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recettore 5-HT

recettore 5-HT

I recettori 5-HT, noti anche come recettori della serotonina, sono un gruppo di recettori accoppiati alle proteine G (GPCR) che mediano gli effetti della serotonina, un neurotrasmettitore coinvolto nella regolazione dell'umore, dell'ansia, del sonno, dell'appetito e di altri processi fisiologici. Questi recettori sono suddivisi in diversi sottotipi, ciascuno con funzioni e proprietà farmacologiche distinte. I modulatori dei recettori 5-HT sono ampiamente studiati per il loro ruolo nel trattamento della depressione, dei disturbi d'ansia e di altre condizioni neuropsichiatriche. Presso CymitQuimica, offriamo una gamma di modulatori dei recettori 5-HT di alta qualità per supportare la tua ricerca in neurofarmacologia, disturbi dell'umore e segnalazione GPCR.

Trovati 1025 prodotti di "recettore 5-HT"

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  • Xaliproden hydrochloride

    CAS:
    Xaliproden is a compound that mimics the effects of nerve growth factor and is also a serotonin 5-HT1A receptor agonist.
    Formula:C24H23ClF3N
    Purezza:99.99%
    Colore e forma:Solid
    Peso molecolare:417.89

    Ref: TM-T9272

    1mg
    38,00€
    5mg
    80,00€
    10mg
    114,00€
    25mg
    222,00€
    50mg
    356,00€
    100mg
    512,00€
    200mg
    735,00€
    1mL*10mM (DMSO)
    92,00€
  • lumateperone Tosylate

    CAS:
    lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors.
    Formula:C31H36FN3O4S
    Purezza:95.83% - 99.95%
    Colore e forma:Solid
    Peso molecolare:565.7

    Ref: TM-TQ0084

    5mg
    49,00€
    10mg
    84,00€
    25mg
    152,00€
    50mg
    219,00€
    100mg
    324,00€
    1mL*10mM (DMSO)
    62,00€
  • Cerlapirdine

    CAS:
    Cerlapirdine (PF-05212365), a 5-HT6 receptor antagonist, is in trials for Alzheimer's and schizophrenia cognition issues.
    Formula:C22H23N3O3S
    Purezza:98.77%
    Colore e forma:Solid
    Peso molecolare:409.5

    Ref: TM-T30798

    1mg
    81,00€
    5mg
    170,00€
    10mg
    274,00€
    25mg
    543,00€
    50mg
    780,00€
    100mg
    1.074,00€
    1mL*10mM (DMSO)
    198,00€
  • Cariprazine hydrochloride

    CAS:
    Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)
    Formula:C21H33Cl3N4O
    Purezza:99.78% - >99.99%
    Colore e forma:Solid
    Peso molecolare:463.87

    Ref: TM-T8382

    5mg
    34,00€
    10mg
    49,00€
    25mg
    79,00€
    50mg
    108,00€
    100mg
    161,00€
    500mg
    385,00€
  • Lerisetron

    CAS:
    Lerisetron is an antagonist of serotonin type 3 (5-HT3) receptor, with antiemetic activity.
    Formula:C18H20N4
    Purezza:99.15% - 99.82%
    Colore e forma:Solid
    Peso molecolare:292.38

    Ref: TM-T8441

    1mg
    57,00€
    5mg
    120,00€
    10mg
    178,00€
    25mg
    314,00€
    50mg
    462,00€
    100mg
    663,00€
    1mL*10mM (DMSO)
    114,00€
  • Indophagolin

    CAS:
    Indophagolin: autophagy inhibitor, IC50 140 nM; blocks P2X4, P2X1, P2X3 receptors, IC50s 2.71, 2.40, 3.49 μM.
    Formula:C19H15BrClF3N2O3S
    Purezza:99.76%
    Colore e forma:Solid
    Peso molecolare:523.75

    Ref: TM-T8946

    1mg
    42,00€
    5mg
    82,00€
    10mg
    116,00€
    25mg
    188,00€
    50mg
    260,00€
    100mg
    366,00€
    200mg
    497,00€
    1mL*10mM (DMSO)
    95,00€
  • Amperozide

    CAS:
    Amperozide (FG 5606), an atypical antipsychotic, antagonizes 5-HT2A and modulates dopamine activity for schizophrenia treatment.
    Formula:C23H29F2N3O
    Purezza:99.68%
    Colore e forma:Solid
    Peso molecolare:401.49

    Ref: TM-T23733

    1mg
    87,00€
    5mg
    178,00€
    10mg
    295,00€
    25mg
    497,00€
    50mg
    708,00€
    100mg
    964,00€
    500mg
    1.918,00€
    1mL*10mM (DMSO)
    321,00€
  • Metoclopramide hydrochloride hydrate

    CAS:
    Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) is a dopamine D2 antagonist that is a drug used for digestive dysfunction.
    Formula:C14H25Cl2N3O3
    Purezza:99.33%
    Colore e forma:Solid
    Peso molecolare:354.27

    Ref: TM-T8385

    1g
    126,00€
    50mg
    38,00€
    100mg
    52,00€
    500mg
    87,00€
  • Eltoprazine hydrochloride

    CAS:
    Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM,
    Formula:C12H17ClN2O2
    Purezza:99.35%
    Colore e forma:Solid
    Peso molecolare:256.73

    Ref: TM-T7498

    5mg
    46,00€
    10mg
    75,00€
    25mg
    137,00€
    50mg
    245,00€
    100mg
    356,00€
    500mg
    835,00€
    1mL*10mM (DMSO)
    49,00€
  • Vortioxetine hydrobromide

