
recettore 5-HT
I recettori 5-HT, noti anche come recettori della serotonina, sono un gruppo di recettori accoppiati alle proteine G (GPCR) che mediano gli effetti della serotonina, un neurotrasmettitore coinvolto nella regolazione dell'umore, dell'ansia, del sonno, dell'appetito e di altri processi fisiologici. Questi recettori sono suddivisi in diversi sottotipi, ciascuno con funzioni e proprietà farmacologiche distinte. I modulatori dei recettori 5-HT sono ampiamente studiati per il loro ruolo nel trattamento della depressione, dei disturbi d'ansia e di altre condizioni neuropsichiatriche. Presso CymitQuimica, offriamo una gamma di modulatori dei recettori 5-HT di alta qualità per supportare la tua ricerca in neurofarmacologia, disturbi dell'umore e segnalazione GPCR.
Trovati 1025 prodotti di "recettore 5-HT"
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(S)-Mirtazapine
CAS:(S)-Mirtazapine ((S)-Org3770) is a 5-HT2 receptor antagonist with pro-nociceptive effects that can be used to study depression.Formula:C17H19N3Purezza:99.37%Colore e forma:SolidPeso molecolare:265.35Rotigotine
CAS:Rotigotine (1-Naphthalenol, 5,6,7,8-tetrahydro-6-[propyl[2-(2-thienyl)ethyl]amino]-) is an antiparkinson agent and dopamine receptor agonist.Formula:C19H25NOSPurezza:99.04% - 99.88%Colore e forma:SolidPeso molecolare:315.47Tandospirone
CAS:Tandospirone (SM-3997) is a 5-HT1A receptor partial agonist with anxiolytic and antidepressant activity used in the study of central nervous system disorders.Formula:C21H29N5O2Purezza:99.94%Colore e forma:SolidPeso molecolare:383.49Ref: TM-TQ0315
2mg34,00€5mg50,00€10mg80,00€25mg130,00€50mg178,00€100mg284,00€200mg408,00€1mL*10mM (DMSO)55,00€Renzapride
CAS:Renzapride (BRL 24924) is a mixed 5-hydroxytryptamine type 4 (5-HT4) agonist and 5-HT3 receptor antagonist used in the study of irritable bowel syndrome.Formula:C16H22ClN3O2Purezza:98.97% - 99.09%Colore e forma:SolidPeso molecolare:323.82Ref: TM-T38507
1mg93,00€2mg124,00€5mg200,00€10mg359,00€25mg692,00€50mg945,00€100mg1.279,00€200mg1.701,00€WAY-100635 maleate
CAS:WAY-100635 Maleate is a specific and effective 5-HT receptor antagonist (IC50=0.95 nM).Formula:C25H34N4O2·xC4H4O4Purezza:99.96%Colore e forma:White SolidPeso molecolare:538.645Ref: TM-T3453
2mg46,00€5mg66,00€10mg95,00€25mg159,00€50mg226,00€100mg334,00€500mg807,00€1mL*10mM (DMSO)79,00€(R)-Mirtazapine
CAS:(R)-Mirtazapine ((R)-Org3770) is a 5-HT3 receptor antagonist, a potential analgesic with anti-injury perception properties.Formula:C17H19N3Purezza:99.75%Colore e forma:SolidPeso molecolare:265.35S1RA
CAS:S1RA (E-52862)(E-52862) is a potent, selective antagonist of the sigma-1 receptor (σ1R, Ki=17 nM), demonstrating significant selectivity over the sigma-2Formula:C20H23N3O2Purezza:99.45%Colore e forma:SolidPeso molecolare:337.42Syk Inhibitor II
CAS:Syk inhibitor II, a cell-permeable, ATP-competitive, pyrimidine-carboxamide compound, selectively and reversibly inhibits Syk (IC50 = 41 nM).Formula:C14H15F3N6OPurezza:97.63%Colore e forma:SolidPeso molecolare:340.3R 59-022
CAS:R 59-022 (DKGI-I) is a DGK inhibitor and a 5-HT Receptor antagonist that blocks filovirus internalization in host cells.Formula:C27H26FN3OSPurezza:98.55%Colore e forma:SolidPeso molecolare:459.58Ref: TM-T16709
1mg35,00€5mg74,00€10mg119,00€25mg269,00€50mg447,00€100mg733,00€200mg973,00€1mL*10mM (DMSO)75,00€Cyproheptadine hydrochloride
CAS:Cyproheptadine hydrochloride (Periactin hydrochloride) is a hydrochloride salt form of cyproheptadine which is a histamine receptor antagonist.
Formula:C21H21N·HClPurezza:99.88% - 99.97%Colore e forma:SolidPeso molecolare:323.86Escitalopram
CAS:Escitalopram (Seroplex), a serotonin inhibitor for depression, curbs alcohol intake and is favored over tricyclics for tardive dyskinesia.Formula:C20H21FN2OPurezza:99.82%Colore e forma:White Or White Crystalline PowderPeso molecolare:324.39Risperidone Mesylate
CAS:Risperidone Mesylate is a selective serotonin 5-HT2 receptor and dopamine D2 receptor blocker.Formula:C24H31FN4O5SPurezza:98%Colore e forma:SolidPeso molecolare:506.59N-Methyl amisulpride
CAS:N-Methyl amisulpride (Amisulpride impurity H) is a 5-HT7 receptor, D2 receptor, and D3 receptor antagonist used in the study of acute schizophrenia.Formula:C18H29N3O4SColore e forma:SolidPeso molecolare:383.51Keto Ziprasidone
CAS:Ziprasidone, an antipsychotic agent, functions as a dual antagonist of 5-HT (serotonin) and dopamine receptors.Formula:C21H19ClN4O2SPurezza:98%Colore e forma:SolidPeso molecolare:426.92Arazasetron HCl
CAS:Arazasetron is an antiemetic which acts as a 5-HT3 receptor antagonist, pKi = 9.27.Formula:C17H20ClN3O3Purezza:98%Colore e forma:SolidPeso molecolare:349.81Mirtazapine D3
CAS:Mirtazapine D3 is a deuterium labeled Mirtazapine. Mirtazapine is an inhibitor of 5-HT receptor .Formula:C17H19N3Purezza:98%Colore e forma:SolidPeso molecolare:268.37Brexpiprazole-d8
CAS:Brexpiprazole D8 is a deuterium-modified partial agonist of 5-HT1A and dopamine receptors, with Ki values of 0.12 nM and 0.3 nM respectively.Formula:C25H27N3O2SPurezza:98%Colore e forma:SolidPeso molecolare:441.62Amitriptyline-d6 Hydrochloride
CAS:Amitriptyline-d6 Hydrochloride is a deuterated compound of Amitriptyline Hydrochloride. Amitriptyline Hydrochloride has a CAS number of 549-18-8. Amitriptyline Hydrochloride is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptive activities.Formula:C20H18D6ClNColore e forma:SolidPeso molecolare:319.90Pardoprunox
CAS:Pardoprunox (SLV-308) is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties.Formula:C12H15N3O2Purezza:98%Colore e forma:SolidPeso molecolare:233.275-Methyltryptamine hydrochloride
CAS:5-Methyltryptamine hydrochloride is a high-affinity 5-HT1C receptor ligand and a partial agonist of 5-HT. 5-Methyltryptamine hydrochloride protects mice subjected to burn, tourniquet and endotoxin shock.Formula:C11H15ClN2Purezza:99.45%Colore e forma:SolidPeso molecolare:210.703
