
recettore 5-HT
I recettori 5-HT, noti anche come recettori della serotonina, sono un gruppo di recettori accoppiati alle proteine G (GPCR) che mediano gli effetti della serotonina, un neurotrasmettitore coinvolto nella regolazione dell'umore, dell'ansia, del sonno, dell'appetito e di altri processi fisiologici. Questi recettori sono suddivisi in diversi sottotipi, ciascuno con funzioni e proprietà farmacologiche distinte. I modulatori dei recettori 5-HT sono ampiamente studiati per il loro ruolo nel trattamento della depressione, dei disturbi d'ansia e di altre condizioni neuropsichiatriche. Presso CymitQuimica, offriamo una gamma di modulatori dei recettori 5-HT di alta qualità per supportare la tua ricerca in neurofarmacologia, disturbi dell'umore e segnalazione GPCR.
Trovati 1025 prodotti di "recettore 5-HT"
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Ondansetron
CAS:Ondansetron (GR 38032) is a serotonin 5-HT3 receptor antagonist used mainly as an antiemetic.Formula:C18H19N3OPurezza:99.92%Colore e forma:White To Yellow CrystalsPeso molecolare:293.368-Hydroxy-DPAT hydrobromide
CAS:8-Hydroxy-DPAT hydrobromide (8-OH-DPAT hydrobromide) (8-OH-DPAT hydrobromide) is a potent and selective 5-HT1A agonist with a pIC50 of 8.19.Formula:C16H26BrNOPurezza:98.90% - 99.96%Colore e forma:SolidPeso molecolare:328.292'-O-Methylisoliquiritigenin
CAS:2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-Formula:C16H14O4Purezza:98.75%Colore e forma:SolidPeso molecolare:270.28Ref: TM-TN1217
1mg109,00€5mg260,00€10mg432,00€25mg692,00€50mgPrezzo su richiesta1mL*10mM (DMSO)358,00€Escitalopram Oxalate
CAS:Escitalopram Oxalate ((S)-(+)Citalopram oxalate) is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.Formula:C22H23FN2O5Purezza:97.39% - 99.73%Colore e forma:White SolidPeso molecolare:414.43Ref: TM-T6493
1g268,00€10mg37,00€25mg52,00€50mg63,00€100mg86,00€200mg118,00€500mg187,00€1mL*10mM (DMSO)42,00€Sarpogrelate hydrochloride
CAS:Sarpogrelate hydrochloride (MCI-9042), a 5-HT2 antagonist with high affinity (Ki=8.39nM), is used as an anti-platelet for PAD, improving vascular function.
Formula:C24H32ClNO6Purezza:99.73%Colore e forma:Colorless LiquidPeso molecolare:465.97Vilazodone Hydrochloride
CAS:Vilazodone Hydrochloride (EMD 68843) , a partial agonist of 5-HT1A receptors and specific serotonin reuptake inhibitor (SSRI), is utilized in treating of theFormula:C26H27N5O2·HClPurezza:99.56% - >99.99%Colore e forma:SolidPeso molecolare:477.99Naluzotan
CAS:Naluzotan(PRX 00023) is a novel and potent 5-HT1A agonist with IC50 and Ki values of approximately 20 nM and 5.1 nM, respectively.Naluzotan is a potent hERG K+Formula:C23H38N4O3SPurezza:>99.99%Colore e forma:SolidPeso molecolare:450.64Dolasetron
CAS:Dolasetron (MDL-73147)(MDL-73147) is a serotonin 5-HT3 receptor antagonist. Dolasetron is used to treat nausea and vomiting following chemotherapy.Formula:C19H20N2O3Purezza:99.84% - 99.86%Colore e forma:White PowderPeso molecolare:324.37AC-90179 HCl
CAS:AC-90179 HCl: selective 5-HT2A inverse agonist, atypical antipsychotic, reduces hallucinogen-induced vasoconstriction.Formula:C23H31ClN2O2Purezza:99.71%Colore e forma:SolidPeso molecolare:402.96Harmine hydrochloride
CAS:Harmine hydrochloride (telepathine hydrochloride) is extracted from Peganum Harmala Genus.Formula:C13H13ClN2OPurezza:99.61% - >99.99%Colore e forma:Yellow To Slightly Green Crystalline PowderPeso molecolare:248.71Cilansetron Hydrochloride
CAS:Cilansetron Hydrochloride can be used for irritable Bowel Syndrome (IBS) with Diarrhea Predominance.Formula:C20H24ClN3O2Colore e forma:SolidPeso molecolare:373.88Ritanserin
CAS:Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.Formula:C27H25F2N3OSPurezza:99.77% - 99.89%Colore e forma:SolidPeso molecolare:477.57Cariprazine
CAS:Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate
Formula:C21H32Cl2N4OPurezza:99.68% - 99.87%Colore e forma:SolidPeso molecolare:427.41Opiranserin hydrochloride
CAS:Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μMFormula:C21H35ClN2O5Purezza:99.33%Colore e forma:SolidPeso molecolare:430.97Ref: TM-T9833
1mg90,00€5mg215,00€10mg340,00€25mg618,00€50mg879,00€100mg1.224,00€500mg2.457,00€1mL*10mM (DMSO)236,00€Eltoprazine dihydrochloride
CAS:Eltoprazine dihydrochloride, a drug developed for aggression, is now studied for L-DOPA-induced dyskinesia in Parkinson's.Formula:C12H18Cl2N2O2Purezza:99.64%Colore e forma:SolidPeso molecolare:293.19NAN-190 hydrobromide
CAS:NAN-190 hydrobromide is an antagonist of serotonin receptor 5-HT.
Formula:C23H28BrN3O3Purezza:95.20%Colore e forma:SolidPeso molecolare:474.39Pardoprunox hydrochloride
CAS:Pardoprunox hydrochloride (SLV-308 hydrochloride) is a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist, D2 (pKi = 8.1)Formula:C12H16ClN3O2Purezza:98.95% - 99.13%Colore e forma:SolidPeso molecolare:269.73Pirenperone
CAS:Pirenperone is a putative 5-HT2 receptor antagonist with the central antiserotonergic and antidopaminergic action.Formula:C23H24FN3O2Purezza:99.2%Colore e forma:SolidPeso molecolare:393.45Nefazodone hydrochloride
CAS:Nefazodone hydrochloride (Serzone) is a serotoninergic modulating antidepressant that is used in therapy of depression, aggressive behavior and panic disorder.Formula:C25H33Cl2N5O2Purezza:99% - 99.86%Colore e forma:White SolidPeso molecolare:506.47Ref: TM-T3275
5mg47,00€10mg70,00€25mg120,00€50mg216,00€100mg325,00€200mg472,00€500mg775,00€1mL*10mM (DMSO)77,00€Olanzapine HCl
CAS:Olanzapine HCl, an FDA-approved atypical antipsychotic for schizophrenia and bipolar disorder, resembles clozapine and quetiapine.Formula:C17H21ClN4SColore e forma:SolidPeso molecolare:348.89
