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Beta amiloide

Beta amiloide

Gli inibitori del beta-amiloide sono composti che mirano specificamente a inibire la formazione o l'aggregazione dei peptidi beta-amiloidi, coinvolti in modo critico nella patogenesi della malattia di Alzheimer. L'accumulo di placche di beta-amiloide nel cervello è uno dei tratti patologici distintivi della malattia, contribuendo alla disfunzione neuronale e al declino cognitivo. Inibendo l'aggregazione del beta-amiloide, questi inibitori sono studiati come potenziali agenti terapeutici per rallentare o prevenire la progressione della malattia di Alzheimer. Presso CymitQuimica, offriamo una gamma di inibitori del beta-amiloide di alta qualità per supportare la tua ricerca nella neurodegenerazione, nell'aggregazione proteica e nella terapia dell'Alzheimer.

Trovati 218 prodotti di "Beta amiloide"

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  • AZD4694

    CAS:
    Flutafuranol (AZD4694/NAV4694) binds beta-amyloid, potential PET tracer for Alzheimer's. Non-F18 version supplied.
    Formula:C14H11FN2O2
    Colore e forma:Solid
    Peso molecolare:258.25
  • (Rac)-Z-Phe-Phe-FMK

    CAS:
    (Rac)-Z-Phe-Phe-FMK (Cathepsin L-IN-2) is a cathepsin L inhibitor that inhibits the tendency of β-amyloid to induce apoptotic changes .
    Formula:C27H27FN2O4
    Purezza:98.27%
    Colore e forma:Solid
    Peso molecolare:462.51
  • Cu(II)GTSM

    CAS:
    Cu(II)GTSM is a cell permeable copper complex inhibits GSK3β activity and suppresses levels of neurotoxic amyloid β-trimers and phosphorylated tau.
    Formula:C6H10CuN6S2
    Purezza:99.21%
    Colore e forma:Solid
    Peso molecolare:293.86
  • JLK6

    CAS:
    JLK6 was a gamma-secretase inhibitor that does not interfere with Notch signalling
    Formula:C10H8ClNO3
    Purezza:96.50%
    Colore e forma:Solid
    Peso molecolare:225.63
  • EUK-134

    CAS:
    EUK-134, a synthetic SOD/catalase mimetic, exhibits potent antioxidant activities, and inhibits the formation of β-amyloid and related amyloid fibril.
    Formula:C18H18ClMnN2O4
    Purezza:98.39%
    Colore e forma:Solid
    Peso molecolare:416.74
  • Dihydroergocristine mesylate

    CAS:
    DHEC mesylate is a vasodilator and α-adrenergic antagonist used for vascular dementia and as a geroprotector.
    Formula:C36H45N5O8S
    Purezza:98.9% - 99.79%
    Colore e forma:Solid
    Peso molecolare:707.84
  • PBD-150

    CAS:
    PBD-150 is an inhibitor of human glutaminyl cyclase (hQC) Y115E-Y117E variant( ki : 490 nM)
    Formula:C15H20N4O2S
    Purezza:99.68%
    Colore e forma:Solid
    Peso molecolare:320.41
  • ARN2966

    CAS:
    ARN2966 is an inhibitor of amyloid precursor protein (APP)and amyloid-β (Aβ) secretion.
    Formula:C12H12N2O
    Purezza:99.52% - 99.86%
    Colore e forma:Solid
    Peso molecolare:200.24
  • Cromoglicic acid

    CAS:
    <p>Cromoglicic acid prevents the release of inflammatory chemicals such as histamine from mast cells.</p>
    Formula:C23H16O11
    Purezza:99.55% - >99.99%
    Colore e forma:Colorless Crystals From Ethanol + Ether Physical Description Solid (Ntp 1992)
    Peso molecolare:468.37
  • Benzenesulfonamide

    CAS:
    Benzenesulfonamide (Benzosulfonamide) ia an inhibitor of carbonic anhydrases.
    Formula:C6H7NO2S
    Purezza:99.42% - 99.99%
    Colore e forma:White Crystalline Powder
    Peso molecolare:157.19
  • CRANAD 2

    CAS:
    CRANAD-2, a near-infrared probe, detects amyloid-beta in vivo, increasing fluorescence 70x and shifting blue 90 nm upon binding.
    Formula:C23H25BF2N2O2
    Purezza:99.44%
    Colore e forma:Dark Blue To Black Powder
    Peso molecolare:410.27
  • Anle138b

    CAS:
    Anle138b: a novel oligomer modulator for disease-modifying therapy of neurodegenerative diseases such as prion and Parkinson's disease
    Formula:C16H11BrN2O2
    Purezza:98.88% - 99.82%
    Colore e forma:Solid
    Peso molecolare:343.17
  • PE859

    CAS:
    PE859 is a potent inhibitor of both tau and Aβ aggregation.
    Formula:C28H24N4O2
    Purezza:98.8% - 99.09%
    Colore e forma:Solid
    Peso molecolare:448.52
  • 1,1'-Methylenedi-2-naphthol

    CAS:
    <p>1,1'-Methylenedi-2-naphthol target CYP2C19 - cytochrome P450 family 2 subfamily C member 19 (human).</p>
    Formula:C21H16O2
    Purezza:98.91%
    Colore e forma:Light Pink To Light Brown Crystalline Powder
    Peso molecolare:300.35
  • MK-0752

    CAS:
    <p>MK-0752, a γ-secretase inhibitor, reduces Aβ40 production(IC50=5 nM).</p>
    Formula:C21H21ClF2O4S
    Purezza:98% - 99.55%
    Colore e forma:Solid
    Peso molecolare:442.9
  • TAE-1

    CAS:
    <p>TAE-1 is an inhibitor of amyloid-β fibril formation and aggregation. It inhibits cholinesterases AChE and BuChE with IC50 of 0.3 μM and 3.9 μM, respectively.</p>
    Formula:C39H51I3N6O9
    Purezza:94.58%
    Colore e forma:Solid
    Peso molecolare:1128.57
  • RO4929097

    CAS:
    <p>RO4929097 (RG-4733), a γ secretase inhibitor (IC50: 4 nM), inhibits cellular processing of Aβ40 and Notch (EC50: 14/5 nM).</p>
    Formula:C22H20F5N3O3
    Purezza:98.5% - 99.51%
    Colore e forma:Solid
    Peso molecolare:469.4
  • Frentizole

    CAS:
    Frentizole, an immunosuppressive agent, is an inhibitor of the Aβ-ABAD interaction
    Formula:C15H13N3O2S
    Purezza:99.82%
    Colore e forma:Solid
    Peso molecolare:299.35
  • Azeliragon

    CAS:
    Azeliragon (TTP488) is an antagonist at the Receptor for Advanced Glycation End products; is evaluated as a potential treatment for patients with mild-to-
    Formula:C32H38ClN3O2
    Purezza:96.7% - 98.33%
    Colore e forma:Solid
    Peso molecolare:532.12
  • Semax acetate(80714-61-0 free base)

    CAS:
    Semax acetate is a synthetic peptide analog of adrenocorticotropic hormone (ACTH) that has neuroprotective, analgesic, and anxiolytic properties.
    Formula:C39H55N9O12S
    Purezza:99.46%
    Colore e forma:Solid
    Peso molecolare:873.98