348 is an effective and orally active 5-HT2C receptor agonist. YM348 also shows a high affinity for the cloned human 5-HT2C receptor (Ki: 0.89 nM).Formula:C14H17N3OPurezza:98%Colore e forma:SolidPeso molecolare:243.3MAO-B-IN-27
CAS:MAO-B-IN-27 (Compound 12c), a monoamine oxidase B (MAO-B) inhibitor, exhibits a potent and selective inhibitory effect on hMAO-B, with an IC50 value of 8.9 nM,Formula:C16H17ClF3NOPurezza:98%Colore e forma:SolidPeso molecolare:331.764-Chloro-L-phenylalanine
CAS:4-Chloro-L-phenalanine (L-PCPA) is an inhibitor of 5-HT biosynthesis and a non-specific antagonist of tryptophan hydroxylases (TPH1 and TPH2).Formula:C9H10ClNO2Purezza:99.76% - 99.96%Colore e forma:SolidPeso molecolare:199.635-HT2C agonist-3
CAS:5-HT2C agonist-3 ((+)-19), a selective 5-HT2C agonist (EC 50: 24 nM, Ki: 78 nM), exhibits antipsychotic-like activity by blocking amphetamine-inducedFormula:C19H23ClFNO2Purezza:98%Colore e forma:SolidPeso molecolare:351.84(S)-Bexicaserin
CAS:(S)-Bexcaserin (compound 2) serves as a 5-HT2C receptor agonist, presenting research possibilities in obesity and psychiatric disorders [1].Formula:C15H19F2N3OPurezza:98%Colore e forma:SolidPeso molecolare:295.33Wf-516
CAS:Wf-516 is a 5-HT reuptake inhibitor (Kis: 5 nM and 40 nM for 5-HT1A receptor and 5-HT2A receptor in humans, respectively), and with potent antidepressantFormula:C25H25Cl2N3O4Purezza:98%Colore e forma:SolidPeso molecolare:502.395-HT2A&5-HT2C agonist-1
CAS:5-HT2A&5-HT2C agonist-1 (Example 2) is a dual-acting agent targeting the 5-HT2A and 5-HT2C receptors with respective IC50 values of 196 nM and 0.9 nM.Formula:C14H20N2OPurezza:98%Colore e forma:SolidPeso molecolare:232.32NCS-382 sodium
CAS:NCS-382 (sodium) is a potent antagonist of the GABA receptor, exhibiting anti-sedative and anti-hypnotic properties, with applications in neurological diseaseFormula:C13H13NaO3Purezza:98%Colore e forma:SolidPeso molecolare:240.23MAO-B-IN-19
CAS:MAO-B-IN-19, a selective MAO-B inhibitor, exhibits neuroprotective and anti-inflammatory properties and demonstrates an IC50 value of 0.67 μM [1].Formula:C15H11FO2Purezza:98%Colore e forma:SolidPeso molecolare:242.255-HT2A receptor agonist-3
CAS:5-HT2A receptor agonist-3 represents the highest selectivity for the human 5-HT2A receptor currently identified, exhibiting a K i of 2.5 nM.Formula:C21H26BrNO3Purezza:98%Colore e forma:SolidPeso molecolare:420.34MAO-IN-3
CAS:MAO-IN-3 (Compound 5), a reversible and competitive monoamine oxidase (MAO) inhibitor with inhibition constants (K i) of 0.6 μM for MAO A and 0.2 μM for MAO B,Formula:C42H54N4O4Purezza:98%Colore e forma:SolidPeso molecolare:678.9JNJ-46281222
CAS:JNJ-46281222: mGlu2-selective, potent PAM, Kd = 1.7 nM, pEC50 = 7.71.Formula:C23H25F3N4Colore e forma:SolidPeso molecolare:414.47BACE1-IN-13
CAS:BACE1-IN-13 (Compound 36), an orally active inhibitor of BACE1, exhibits high potency with an IC50 of 2.9 nM and demonstrates greater efficacy in hAβ42 cells (Formula:C20H17FN8O2Purezza:98%Colore e forma:SolidPeso molecolare:420.4Osemozotan Free Base