    CAS:
    Vortioxetine hydrobromide (Lu AA21004 hydrobromide) is a serotonin (5-HT) modulator and stimulator (SMS), inhibits 5-HT1A/1B/3A/7 receptor and SERT (IC50: 15/33
    Formula:C18H22N2S·HBr
    Purezza:98.85% - 99.98%
    Colore e forma:Solid
    Peso molecolare:379.36

    Ref: TM-T2395L

    25mg
    39,00€
    50mg
    55,00€
    100mg
    79,00€
    500mg
    198,00€
    1mL*10mM (DMSO)
    33,00€
  • Azaphen dihydrochloride monohydrate

    CAS:
    Azaphen dihydrochloride monohydrate is a 5-hydroxytryptamine reabsorption inhibitor with antidepressant activity and can be used to study neurological diseases.
    Formula:C16H23Cl2N5O2
    Purezza:99.85%
    Colore e forma:Solid
    Peso molecolare:388.29

    Ref: TM-T61741

    10mg
    42,00€
    25mg
    62,00€
    50mg
    89,00€
    100mg
    117,00€
  • RS-67333

    CAS:
    RS-67333 is a partial agonist of 5-HT4R with neuroprotective effects.
    Formula:C19H29ClN2O2
    Purezza:99.24%
    Colore e forma:Solid
    Peso molecolare:352.9

    Ref: TM-T24742

    1mg
    285,00€
    5mg
    692,00€
  • SB 243213

    CAS:
    SB 243213 is a 5-HT2C receptor antagonist with anxiolytic and antidepressant activity used in schizophrenia and movement disorders.
    Formula:C22H19F3N4O2
    Purezza:98.78% - 99.86%
    Colore e forma:Solid
    Peso molecolare:428.41

    Ref: TM-T37816

    1mg
    35,00€
    5mg
    75,00€
    10mg
    114,00€
    25mg
    260,00€
    50mg
    485,00€
    100mg
    893,00€
    1mL*10mM (DMSO)
    84,00€
  • Jatrorrhizine chloride

    CAS:
    Jatrorrhizine chloride (Neprotine chloride) is an alkaloid isolated from Rhizoma coptidis with neuroprotective, antimicrobial, and antiplasmodial activities.
    Formula:C20H20ClNO4
    Purezza:99.79%
    Colore e forma:Solid
    Peso molecolare:373.8

    Ref: TM-T4912

    5mg
    37,00€
    10mg
    56,00€
    25mg
    90,00€
    50mg
    155,00€
    100mg
    221,00€
    500mg
    525,00€
    1mL*10mM (DMSO)
    42,00€
  • Ketanserin tartrate

    CAS:
    Ketanserin tartrate (KJK-945 tartrate) is a 5-HT2A receptor and α1-adrenergic receptor antagonist for the study of systemic sclerosis.
    Formula:C26H28FN3O9
    Purezza:99.68%
    Colore e forma:Solid
    Peso molecolare:545.51

    Ref: TM-T1066L

    25mg
    34,00€
    50mg
    49,00€
    100mg
    64,00€
    1mL*10mM (DMSO)
    34,00€
  • Latrepirdine dihydrochloride

    CAS:
    Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets.
    Formula:C21H25N3·2HCl
    Purezza:98.45%
    Colore e forma:Solid
    Peso molecolare:392.37

    Ref: TM-T6562

    2mg
    34,00€
    1mL*10mM (DMSO)
    50,00€
  • LP-533401 hydrochloride

    CAS:
    LP-533401 hydrochloride is a peripheral Tph inhibitor that does not cross the BBB and can be used to study periodontal disease and hepatic steatosis.
    Formula:C27H23ClF4N4O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:562.94

    Ref: TM-T15779

    1mg
    38,00€
    5mg
    84,00€
    10mg
    114,00€
    25mg
    Prezzo su richiesta
    1mL*10mM (DMSO)
    92,00€
  • Rizatriptan

    CAS:
    Rizatriptan (Risatriptan) is a selective 5-hydroxytryptamine 1B/1D receptor agonist used in the study of migraine.
    Formula:C15H19N5
    Purezza:99.74%
    Colore e forma:Solid
    Peso molecolare:269.35

    Ref: TM-T1734L

    5mg
    34,00€
    10mg
    46,00€
    25mg
    65,00€
    50mg
    94,00€
    100mg
    126,00€
  • Setiptiline

    CAS:
    Setiptiline (Org-8282) is a norepinephrine reuptake inhibitor, 2-adrenergic receptor antagonist, H1 receptor inverse agonist with antidepressant activity.
    Formula:C19H19N
    Purezza:98.05% - 98.07%
    Colore e forma:Solid
    Peso molecolare:261.36

    Ref: TM-T12900

    5mg
    33,00€
    1mL*10mM (DMSO)
    60,00€
  • Citalopram

    CAS:
    Citalopram (Lu 10-171), a serotonin and 5-HT reuptake inhibitor.Citalopram has antidepressant activity and may be used to study dementia.
    Formula:C20H21FN2O
    Purezza:99.78% - 99.89%
    Colore e forma:Solid
    Peso molecolare:324.39

    Ref: TM-T20828

    25mg
    35,00€
    50mg
    48,00€
    100mg
    70,00€
    500mg
    150,00€
    1mL*10mM (DMSO)
    50,00€