
recettore 5-HT
I recettori 5-HT, noti anche come recettori della serotonina, sono un gruppo di recettori accoppiati alle proteine G (GPCR) che mediano gli effetti della serotonina, un neurotrasmettitore coinvolto nella regolazione dell'umore, dell'ansia, del sonno, dell'appetito e di altri processi fisiologici. Questi recettori sono suddivisi in diversi sottotipi, ciascuno con funzioni e proprietà farmacologiche distinte. I modulatori dei recettori 5-HT sono ampiamente studiati per il loro ruolo nel trattamento della depressione, dei disturbi d'ansia e di altre condizioni neuropsichiatriche. Presso CymitQuimica, offriamo una gamma di modulatori dei recettori 5-HT di alta qualità per supportare la tua ricerca in neurofarmacologia, disturbi dell'umore e segnalazione GPCR.
Trovati 1025 prodotti di "recettore 5-HT"
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Eltoprazine dihydrochloride
CAS:Eltoprazine dihydrochloride, a drug developed for aggression, is now studied for L-DOPA-induced dyskinesia in Parkinson's.Formula:C12H18Cl2N2O2Purezza:99.64%Colore e forma:SolidPeso molecolare:293.19Indophagolin
CAS:Indophagolin: autophagy inhibitor, IC50 140 nM; blocks P2X4, P2X1, P2X3 receptors, IC50s 2.71, 2.40, 3.49 μM.Formula:C19H15BrClF3N2O3SPurezza:99.76%Colore e forma:SolidPeso molecolare:523.75Ref: TM-T8946
1mg42,00€5mg82,00€10mg116,00€25mg188,00€50mg260,00€100mg366,00€200mg497,00€1mL*10mM (DMSO)95,00€Adoprazine hydrochloride
CAS:Adoprazine hydrochloride is a dopamine D2 receptor antagonist and 5-HT1A receptor agonist potential antipsychotic drug.Formula:C24H25ClFN3O2Colore e forma:SolidPeso molecolare:441.93Nefazodone hydrochloride
CAS:Nefazodone hydrochloride (Serzone) is a serotoninergic modulating antidepressant that is used in therapy of depression, aggressive behavior and panic disorder.Formula:C25H33Cl2N5O2Purezza:99% - 99.86%Colore e forma:White SolidPeso molecolare:506.47Ref: TM-T3275
5mg47,00€10mg70,00€25mg120,00€50mg216,00€100mg325,00€200mg472,00€500mg775,00€1mL*10mM (DMSO)77,00€NLX-204 hydrochloride(2170405-10-2 free base)
NLX-204 hydrochloride is a potent and selective ERK1/2 phosphorylation-preferring serotonin 5 HT1A receptor agonist(pKi = 10.19).Formula:C20H23Cl2F2N3O2Purezza:99.59%Colore e forma:SolidPeso molecolare:446.32Idalopirdine Hydrochloride
CAS:Idalopirdine Hydrochloride (Lu AE58054 Hydrochloride) is an in-vivo binding affinity and effect, in-vitro selectivity and potency of 5-HT(6)R antagonist (Ki: 0.
Formula:C20H20ClF5N2OPurezza:99.77%Colore e forma:SolidPeso molecolare:434.83Almotriptan Malate
CAS:Almotriptan Malate (PNU180638), a selective 5-HT1B/1D receptor agonist, is used in the therapy of Migraine attacks in adults.Formula:C17H25N3O2S·C4H6O5Purezza:99.95%Colore e forma:Pale Yellow SolidPeso molecolare:469.55Anpirtoline free base
CAS:Anpirtoline: potent 5-HT1B agonist; lowers serotonin synthesis; reduces aggression; 5-HT3 antagonist; crosses blood-brain barrier.Formula:C10H13ClN2SColore e forma:SolidPeso molecolare:228.74Naratriptan
CAS:Naratriptan is a selective agonist of 5-HT1 receptor and is is used for the treatment of migraine headaches.Formula:C17H25N3O2SPurezza:99.08%Colore e forma:SolidPeso molecolare:335.47Ref: TM-T8666
1mg39,00€2mg50,00€5mg73,00€10mg92,00€25mg166,00€50mg240,00€100mg360,00€1mL*10mM (DMSO)88,00€SB 204741
CAS:SB 204741 is a selective 5-HT2B antagonist with high affinity and pKi value of 7.1.Formula:C14H14N4OSPurezza:99.83%Colore e forma:SolidPeso molecolare:286.35Ref: TM-T23312
1mg38,00€2mg50,00€5mg84,00€10mg119,00€25mg234,00€50mg439,00€100mg600,00€200mg837,00€1mL*10mM (DMSO)84,00€Serotonin hydrochloride
CAS:Serotonin hydrochloride (Serotonin HCl) is an endogenous 5-HT receptor agonist, a monoamine neurotransmitter in the CNS, and a catechol O-methyltransferase (Formula:C10H13ClN2OPurezza:98.05% - 99.93%Colore e forma:White To Cream PowderPeso molecolare:212.676Cerlapirdine hydrochloride
CAS:Cerlapirdine/SAM-531, potent 5-HT6 antagonist, targets Alzheimer's and schizophrenia cognitive issues; phase II trials, promising efficacy, safe profile.Formula:C22H24ClN3O3SColore e forma:SolidPeso molecolare:445.96Cilansetron Hydrochloride
CAS:Cilansetron Hydrochloride can be used for irritable Bowel Syndrome (IBS) with Diarrhea Predominance.Formula:C20H24ClN3O2Colore e forma:SolidPeso molecolare:373.88Naratriptan hydrochloride
CAS:Naratriptan Hydrochloride, a selective 5-HT1 receptor agonist with anti-migraine effect, induces vasoconstriction and reduces inflammation in migraines.Formula:C17H25N3O2S·HClPurezza:99.17% - 99.93%Colore e forma:Beige SolidPeso molecolare:371.93Rizatriptan sulfate
CAS:Rizatriptan sulfate is a selective serotonin 5-HTID receptor agonist derived from tryptamine.Formula:C15H21N5O4SColore e forma:SolidPeso molecolare:367.42Ralmitaront
CAS:Ralmitaront (RO6889450) is a potent, orally active partial agonist of the trace amine-associated receptor 1 (TAAR1).Formula:C17H22N4O2Purezza:99.71% - 99.79%Colore e forma:SolidPeso molecolare:314.38Ref: TM-T9183
1mg105,00€5mg260,00€10mg401,00€25mg668,00€50mg897,00€100mg1.243,00€200mg1.693,00€1mL*10mM (DMSO)286,00€Mosapride Citrate
CAS:Mosapride Citrate (TAK-370 citrate), a gastroprokinetic agent, utilizes as a selective 5HT4 agonist.Formula:C21H25ClFN3O3·C6H8O7Purezza:99.70%Colore e forma:White PowderPeso molecolare:614.02Cariprazine
CAS:Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate
Formula:C21H32Cl2N4OPurezza:99.68% - 99.87%Colore e forma:SolidPeso molecolare:427.41Pipamperone HCl
CAS:Pipamperone blocks 5-HT2A/B/C, D2/D3/D4, α1/α2 receptors; favors 5-HT2A/D4 over D2; negligible affinity for H1, mACh. Highly selective at low doses.Formula:C21H31ClFN3O2Colore e forma:SolidPeso molecolare:411.95Intepirdine
CAS:Intepirdine (GSK-742457) is a highly selective 5-HT6 receptor antagonist, used in trials studying the treatment of Alzheimer's Disease.Formula:C19H19N3O2SPurezza:98% - 98.63%Colore e forma:SolidPeso molecolare:353.44