CAS:Osemozotan Free Base is a 5-HT(1A) receptor agonist.Formula:C19H21NO5Colore e forma:SolidPeso molecolare:343.37mGAT3/4-IN-2
CAS:mGAT3/4-IN-2 are potent inhibitors of mGAT3/mGAT4 with their pIC50 values of 5.44 and 5.25, respectively.Formula:C26H32ClN3OS2Colore e forma:SolidPeso molecolare:502.13VU6005649
CAS:VU6005649 is an agonist of CNS penetrant mGlu7/8 receptor (EC50s: 0.65 μM and 2.6 μM for mGlu7 receptor and mGlu8 receptor, respectively).Formula:C16H12F5N3OPurezza:99.87%Colore e forma:SolidPeso molecolare:357.28AAK1-IN-5
CAS:AAK1-IN-5: Potent, selective AAK1 inhibitor; CNS-penetrant; oral; IC50: 1.2 nM; Ki: 0.05 nM; cell IC50: 0.5 nM. Useful in neuropathic pain research.Formula:C19H23F4N3OColore e forma:SolidPeso molecolare:385.4(S)-Renzapride
(S)-Renzapride (BRL 24924), 5-HT4 agonist (Ki 115 nM), 5HT2b/5HT3 antagonist, for C-IBS study.Formula:C16H22ClN3O2Colore e forma:SolidPeso molecolare:323.82Octahydroaminoacridine succinate
CAS:Octahydroaminoacridine succinate, an acetylcholinesterase inhibitor, is used potentially for the treatment of Alzheimer's disease.Formula:C17H24N2O4Purezza:99.91%Colore e forma:SolidPeso molecolare:320.38BT-GSI
BT-GSI: γ-secretase inhibitor targeting Notch, anti-myeloma & anti-resorptive for multiple myeloma/bone disease research.Formula:C26H46BrN5O10P2Colore e forma:SolidPeso molecolare:730.52Biphenylindanone A
CAS:Biphenylindanone A is a selective potentiator of human mGluR2 (hmGluR2),and for the treatment of neurological disorders.Formula:C30H30O4Purezza:98%Colore e forma:SolidPeso molecolare:454.56eeAChE-IN-2
CAS:eeAChE-IN-2 is a potent inhibitor of eeAChE, exhibiting inhibitory potency with an IC50 of 2 nM.Formula:C37H40N8O5SColore e forma:SolidPeso molecolare:708.83FGIN-1-27
CAS:FGIN-1-27 is a high-affinity agonist of the translocator protein and a specific peripheral benzodiazepine receptor (PBR) ligand(Ki = 5.0 nM).Formula:C28H37FN2OPurezza:99.86%Colore e forma:SolidPeso molecolare:436.6GR-127935
CAS:GR-127935 is a potent and selective 5-HT1B/1D receptor antagonist.Formula:C29H31N5O3Colore e forma:SolidPeso molecolare:497.59Quinolactacin A1
CAS:Quinolactacin A1, a strong AChE inhibitor from Penicillium citrinum, aids Alzheimer's research.Formula:C16H18N2O2Colore e forma:SolidPeso molecolare:270.33BMS-933043
CAS:BMS-933043: α7 nAChR partial agonist, binds rat (Ki=3.3 nM) & human (Ki=8.1 nM), agonist with EC50=23.4 nM (calcium assay), 0.14-0.29 μM (electrophysiology).Formula:C16H19N7OPurezza:98%Colore e forma:SolidPeso molecolare:325.375-HT3 antagonist 1
CAS:5-HT3 antagonist 1 is a potent and selective antagonist of 5-HT3 receptor.Formula:C22H27N5OPurezza:98%Colore e forma:SolidPeso molecolare:377.48ABT-418 hydrochloride
CAS:ABT-418 HCl enhances cognition and reduces anxiety as a selective nAChRs agonist, researched for Alzheimer's.Formula:C9H15ClN2OColore e forma:SolidPeso molecolare:202.68Dothiepin
CAS:Dothiepin (Dosulepin; Dothep), an antidepressant with sedative/anxiolytic properties, preferentially inhibits noradrenaline over serotonin uptake, enhancingFormula:C19H21NSPurezza:98%Colore e forma:SolidPeso molecolare:295.44QM-FN-SO3
CAS:QM-FN-SO3 is a blood-brain barrier (BBB)-penetrable, near-infrared (NIR) probe with aggregation-induced emission (AIE) activity, specifically designed for the detection of Aβ plaques. It exhibits ultra-high signal-to-noise (S/N) ratio, binding affinity, and high-performance NIR emission, making it suitable for in vivo detection of Aβ plaques [1].Formula:C29H25N4NaO3S2Colore e forma:SolidPeso molecolare:564.65LY108742
CAS:LY108742 is an antagonist of 5-HT2.Formula:C21H28N2O3Purezza:98%Colore e forma:SolidPeso molecolare:356.46AMG-8718
CAS:AMG-8718, an oral BACE1 blocker (IC50: 0.0007 μM), also inhibits BACE2 (IC50: 0.005 μM), lowering CSF and Aβ40 brain levels.Formula:C25H19FN4O3Colore e forma:SolidPeso molecolare:442.44BMS 433796
CAS:BMS 433796 is a γ-secretase inhibitor that demonstrates Aβ-lowering activity within a transgenic mouse model of Alzheimer's disease.Formula:C21H20F2N4O4Purezza:99.17%Colore e forma:SolidPeso molecolare:430.4Befiradol
CAS:Befiradol (NLX-112) is an agonist of 5-HT1A receptor.Formula:C20H22ClF2N3OColore e forma:SolidPeso molecolare:393.86UNC9994
CAS:UNC9994 is a β-arrestin-biased dopamine D₂ receptor agonist (β-arrestin EC50 = 50 nM; Emax = 97%) with robust in vivo antipsychotic drug-like activities.Formula:C21H22Cl2N2OSColore e forma:SolidPeso molecolare:421.38Zamifenacin fumarate
CAS:Zamifenacin fumarate (UK-76654 fumarate) is a potent and gut-selective antagonist of muscarinic M3 receptor.Formula:C31H33NO7Purezza:99.88%Colore e forma:SolidPeso molecolare:531.6Ref: TM-T13385
2mg34,00€5mg50,00€10mg75,00€25mg128,00€50mg200,00€100mg304,00€200mg424,00€1mL*10mM (DMSO)58,00€5-HT3-In-1
CAS:5-HT3-In-1 (compound example 8) exhabits with 5-HT3 inhibition activity.Formula:C16H21ClN4O3Purezza:98%Colore e forma:SolidPeso molecolare:352.82Muscarine tosylate
CAS:Muscarine ((+)-Muscarine) tosylate, a prototype mAChR agonist, serves as a parasympathetic nervous system stimulant and is recognized for its toxic properties [1] [2].Formula:C16H27NO5SColore e forma:SolidPeso molecolare:345.45R-96544
CAS:R-96544 is an orally active antagonist of the 5-HT2A receptor that has demonstrated the ability to inhibit platelet aggregation in vitro [1].Formula:C22H30ClNO3Colore e forma:SolidPeso molecolare:391.93NAS-181
CAS:NAS-181 is a potent and selective rat 5-hydroxytryptamine 1B (r5-HT1B) antagonist (Ki: 47 nM).NAS-181 enhances the accumulation of 5-HTP in rat brain regions.Formula:C20H30N2O7SColore e forma:SolidPeso molecolare:442.53PZ-II-029
CAS:PZ-II-029 is a modulator of α6β3γ2-selective GABAA channel.Formula:C18H15N3O3Purezza:99.79%Colore e forma:SolidPeso molecolare:321.33Ref: TM-T28479
1mg50,00€5mg105,00€10mg167,00€25mg289,00€50mg447,00€100mg685,00€500mg1.378,00€1mL*10mM (DMSO)192,00€SB 649915
CAS:SB 649915 is a serotonin reuptake inhibitor and 5-HT1A and 5-HT1B receptor antagonist.Formula:C26H29N3O3Colore e forma:SolidPeso molecolare:431.53
